3-AMINO-1,2-BENZISOTHIAZOLE COMPOUNDS FOR COMBATING ANIMAL PEST II
    4.
    发明申请
    3-AMINO-1,2-BENZISOTHIAZOLE COMPOUNDS FOR COMBATING ANIMAL PEST II 审中-公开
    3-氨基-1,2-苯并二硫唑化合物治疗动物瘟疫II

    公开(公告)号:WO2008090048A3

    公开(公告)日:2008-11-20

    申请号:PCT/EP2008050337

    申请日:2008-01-14

    Abstract: The invention provides 3-amino-1,2-benzisothiazole compounds of formula (I) wherein n, R 1 , R 2 , R 3 , R 4 and A are defined as in the description. The invention provides further agricultural compositions comprising an amount of at least one compound of the formula (I) or an enantiomer, diasteromer or salt thereof; the use of a compound of formula (I) or an enantiomer, diasteromer or salt thereof for combating animal pests; a method of combating animal pests which comprises contacting the animal pests, their habit, breeding ground, food supply, plant, seed, soil, area, material or environment in which the animal pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from animal attack or infestation with a pesticidally effective amount of at least one compound of the formula (I) or an enantiomer, diasteromer or salt thereof; a method for protecting crops from attack or infestation by animal pests, which comprises contacting a crop with a pesticidally effective amount of at least one compound of the formula (I) or an enantiomer, diasteromer or salt thereof; a method for the protection of seeds from soil insects and of the seedlings' roots and shoots from soil and foliar insects comprising contacting the seeds before sowing and/or after pregermination with at least one compound of the formula (I), or the enantiomers, diastereomers or salts thereof; and seeds comprising a compound of the formula I or an enantiomer, diasteromer or salt thereof.

    Abstract translation: 本发明提供了式(I)的3-氨基-1,2-苯并异噻唑化合物,其中n,R 1,R 2,R 3, R 4和A如说明书中所定义。 本发明提供了另外的农业组合物,其包含一定量的至少一种式(I)化合物或其对映异构体,非对映异构体或盐; 式(I)化合物或其对映体,非对映体或盐用于对抗动物害虫的用途; 一种防治动物害虫的方法,其包括使动物害虫,其习性,繁殖场,食物供应,植物,种子,土壤,面积,动物害虫正在生长或可能生长的材料或环境,或材料,植物, (I)化合物或其对映异构体,非对映异构体或盐的动物攻击或侵染的种子,土壤,表面或空间; 该方法包括使农作物与杀虫有效量的至少一种式(I)化合物或其对映异构体,非对映异构体或盐接触; 一种保护种子免受土壤昆虫以及幼苗的根和芽以及土壤和叶面昆虫的方法,包括在播种前和/或发芽后使种子与至少一种式(I)化合物或对映异构体接触, 非对映异构体或其盐; 和包含式I化合物或其对映体,非对映体或盐的种子。

    RESORCINE DERIVATIVES AND THEIR USE AS PESTICIDES
    5.
    发明申请
    RESORCINE DERIVATIVES AND THEIR USE AS PESTICIDES 审中-公开
    RESORCINE衍生物及其作为杀虫剂的用途

    公开(公告)号:WO2007054558A2

    公开(公告)日:2007-05-18

    申请号:PCT/EP2006068329

    申请日:2006-11-10

    CPC classification number: C07D213/64 C07D277/34 C07D307/80

    Abstract: This invention relates to resorcine derivatives of formula (I) wherein R 1 is phenyl or a 5- to 6-membered heteroaromatic ring which may contain 1 to 3 heteroatoms selected from oxygen, nitrogen and sulfur, wherein phenyl or the heteroaromatic ring may be fused to a ring selected from phenyl and a 5- to 6-membered saturated, partially unsaturated or aromatic heterocyclic ring which may contain 1 to 3 heteroatoms selected from oxygen, nitrogen and sulfur, wherein phenyl or the 5- to 6-membered heteroaromatic ring or the respective fused ring systems may be unsubstituted or substituted by any combination of 1 to 6 optionally substituted groups R 3 , wherein R 3 is halogen, cyano, nitro, hydroxy, mercapto, amino, alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, haloalkyl, haloalkenyl, haloalkynyl, halocycloalkyl, halocycloalkenyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, haloalkenyloxy, haloalkynyloxy, alkylthio, alkenylthio, alkynylthio, haloalkylthio, haloalkenylthio, haloalkynylthio, alkylamino, alkenylamino, alkynylamino, dialkylamino, dialkenylamino, dialkynylamino, alkyl-alkenylamino, alkyl-alkynylamino, alkenyl- alkynylamino, trialkylsilyl, or phenyl or a 5-to 7-membered saturated or partially unsaturated heterocyclic ring which may contain 1 to 3 heteroatoms selected from oxygen, sulfur and nitrogen or a 5- to 6-membered heteraromatic ring system which may contain 1 to 4 heteroatoms selected from oxygen, nitrogen and sulfur, which phenyl and which heteroaromatic ring may be bonded via an oxygen or a sulfur atom, or -C(=G)Ra, -C(=G)ORa, -C(=G)NRa2, -C(=G)[N=SRa2], -C(=NORa)Ra, -C(=NORa)NRa2, -C(=NNRa2)Ra , -OC(=G)-OC(=G)ORa, N=SRa2, -NRaC(=G)Ra, -N[C(=G)Ra]2, - NRaC(=G)ORa, -C(=G)NRa-NRa2, -C(=G)NRa-NRa [C(=G)Ra], -NRa-C(=G)NRa2, -NRa-NRaC(=G)Ra, -NRa-N[C(=G)Ra]2, -N[(C=G)Ra]-NRa2, -NRa-NRa[(C=G)GRa], -NRa[(C=G)NRa2, -NRa[C=NRa]Ra, -NRa(C=NRa)NRa2, -O-NRa2, -O-NRa(C=G)Ra, - SO2NRa2, -NRaSO2Ra, -S(=O)Ra, -S(=O)2Ra, -SO2ORa, or -OSO2Ra, wherein G is oxygen or sulfur and Ra is as defined in the description, R 2 is hydrogen, halogen, cyano, alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, haloalkynyl, alkoxy, or haloalkoxy, x is 2, 3, 4, 5, 6, or 7, or the diastereomers, enantiomers, salts or N-oxides thereof, with the proviso that R 1 is not 5-chloro-2,2,-dimethyl-2,3-dihydrobenzo[b]furan-7-yl when R 2 is hydrogen and x is 3 or 4, processes and intermediates for the preparation of compounds I, use of compounds I for combating insects, acarids, or nematodes, and a method for treating, controlling, preventing or protecting animals against infestation or infection by parasites using compounds I.

    Abstract translation: 本发明涉及其中R 1为苯基或可含有1-3个选自氧,氮和硫的杂原子的5至6元杂芳环的式(I)的间苯二酚衍生物,其中苯基 或杂芳环可以与选自苯基和5-至6-元饱和,部分不饱和或芳族杂环的环稠合,所述杂环可以含有1-3个选自氧,氮和硫的杂原子,其中苯基或5- 至6元杂芳环或相应的稠环体系可以是未取代的或被1至6个任选取代的基团R 3 3的任何组合取代,其中R 3是卤素, 氰基,硝基,羟基,巯基,氨基,烷基,烯基,炔基,环烷基,环烯基,卤代烷基,卤代烯基,卤代炔基,卤代环烷基,卤代环烯基,烷氧基,烯氧基,炔氧基,卤代烷氧基,卤代烯氧基,卤代炔氧基,烷硫基,烯硫基,炔硫基,卤代烷硫基, H 烯基氨基,炔基氨基,二烷基氨基,二链烷基氨基,二炔基氨基,烷基 - 链烯基氨基,烷基 - 炔基氨基,烯基 - 炔基氨基,三烷基甲硅烷基或苯基或5至7元饱和或部分不饱和的杂环, 至3个选自氧,硫和氮的杂原子或5至6元杂芳环体系,其可以含有1至4个选自氧,氮和硫的杂原子,该苯基和杂芳环可以通过氧或 硫原子或-C(= G)R a,-C(= G)OR a,-C(= G)NR a 2,-C(= G)[N = SR a 2] (= NORa)NRa2,-C(= NNRa2)Ra,-OC(= G)-OC(= G)ORa,N = SRa2,-NRaC(= G)Ra,-N [C(= G)Ra] 2,-NR a C(= G)OR a,-C(= G)NR a -NR a 2,-C(= G)NR a -NR a [C(= G)R a] -NRaC(= G)Ra,-NRa-N [C(= G)Ra] 2,-N [(C = G)Ra] -NRa2,-NRa-NRa [(C = G) [(C = G)NRa2,-NRa [C = NRa] Ra,-NRa(C = NRa)NRa2,-O-NRa2,-O-NRa(C = G)Ra,-SO2NRa2,-NRaSO2Ra,-S (= O)R a,-S(= O)2 R a,-SO 2 OR a或-O SO 2 R a,其中G是氧或硫,Ra如说明书中所定义,R 2是氢,卤素,氰基,烷基,卤代烷基,烯基,卤代烯基,炔基,卤代炔基,烷氧基或卤代烷氧基, x是2,3,4,5,6或7,或其非对映异构体,对映异构体,盐或N-氧化物,条件是R 1不是5-氯-2,2 ,当R 2是氢并且x是3或4时,制备化合物I的方法和中间体,使用化合物I,其中R 1,R 2,R 3, 用于防治昆虫,螨虫或线虫,以及用化合物I治疗,控制,预防或保护动物免受寄生虫侵袭或感染的方法。

    NOVEL 2-CYANO-3-(HALO)ALKOXY-BENZENESULFONAMIDE COMPOUNDS FOR COMBATING ANIMAL PESTS
    6.
    发明申请
    NOVEL 2-CYANO-3-(HALO)ALKOXY-BENZENESULFONAMIDE COMPOUNDS FOR COMBATING ANIMAL PESTS 审中-公开
    新型2-氰基-3-(卤代)烷氧基苯磺酰胺化合物用于防治动物病虫害

    公开(公告)号:WO2006056433A2

    公开(公告)日:2006-06-01

    申请号:PCT/EP2005012561

    申请日:2005-11-24

    CPC classification number: C07C319/20 A01N41/06 C07C311/29 C07C323/62

    Abstract: The invention relates to 2-cyano-3-(halo)alkoxy-benzenesulfonamide compounds (I), where the variables Alk and R1 to R5 are as defined in claim 1, and/or to their agriculturally useful salts. Moreover, the present invention relates to: the use of compounds (I) and/or their salts for combating animal pests; agricultural compositions comprising such an amount of at least one compound of the general formula (I) and/or at least one agriculturally useful salt of (I) and at least one inert liquid and/or solid agronomically acceptable carrier that it has a pesticidal action and, if desired, at least one surfactant; and a method of combating animal pests which comprises contacting the animal pests, their habit, breeding ground, food supply, plant, seed, soil, area, material or environment in which the animal pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from animal attack or infestation with a pesticidally effective amount of at least one2-cyano-3-(halo)alkoxy-benzenesulfonamide compound of the formula (I) and/or at least one agriculturally acceptable salt thereof; a method for the for the protection of seeds from soil insects and of the resulting plant's roots and shoots from soil and foliar insects comprising contacting the seeds before sowing and/or after pregermination with a 2-cyano-3-(halo)alkoxy-benzenesulfonamide compound of the general formula (I).

    Abstract translation: 本发明涉及2-氰基-3-(卤代)烷氧基 - 苯磺酰胺化合物(I),其中变量Alk和R1-R5如权利要求1中所定义,和/或其可农用盐。 此外,本发明涉及:化合物(I)和/或其盐用于对抗动物害虫的用途; 包含这种量的至少一种通式(I)的化合物和/或至少一种(I)的农业上有用的盐和至少一种惰性液体和/或固体农艺上可接受的载体的农业组合物,其具有杀虫作用 和如果需要的话,至少一种表面活性剂; 以及防治动物害虫的方法,其包括使动物害虫,其习性,繁殖场,食物供应,植物,种子,土壤,面积,动物害虫正在生长或可能生长的材料或环境,或材料,植物 (I)的至少一种2-氰基-3-(卤代)烷氧基 - 苯磺酰胺化合物和/或至少一种农业上受到保护的种子,土壤,表面或空间免于动物攻击或侵染 其可接受的盐; 一种用于保护种子免受土壤昆虫以及所得植物的根和茎由土壤和叶面昆虫引起的方法,包括在播种之前和/或在萌芽后使种子与2-氰基-3-(卤代)烷氧基 - 苯磺酰胺 通式(I)的化合物。

    COMPUESTOS DERIVADOS DE 3-AMINO-1,2-BENCISOTIAZOL COMO INSECTICIDAS

    公开(公告)号:PE20070847A1

    公开(公告)日:2007-09-21

    申请号:PE2006001454

    申请日:2006-11-15

    Applicant: BASF AG

    Abstract: SE REFIERE A COMPUESTOS DERIVADOS DE 3-AMINO-1,2-BENCISOTIAZOL DE FORMULA (I) DONDE n ES DE 0 A 2; R1 ES H, NITRO, AZIDO, AMINO, ENTRE OTROS; R2, R3 Y R4 SON CADA UNO H, HALOGENO, CIANO, AZIDO, ALQUILO(C1-C6), ENTRE OTROS; R5 ES ALQUILO(C1-C10), ALQUENILO(C2-C10), CICLOALQUILO(C3-C10), ENTRE OTROS, OPCIONALMENTE SUSTITUIDOS CON ALCOXI(C1-C10), ALQUILTIO(C1-C10), ALQUILSULFINILO(C1-C10), ENTRE OTROS SUSTITUYENTES; R6 ES ALQUILO(C1-C10), ALQUENILO(C2-C10), ALQUINILO(C2-C10), ENTRE OTROS. SON COMPUESTOS PREFERIDOS: (4-CLORO-1,1-DIOXO-1H-1?6-BENZO[d]ISOTIAZOL-3-IL)ISO-BUTIL-METIL-AMINA, ETIL-(4-METOXI-1,1-DIOXO-1H-1?6-BENZO[d]ISOTIAZOL-3-IL)-METIL-AMINA, (4-DIFLUOROMETOXI-1,1-DIOXO-1H-1?6-BENZO[d]ISOTIAZOL-3-IL)-DIETIL-AMINA, ENTRE OTROS. SE REFIERE TAMBIEN A UNA COMPOSICION. DICHOS COMPUESTOS ACTUAN COMO PLAGUICIDAS SIENDO UTILES PARA COMBATIR INSECTOS TAL COMO LOS LEPIDOPTEROS, COLEOPTEROS, DIPTEROS, ENTRE OTROS, ARACNIDOS O NEMATODOS PARASITOS DE LAS PLANTAS Y LOS QUE VIVEN EN EL SUELO

    9.
    发明专利
    未知

    公开(公告)号:BRPI0517879A

    公开(公告)日:2008-10-21

    申请号:BRPI0517879

    申请日:2005-11-24

    Applicant: BASF AG

    Abstract: The invention relates to 2-cyano-3-(halo)alkoxy-benzenesulfonamide compounds I where the variables Alk and R1 to R5 are as defined in claim 1, and/or to their agriculturally useful salts. Moreover, the present invention relates to the use of compounds I and/or their salts for combating animal pests; agricultural compositions comprising such an amount of at least one compound of the general formula I and/or at least one agriculturally useful salt of I and at least one inert liquid and/or solid agronomically acceptable carrier that it has a pesticidal action and, if desired, at least one surfactant; and a method of combating animal pests which comprises contacting the animal pests, their habit, breeding ground, food supply, plant, seed, soil, area, material or environment in which the animal pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from animal attack or infestation with a pesticidally effective amount of at least one 2-cyano-3-(halo)alkoxy-benzenesulfonamide compound of the formula I and/or at least one agriculturally acceptable salt thereof. a method for the for the protection of seeds from soil insects and of the resulting plant's roots and shoots from soil and foliar insects comprising contacting the seeds before sowing and/or after pregermination with a 2-cyano-3-(halo)alkoxy-benzenesulfonamide compound of the general formula I.

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