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公开(公告)号:BR0210703A
公开(公告)日:2004-07-20
申请号:BR0210703
申请日:2002-06-25
Applicant: SYNGENTA PARTICIPATIONS AG
Inventor: JEANGUENAT ANDRE , LAMBERTH CLEMENS , ZELLER MARTIN
IPC: A01N41/06 , A01N55/00 , A01N55/10 , C07C217/74 , C07C307/06 , C07C311/06 , C07F7/18 , A01N41/02
Abstract: The invention relates to novel pesticidally active N-bisaryl-and N-aryl-cycloalkylidenyl-alpha-sulfin-and alpha-sulfonamino acid amides of the general formula I, including the optical isomers thereof and mixtures of such isomers, wherein n is a number zero or one; R1 is C1-C12alkyl; C1-C12alkyl substituted with C1-C4alkoxy, C1-C4alkylthio, C1-C4alkylsulfonyl, C3-C8cycloalkyl, cyano, C1-C6alkoxycarbonyl, C3-C6alkoxycarbonyl, C3-C6alkenyloxycarbonyl or C3-C6alkynyloxycarbonyl; C2-C12alkenyl; C2-C12alkynyl; C1-C12haloalkyl; or a group NR11R12 wherein R11 and R12 are each independently of the other C1-C6alkyl, or together are tetra- or penta-methylene; R2 and R3 ae each independently hydrogen; C1-C8alkyl; C1-C8alkyl substituted with hydroxy, mercapto, C1-C4alkoxy or C1-C4alkylthio; C3-C8alkenyl; C3-C8alkynyl; C3-C8cycloalkyl; C3-C8cycloalkyl-C1-C4alkyl; optionally substituted aryl; optionally substituted heteroaryl; or the two groups R2 and R3 together with the carbon atom to which they are bonded form a three- to eight-membered hydrocarbon ring; A is an optionally substituted saturated or unsaturated C3-C8-cycloalkylidene, optionally substituted phenylidene or optionally substituted saturated or unsaturated heterocyclylidene bridge, R4 and R5 are each independently hydrogen or an organic radicak, and R6 is hydr
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公开(公告)号:AT271031T
公开(公告)日:2004-07-15
申请号:AT01933967
申请日:2001-05-15
Applicant: SYNGENTA PARTICIPATIONS AG
Inventor: LAMBERTH CLEMENS , ZELLER MARTIN , KUNZ WALTER , CEDERBAUM FREDRIK
IPC: A01N37/18 , A01N37/30 , A01N37/36 , A01N41/06 , A01N41/12 , A01N43/00 , A01N43/12 , A01N43/30 , A01N43/32 , A01P3/00 , C07C231/02 , C07C231/12 , C07C233/22 , C07C235/34 , C07C239/12 , C07C239/22 , C07C313/04 , C07C323/56 , C07C323/60 , C07C323/62 , C07D213/02 , C07D213/56 , C07D215/14 , C07D239/02 , C07D239/26 , C07D241/42 , C07D261/08 , C07D277/64 , C07D307/16 , C07D307/79 , C07D307/80 , C07D317/60 , C07D319/18 , C07D333/00 , C07D333/24 , C07D333/28 , C07D333/52 , C07D333/60
Abstract: The invention relates to phenyl-propargylether derivatives of the general formula Iincluding the optical isomers thereof and mixtures of such isomers, whereinR1 is hydrogen, alkyl, cycloalkyl or optionally substituted aryl,R2 and R3 are each independently hydrogen or alkyl,R4 is alkyl, alkenyl or alkynyl,R5, R6, R7, and R8 are each independently hydrogen or alkyl,R9 is hydrogen, optionally substituted alkyl, optionally substituted alkenyl or optionally substituted alkynyl,R10 is optionally substituted aryl or optionally substituted heteroaryl, andZ is halogen, optionally substituted aryloxy, optionally substituted alkoxy, optionally substituted alkenyloxy, optionally substituted alkynyloxy, optionally substituted arylthio, optionally substituted alkylthio, optionally substituted alkenylthio; optionally substituted alkynylthio, optionally substituted alkylsulfinyl, optionally substituted alkenylsulfinyl, optionally substituted alkynylsulfinyl, optionally substituted alkylsulfonyl, optionally substituted alkenylsulfonyl or optionally substituted alkynylsulfonyl. These compounds possess useful plant protecting properties and may advantageously be employed in agricultural practice for controlling or preventing the infestation of plants by phytopathogenic microorganisms, especially fungi.
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公开(公告)号:PL357011A1
公开(公告)日:2004-07-12
申请号:PL35701101
申请日:2001-04-11
Applicant: SYNGENTA PARTICIPATIONS AG
Inventor: ZELLER MARTIN , LAMBERTH CLEMENS , SZCZEPANSKI HENRY , DE MESMAEKER ALAIN
IPC: C07D295/22 , A01N41/06 , A01N43/10 , A01N43/36 , A01N43/40 , A01N43/42 , A01N43/60 , C07C303/34 , C07C303/38 , C07C307/06 , C07C311/06 , C07C313/06 , C07D213/30 , C07D213/61 , C07D215/14 , C07D241/12 , C07D333/16 , C07D333/28
Abstract: The invention relates to novel pesticidally active alpha-sulfin- and alpha-sulfonamino acid amides of the general formula (I) including the optical isomers thereof and mixtures of such isomers, wherein n is a number zero or one, R1-R7 have the meanings given in the specification. R8 is either hydrogen, (a), (b), (c), (d) or (e) wherein R11, R12, R14, R15 and R17 are each independently hydrogen or C1-C4alkyl, R13 is C4-C12alkyl; C1-C12 halogenalkyl; C3-C8 cycloalkyl; optionally substituted aryl or optionally substituted heteroaryl, R16 is optionally substituted aryl or optionally substituted heteroaryl; and Z is oxygen, sulfur -CR18R19- or -NR20-, wherein R18, R19, R20 independently of each other are hydrogen or C1-C4alkyl. The novel compounds possess plant-protecting properties and are suitable for protecting plants against infestation by phytopathogenic microorganisms
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公开(公告)号:DE60103292D1
公开(公告)日:2004-06-17
申请号:DE60103292
申请日:2001-09-10
Applicant: SYNGENTA PARTICIPATIONS AG
Inventor: NUNINGER COSIMA , ZELLER MARTIN
IPC: C07C311/06 , A01N37/18 , A01N37/22 , A01N37/34 , A01N37/50 , A01N41/06 , A01N43/36 , A01N43/40 , A01N43/50 , A01N43/54 , A01N43/56 , A01N43/828 , A01N43/84 , A01N47/14
Abstract: It has now been found that the use of: A) a N-sulfonyl-valine-amide of formula (I) wherein R1 is hydrogen, C1-4alkyl, C3-6cycloalkyl or halophenyl, and R2 is C1-4alkyl; in association with B) either compounds of formulae II to XII is particularly effective in combating or preventing fungal diseases of crop plants. These combinations exhibit synergistic fungicidal activity. Prominent examples for the compounds of formulae II to XII are: acibenzolar-S-methyl, azoxystrobin, chlorothalonil, cymoxanil, dimethomorph, fluazinam, fludioxonil, imazalil, S-imazalil, mancozeb, metalaxyl, metalaxyl-M, picoxystrobin, pyraclostrobin (BAS 500F) and trifloxystrobin.
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公开(公告)号:CA2503558A1
公开(公告)日:2004-06-17
申请号:CA2503558
申请日:2003-12-04
Applicant: SYNGENTA PARTICIPATIONS AG
Inventor: ZELLER MARTIN
IPC: C07C253/30 , C07C255/33
Abstract: Phenylmalonic acid dinitriles are prepared by reaction of, for example, phen yl Kalides with malonic acid dinitrile in the presence of palladium catalysts a nd bases.
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公开(公告)号:AT260249T
公开(公告)日:2004-03-15
申请号:AT99961032
申请日:1999-12-01
Applicant: SYNGENTA PARTICIPATIONS AG
Inventor: ZELLER MARTIN , JEANGUENAT ANDRE , LAMBERTH CLEMENS
IPC: A01N41/06 , C07B61/00 , C07C303/34 , C07C303/38 , C07C303/40 , C07C307/06 , C07C311/06 , C07C311/11 , C07C323/12 , C07C311/00
Abstract: The invention relates to alpha-sulfin- and alpha-sulfonamino acid amides of the general formula Iincluding the optical isomers thereof and mixtures of such isomers,whereinn is a number zero or one;R1 is C1-C12alkyl, C1-C12alkyl substituted with C1-C4alkoxy, C1-C4alkylthio, C1-C4alkylsulfonyl, C3-C8cycloalkyl, cyano, C1-C6alkoxycarbonyl, C3-C6alkenyloxycarbonyl or C3-C6alkynyloxycarbonyl; C3-C8cycloalkyl; C2-C12alkenyl; C2-C12alkynyl; C1-C12haloalkyl; or a group NR12R13 wherein R12 and R13 are each independently of the other hydrogen or C1-C6-alkyl, or together are tetra- or penta-methylene;R2 and R3 are each independently hydrogen; C1-C8alkyl; C1-C8alkyl substituted with hydroxy, mercapto, C1-C4alkoxy or C1-C4alkylthio; C3-C8alkenyl; C3-C8alkynyl; C3-C8cycloalkyl; C3-C8cycloalkyl-C1-C4alkyl; or the two groups R2 and R3 together with the carbon atom to which they are bonded form a three- to eight-membered hydrocarbon ring;R4, R5, R6 and R7 are each independently hydrogen or C1-C4alkyl;R8 is C1-C6alkyl, C3-C6alkenyl or C3-C6alkynyl;R9 and R10 are each independently hydrogen or C1-C4alkyl; andR11 is either in whereinR14, R,15, R16 and R17 are each independently hydrogen or C1-C4alkyl,X is oxygen, sulfur or -NR18-, wherein R18 is hydrogen or C1-C4alkyl, andA is optionally substituted mono- or polycylic aryl or heteroaryl, andto the preparation of those substances and to agrochemical compositions comprising at least one of those compounds as active ingredient. The invention relates also to the preparation of compositions and to the use of the compounds or of the compositions in controlling or preventing the infestation of plants by phytopathogenic microorganisms, especially fungi.
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公开(公告)号:DE69905027T2
公开(公告)日:2003-10-09
申请号:DE69905027
申请日:1999-02-25
Applicant: SYNGENTA PARTICIPATIONS AG
Inventor: JEANGUENAT ANDRE , ZELLER MARTIN
IPC: C07D295/14 , A01N41/02 , A01N41/06 , C07C237/08 , C07C307/06 , C07C311/06 , C07C311/19 , C07C323/63 , C07D209/20 , C07D213/56 , C07D235/16 , C07D277/64 , C07D307/54 , C07D311/80 , C07D317/60 , C07D333/24 , C07D333/28
Abstract: Novel alpha-amino acid amides of formula (I) as well as possible isomers and mixtures of isomers thereof, wherein the substituents are defined as follows: n is the number zero or one; R1 is optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkylalkyl, aryl or arylalkyl; or a group NRaRb wherein Ra and Rb are each independently of the other hydrogen, alkyl or form together an alkylene bridge; R2 is hydrogen or alkyl; R3 is optionally substituted aryl or heteroaryl; A is alkylene; and B is optionally substituted aryl; with the exception of the following compounds 2-phenyl-N-(1-phenyl-ethyl)-2-(4-methylphenyl)-sulfonylamino-acetamide, 2-phenyl-N-(1-phenyl-ethyl)-2-(4-chlorophenyl)-sulfonylamino-acetamide, 2-phenyl-N-(1-phenyl-ethyl)-2-(4-nitrolphenyl)-sulfonylamino-acetamide, 2-phenyl-N-(1-phenyl-ethyl)-2-(4-methoxyphenyl)-sulfonylamino-acetamide, 2-phenyl-N-(1-phenyl-ethyl)-2-(4-fluorophenyl)-sulfonylamino-acetamide, 2-phenyl-N-(1-phenyl-ethyl)-2-phenyl-sulfonylamino-acetamide and 2-phenyl-N-(1-phenyl-ethyl)-2-methane-sulfonylamino-acetamide. The novel compounds have plant-protective properties and are suitable for protecting plants against infestations by phytopathogenic microorganisms, in particular fungi.
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公开(公告)号:GT200200231A
公开(公告)日:2003-06-18
申请号:GT200200231
申请日:2002-11-13
Applicant: SYNGENTA PARTICIPATIONS AG
Inventor: ZELLER MARTIN , LAMBERTH CLEMENS , KRIZ MIROSLAV
IPC: A01N20060101 , A01N37/18 , A01N37/36 , A01N37/38 , C07D237/08 , A01N37/42 , A01N41/10 , A01N41/12 , A01N43/00 , A61K31/16 , C07C20060101 , C07C231/02 , C07C233/02 , C07C233/08 , C07C233/11 , C07C235/34 , C07C237/20 , C07C317/22 , C07C323/22 , C07C323/58 , C07C323/63 , C07C327/44 , C07D213/24 , C07D213/60 , C07D215/06 , C07D215/08 , C07D237/10 , C07D239/26 , C07D239/28 , C07D241/12 , C07D241/14 , C07D261/08 , C07D261/10 , C07D277/20 , C07D277/22 , C07D277/32 , C07D307/38 , C07D307/56 , C07D307/78 , C07D317/50 , C07D317/62 , C07D319/18 , C07D333/06 , C07D333/26
Abstract: LA PRESENTE INVENCION SE REFIERE A NOVEDOSOS DERIVADOS DE FENETILAMIDA DE ACIDO CARBOXILICO ALFAOXIGENADOS O ALFATIOLADOS DE FORMULA GENERAL (I) EN DONDE A,B1,Y,X,R1,R2,R5,B2,R4,N,R3,SON GRUPOS FUNCIONALES DESCRITOS EN EL EXPEDIENTE. ESTOS COMPUESTOS SON DE UTILIDAD PARA CONTROLAR O EVITAR LA INFESTACION DE PLANTAS POR MICROORGANISMOS FITOPATOGENOS, ESPECIALMENTE HONGOS. ENTRE LAS PLANTAS QUE TIENEN POR OBJETO EL SER PROTEGIDAS POR LA PRESENTE SOLICITUD DESTACAN TRIGO, CEBADA,CENTENO,AVENA,ARROZ,MAIZ,SORGO,REMOLACHA,PLANTAS OLEAGINOSAS, ENTRE OTRAS QUE SE MENCIONAN.
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公开(公告)号:BR0109999A
公开(公告)日:2003-05-27
申请号:BR0109999
申请日:2001-04-11
Applicant: SYNGENTA PARTICIPATIONS AG
Inventor: ZELLER MARTIN , LAMBERTH CLEMENS , SZCZEPANSKI HENRY , MESMAEKER ALAIN DE
IPC: C07D239/34 , A01N41/02 , A01N41/06 , C07C303/38 , C07C303/40 , C07C307/06 , C07C311/06 , C07C313/06 , C07D207/06 , C07D213/30 , C07D213/61 , C07D215/14 , C07D333/16 , C07D333/28
Abstract: The invention relates to novel pesticidally active alpha-sulfin- and alpha-sulfonamino acid amides of the general formula (I) including the optical isomers thereof and mixtures of such isomers, wherein n is a number zero or one; R1-R9 have the meanings given in the specification R10 is either hydrogen, (a), (b), (c), (d) or (e) wherein R13, R14, R16, R17 and R19 are each independently hydrogen or C1-C4 alkyl, R15 is C4-C12 alkyl; C1-C12 halogenalkyl; C3-C8 cycloalkyl; optionally substituted aryl or optionally substituted heteroaryl, R18 is optionally substituted aryl or optionally substituted heteroaryl; and Z is oxygen, sulfur -CR20R21- or -NR22-, wherein R20, R21 and R22 independently of each other are hydrogen of C1-C4 alkyl; provided that when R8 is hydrogen, R9 is not C1-C6-alkoxy, C3-C6 alkenyloxy or C3-C6-alkynyloxy in position 3 of the phenyl ring carrying these radicals. The novel compounds possess plant-protecting properties and are suitable for protecting plants against infestation by phytopathogenic microorganisms.
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公开(公告)号:BR0109977A
公开(公告)日:2003-05-27
申请号:BR0109977
申请日:2001-04-11
Applicant: SYNGENTA PARTICIPATIONS AG
Inventor: ZELLER MARTIN , LAMBERTH CLEMENS , SZCZEPANSKI HENRY , MESMAEKER ALAIN DE
IPC: C07D295/22 , A01N41/06 , C07C303/38 , C07C303/40 , C07C307/06 , C07C311/06 , C07C313/06 , C07D213/30 , C07D241/20
Abstract: The invention relates to novel pesticidally active alpha-sulfin and alpha-sulfonamino acid amides of the general formula (I) including the optical isomers thereof and mixtures of such isomers, wherein n is a number zero or one; R1, R2, R3, R4, R5, R6 and R7 have the meanings given in the specification, and R8 is either hydrogen, (a), (b), (c), (d) or (e) wherein R11, R12, R13, R15 and R17 are each independently hydrogen or C1-C4 alkyl, R13 is C4-C12 alkyl, C1-C12 halogenalkyl; C3-C8 cycloalkyl; optionally substituted aryl or optionally substituted heteroaryl, R16 is optionally substituted aryl or optionally substituted heteroaryl; and Z is oxygen, sulfur -CR18R19- or -NR2O-, wherein R18, R19 and R20 independently of each other are hydrogen or C1-C4 alkyl. The novel compounds possess plant-protecting properties and are suitable for protecting plants against infestation by phytopathogenic microorganisms.
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