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公开(公告)号:BG48681A3
公开(公告)日:1991-04-15
申请号:BG6333283
申请日:1983-12-06
Applicant: CIBA GEIGY AG
Inventor: STURM ELMAR , MEYER ALFRED
IPC: A01N43/50 , A01N43/653 , A01P3/00 , C07C39/00 , C07C45/63 , C07C45/71 , C07D233/60 , C07D233/64 , C07D249/08 , C07D303/08 , C07D303/22 , C07D303/34 , C07D521/00 , A01N29/02
Abstract: 1-Azolyl-2-aryl-3-fluoro-alkan-2- ols of the general formula I in which Az is 1H-1,2,4-triazole, 4H-1,2,4-triazole or 1H-imidazole; Ar is an unsubstituted or substituted aromatic radical from the series comprising phenyl, biphenyl, phenoxyphenyl and naphthyl; R1 is hydrogen, C1-C4-alkyl, C3-C5-alkenyl or benzyl; R2 is hydrogen, fluorine or C1-C6-alkyl and R3 is hydrogen, fluorine, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy, C1-C6-alkylthio, phenyl, phenoxy, phenylthio or C3-C7-cycloalkyl, and each aromatic substituent or aromatic moiety of a substituent is unsubstituted or mono- or poly-substituted by halogen, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, nitro and/or cyano; including the acid addition salts, quaternary azolium salts and metal complexes, are useful for controlling phytopathogenic microorganisms.
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公开(公告)号:DK159093C
公开(公告)日:1991-03-11
申请号:DK380682
申请日:1982-08-25
Applicant: CIBA GEIGY AG
Inventor: FANKHAUSER ERNST , STURM ELMAR
IPC: A01N20060101 , A01N41/10 , A01N53/00 , C07C20060101 , C07C317/22
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公开(公告)号:DK159774B
公开(公告)日:1990-12-03
申请号:DK528382
申请日:1982-11-26
Applicant: CIBA GEIGY AG
Inventor: NYFELER ROBERT , MEYER ALFRED , STURM ELMAR
IPC: A01N43/50 , A01N43/64 , A01N43/653 , C07D233/60 , C07D249/08 , C07D521/00
Abstract: Novel substituted azolyl-ethyl ethers of the general formula I wherein R1 is phenyl, phenyl mono- to trisubstituted by halogen, C1-C3- haloalkyl, nitro, C1-C3-alkoxy, C1-C8-alkyl and/or cyano, or phenyl substituted by phenyl or phenoxy, naphthyl, or naphthyl mono- or -disubstituted by halogen, nitro and/or C1-C3-alkyl, benzyl, or benzyl mono- or disubstituted by halogen, nitro and/or C1-C3-alkyl; R2 is phenyl, phenyl mono- to trisubstituted by halogen, C1-C3-haloalkyl, nitro, C1-C3-alkoxy, C1-C8-alkyl and/or cyano, or phenyl substituted by phenyl or phenoxy, or it is C1-C10-alkyl, C3-C8-cycloalkyl or C3-C8- cycloalkyl-(C1-C4-alkyl); R3 is C1-C12-alkyl, C2-C4-alkenyl, C3-C4-alkynyl, benzyl, or benzyl mono- or disubstituted by halogen, nitro and/or C1-C3-alkyl; and R4 is an azolyl group; including acid addition salts thereof, quaternary azolium salts and metal complexes, are used in agrochemical compositions for the preventive and curative combating of harmful microorganisms.
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公开(公告)号:CA1271753A
公开(公告)日:1990-07-17
申请号:CA501751
申请日:1986-02-13
Applicant: CIBA GEIGY AG
Inventor: STURM ELMAR , GALLAY JEAN J , PISSIOTAS GEORG
IPC: A61K31/515 , A61K31/517 , A61K31/53 , A61P33/00 , A61P33/10 , C07D215/20 , C07D215/22 , C07D215/227 , C07D237/00 , C07D237/14 , C07D237/16 , C07D237/32 , C07D239/34 , C07D239/56 , C07D239/62 , C07D239/66 , C07D239/80 , C07D239/88 , C07D241/18 , C07D241/44 , C07D251/34 , C07D251/38 , C07D251/42 , C07D401/12 , C07D403/12 , A01N43/00 , A61K31/395
Abstract: Barbituric acid derivatives The invention relates to novel phenylcarbamoylbarbituric acid derivatives of the general formula wherein R1 is C1-C4alkyl, C1-C3alkoxy, allyl or C3-C6cycloalkyl, R2 is C1-C4a1kyl or allyl, R3 is an unsubstituted or substituted heteroaromatic 6-membered ring which contains 2 or 3 nitrogen atoms, or is sn unsubstituted or substituted heteroaromatic 6-membered ring which is fused to a benzene ring and which contains 1 to 3 nitrogen atoms, R4 and R5 are each independently of the other hydrogen, C1-C4alkyl, C1-C4alkoxy or C1-C3haloalkyl and X is an oxygen or sulfur atom, and to the tautomers and salts thereof. These compounds may be used for controlling helminths which are parasites of animals.
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公开(公告)号:CA1254560A
公开(公告)日:1989-05-23
申请号:CA461860
申请日:1984-08-27
Applicant: CIBA GEIGY AG
Inventor: HUBELE ADOLF , ECKHARDT WOLFGANG , STURM ELMAR , ZONDLER HELMUT
IPC: A01N43/54 , C07D239/42 , C07D239/46 , C07D239/47 , C07D239/48 , C07D239/50 , C07D239/52 , C07D239/56 , C07D401/12 , C07D405/12 , C07D239/28 , C07D401/04
Abstract: Novel N-(2-nitrophenyl)-4-aminopyrimidine derivatives of the general formula I (I) wherein R1 is NO2 or CF3, R2 is NO2 or CF3, R3 is hydrogen or halogen, R4 is hydrogen or the -C(O)R7 group, in which R7 is an unsubstituted or substituted radical selected from the group consisting of C1-C12alkyl, C2-C6alkenyl, C3-C7cyclo-alkyl, phenyl and heterocyclyl, R5, R6 and R7 are each independently halogen, cyano, thiocyano, nitro or a group selected from -N(R9)(R10), -R11, R12-O- or R13-S(O)n, in which R9 and R10 are each independently hydrogen or an unsubstituted or substituted radical selected from the group consisting of C1-C12alkyl, C3-C6alkenyl and phenyl, or together with the nitrogen atom form an unsubstituted or substituted heterocyclic ring, n is 0, 1 or 2, R11, R12 and R13 are each independently an unsubstituted or substituted radical selected from the group consisting of C1-C12 alkyl, C2-C6alkenyl, C3-C6cycloalkyl, phenyl or heterocyclyl; and in addition R5 can be hydrogen, R6 can be hydrogen, or two of R5, R6 and R8 may be hydrogen. Methods of preparing these compounds are disclosed, as are also agrochemical compositions which contain one of said compounds active ingredient. The use of the novel compounds and the compositions containing them in agriculture are also described. The novel compounds or the compositions containing them are used for the control of harmful micro-organisms.
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公开(公告)号:DD267037A5
公开(公告)日:1989-04-19
申请号:DD30793886
申请日:1986-02-13
Applicant: CIBA GEIGY AG
Inventor: STURM ELMAR , GALLAY JEAN J , PISSIOTAS GEORG
IPC: A61K31/515 , A61K31/517 , A61K31/53 , A61P33/00 , A61P33/10 , C07D215/20 , C07D215/22 , C07D215/227 , C07D237/00 , C07D237/14 , C07D237/16 , C07D237/32 , C07D239/34 , C07D239/56 , C07D239/62 , C07D239/66 , C07D239/80 , C07D239/88 , C07D241/18 , C07D241/44 , C07D251/34 , C07D251/38 , C07D251/42 , C07D401/12 , C07D403/12 , C07D251/26 , C07D237/10 , C07D239/28 , C07D241/14
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公开(公告)号:DD264211A5
公开(公告)日:1989-01-25
申请号:DD30793986
申请日:1986-02-13
Applicant: CIBA GEIGY AG
Inventor: STURM ELMAR , GALLAY JEAN J , PISSIOTAS GEORG
IPC: A61K31/515 , A61K31/517 , A61K31/53 , A61P33/00 , A61P33/10 , C07D215/20 , C07D215/22 , C07D215/227 , C07D237/00 , C07D237/14 , C07D237/16 , C07D237/32 , C07D239/34 , C07D239/56 , C07D239/62 , C07D239/66 , C07D239/80 , C07D239/88 , C07D241/18 , C07D241/44 , C07D251/34 , C07D251/38 , C07D251/42 , C07D401/12 , C07D403/12
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公开(公告)号:GB2174388B
公开(公告)日:1988-10-19
申请号:GB8603353
申请日:1986-02-11
Applicant: CIBA GEIGY AG
Inventor: STURM ELMAR , GALLAY JEAN JACQUES , PISSIOTAS GEORG
IPC: A61K31/515 , A61K31/517 , A61K31/53 , A61P33/00 , A61P33/10 , C07D215/20 , C07D215/22 , C07D215/227 , C07D237/00 , C07D237/14 , C07D237/16 , C07D237/32 , C07D239/34 , C07D239/56 , C07D239/62 , C07D239/66 , C07D239/80 , C07D239/88 , C07D241/18 , C07D241/44 , C07D251/34 , C07D251/38 , C07D251/42 , C07D401/12 , C07D403/12 , C07D215/16 , C07D237/10 , C07D239/28 , C07D239/60 , C07D241/14
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公开(公告)号:GB2179659A
公开(公告)日:1987-03-11
申请号:GB8622763
申请日:1986-09-22
Applicant: CIBA GEIGY AG
Inventor: NYFELER ROBERT , ZONDLER HELMUT , STURM ELMAR
IPC: A01N31/04 , A01N31/14 , A01N43/64 , C07D249/08 , A01N43/653 , B01J27/10 , B01J31/10 , B01J31/22 , C07B61/00 , C07C20060101 , C07C33/20 , C07C41/00 , C07C41/03 , C07C43/13 , C07C43/178 , C07C43/23 , C07C43/295 , C07C43/315 , C07C67/00 , C07C201/00 , C07C201/12 , C07C205/34 , C07C253/00 , C07C253/30 , C07C255/54 , C07D253/00 , C07D521/00 , C07C33/025
Abstract: New glycol monoethers have the formula I: in which R1 is C1-C6-alkyl which is substituted by C1-C6-alkoxy or C3-C6-cycloalkyl, C3-C8-cycloalkyl, phenyl, phenyl which is monosubstituted to trisubstituted by halogen, C1-C6-halogenoalkyl, C1-C6-halogenoalkoxy, C1-C6-alkoxy, C1-C6-alkyl, nitro and/or cyano, phenyl which is substituted by phenoxy, halogenophenoxy, phenyl, halogenophenyl, benzyl or halogenobenzyl, benzyl or benzyl which is monosubstituted to trisubstituted by halogen, C1-C6-halogenoalkyl, C1-C6-halogenoalkoxy, C1-C6-alkoxy, C1-C6-alkyl, nitro and/or cyano; R2 is C1-C12-alkyl or a radical indicated under R1; and R3 is C1-C6-alkyl, C1-C6-alkyl which is substituted by C1-C3-alkoxy, C3-C4-alkenyl, benzyl or halogenobenzyl. Process for producing the new ethers is also described. The ethers are useful e.g. as intermediates for 1-triazolylethyl ethers having value as agrochemically active materials.
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公开(公告)号:CS247179B2
公开(公告)日:1986-12-18
申请号:CS376984
申请日:1984-05-18
Applicant: CIBA GEIGY AG
Inventor: NYFELER ROBERT , ZONDLER HELMUT , STURM ELMAR
IPC: C07D249/08 , A01N31/04 , A01N31/14 , A01N43/64 , A01N43/653 , B01J27/10 , B01J31/10 , B01J31/22 , C07B61/00 , C07C20060101 , C07C33/20 , C07C41/00 , C07C41/03 , C07C43/13 , C07C43/178 , C07C43/23 , C07C43/295 , C07C43/315 , C07C67/00 , C07C201/00 , C07C201/12 , C07C205/34 , C07C253/00 , C07C253/30 , C07C255/54 , C07D253/00 , C07D521/00
Abstract: Essentially, a process is described for the preparation of the 1-triazolylethyl ether derivatives, defined in claim 1, of the general formula I (I) which consists in (a) reacting an oxirane of the formula II (II) at temperatures of -20 DEG to +100 DEG C., in the presence of an acid catalyst or an acid condensation agent, with an alcohol of the formula III R3-OH (III) to give a glycol monoether of the formula IV (IV) and (b) subsequently reacting the glycol monoether of the formula IV or one of its esters, in the presence of an acid-binding agent or condensation agent, at temperatures of 0 DEG to 150 DEG C., with a triazole of the formula V (V) the substituents R1, R2 ; amd R3 in the formula II to IV being as defined under formula I and M in formula V being hydrogen or a metal atom. The novel compounds within the scope of formula I and their use are also described.
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