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公开(公告)号:WO2006043149A2
公开(公告)日:2006-04-27
申请号:PCT/IB2005/003113
申请日:2005-10-18
Applicant: BIOPROJET , SUN PHARMACEUTICAL INDUSTRIES LTD , CAPET, Marc , LEVOIN, Nicolas , BERREBI-BERTRAND, Isabelle , POUPARDIN, Olivia , ROBERT, Philippe , SCHWARTZ, Jean-charles , LECOMTE, Jeanne-marie , RAJAMANNAR, Thennati , PAL, Ranjan Kumar , SAMANTA, Biswajit , JIVANI, Jignesh K , PANCHAL, Bhavesh M. , BHATT, Isha H. , ARADHYE, Jayraj D.
Inventor: CAPET, Marc , LEVOIN, Nicolas , BERREBI-BERTRAND, Isabelle , POUPARDIN, Olivia , ROBERT, Philippe , SCHWARTZ, Jean-charles , LECOMTE, Jeanne-marie , RAJAMANNAR, Thennati , PAL, Ranjan Kumar , SAMANTA, Biswajit , JIVANI, Jignesh K , PANCHAL, Bhavesh M. , BHATT, Isha H. , ARADHYE, Jayraj D.
CPC classification number: C07C237/24 , C07C229/30 , C07C229/48 , C07C323/12 , C07C2601/08
Abstract: The present patent application concerns new compounds of formula (I): displaying agonistic activity at sphingosine-1-phosphate (S1P) receptors, their process of preparation and their use as immunosuppressive agents.
Abstract translation: 本专利申请涉及式(I)的新化合物:在鞘氨醇-1-磷酸(S1P)受体显示激动活性,其制备方法及其作为免疫抑制剂的用途。
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2.NOVEL PIPERIDINYL MONOCARBOXYLIC ACIDS AS S1P1 RECEPTOR AGONISTS 审中-公开
Title translation: 新型PIPERIDINYL单羧酸作为S1P1受体激动剂公开(公告)号:WO2012140020A1
公开(公告)日:2012-10-18
申请号:PCT/EP2012/056470
申请日:2012-04-10
Applicant: BIOPROJET , SUN PHARMA ADVANCED RESEARCH COMPANY LTD , CAPET, Marc , BERREBI-BERTRAND, Isabelle , ROBERT, Philippe , SCHWARTZ, Jean-Charles , LECOMTE, Jeanne-Marie , THENNATI, Rajamannar , PAL, Ranjan, Kumar , SAMANTA, Biswajit , PILLAI, Muthukumaran, Natarajan , DESAI, Japan, Nitinkumar , RANA, Dijixa, Chandubhai , PRAJAPATI, Kaushik, Dhanjubhai , PATHAK, Sandeep, Pankajbhai , PANCHAL, Bhavesh, M. , ARADHYE, Jayraj, D.
Inventor: CAPET, Marc , BERREBI-BERTRAND, Isabelle , ROBERT, Philippe , SCHWARTZ, Jean-Charles , LECOMTE, Jeanne-Marie , THENNATI, Rajamannar , PAL, Ranjan, Kumar , SAMANTA, Biswajit , PILLAI, Muthukumaran, Natarajan , DESAI, Japan, Nitinkumar , RANA, Dijixa, Chandubhai , PRAJAPATI, Kaushik, Dhanjubhai , PATHAK, Sandeep, Pankajbhai , PANCHAL, Bhavesh, M. , ARADHYE, Jayraj, D.
IPC: C07D413/10 , A61K31/454 , A61P9/10 , A61P29/00 , A61P37/06 , A61P35/00 , C07D413/14 , A61K31/5377
CPC classification number: C07D413/10 , A61K31/454 , A61K45/06 , C07D271/06
Abstract: The present invention relates to novel compounds acting as agonists at S1P (sphingosine-1-phosphate) receptors, compositions containing these compounds, use of these compounds in medicine and their process of preparation.
Abstract translation: 本发明涉及作为S1P(鞘氨醇-1-磷酸)受体的激动剂的新化合物,含有这些化合物的组合物,这些化合物在医药中的应用及其制备方法。
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公开(公告)号:WO2006043149A9
公开(公告)日:2006-08-10
申请号:PCT/IB2005003113
申请日:2005-10-18
Applicant: BIOPROJET SOC CIV , SUN PHARMACEUTICAL IND LTD , CAPET MARC , LEVOIN NICOLAS , BERREBI-BERTRAND ISABELLE , POUPARDIN OLIVIA , ROBERT PHILIPPE , SCHWARTZ JEAN-CHARLES , LECOMTE JEANNE-MARIE , RAJAMANNAR THENNATI , PAL RANJAN KUMAR , SAMANTA BISWAJIT , JIVANI JIGNESH K , PANCHAL BHAVESH M , BHATT ISHA H , ARADHYE JAYRAJ D
Inventor: CAPET MARC , LEVOIN NICOLAS , BERREBI-BERTRAND ISABELLE , POUPARDIN OLIVIA , ROBERT PHILIPPE , SCHWARTZ JEAN-CHARLES , LECOMTE JEANNE-MARIE , RAJAMANNAR THENNATI , PAL RANJAN KUMAR , SAMANTA BISWAJIT , JIVANI JIGNESH K , PANCHAL BHAVESH M , BHATT ISHA H , ARADHYE JAYRAJ D
IPC: C07C229/30 , A61K31/10 , A61K31/165 , A61K31/196 , A61K31/197 , A61K31/216 , A61P37/06 , C07C229/48 , C07C237/24 , C07C323/12
CPC classification number: C07C237/24 , C07C229/30 , C07C229/48 , C07C323/12 , C07C2601/08
Abstract: The present patent application concerns new compounds of formula (I): displaying agonistic activity at sphingosine-1-phosphate (S1P) receptors, their process of preparation and their use as immunosuppressive agents.
Abstract translation: 本专利申请涉及式(I)的新化合物:显示对1-磷酸鞘氨醇(S1P)受体的激动活性,其制备过程及其作为免疫抑制剂的用途。
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公开(公告)号:WO2006043149A3
公开(公告)日:2006-07-13
申请号:PCT/IB2005003113
申请日:2005-10-18
Applicant: BIOPROJET SOC CIV , SUN PHARMACEUTICAL IND LTD , CAPET MARC , LEVOIN NICOLAS , BERREBI-BERTRAND ISABELLE , POUPARDIN OLIVIA , ROBERT PHILIPPE , SCHWARTZ JEAN-CHARLES , LECOMTE JEANNE-MARIE , RAJAMANNAR THENNATI , PAL RANJAN KUMAR , SAMANTA BISWAJIT , JIVANI JIGNESH K , PANCHAL BHAVESH M , BHATT ISHA H , ARADHYE JAYRAJ D
Inventor: CAPET MARC , LEVOIN NICOLAS , BERREBI-BERTRAND ISABELLE , POUPARDIN OLIVIA , ROBERT PHILIPPE , SCHWARTZ JEAN-CHARLES , LECOMTE JEANNE-MARIE , RAJAMANNAR THENNATI , PAL RANJAN KUMAR , SAMANTA BISWAJIT , JIVANI JIGNESH K , PANCHAL BHAVESH M , BHATT ISHA H , ARADHYE JAYRAJ D
IPC: C07C229/30 , A61K31/10 , A61K31/165 , A61K31/196 , A61K31/197 , A61K31/216 , A61P37/06 , C07C229/48 , C07C237/24 , C07C323/12
CPC classification number: C07C237/24 , C07C229/30 , C07C229/48 , C07C323/12 , C07C2601/08
Abstract: The present patent application concerns new compounds of formula (I): displaying agonistic activity at sphingosine-1-phosphate (S1P) receptors, their process of preparation and their use as immunosuppressive agents.
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