公开(公告)号：DK573883A

公开(公告)日：1984-06-15

申请号：DK573883

申请日：1983-12-13

Applicant: CIBA GEIGY AG

Inventor： STURM ELMAR ,  MEYER ALFRED

IPC: A01N43/50 ,  A01N43/653 ,  A01P3/00 ,  C07C39/00 ,  C07C45/63 ,  C07C45/71 ,  C07D233/60 ,  C07D233/64 ,  C07D249/08 ,  C07D303/08 ,  C07D303/22 ,  C07D303/34 ,  C07D521/00 ,  C07D ,  A01N

Abstract: 1-Azolyl-2-aryl-3-fluoro-alkan-2- ols of the general formula I in which Az is 1H-1,2,4-triazole, 4H-1,2,4-triazole or 1H-imidazole; Ar is an unsubstituted or substituted aromatic radical from the series comprising phenyl, biphenyl, phenoxyphenyl and naphthyl; R1 is hydrogen, C1-C4-alkyl, C3-C5-alkenyl or benzyl; R2 is hydrogen, fluorine or C1-C6-alkyl and R3 is hydrogen, fluorine, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy, C1-C6-alkylthio, phenyl, phenoxy, phenylthio or C3-C7-cycloalkyl, and each aromatic substituent or aromatic moiety of a substituent is unsubstituted or mono- or poly-substituted by halogen, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, nitro and/or cyano; including the acid addition salts, quaternary azolium salts and metal complexes, are useful for controlling phytopathogenic microorganisms.

公开(公告)号：DK573883D0

公开(公告)日：1983-12-13

申请号：DK573883

申请日：1983-12-13

Applicant: CIBA GEIGY AG

Inventor： STURM ELMAR ,  MEYER ALFRED

IPC: A01N43/50 ,  A01N43/653 ,  A01P3/00 ,  C07C39/00 ,  C07C45/63 ,  C07C45/71 ,  C07D233/60 ,  C07D233/64 ,  C07D249/08 ,  C07D303/08 ,  C07D303/22 ,  C07D303/34 ,  C07D521/00 ,  C07D249

Abstract: 1-Azolyl-2-aryl-3-fluoro-alkan-2- ols of the general formula I in which Az is 1H-1,2,4-triazole, 4H-1,2,4-triazole or 1H-imidazole; Ar is an unsubstituted or substituted aromatic radical from the series comprising phenyl, biphenyl, phenoxyphenyl and naphthyl; R1 is hydrogen, C1-C4-alkyl, C3-C5-alkenyl or benzyl; R2 is hydrogen, fluorine or C1-C6-alkyl and R3 is hydrogen, fluorine, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy, C1-C6-alkylthio, phenyl, phenoxy, phenylthio or C3-C7-cycloalkyl, and each aromatic substituent or aromatic moiety of a substituent is unsubstituted or mono- or poly-substituted by halogen, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, nitro and/or cyano; including the acid addition salts, quaternary azolium salts and metal complexes, are useful for controlling phytopathogenic microorganisms.

公开(公告)号：FI834522A0

公开(公告)日：1983-12-09

申请号：FI834522

申请日：1983-12-09

Applicant: CIBA GEIGY AG

Inventor： STURM ELMAR ,  MEYER ALFRED

IPC: A01N43/50 ,  A01N43/653 ,  A01P3/00 ,  C07C39/00 ,  C07C45/63 ,  C07C45/71 ,  C07D233/60 ,  C07D233/64 ,  C07D249/08 ,  C07D303/08 ,  C07D303/22 ,  C07D303/34 ,  C07D521/00 ,  C07D

Abstract: 1-Azolyl-2-aryl-3-fluoro-alkan-2- ols of the general formula I in which Az is 1H-1,2,4-triazole, 4H-1,2,4-triazole or 1H-imidazole; Ar is an unsubstituted or substituted aromatic radical from the series comprising phenyl, biphenyl, phenoxyphenyl and naphthyl; R1 is hydrogen, C1-C4-alkyl, C3-C5-alkenyl or benzyl; R2 is hydrogen, fluorine or C1-C6-alkyl and R3 is hydrogen, fluorine, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy, C1-C6-alkylthio, phenyl, phenoxy, phenylthio or C3-C7-cycloalkyl, and each aromatic substituent or aromatic moiety of a substituent is unsubstituted or mono- or poly-substituted by halogen, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, nitro and/or cyano; including the acid addition salts, quaternary azolium salts and metal complexes, are useful for controlling phytopathogenic microorganisms.

公开(公告)号：HU181860B

公开(公告)日：1983-11-28

申请号：HUCI001823

申请日：1978-04-11

Applicant: CIBA GEIGY AG

Inventor： AUFDERHAAR ERNST ,  GALLAY JEAN J ,  KUEHNE MANFRED ,  MEYER ALFRED ,  RECHSTEINER OSWALD ,  SCHELLENBAUM MAX ,  FUMEAUX JEAN-PAUL

IPC: A01N43/52 ,  A61K31/415 ,  A61K31/4184 ,  A61P33/00 ,  C07D235/28

Abstract: Benzimidazole derivatives of the formula in which R and R1 independently of one another are each hydrogen, an alkanoyl group having 1 to 4 carbon atoms, an alkoxycarbonyl group having 1 to 4 carbon atoms, an alkylsulphonyl group having 1 to 4 carbon atoms, a benzoyl group, a phenylsulphonyl group or a p-methylphenylsulphonyl group; R2 and R4 independently of one another are each hydrogen, halogen or a methyl group, R3 is hydrogen, halogen, a methyl group or a methoxy group; X is oxygen or sulphur; Y is halogen, an alkyl group having 1 to 4 carbon atoms, an alkoxy group having 1 to 4 carbon atoms, a methylthio group, a methylsulphinyl group, a methylsulphonyl group, a trifluoromethyl group, a nitro group, a hydroxyl group, a cyano group or an acetyl group; and m is 0, 1, 2 or 3; and if one of the two radicals R or R1 is hydrogen, the position of the other of these radicals on the N atoms cannot be clearly established, including, when at least one of the two radicals R or R1 is hydrogen, the possible tautomeric compounds of the formula I; and the disulphides obtainable by oxidation of compounds of the formula I. The compounds are useful for combating helminths in domestic animals and productive animals.

公开(公告)号：GB2103210A

公开(公告)日：1983-02-16

申请号：GB8218714

申请日：1982-06-29

Applicant: CIBA GEIGY AG

Inventor： NYFELER ROBERT ,  MEYER ALFRED ,  STURM ELMAR ,  MULLER URS

IPC: A01N43/50 ,  A01N43/653 ,  C07D303/22 ,  C07D303/34 ,  C07D521/00 ,  C07D249/08 ,  C07D233/60

Abstract: Novel 2-hydroxy-3-azolylpropane derivatives of the general formula I wherein R1 is an azolyl group, R2 is C1-C4alkyl or an aryl group which is unsubstituted or substituted by halogen, cyano, C1-C3alkyl, C1-C3alkoxy, nitro, thiocyano, C1-C3alkylthio and/or C1-C3haloalkyl, R3 and R4, each independently of the other, are hydrogen or C1-C4alkyl, R5 is an unsubstituted or mono- or polysubstituted radical selected from C1-C8alkyl, C3-C8cycloalkyl, C3-C6alkenyl, C3-C6alkynyl and aralkyl, said substituents being selected from the group consisting of halogen, cyano, C1-C3alkyl, C1-C5alkoxy, C1-C5haloalkoxy, C1-C3alkylthio, C1-C3haloalkyl, C1-C3haloalkylthio, nitro and/or thiocyano; and X is oxygen or sulfur, and the acid addition salts, quaternary azolium salts and metal complexes thereof, are useful in controlling phytopathogenic microorganisms and/or of regulating plant growth.

公开(公告)号：BR8201264A

公开(公告)日：1983-01-18

申请号：BR8201264

申请日：1982-03-09

Applicant: CIBA GEIGY AG

Inventor： KUNZ WALTER ,  NYFELER ROBERT ,  MEYER ALFRED ,  FRICK WILLY ,  MAIER LUDWIG ,  STURM ELMAR

IPC: C07D249/08 ,  C07D521/00 ,  C07F9/6518 ,  C07D233/56 ,  A01N43/50 ,  A01N43/64 ,  C07D401/06 ,  C07D409/06

公开(公告)号：DK422582A

公开(公告)日：1983-01-03

申请号：DK422582

申请日：1982-09-22

Applicant: CIBA GEIGY AG

Inventor： MEYER ALFRED ,  NYFELER ROBERT ,  STURM ELMAR ,  MUELLER URS

IPC: C07D20060101 ,  C07D

公开(公告)号：CA1105034A

公开(公告)日：1981-07-14

申请号：CA300973

申请日：1978-04-12

Applicant: CIBA GEIGY AG

Inventor： GALLAY JEAN J ,  KUEHNE MANFRED ,  MEYER ALFRED ,  RECHSTEINER OSWALD ,  SCHELLENBAUM MAX

IPC: A61K31/415 ,  A61K31/4184 ,  A61P33/00 ,  A61P33/10 ,  C07D235/28

Abstract: Benzimidazole derivatives of the formula in which R is an alkyl group having 1 to 6 carbon atoms, an alkenyl group having 3 to 5 carbon atoms, an alkynyl group having 3 to 5 carbon atoms or a benzyl group, which is unsubstituted monosubstituted to disubstituted by a methyl group, halogen or a nitro group, R1 is hydrogen, an alkanoyl group having 1 to 4 carbon atoms, an alkoxycarbonyl group having 1 to 4 carbon atoms, a N,N-dialkylcarbamoyl group or N,N-dialkyl-thiocarbamoyl group, each having 1 to 4 carbon atoms in the alkyl groups, an alkylsulphonyl group having 1 to 4 carbon atoms, a benzoyl group, a a phenylsulphonyl group, a 4-methylphenyl-sulphonyl group or the radical, in which Q is a carbonyl group, a thiocarbonyl group or an oxalyl group, R2 is hydrogen, halogen or a methyl group, R3 is hydrogen, halogen, a methyl group or an alkoxy group having 1 to 4 carbon atoms, R4 is hydrogen, halogen or a methyl group, X is oxygen or sulphur, Y is halogen, an alkyl group having 1 to 4 carbon atoms, an alkoxy group having 1 to 4 carbon atoms, a methylthio group, a methylsulphinyl group, a methylsulphonyl group, a trifluoromethyl group, a nitro group, a hydroxyl group, a cyano group or an alkanoyl group having 1 to 4 carbon atoms in the alkyl moiety and m is 0, 1, 2 or 3 and n is 0, 1 or 2, including, if R1 is not hydrogen, the tautomeric compounds of the formula I, for combating helminths in domestic and useful animals. - 1a

公开(公告)号：AU3502278A

公开(公告)日：1979-10-18

申请号：AU3502278

申请日：1978-04-12

Applicant: CIBA GEIGY AG

Inventor： GALLAY JEAN JACQUES ,  SCHELLENBAUM MAX ,  KUHNE MANFRED ,  MEYER ALFRED ,  RECHSTEINER OSWALD

IPC: A61K31/415 ,  A61K31/4184 ,  A61P33/00 ,  A61P33/10 ,  C07D235/28

Abstract: Benzimidazole derivatives of the formula in which R is an alkyl group having 1 to 6 carbon atoms, an alkenyl group having 3 to 5 carbon atoms, an alkynyl group having 3 to 5 carbon atoms or a benzyl group, which is unsubstituted or monosubstituted to disubstituted by a methyl group, halogen or a nitro group; R1 is hydrogen, an alkanoyl group having 1 to 4 carbon atoms, an alkoxycarbonyl group having 1 to 4 carbon atoms, a N,N-dialkylcarbamoyl group or N,N-dialkylthiocarbamoyl group, each having 1 to 4 carbon atoms in the alkyl groups, an alkylsulphonyl group having 1 to 4 carbon atoms, a benzoyl group, a phenylsulphonyl group, a 4-methylphenylsulphonyl group or the radical, in which Q is a carbonyl group, a thiocarbonyl group or an oxalyl group; R2 is hydrogen, halogen or a methyl group; R3 is hydrogen, halogen, a methyl group or an alkoxy group having 1 to 4 carbon atoms; R4 is hydrogen, halogen or a methyl group; X is oxygen or sulphur; Y is halogen, an alkyl group having 1 to 4 carbon atoms, an alkoxy group having 1 to 4 carbon atoms, a methylthio group, a methylsulphinyl group, a methylsulphonyl group, a trifluoromethyl group, a nitro group, a hydroxyl group, a cyano group or an alkanoyl group having 1 to 4 carbon atoms in the alkyl moiety m is 0, 1, 2 or 3; and n is 0, 1 or 2. Included are, if R1 is not hydrogen, the tautomeric compounds of the formula I. The compounds are effective for combating helminths in domestic and useful animals.

公开(公告)号：BG48681A3

公开(公告)日：1991-04-15

申请号：BG6333283

申请日：1983-12-06

Applicant: CIBA GEIGY AG

Inventor： STURM ELMAR ,  MEYER ALFRED

IPC: A01N43/50 ,  A01N43/653 ,  A01P3/00 ,  C07C39/00 ,  C07C45/63 ,  C07C45/71 ,  C07D233/60 ,  C07D233/64 ,  C07D249/08 ,  C07D303/08 ,  C07D303/22 ,  C07D303/34 ,  C07D521/00 ,  A01N29/02

Abstract: 1-Azolyl-2-aryl-3-fluoro-alkan-2- ols of the general formula I in which Az is 1H-1,2,4-triazole, 4H-1,2,4-triazole or 1H-imidazole; Ar is an unsubstituted or substituted aromatic radical from the series comprising phenyl, biphenyl, phenoxyphenyl and naphthyl; R1 is hydrogen, C1-C4-alkyl, C3-C5-alkenyl or benzyl; R2 is hydrogen, fluorine or C1-C6-alkyl and R3 is hydrogen, fluorine, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy, C1-C6-alkylthio, phenyl, phenoxy, phenylthio or C3-C7-cycloalkyl, and each aromatic substituent or aromatic moiety of a substituent is unsubstituted or mono- or poly-substituted by halogen, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, nitro and/or cyano; including the acid addition salts, quaternary azolium salts and metal complexes, are useful for controlling phytopathogenic microorganisms.