거대분자를 포함하는 세포투과성 펩티드가 도입된 약물전달담체
    41.
    发明公开
    거대분자를 포함하는 세포투과성 펩티드가 도입된 약물전달담체 审中-实审
    细胞穿刺肽介绍包含大分子的药物递送载体

    公开(公告)号:KR1020160044408A

    公开(公告)日:2016-04-25

    申请号:KR1020150130127

    申请日:2015-09-15

    Abstract: 본명세서는세포투과펩티드인 AP-GRR 펩티드(서열번호 1) 또는상기펩티드를포함하는펩티드사슬과공유결합되거나상기펩티드를포함하는펩티드사슬로변형된지질구조체또는고분자입자를포함하는약물전달담체에관한것이다. 또한, 본명세서는약물전달담체와그 담체내부에포집된생리활성성분을포함하는조성물에관한것이다. 본명세서의약물전달담체의경우세포내로투입이어려운거대분자들을생체의세포내로효과적으로전달하여거대분자들의생체이용률을높일수 있다.

    Abstract translation: 本发明涉及包含聚合物颗粒或脂质结构的药物递送载体,所述聚合物颗粒或脂质结构与AP-GRR肽(SEQ ID NO:1)共价结合,作为细胞穿透肽或包含肽的肽链,或修饰为 包括肽的肽链。 此外,本发明涉及包含药物递送载体和收集在载体内部的生理活性成分的组合物。 在本发明的药物递送载体的情况下,通过将难以插入细胞内的大分子有效地输送到活体的细胞中,可以提高大分子的生物利用度。

    피부 미백용 물질을 스크리닝하는 방법
    44.
    发明公开
    피부 미백용 물질을 스크리닝하는 방법 审中-实审
    用于筛选皮肤白色材料的方法

    公开(公告)号:KR1020140064272A

    公开(公告)日:2014-05-28

    申请号:KR1020120131433

    申请日:2012-11-20

    CPC classification number: G01N33/5308 C12Q1/6851 G01N33/15 G01N33/5008

    Abstract: The present invention relates to a method for screening effective substances related to skin-whitening, and more specifically, to a method which checks reduction of PGE_2 (prostaglandin E_2) generation related to melanin production and movement through measurement of a TRPM8 gene expression amount and screens substances effective to skin-whitening using the same.

    Abstract translation: 本发明涉及一种筛选与皮肤美白相关的有效物质的方法,更具体地说,涉及通过测定TRPM8基因表达量和筛选来检查与黑色素产生和运动相关的PGE_2(前列腺素E_2)生成减少的方法 使用该物质对皮肤美白有效的物质。

    비타민 B군 및 피리미딘옥사이드 유도체를 함유하는 모발성장 촉진용 조성물
    46.
    发明公开
    비타민 B군 및 피리미딘옥사이드 유도체를 함유하는 모발성장 촉진용 조성물 有权
    含有维生素B和氧化吡啶衍生物的头发生长材料的组合物

    公开(公告)号:KR1020070065950A

    公开(公告)日:2007-06-27

    申请号:KR1020050113387

    申请日:2005-11-25

    CPC classification number: A61Q7/00 A61K8/4953 A61K8/673 A61K2800/59

    Abstract: A composition comprising a vitamin B and pyrimidine oxide is provided to prevent hair loss and promote hair growth due to potassium channel opening effect of the active ingredients. The composition for promoting hair growth and preventing hair loss comprises 0.00001-5 wt.% of a water-soluble vitamin selected from the group consisting of vitamin B1(thiamine), vitamin B2(riboflavin), vitamin B6(pyridoxine), vitamin B12(cyanocobalamine), vitamin B9(folic acid) and biotin, and a pyrimidine oxide derivative which has at least one pyrimidine derivative represented by the formula(2) and is in the form of an acid addition salt. In the formula(2), R1 is a group represented by the formula(3) of NR3R4, and R2 is lower alkoxy, lower alkyl, alkenyl, alkoxyalkyl, cycloalkyl, aryl, alkylaryl, arylalkyl, alkylarylalkyl, alkoxyarylalkyl or haloarylalkyl. In the formula(3), each R3 and R4 is independently H, lower alkyl, alkenyl, alkylaryl or cycloalkyl, or R3 and R4 together with a nitrogen atom coupled thereto form a hetero-cycle such as aziridinyl, azetidinyl, pyrrolidinyl, piperidino, hexahydrozepinyl, heptamethylenimino, octamethylenimino, morpholine and 4-(lower alkyl)piperazinyl group(wherein the hetero-cycle is substituted or unsubstituted by 1-3 lower alkyl, hydroxy or alkoxy). The composition is in the form of hair-tonic, scalp treatment, hair shampoo, hair cream, general ointment, skin, lotion, eye cream, nutritive cream, massage cream, cleansing cream, cleansing foam or powder.

    Abstract translation: 提供了包含维生素B和嘧啶氧化物的组合物,以防止由于活性成分的钾通道开放作用引起的脱发和促进毛发生长。 用于促进毛发生长和防止脱发的组合物包含0.00001-5重量%的选自维生素B1(硫胺素),维生素B2(核黄素),维生素B6(吡哆醇)),维生素B12(维生素B 2 氰钴胺),维生素B9(叶酸)和生物素,以及具有至少一个式(2)所示的嘧啶衍生物并且为酸加成盐形式的嘧啶氧化物衍生物。 式(2)中,R 1为NR 3 R 4式(3)所示的基团,R 2为低级烷氧基,低级烷基,烯基,烷氧基烷基,环烷基,芳基,烷基芳基,芳基烷基,烷基芳基烷基,烷氧基芳基烷基或卤代芳基烷基。 在式(3)中,R 3和R 4各自独立地为H,低级烷基,烯基,烷基芳基或环烷基,或者R 3和R 4与与其偶联的氮原子一起形成杂环,例如氮杂环丙烷基,氮杂环丁烷基,吡咯烷基,哌啶子基, 六氢吖庚因,七亚甲基亚氨基,八亚甲基亚氨基,吗啉和4-(低级烷基)哌嗪基(其中异环由1-3个低级烷基,羟基或烷氧基取代或未取代)。 组合物为头发补品,头皮治疗,洗发剂,发霜,一般软膏,皮肤,洗剂,眼霜,营养霜,按摩膏,清洁霜,清洁泡沫或粉末的形式。

    인삼 꽃 추출물을 함유하는 피부 외용제 조성물
    50.
    发明公开
    인삼 꽃 추출물을 함유하는 피부 외용제 조성물 有权
    含有人参花提取物的皮肤外用组合物

    公开(公告)号:KR1020160070732A

    公开(公告)日:2016-06-20

    申请号:KR1020160065735

    申请日:2016-05-27

    CPC classification number: A61K8/97 A61Q5/006 A61Q19/00 A61Q19/08

    Abstract: 본발명은인삼꽃 추출물의용도에관한것으로서, 상기용도는피부보호용도, 항노화, 항주름, 피부탄력개선, 미백, 피부보습, 아토피등의피부건조질환의예방및 개선, 피지조절, 항염증, 여드름등의피부트러블예방또는개선, 각질제거, 피부혈색개선, 탈모예방, 항비듬, 모발의광택및 부드러움개선, 얼굴또는바디의볼륨및 탄력증진, 얼굴또는바디의라인개선을포함한다.

    Abstract translation: 本发明涉及使用人参花提取物,使用该皮肤保护的目的,抗老化,抗皱纹,改善皮肤弹性,美白,皮肤保湿,预防和改善,皮肤干燥性疾病如特应性皮炎,抗炎的皮脂控制的 例如痤疮和皮肤问题,包括预防或改善,去角质,皮肤肤色的改善,防止损失,抗头皮屑,光泽性和柔软性的改善,面部或的体积和弹性增加,脸或头发线改善的身体机构。

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