N-SUBSTITUTED IMINO HETEROCYCLIC COMPOUNDS
    53.
    发明公开
    N-SUBSTITUTED IMINO HETEROCYCLIC COMPOUNDS 审中-公开
    的N-取代的杂环亚氨基

    公开(公告)号:EP3083581A1

    公开(公告)日:2016-10-26

    申请号:EP14820824.2

    申请日:2014-12-17

    Applicant: BASF SE

    Abstract: The present invention relates to N-substituted imino compound of formula (I), wherein Y is a radical Y
    1 , Y
    2 , Y
    3 , Y
    4 or Y
    5 , where Y
    1 is O-C(=X)-R
    3 ; Y
    2 is S-C(=X)-R
    3 ; Y
    3 is N(R
    5 )-C(=X)-R
    3 ; Y
    4 is N(R
    5 )-S(=O)-R
    4 ; Y
    5 is N(R
    5 )-S(=O)
    2 -R
    4 ; and where X is O or S; Het is a 5 or 6 membered carbon-bound or nitrogen-bound heterocyclic ring, W
    1 -W
    2 -W
    3 -W
    4 represents a carbon chain group connected to N and C=N, and thus forming a saturated, unsaturated, or partially unsaturated 5 or 6 membered nitrogen containing heterocycle, wherein W
    1 , W
    2 , W
    3 and W
    4 each individually represent CR
    V R
    W ; R
    1 , R
    2 may be hydrogen, halogen, C
    1 -C
    6 -alkyl etc.; and where R
    3 , R
    4 and R
    5 are as defined herein. The invention also relates to the use of the N-acylimino heterocyclic compounds, their stereoisomers, their tautomers and their salts, for combating invertebrate pests. Furthermore the invention relates also to methods of combating invertebrate pests, which comprises applying such compounds.

    PROCESS FOR PREPARING PYRAZOLES
    57.
    发明公开
    PROCESS FOR PREPARING PYRAZOLES 审中-公开
    制备吡唑的方法

    公开(公告)号:EP3174858A1

    公开(公告)日:2017-06-07

    申请号:EP15750664.3

    申请日:2015-07-30

    Applicant: BASF SE

    CPC classification number: C07D231/14 C07D401/12 C07D403/12 C07D405/06

    Abstract: The present invention relates to a process for preparing a pyrazole compound of formula V, the process including cyclizing a hydrazone substituted α,β-unsaturated carbonyl compound of formula IV by reacting it with a suitable reagent, e.g. a reducing agent, an organometallic reagent or a nucleophilic reagent. The compounds of formula V are versatile reaction tools for the preparation of pyrazole derived fine chemicals. The present invention also relates to pyrazole compounds of formulae Va, Vb, Vc, and VI.

    Abstract translation: 本发明涉及制备式V的吡唑化合物的方法,该方法包括通过使式IV的腙取代的α,β-不饱和羰基化合物与合适的试剂例如环己烷反应来环化。 还原剂,有机金属试剂或亲核试剂。 式V化合物是用于制备吡唑衍生的精细化学品的通用反应工具。 本发明还涉及式Va,Vb,Vc和VI的吡唑化合物。

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