FERREDOXIN: NADP REDUCTASE INHIBITOR

    公开(公告)号:JP2000080089A

    公开(公告)日:2000-03-21

    申请号:JP18237199

    申请日:1999-06-28

    Applicant: BASF AG

    Abstract: PROBLEM TO BE SOLVED: To obtain a new ferredoxin: NADP reductase inhibitor expressed by a specific chemical structural formula, capable of being used by mixing with a noxious insecticide, a bactericide for plant pathogenic bacteria or the like, and useful as a herbicide, etc. SOLUTION: This ferredoxin: NADP reductase inhibitor is a compound of formula I [formula II expresses E/Z isomers; Y is CO or SO2; R1 to R3 are each H, a halogen, a 1-6C (halo)alkyl, a 1-6C (halo)alkoxy, a 1-6C alkoxyalkyl, a 1-6C alkylthio or the like; R4 is H or a 1-6C alkyl; R5 to R7 are each H, a halogen, cyano, a 1-30C alkyl, a 1-30C alkoxyalkyl, a 1-10C alkylthio, SO3H or the like]. Further, the compound of formula I is obtained e.g. by reacting a compound of formula III with a compound of formula IV in an inert organic solvent in the presence of a base such as triethylamine.

    7-AMINO-6-HETARYLIMIDAZOLO[1,2-A]PYRIMIDINE COMPOUNDS AND USE THEREOF FOR CONTROLLING HARMFUL FUNGI
    2.
    发明申请
    7-AMINO-6-HETARYLIMIDAZOLO[1,2-A]PYRIMIDINE COMPOUNDS AND USE THEREOF FOR CONTROLLING HARMFUL FUNGI 审中-公开
    7-氨基-6- HETARYLIMIDAZOLO并[1,2-a]嘧啶化合物和使用它们在防治有害真菌

    公开(公告)号:WO2006122740A3

    公开(公告)日:2007-02-22

    申请号:PCT/EP2006004573

    申请日:2006-05-15

    Inventor: WAGNER OLIVER

    CPC classification number: C07D487/04 A01N43/90

    Abstract: The invention relates to novel 7-amino-6-hetarylimidazolo[1,2-a]pyrimidine compounds of formula (I), the salts thereof, the use of said compounds for controlling harmful fungi, and agricultural pesticides containing at least one such compound as an active component. The substituents Het, X, Y 1 , and Y 2 in formula (I) have the following meanings: Het represents a five-membered or six-membered heteroaromatic radical which can contain one, two, three, or four heteroatoms selected among O, S, and N as ring members, said five-membered or six-membered heteroaromatic radical being optionally provided with one, two, three, or four identical or different substituents L; X represents hydrogen, OH, halogen, cyano, NR 3 R 4 , C 1 -C 8 alkyl, C 1 -C 8 alkoxy, C 1 -C 8 alkylthio, C 1 -C 8 alkylsulfinyl, C 1 -C 8 alkylsulfonyl, C 2 -C 8 alkenyl, or C 2 -C 8 alkinyl, the seven latter radicals being optionally halogenated in full or in part and/or optionally carrying one, two, or three substituents selected among nitro, cyano, C 1 -C 2 alkoxy, C 1 -C 4 alkoxycarbonyl, amino, C 1 -C 4 alkylamino, and di-C 1 -C 4 alkylamino. R 3 and R 4 independently have the meanings indicated for R 1 or R 2 ; Y 1 , Y 2 independently represent hydrogen, halogen, cyano, C 1 -C 4 alkyl, C 1 -C 4 alkyl halide, C 3 -C 7 cycloalkyl, C 1 -C 4 alkoxy, C 1 -C 4 alkylthio, C 1 -C 4 alkylsulfinyl, C 1 -C 4 alkylsulfonyl, or C 1 -C 4 haloalkoxy; and R 1 , R 2 have the meanings indicated in the claims and the description.

    Abstract translation: 本发明涉及新颖的7-氨基-6- hetarylimidazolo [1,2-A]下式的嘧啶化合物,其包含至少一种这样的化合物作为有效成分的I和其盐以及在防治有害真菌中使用这些化合物中,和植物保护剂 , 在式I中,取代基的Het,X,Y 1 和Y 2 具有以下含义:的Het:含有5-或6-元杂芳基1,2 ,3或4个可以是O,S和N的已选择的杂原子作为环成员,其中所述5元或6元杂芳族残基1,2,3或4个相同或不同的取代基L可以包括,X:氢,OH,卤素, 氰基,NR 3 - [R 4 ,C 1 -C 8 烷基,C 1 -C 8 烷氧基,C 1 -C 8 烷硫基,C 1 -C 8 烷基亚磺酰基,C 1 -C 8 烷基磺酰基,C 2 -C 8 链烯基或C 2 -C 8 炔基,其中所述7最后提到的基团可以部分或完全卤化和/或一个,两个或三个选自硝基取代基取代, 氰基,C 1 -C 2 烷氧基,C 1 -C 4 烷氧基羰基,氨基,C < SUB> 1 -C 4 -A lkylamino和二C 1 -C 4可以烷基氨基磨损,且其中R 3 和R 4 独立地 从对方, 2 具有对于R所给出的含义 1 或R; ÿ 1 ,Y 2 彼此独立地为氢,卤素,氰基,C 1 -C 4 烷基, ç 1 -C 4 卤代烷基,C 3 -C 7 环烷基,C 1 < / SUB> -C 4 烷氧基,C 1 -C 4 烷硫基,C 1 -C < SUB> 4 烷基亚磺酰基,C 1 -C 4 烷基磺酰基或C 1 -C 4 卤代烷氧基; [R 1 ,R 2 具有权利要求书和说明书中给出的含义。

    3-HETEROARYL SUBSTITUTED 5-METHYLOXYMETHYL ISOXAZOLINES USED AS HERBICIDES
    9.
    发明申请
    3-HETEROARYL SUBSTITUTED 5-METHYLOXYMETHYL ISOXAZOLINES USED AS HERBICIDES 审中-公开
    3 - 杂芳基 - 取代的异恶唑啉5甲氧基甲基-AS除草剂

    公开(公告)号:WO03090539A8

    公开(公告)日:2004-12-16

    申请号:PCT/EP0304136

    申请日:2003-04-22

    Abstract: The invention relates to 3-heteroaryl substituted isoxazolines of formula (I), or to their salts that can be used for agricultural purposes. In said formula, the variables are defined as follows: X represents a substituted 5-membered heteroaryl comprising between one and four nitrogen atoms, or between one and three nitrogen atoms and one oxygen or sulphur atom, or one oxygen or sulphur atom, or represents a substituted 6-membered heteroaryl comprising between one and four nitrogen atoms, whereby the aforementioned 5-membered heteroaryl is not pyrazolyl or thienyl; R - R represent hydrogen, alkyl or haloalkyl; Y represents an optionally substituted aryl, or benzo[1,4]dioxonyl, benzo[1,3]dioxolanyl, 2,3-dihydrobenzofuranyl or benzimidazole, or an optionally substituted 5- to 6-membered heteroaryl. The invention also relates to methods and intermediate products for the production of said compounds, in addition to the use thereof or of agents containing the compounds for controlling undesired plants.

    Abstract translation: 本发明涉及式(I)的3- heteroarylsubstituerte异恶唑啉:其中各变量具有以下含义:X为取代的具有一至四个氮原子或具有一至三个氮原子和一个氧或硫原子,或具有5元杂芳基 一个氧或硫原子; 的或取代的具有一至四个氮原子的6元杂芳基; 其中,上述的5元杂芳基未被吡唑基或噻吩基; [R <1> - R的<7>是氢,烷基或卤代烷基; Y是任选取代的芳基,或苯并[1,4] dioxonyl,苯并[1,3]二氧戊环基,2,3-二氢苯并呋喃基或苯并咪唑; 或任选取代的5-至6-元杂芳基; 及其可农用盐,它们的制备方法和中间体; 和使用这些化合物或包含用于控制不希望的植物的装置这些化合物。

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