-
公开(公告)号:NO992492A
公开(公告)日:1999-05-25
申请号:NO992492
申请日:1999-05-25
Applicant: BASF AG
Inventor: LUBISCH WILFRIED , M LLER ACHIM , TREIBER HANS-J RG
IPC: A61K31/16 , A61K31/166 , A61K31/18 , A61K31/4045 , A61K31/435 , A61K31/4402 , A61K31/4406 , A61K31/4409 , A61K31/47 , A61P9/10 , A61P21/00 , A61P25/00 , A61P25/08 , A61P25/28 , A61P27/00 , A61P35/00 , A61P35/04 , A61P43/00 , C07C233/76 , C07C235/42 , C07C235/46 , C07C235/58 , C07C235/60 , C07C235/84 , C07C237/42 , C07C311/08 , C07C311/21 , C07C317/44 , C07C323/42 , C07C323/60 , C07D209/14 , C07D209/16 , C07D213/30 , C07D213/56 , C07D213/71 , C07D213/82 , C07D215/36
CPC classification number: C07D213/82 , C07C233/76 , C07C235/42 , C07C235/46 , C07C235/60 , C07C235/84 , C07C237/42 , C07C311/21 , C07C317/44 , C07C323/42 , C07C323/60 , C07C2601/14 , C07D209/16 , C07D215/36
-
公开(公告)号:NO991761D0
公开(公告)日:1999-04-14
申请号:NO991761
申请日:1999-04-14
Applicant: BASF AG
Inventor: LUBISCH WILFRIED , M LLER ACHIM , DELZER J RGEN
IPC: A61K31/445 , A61K31/4523 , A61K31/4545 , A61K31/4709 , A61K31/498 , A61K31/5355 , A61P9/10 , A61P25/14 , A61P25/28 , A61P35/00 , A61P43/00 , C07D211/62 , C07D213/40 , C07D295/04 , C07D401/06 , C07D401/12 , C07D401/14 , C07D409/06 , C07D413/12 , C07D413/14
Abstract: Piperidineketocarboxylic acid derivatives of the general formula Iand their tautomeric and isomeric forms, and physiologically tolerable salts thereof, where the variables have the meanings given in the description, preparation of these compounds and their use as drugs.
-
公开(公告)号:NO991761A
公开(公告)日:1999-04-14
申请号:NO991761
申请日:1999-04-14
Applicant: BASF AG
Inventor: LUBISCH WILFRIED , M LLER ACHIM , DELZER J RGEN
IPC: A61K31/445 , A61K31/4523 , A61K31/4545 , A61K31/4709 , A61K31/498 , A61K31/5355 , A61P9/10 , A61P25/14 , A61P25/28 , A61P35/00 , A61P43/00 , C07D211/62 , C07D213/40 , C07D295/04 , C07D401/06 , C07D401/12 , C07D401/14 , C07D409/06 , C07D413/12 , C07D413/14
CPC classification number: C07D401/06 , C07D211/62 , C07D401/12
-
公开(公告)号:NO992821L
公开(公告)日:1999-06-11
申请号:NO992821
申请日:1999-06-10
Applicant: BASF AG
Inventor: LUBISCH WILFRIED , M LLER ACHIM , TREIBER HANS-J RG
IPC: C07D295/12 , A61K31/16 , A61K31/166 , A61K31/381 , A61K31/40 , A61K31/4164 , A61K31/4402 , A61K31/4409 , A61K31/4439 , A61K31/4453 , A61K31/4468 , A61K31/4545 , A61K31/47 , A61K31/4709 , A61K31/495 , A61K31/496 , A61K31/498 , A61K31/5355 , A61K31/5375 , A61K31/5377 , A61P9/10 , A61P25/00 , A61P25/08 , A61P25/28 , A61P35/00 , A61P43/00 , C07C233/87 , C07C237/22 , C07C237/36 , C07C237/42 , C07C311/19 , C07C311/21 , C07D211/58 , C07D213/56 , C07D215/12 , C07D215/36 , C07D215/48 , C07D233/54 , C07D233/61 , C07D241/42 , C07D241/44 , C07D295/02 , C07D295/13 , C07D333/38 , C07D333/56 , C07D333/60 , C07D401/12 , C07D521/00 , C07K5/02
Abstract: PCT No. PCT/EP97/06655 Sec. 371 Date Jun. 8, 1999 Sec. 102(e) Date Jun. 8, 1999 PCT Filed Nov. 28, 1997 PCT Pub. No. WO98/25883 PCT Pub. Date Jun. 18, 1998The patent describes ketobenzamides of the formula where R1, R2, R3, R4, X and n have the meanings given in the description, and their preparation. The novel compounds are useful for controlling disorders.
-
公开(公告)号:NO992492L
公开(公告)日:1999-05-25
申请号:NO992492
申请日:1999-05-25
Applicant: BASF AG
Inventor: LUBISCH WILFRIED , M LLER ACHIM , TREIBER HANS-J RG
IPC: A61K31/16 , A61K31/166 , A61K31/18 , A61K31/4045 , A61K31/435 , A61K31/4402 , A61K31/4406 , A61K31/4409 , A61K31/47 , A61P9/10 , A61P21/00 , A61P25/00 , A61P25/08 , A61P25/28 , A61P27/00 , A61P35/00 , A61P35/04 , A61P43/00 , C07C233/76 , C07C235/42 , C07C235/46 , C07C235/58 , C07C235/60 , C07C235/84 , C07C237/42 , C07C311/08 , C07C311/21 , C07C317/44 , C07C323/42 , C07C323/60 , C07D209/14 , C07D209/16 , C07D213/30 , C07D213/56 , C07D213/71 , C07D213/82 , C07D215/36
Abstract: Compounds of the formulawhere R1, R2, R3, X and n are as defined in the description, are inhibitors of cysteine protease.
-
公开(公告)号:NO992492D0
公开(公告)日:1999-05-25
申请号:NO992492
申请日:1999-05-25
Applicant: BASF AG
Inventor: LUBISCH WILFRIED , M LLER ACHIM , TREIBER HANS-J RG
IPC: A61K31/16 , A61K31/166 , A61K31/18 , A61K31/4045 , A61K31/435 , A61K31/4402 , A61K31/4406 , A61K31/4409 , A61K31/47 , A61P9/10 , A61P21/00 , A61P25/00 , A61P25/08 , A61P25/28 , A61P27/00 , A61P35/00 , A61P35/04 , A61P43/00 , C07C233/76 , C07C235/42 , C07C235/46 , C07C235/58 , C07C235/60 , C07C235/84 , C07C237/42 , C07C311/08 , C07C311/21 , C07C317/44 , C07C323/42 , C07C323/60 , C07D209/14 , C07D209/16 , C07D213/30 , C07D213/56 , C07D213/71 , C07D213/82 , C07D215/36 , C07C
Abstract: Compounds of the formulawhere R1, R2, R3, X and n are as defined in the description, are inhibitors of cysteine protease.
-
公开(公告)号:NO992821A
公开(公告)日:1999-06-11
申请号:NO992821
申请日:1999-06-10
Applicant: BASF AG
Inventor: LUBISCH WILFRIED , M LLER ACHIM , TREIBER HANS-J RG
IPC: C07D295/12 , A61K31/16 , A61K31/166 , A61K31/381 , A61K31/40 , A61K31/4164 , A61K31/4402 , A61K31/4409 , A61K31/4439 , A61K31/4453 , A61K31/4468 , A61K31/4545 , A61K31/47 , A61K31/4709 , A61K31/495 , A61K31/496 , A61K31/498 , A61K31/5355 , A61K31/5375 , A61K31/5377 , A61P9/10 , A61P25/00 , A61P25/08 , A61P25/28 , A61P35/00 , A61P43/00 , C07C233/87 , C07C237/22 , C07C237/36 , C07C237/42 , C07C311/19 , C07C311/21 , C07D211/58 , C07D213/56 , C07D215/12 , C07D215/36 , C07D215/48 , C07D233/54 , C07D233/61 , C07D241/42 , C07D241/44 , C07D295/02 , C07D295/13 , C07D333/38 , C07D333/56 , C07D333/60 , C07D401/12 , C07D521/00 , C07K5/02
CPC classification number: C07D295/13 , C07C237/36 , C07C311/19 , C07C311/21 , C07D211/58 , C07D213/56 , C07D215/12 , C07D215/36 , C07D215/48 , C07D231/12 , C07D233/56 , C07D241/42 , C07D241/44 , C07D249/08 , C07D333/38 , C07D333/60 , C07K5/0205
-
公开(公告)号:NO992770L
公开(公告)日:1999-06-08
申请号:NO992770
申请日:1999-06-08
Applicant: BASF AG
Inventor: LUBISCH WILFRIED , M LLER ACHIM , TREIBER HANS-J RG
IPC: A61K31/403 , A61K31/4035 , A61K31/405 , A61K31/4439 , A61K31/496 , A61K31/517 , A61K31/519 , A61K31/5377 , A61P9/00 , A61P25/00 , A61P25/08 , A61P25/14 , A61P25/28 , A61P35/00 , A61P35/04 , A61P43/00 , C07D209/48 , C07D209/66 , C07D239/70 , C07D239/96 , C07D401/12 , C07D471/04 , C07D475/02 , A61K31/40
Abstract: Heterocyclically substituted benzamides of the formula Iare described, where R1, R2, R3, R4, R5, X, m and n have the meanings given in the description. The novel compounds are useful for controlling diseases.
-
公开(公告)号:NO992770A
公开(公告)日:1999-06-08
申请号:NO992770
申请日:1999-06-08
Applicant: BASF AG
Inventor: LUBISCH WILFRIED , M LLER ACHIM , TREIBER HANS-J RG
IPC: A61K31/403 , A61K31/4035 , A61K31/405 , A61K31/4439 , A61K31/496 , A61K31/517 , A61K31/519 , A61K31/5377 , A61P9/00 , A61P25/00 , A61P25/08 , A61P25/14 , A61P25/28 , A61P35/00 , A61P35/04 , A61P43/00 , C07D209/48 , C07D209/66 , C07D239/70 , C07D239/96 , C07D401/12 , C07D471/04 , C07D475/02 , A61K31/40
CPC classification number: C07D471/04 , C07D209/66 , C07D239/70 , C07D239/96 , C07D475/02
-
公开(公告)号:NO991761L
公开(公告)日:1999-04-14
申请号:NO991761
申请日:1999-04-14
Applicant: BASF AG
Inventor: LUBISCH WILFRIED , M LLER ACHIM , DELZER J RGEN
IPC: A61K31/445 , A61K31/4523 , A61K31/4545 , A61K31/4709 , A61K31/498 , A61K31/5355 , A61P9/10 , A61P25/14 , A61P25/28 , A61P35/00 , A61P43/00 , C07D211/62 , C07D213/40 , C07D295/04 , C07D401/06 , C07D401/12 , C07D401/14 , C07D409/06 , C07D413/12 , C07D413/14
Abstract: Piperidineketocarboxylic acid derivatives of the general formula Iand their tautomeric and isomeric forms, and physiologically tolerable salts thereof, where the variables have the meanings given in the description, preparation of these compounds and their use as drugs.
-
-
-
-
-
-
-
-
-