-
1.INHIBITORS OF DIACYLGLYCEROL O-ACYLTRANSFERASE TYPE 1 ENZYME 审中-公开
Title translation: 二乙酰胆碱酯酶1型酶的抑制剂公开(公告)号:WO2008134693A1
公开(公告)日:2008-11-06
申请号:PCT/US2008/061951
申请日:2008-04-30
Applicant: ABBOTT LABORATORIES , JUDD, Andrew S , MULHERN, Mathew M , IYENGAR, Rajesh R , KYM, Philip R , SOUERS, Andrew J
Inventor: JUDD, Andrew S , MULHERN, Mathew M , IYENGAR, Rajesh R , KYM, Philip R , SOUERS, Andrew J
IPC: C07D277/20 , C07D401/04 , C07D401/12 , C07D401/14 , C07D417/04 , C07D417/12 , C07D417/14 , C07D493/08 , A61K31/427 , A61K31/44 , A61P3/04 , A61P3/10
CPC classification number: C07D417/04 , C07D213/40 , C07D213/75 , C07D277/28 , C07D277/82 , C07D405/04 , C07D417/12 , C07D417/14 , C07D498/08
Abstract: The present invention relates to compounds of formula (I): wherein Q, G 1 , G 2 , and G 3 , are defined herein. Pharmaceutical compositions and methods for treating DGAT-1 related diseases or conditions are also disclosed.
Abstract translation: 本发明涉及式(I)的化合物:其中Q,G 1,G 2和G 3在本文中定义。 还公开了治疗DGAT-1相关疾病或病症的药物组合物和方法。
-
2.INHIBITORS OF DIACYLGLYCEROL O-ACYLTRANSFERASE TYPE 1 ENZYME 审中-公开
Title translation: 作者二酰基甘油O-酰基转移酶1酶抑制剂公开(公告)号:EP2142521A1
公开(公告)日:2010-01-13
申请号:EP08795827.8
申请日:2008-04-30
Applicant: Abbott Laboratories
Inventor: JUDD, Andrew S , MULHERN, Mathew M , IYENGAR, Rajesh R , KYM, Philip R , SOUERS, Andrew J
IPC: C07D277/20 , C07D401/04 , C07D401/12 , C07D401/14 , C07D417/04 , C07D417/12 , C07D417/14 , C07D493/08 , A61K31/427 , A61K31/44 , A61P3/04 , A61P3/10
CPC classification number: C07D417/04 , C07D213/40 , C07D213/75 , C07D277/28 , C07D277/82 , C07D405/04 , C07D417/12 , C07D417/14 , C07D498/08
Abstract: The present invention relates to compounds of formula (I): wherein Q, G1, G2, and G3, are defined herein. Pharmaceutical compositions and methods for treating DGAT-1 related diseases or conditions are also disclosed.
-