-
公开(公告)号:AU599014B2
公开(公告)日:1990-07-12
申请号:AU5349286
申请日:1986-02-14
Applicant: CIBA GEIGY AG
Inventor: STURM ELMAR , GALLAY JEAN JACQUES , KRISTINSSON HAUKUR , PISSIOTAS GEORG
IPC: C07D263/58 , A61K31/496 , A61K31/515 , A61P33/10 , C07D233/70 , C07D235/26 , C07D239/62 , C07D239/66 , C07D249/08 , C07D249/12 , C07D263/34 , C07D271/06 , C07D271/10 , C07D271/113 , C07D277/24 , C07D277/34 , C07D277/58 , C07D277/68 , C07D285/08 , C07D285/12 , C07D285/13 , C07D403/12 , C07D413/12 , C07D417/12 , A61K31/505
Abstract: The invention relates to novel 5-(azolyloxyphenylcarbamoyl)barbituric acid derivatives of the general formula I (I) wherein X is oxygen or sulfur; R1 is C1-C6alkyl, C1-C6alkoxy, C3-C6cycloalkyl or allyl; R2 is C1-C6alkyl or allyl; R3 is an unsubstituted or substituted five-membered azole ring which is bound through carbon and is selected from the group consisting of benzimadazole, benzoxazole, benzothiazole, imidazole, oxazole, thiazole, oxadiazole, thiadiazole and triazole; and R4 and R5 are each independently of the other hydrogen, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkoxy or C1-C6haloalkoxy; and to the tautomers and salts thereof, as anthelmintic compounds. Together with suitable carriers and further assistants, these compounds may be used in particular for controlling helminths which are parasites of animals.
-
公开(公告)号:PH24447A
公开(公告)日:1990-06-25
申请号:PH37183
申请日:1988-07-06
Applicant: CIBA GEIGY AG
Inventor: STURM ELMAR , GALLAY JEAN JAQUES , KRISTINSSON HAUKUR , PISSIOTAS GEORG
IPC: C07D263/58 , A61K31/496 , A61K31/515 , A61P33/10 , C07D233/70 , C07D235/26 , C07D239/62 , C07D239/66 , C07D249/08 , C07D249/12 , C07D263/34 , C07D271/06 , C07D271/10 , C07D271/113 , C07D277/24 , C07D277/34 , C07D277/58 , C07D277/68 , C07D285/08 , C07D285/12 , C07D285/13 , C07D403/12 , C07D413/12 , C07D417/12
Abstract: The invention relates to novel 5-(azolyloxyphenylcarbamoyl)barbituric acid derivatives of the general formula I (I) wherein X is oxygen or sulfur; R1 is C1-C6alkyl, C1-C6alkoxy, C3-C6cycloalkyl or allyl; R2 is C1-C6alkyl or allyl; R3 is an unsubstituted or substituted five-membered azole ring which is bound through carbon and is selected from the group consisting of benzimadazole, benzoxazole, benzothiazole, imidazole, oxazole, thiazole, oxadiazole, thiadiazole and triazole; and R4 and R5 are each independently of the other hydrogen, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkoxy or C1-C6haloalkoxy; and to the tautomers and salts thereof, as anthelmintic compounds. Together with suitable carriers and further assistants, these compounds may be used in particular for controlling helminths which are parasites of animals.
-
公开(公告)号:NO161256C
公开(公告)日:1989-07-26
申请号:NO834592
申请日:1983-12-13
Applicant: CIBA GEIGY AG
Inventor: STURM ELMAR , MEYER ALFRED
IPC: A01N43/50 , A01N43/653 , A01P3/00 , C07C39/00 , C07C45/63 , C07C45/71 , C07D233/60 , C07D233/64 , C07D249/08 , C07D303/08 , C07D303/22 , C07D303/34 , C07D521/00
Abstract: 1-Azolyl-2-aryl-3-fluoro-alkan-2- ols of the general formula I in which Az is 1H-1,2,4-triazole, 4H-1,2,4-triazole or 1H-imidazole; Ar is an unsubstituted or substituted aromatic radical from the series comprising phenyl, biphenyl, phenoxyphenyl and naphthyl; R1 is hydrogen, C1-C4-alkyl, C3-C5-alkenyl or benzyl; R2 is hydrogen, fluorine or C1-C6-alkyl and R3 is hydrogen, fluorine, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy, C1-C6-alkylthio, phenyl, phenoxy, phenylthio or C3-C7-cycloalkyl, and each aromatic substituent or aromatic moiety of a substituent is unsubstituted or mono- or poly-substituted by halogen, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, nitro and/or cyano; including the acid addition salts, quaternary azolium salts and metal complexes, are useful for controlling phytopathogenic microorganisms.
-
公开(公告)号:HU196891B
公开(公告)日:1989-02-28
申请号:HU424683
申请日:1983-12-13
Applicant: CIBA GEIGY AG
Inventor: STURM ELMAR , MEYER ALFRED
IPC: A01N43/50 , A01N43/653 , A01P3/00 , C07C39/00 , C07C45/63 , C07C45/71 , C07D233/60 , C07D233/64 , C07D249/08 , C07D303/08 , C07D303/22 , C07D303/34 , C07D521/00
Abstract: 1-Azolyl-2-aryl-3-fluoro-alkan-2- ols of the general formula I in which Az is 1H-1,2,4-triazole, 4H-1,2,4-triazole or 1H-imidazole; Ar is an unsubstituted or substituted aromatic radical from the series comprising phenyl, biphenyl, phenoxyphenyl and naphthyl; R1 is hydrogen, C1-C4-alkyl, C3-C5-alkenyl or benzyl; R2 is hydrogen, fluorine or C1-C6-alkyl and R3 is hydrogen, fluorine, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy, C1-C6-alkylthio, phenyl, phenoxy, phenylthio or C3-C7-cycloalkyl, and each aromatic substituent or aromatic moiety of a substituent is unsubstituted or mono- or poly-substituted by halogen, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, nitro and/or cyano; including the acid addition salts, quaternary azolium salts and metal complexes, are useful for controlling phytopathogenic microorganisms.
-
公开(公告)号:GB2171099B
公开(公告)日:1988-10-19
申请号:GB8603352
申请日:1986-02-11
Applicant: CIBA GEIGY AG
Inventor: STURM ELMAR , GALLAY JEAN JACQUES , KRISTINSSON HAUKUR , PISSIOTAS GEORG
IPC: C07D263/58 , A61K31/496 , A61K31/515 , A61P33/10 , C07D233/70 , C07D235/26 , C07D239/62 , C07D239/66 , C07D249/08 , C07D249/12 , C07D263/34 , C07D271/06 , C07D271/10 , C07D271/113 , C07D277/24 , C07D277/34 , C07D277/58 , C07D277/68 , C07D285/08 , C07D285/12 , C07D285/13 , C07D403/12 , C07D413/12 , C07D417/12
Abstract: The invention relates to novel 5-(azolyloxyphenylcarbamoyl)barbituric acid derivatives of the general formula I (I) wherein X is oxygen or sulfur; R1 is C1-C6alkyl, C1-C6alkoxy, C3-C6cycloalkyl or allyl; R2 is C1-C6alkyl or allyl; R3 is an unsubstituted or substituted five-membered azole ring which is bound through carbon and is selected from the group consisting of benzimadazole, benzoxazole, benzothiazole, imidazole, oxazole, thiazole, oxadiazole, thiadiazole and triazole; and R4 and R5 are each independently of the other hydrogen, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkoxy or C1-C6haloalkoxy; and to the tautomers and salts thereof, as anthelmintic compounds. Together with suitable carriers and further assistants, these compounds may be used in particular for controlling helminths which are parasites of animals.
-
公开(公告)号:AU576029B2
公开(公告)日:1988-08-11
申请号:AU5031685
申请日:1985-11-25
Applicant: CIBA GEIGY AG
Inventor: STURM ELMAR , MAIENFISCH PETER
IPC: A01N43/90 , A61K31/365 , A61P33/10 , C07D493/22 , C07H19/01 , A61K31/41 , A01N33/26 , A61K31/415 , A61K31/35 , A61K31/655 , A01N43/16 , A01N43/50 , A01N43/64 , A01N43/713
Abstract: The present invention relates to milbemycin derivatives of the formula I (I) wherein X is hydrogen or beta -halogen, R is methyl, ethyl, isopropyl or sec-butyl and Az is a 5 membered heterocyclic aromatic ring which contains 2-4 nitrogen atoms and is attached in the 1-position and which is unsubstituted or substituted by one or two C1-C6alkyl groups. These compounds, and the acid addition salts and metal complexes thereof, are effective pesticides for controlling endo-and ectoparasites, especially for controlling neamatodes which are parasites of animals. The may be obtained by appropriate esterification in 5-position of milbemycin derivatives. The selective beta -halogenation of 14,15-epoxymilbemycin derivatives can be effected via the intermediate DELTA 13,14-15-hydroxymilbemycins with appropriate halogenating agents.
-
公开(公告)号:HU195807B
公开(公告)日:1988-07-28
申请号:HU63686
申请日:1986-02-14
Applicant: CIBA GEIGY AG
Inventor: STURM ELMAR , GALLAY JEAN J , PISSIOTAS GEORG , KRISTINSSON HAUKUR
IPC: C07D263/58 , A61K31/496 , A61K31/515 , A61P33/10 , C07D233/70 , C07D235/26 , C07D239/62 , C07D239/66 , C07D249/08 , C07D249/12 , C07D263/34 , C07D271/06 , C07D271/10 , C07D271/113 , C07D277/24 , C07D277/34 , C07D277/58 , C07D277/68 , C07D285/08 , C07D285/12 , C07D285/13 , C07D403/12 , C07D413/12 , C07D417/12
Abstract: The invention relates to novel 5-(azolyloxyphenylcarbamoyl)barbituric acid derivatives of the general formula I (I) wherein X is oxygen or sulfur; R1 is C1-C6alkyl, C1-C6alkoxy, C3-C6cycloalkyl or allyl; R2 is C1-C6alkyl or allyl; R3 is an unsubstituted or substituted five-membered azole ring which is bound through carbon and is selected from the group consisting of benzimadazole, benzoxazole, benzothiazole, imidazole, oxazole, thiazole, oxadiazole, thiadiazole and triazole; and R4 and R5 are each independently of the other hydrogen, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkoxy or C1-C6haloalkoxy; and to the tautomers and salts thereof, as anthelmintic compounds. Together with suitable carriers and further assistants, these compounds may be used in particular for controlling helminths which are parasites of animals.
-
公开(公告)号:ZA876303B
公开(公告)日:1988-05-25
申请号:ZA876303
申请日:1987-08-25
Applicant: CIBA GEIGY AG
Inventor: STURM ELMAR , ELMAR STURM , LANG ROBERT WERNER , ROBERT WERNER LANG , KRISTIANSEN ODD , ODD KRISTIANSEN
IPC: A01N47/34 , A01N20060101 , C07D20060101 , C07D239/34 , C07D , A01N
-
公开(公告)号:BR8704368A
公开(公告)日:1988-04-19
申请号:BR8704368
申请日:1987-08-25
Applicant: CIBA GEIGY AG
Inventor: STURM ELMAR , LANG ROBERT WERNER , KRISTIANSEN ODD
IPC: A01N47/34 , C07D239/34 , A01N47/36
Abstract: The invention relates to novel N-benzoyl-N,-4-(5-phenylpyrimid-2-yloxy)phenylureas of formula +TR wherein X1 is hydrogen, halogen, C1-C3alkoxy or C1-C3alkylthio, X2 is halogen, methyl, C1-C3alkoxy or C1-C3alkylthio, Y1, Y2, Y3 and Y4 are each independently hydrogen, halogen, methyl, trifluoromethyl or methoxy, Z is methyl, halomethyl containing 1 to 3 halogen atoms or pentafluoroethyl; and R1, R2 and R3 are each independently hydrogen, halogen, C1-C3alkyl, trifluoromethyl or C1-C3alkoxy, to the preparation thereof and to intermediates for the synthesis of these compounds, as well as to compositions containing them for use in pest control, especially for controlling representatives of the order Acarina that attack plants and animals and for controlling insects. The novel compounds exhibit especially pronounced activity against plant-destructive mites.
-
公开(公告)号:MX155538A
公开(公告)日:1988-03-25
申请号:MX568782
申请日:1982-11-26
Applicant: CIBA GEIGY AG
Inventor: NYFELER ROBERT , MEYER ALFRED , STURM ELMAR
IPC: A01N43/64 , C07D249/08
-
-
-
-
-
-
-
-
-