RESORCINE DERIVATIVES AND THEIR USE AS PESTICIDES

    公开(公告)号:WO2007054558A3

    公开(公告)日:2007-05-18

    申请号:PCT/EP2006/068329

    申请日:2006-11-10

    Abstract: This invention relates to resorcine derivatives of formula (I) wherein R 1 is phenyl or a 5- to 6-membered heteroaromatic ring which may contain 1 to 3 heteroatoms selected from oxygen, nitrogen and sulfur, wherein phenyl or the heteroaromatic ring may be fused to a ring selected from phenyl and a 5- to 6-membered saturated, partially unsaturated or aromatic heterocyclic ring which may contain 1 to 3 heteroatoms selected from oxygen, nitrogen and sulfur, wherein phenyl or the 5- to 6-membered heteroaromatic ring or the respective fused ring systems may be unsubstituted or substituted by any combination of 1 to 6 optionally substituted groups R 3 , wherein R 3 is halogen, cyano, nitro, hydroxy, mercapto, amino, alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, haloalkyl, haloalkenyl, haloalkynyl, halocycloalkyl, halocycloalkenyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, haloalkenyloxy, haloalkynyloxy, alkylthio, alkenylthio, alkynylthio, haloalkylthio, haloalkenylthio, haloalkynylthio, alkylamino, alkenylamino, alkynylamino, dialkylamino, dialkenylamino, dialkynylamino, alkyl-alkenylamino, alkyl-alkynylamino, alkenyl- alkynylamino, trialkylsilyl, or phenyl or a 5-to 7-membered saturated or partially unsaturated heterocyclic ring which may contain 1 to 3 heteroatoms selected from oxygen, sulfur and nitrogen or a 5- to 6-membered heteraromatic ring system which may contain 1 to 4 heteroatoms selected from oxygen, nitrogen and sulfur, which phenyl and which heteroaromatic ring may be bonded via an oxygen or a sulfur atom, or -C(=G)R a , -C(=G)OR a , -C(=G)NR a 2 , -C(=G)[N=SR a 2 ], -C(=NOR a )R a , -C(=NOR a )NR a 2 , -C(=NNR a 2 )R a , -OC(=G)-OC(=G)OR a , N=SR a 2 , -NR a C(=G)R a , -N[C(=G)R a ] 2 , - NR a C(=G)OR a , -C(=G)NR a -NR a 2 , -C(=G)NR a -NR a [C(=G)R a ], -NR a -C(=G)NR a 2 , -NR a -NR a C(=G)R a , -NR a -N[C(=G)R a ] 2 , -N[(C=G)R a ]-NR a 2 , -NR a -NR a [(C=G)GR a ], -NR a [(C=G)NR a 2 , -NR a [C=NR a ]R a , -NR a (C=NR a )NR a 2 , -O-NR a 2 , -O-NR a (C=G)R a , - SO 2 NR a 2 , -NR a SO 2 R a , -S(=O)R a , -S(=O) 2 R a , -SO 2 OR a , or -OSO 2 R a , wherein G is oxygen or sulfur and Ra is as defined in the description, R 2 is hydrogen, halogen, cyano, alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, haloalkynyl, alkoxy, or haloalkoxy, x is 2, 3, 4, 5, 6, or 7, or the diastereomers, enantiomers, salts or N-oxides thereof, with the proviso that R 1 is not 5-chloro-2,2,-dimethyl-2,3-dihydrobenzo[b]furan-7-yl when R 2 is hydrogen and x is 3 or 4, processes and intermediates for the preparation of compounds I, use of compounds I for combating insects, acarids, or nematodes, and a method for treating, controlling, preventing or protecting animals against infestation or infection by parasites using compounds I.

    PESTICIDAL MIXTURE
    2.
    发明申请
    PESTICIDAL MIXTURE 审中-公开
    杀菌混合物

    公开(公告)号:WO2006128863A1

    公开(公告)日:2006-12-07

    申请号:PCT/EP2006/062714

    申请日:2006-05-30

    CPC classification number: A01N37/52 A01N2300/00

    Abstract: Pesticidal mixtures comprising, as active components 1 ) a compound of the formula I wherein W is CI or CF 3 ; X and Y are each independently CI or Br; R 1 is alkyl, alkenyl, alkynyl, or cycloalkyl optionally substituted with 1 to 3 halogens, or alkyl which is substituted by alkoxy; R 2 and R 3 are alkyl or may be taken together to form cycloalkyl optionally substituted by 1 to 3 halogens; R 4 is H or C 1 -C 8 -alkyl, or the enantiomers or salts thereof, and a Compound II selected from organo(thio)phosphates, carbamates, pyrethroids, growth regulators, nicotinic receptor agonists/antagonists Compounds, GABA antagonist compounds, macrocyclic lactone insecticides, METI I acaricides, METI II and III compounds, uncoupler compounds, oxidative phosphorylation inhibitor compounds, moulting disruptor compounds, mixed function oxidase inhibitor compounds, sodium channel blocker compounds, and other various pesticide compounds. In synergistically effective amounts, methods for the control of insects or acarids by contacting them or their food suppiy, habitat, breeding grounds or their locus with mixtures of the compound I with a compound II, a method of protecting plants from attack or infestation by insects or acarids employing mixtures of the compound I with a compound II, and a process for the preparation of a composition for treating, controlling, preventing or protecting a warm-blooded animal or a fish against infestation or infection by insects or acarids which comprises a pesticidally effective amount of a mixture of the compound I with a compound II.

    Abstract translation: 包含作为活性组分的农药混合物1)式I化合物,其中W是Cl或CF 3; X和Y各自独立地为Cl或Br; R 1是任选被1至3个卤素取代的烷基,烯基,炔基或环烷基,或被烷氧基取代的烷基; R 2和R 3是烷基或可以一起形成任选被1至3个卤素取代的环烷基; R 4是H或C 1 -C 8 - 烷基,或其对映异构体或盐,和选自有机(硫代) )磷酸盐,氨基甲酸盐,拟除虫菊酯,生长调节剂,烟碱受体激动剂/拮抗剂化合物,GABA拮抗剂化合物,大环内酯杀虫剂,METI I杀螨剂,METI II和III化合物,解偶联剂化合物,氧化磷酸化抑制剂化合物,蜕皮破坏剂化合物,混合功能氧化酶 抑制剂化合物,钠通道阻断剂化合物等各种农药化合物。 通过协同有效的量,通过将化合物I与化合物II的混合物接触或控制昆虫或螨的食物,栖息地,繁殖地或其位点与昆虫或螨虫的控制方法,保护植物免受昆虫侵袭或侵袭的方法 或使用化合物I与化合物II的混合物的吖啶,以及制备用于治疗,控制,预防或保护温血动物或鱼类以防止昆虫或螨虫侵染或感染的组合物的方法,其包括农药 有效量的化合物I与化合物II的混合物。

    PESTICIDAL MIXTURES
    3.
    发明申请
    PESTICIDAL MIXTURES 审中-公开
    农药混合物

    公开(公告)号:WO2007082841A2

    公开(公告)日:2007-07-26

    申请号:PCT/EP2007/050280

    申请日:2007-01-12

    CPC classification number: A01N43/56 A01N2300/00

    Abstract: Pesticidal mixtures comprising, as active components, 1 ) an anthranilamid compound of the formula I wherein Q is H, Cl, Cr, I, CN or methyl; B 1 is halogen, alkyl, haloalkyl, or haloalkoxy; B 2 is halogen, haloalkyl, alkoxy, haloalkoxy, alkenyloxy, alkynyloxy, alkylthio, haloalkylthio, alkylsulfinyl, haloalkylsulfinyl, alkylsulfonyl, haloalkylsulfonyl, alkyl- S(=O) x -O- or haloalkyl S(O) x -O-, wherein x is 1 or 2 and the alkoxy radical may be substituted, or C(R i )=N-OR j , C(R i )=N(R j R k ), wherein R i , R j and R k are hydrogen or alkyl; R is hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, alkylene-cycloalkyl, wherein these groups are optionally substituted; R 1 is F, CI, Br, methyl or trifluoromethyl; or the enantiomers or salts or N-oxides thereof, n is 1 , 2 or 3; and 2) one or more compounds II selected from group A consisting of organo(thio)- phosphates, carbamates, pyrethroids, growth regulators, nicotinic receptor agonists/antagonists compounds, GABA antagonist compounds, macrocyclic lactone insecticides, METI I acaricides, METI II and III compounds, uncoupler compounds, oxidative phosphorylation inhibitor compounds, mixed function oxidase inhibitor compounds, sodium channel blocker compounds and others, all as defined in the description, in synergistically effective amounts, use of these mixture for combating insects, arachnids or nematodes in and on plants and for the protection of seeds, and for treating, controlling, preventing or protecting a warm-blooded animal or a fish against infestation or infection by parasites.

    Abstract translation: 作为活性组分的农药混合物,1)式I的氨基甲酰胺化合物,其中Q是H,Cl,Cr,I,CN或甲基; B 1是卤素,烷基,卤代烷基或卤代烷氧基; B 2是卤素,卤代烷基,烷氧基,卤代烷氧基,烯氧基,炔氧基,烷硫基,卤代烷硫基,烷基亚磺酰基,卤代烷基亚磺酰基,烷基磺酰基,卤代烷基磺酰基,烷基-S(= O) O-或卤代烷基S(O)x -O-,其中x为1或2,烷氧基可以被取代,或C(R i)= N- C(R i,R i)= N(R i,R k)),其中R 0, R i,R j和R k都是氢或烷基; R是氢,烷基,烯基,炔基,环烷基,亚烷基 - 环烷基,其中这些基团是任选取代的; R 1是F,Cl,Br,甲基或三氟甲基; 或其对映异构体或其盐或N-氧化物,n为1,2或3; 和2)一种或多种选自有机(硫代) - 磷酸酯,氨基甲酸酯,拟除虫菊酯,生长调节剂,烟碱受体激动剂/拮抗剂化合物,GABA拮抗剂化合物,大环内酯杀虫剂,METI I杀螨剂,METI II和 III化合物,非偶联剂化合物,氧化磷酸化抑制剂化合物,混合功能氧化酶抑制剂化合物,钠通道阻断剂化合物和其他,如描述中所定义的,协同有效量的这些混合物用于对抗昆虫,蜘蛛或线虫 植物和保护种子,以及用于治疗,控制,预防或保护温血动物或鱼类免受寄生虫感染或感染。

    METHOD OF COMBATING ROOT WEEVILS
    4.
    发明申请
    METHOD OF COMBATING ROOT WEEVILS 审中-公开
    组合根部周围的方法

    公开(公告)号:WO2007077147A1

    公开(公告)日:2007-07-12

    申请号:PCT/EP2006/070073

    申请日:2006-12-21

    CPC classification number: A01N37/52

    Abstract: A method of combating root weevils comprising contacting the root weevils or their food supply, habitat, breeding grounds or their locus with a pesticidally effective amount of a compound of the formula (I) wherein W is Cl or CF 3 ; X and Y are each independently Cl or Br; R 1 is alkyl, alkenyl, alkynyl, or cycloalkyl optionally substituted with 1 to 3 halogens, or alkyl which is substituted by alkoxy; R 2 and R 3 are alkyl or may be taken together to form cycloalkyl optionally substituted by 1 to 3 halogens; R 4 is H or C 1 -C 6 -alkyl, or the enantiomers or salts thereof.

    Abstract translation: 一种防治根象鼻虫的方法,包括使根象鼻虫或其食物供应,栖息地,繁殖地或其基因座与杀虫有效量的式(I)化合物(其中W是Cl或CF 3) >; X和Y各自独立地为Cl或Br; R 1是被1至3个卤素任选取代的烷基,烯基,炔基或环烷基,或被烷氧基取代的烷基; R 2和R 3是烷基或可以一起形成任选被1至3个卤素取代的环烷基; R 4是H或C 1 -C 6 - 烷基,或其对映异构体或盐。

    1-(1,2-DIPHENYL-ETHYL)-3-(2-HYDROXYETHYL)-THIOUREA COMPOUNDS FOR COMBATING ANIMAL PESTS
    5.
    发明申请
    1-(1,2-DIPHENYL-ETHYL)-3-(2-HYDROXYETHYL)-THIOUREA COMPOUNDS FOR COMBATING ANIMAL PESTS 审中-公开
    1-(1,2-二苯基乙基)-3-(2-羟基乙基) - 硫脲化合物,用于组合动物饲料

    公开(公告)号:WO2006125745A2

    公开(公告)日:2006-11-30

    申请号:PCT/EP2006/062413

    申请日:2006-05-18

    CPC classification number: C07C335/12 A01N47/28

    Abstract: The present invention relates to a method of combating animal pests which comprises contacting the animal pest, their habit, breeding ground, food supply, plant, seed, soil, area, material or environment in which the animal pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from animal at- tack or infestation, with a pesticidally effective amount of at least one 1-(1 ,2-diphenyl- ethyl)-3-(2-hydroxyethyl)-thiourea compound I or an agriculturally acceptable salt thereof, wherein m is 0 to 5, n is 0 to 5, R 3 and R 4 are H or optionally substituted alkyl, haloalkyl, cycloalkyl, phenyl or benzyl, R 7 , R 8 , R 9 and R 10 are H or optionally substituted C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, C 1 -C 6 - alkylamino, C 1 -C 6 -alkoxy, C 3 -C 6 -cycloalkyl, phenyl or benzyl and the variables R 1 , R 2 , R 5 and R 6 are as defined in the claims. The invention relates also to a method for protecting crops from attack or infestation by animal pests, a method for protecting non-living materials from attack or infestation by animal pests, novel 1-(1 ,2-diphenyl-ethyl)-3-(2-hydroxyethyl)-thiourea compounds I and their agriculturally acceptable salts as well as to an agricultural composition comprising a 1-(1 ,2-diphenyl-ethyl)-3-(2-hydroxyethyl)-thiourea compound I or a salt thereof.

    Abstract translation: 本发明涉及一种防治动物害虫的方法,包括使动物害虫,其习惯,繁殖地,食物供应,植物,种子,土壤,区域,动物害虫生长或可能生长的物质或环境接触,或 防止动物死亡或侵染的材料,植物,种子,土壤,表面或空间,具有杀虫有效量的至少一种1-(1,2-二苯基 - 乙基)-3-(2-羟乙基 ) - 硫脲化合物I或其农业上可接受的盐,其中m为0至5,n为0至5,R 3和R 4为H或任选取代的烷基 ,卤代烷基,环烷基,苯基或苄基,R 7,R 8,R 9和R 10是H 或任选取代的C 1 -C 6 - 烷基,C 1 -C 6 - 卤代烷基,C 1,R 2,R 5和R 6如权利要求中所定义。 本发明还涉及一种保护作物免受动物害虫侵袭或侵袭的方法,一种保护非生物材料免受动物害虫侵袭或侵染的方法,新的1-(1,2-二苯基 - 乙基)-3-( 2-羟乙基) - 硫脲化合物I及其农业上可接受的盐,以及包含1-(1,2-二苯基 - 乙基)-3-(2-羟乙基) - 硫脲化合物I或其盐的农业组合物。

    O-CARBOXYMETHYL OXIME ETHER COMPOUNDS FOR COMBATING ARTHROPOD PESTS
    7.
    发明申请
    O-CARBOXYMETHYL OXIME ETHER COMPOUNDS FOR COMBATING ARTHROPOD PESTS 审中-公开
    用于组合牙周病的O-羧甲氧基醚化合物

    公开(公告)号:WO2007118896A1

    公开(公告)日:2007-10-25

    申请号:PCT/EP2007/053803

    申请日:2007-04-18

    CPC classification number: C07C251/60 A01N37/26 C07D307/81 C07D333/58

    Abstract: The present invention relates to new O-carboxymethyl oxime ether compounds which are useful for combating arthropod pests, in particular insects or arachnids. This object is achieved by compounds of formula (I) as defined below and by the agriculturally or veterinably acceptable salts thereof. The invention also relates to a method for combating arthropod pests. In formula (I) ..... is absent or a covalent bond; k is 0, 1, 2, 3 or 4; Cy is a 5- or 6-membered carbocyclic radical or a heterocyclic radical with 1, 2, 3 or 4 heteroatoms which are selected, from O, N and S; R a is inter alia halogen, cyano, nitro, hydroxy, C 1 -C 10 -alkyl, C 1 -C 10 -haloalkyl, C 1 -C 10 -alkoxy, (C 1 -C 10 -alkyl)carbonyl, NR 7 R 8 , CO-NR 7 R 8 and phenoxy, which may be unsubstituted or may carry 1, 2, 3, 4 or 5 substituents, or two vicinal radicals R a together may also be a bivalent radical, thereby forming a 5- to 7-membered fused heterocycle; R 1 , R 2 and R 3 are inter alia hydrogen, C 1 -C 10 -alkyl, C 1 -C 10 -haloalkyl, C 3 -C 10 -cycloalkyl, C 2 -C 10 -alkenyl, cyano, nitro, hydroxy, C 1 -C 10 -alkoxy, phenyl and pyridyl, wherein the aromatic ring of the 2 last mentioned radicals may be unsubstituted or may carry 1, 2, 3, 4 or substituents; R 4 is inter alia hydrogen, halogen, cyano, nitro, hydroxy, C 1 -C 10 -alkyl, C 1 -C 10 -haloalkyl, C 3 -C 10 -cylcoalkyl, C 2 -C 10 -alkenyl, C 1 -C 10 -alkoxy, (C 1 -C 10 -alkyl)carbonyl, NR 17 R 18 , CO-NR 17 R 18 or phenoxy, which may be unsubstituted or may carry 1, 2, 3, 4 or 5 substituents R e ; or if Cy is phenyl, R 2 and R 4 together can also form a bivalent radical Z, which is selected inter alia from -O-, -S-, -N(R b1 )-, -O-C(O)-, -O-CH(R b2 )-, -C(O)-N(R b3 )-, -C(R b5 )=N-; R 5a is inter alia hydrogen, halogen, cyano, nitro, C 1 -C 10 - alkyl, C 1 -C 10 -haloalkyl, (C 1 -C 4 -alkoxy)-C 1 -C 4 -alkyl, C 3 -C 10 -cylcoalkyl, C 2 -C 10 -alkenyl, C 1 -C 10 - alkoxy, pyridyl, phenyl, benzyl and phenoxy, wherein the aromatic ring of the 6 last mentioned radicals may be unsubstituted or may carry 1, 2, 3, 4 or substituents R f ; R 5b is hydrogen, halogen, C 1 -C 4 -alkyl or C 1 -C 4 -alkoxy; or R 5a and R 5b together can also form a bivalent radical Y; R 6 is inter alia hydrogen, C 1 -C 10 -alkyl, C 1 -C 10 -haloalkyl, C 3 -C 10 -cycloalkyl, C 1 -C 4 -alkoxy-C 1 -C 10 -alkyl, benzyl and hetaryl-C 1 -C 4 -alkyl wherein the aromatic ring of the 2 last mentioned radicals may be unsubstituted or may carry 1, 2, 3, 4 or substituents R h .

    Abstract translation: 本发明涉及新的O-羧甲基肟醚化合物,其可用于防治节肢动物害虫,特别是昆虫或蛛形纲虫。 该目的通过如下定义的式(I)化合物和其农业上或可兽医学上可接受的盐来实现。 本发明还涉及一种防治节肢动物害虫的方法。 式(I)中不存在或共价键; k为0,1,2,3或4; Cy是选自O,N和S的5或6元碳环基或具有1,2,3或4个杂原子的杂环基; 卤素,氰基,硝基,羟基,C 1 -C 10 - 烷基,C 1〜 C 1 -C 10 - 卤代烷基,C 1 -C 10 - 烷氧基,(C 1 -C 3 - 亚烷基) C 10 -C 10 - 烷基)羰基,NR 7 R 8,CO-NR 7 R 8, 和苯氧基,其可以是未取代的或可以带有1,2,3,4或5个取代基,或两个连环基R a一起也可以是二价基团,从而形成5-至7- 元稠合杂环; R 1,R 2和R 3特别是氢,C 1 -C 10烷基, C 1 -C 10烷基,C 1 -C 10 - 卤代烷基,C 3 -C 10 - 环烷基,C 1 -C 10 - C 2 -C 10 - 烯基,氰基,硝基,羟基,C 1 -C 10 - 烷氧基,C 1 -C 10 - 苯基和吡啶基,其中最后提到的2个基团的芳环可以是未取代的或可以带有1,2,3,4或取代基; R 4尤其是氢,卤素,氰基,硝基,羟基,C 1 -C 10 - 烷基,C 1 - C 1 -C 10 - 卤代烷基,C 3 -C 10 - 环烷基,C 2 -C 3 - C 1 -C 10烷基,C 1 -C 10 - 烷氧基,(C 1 -C 10 - C 1-4烷基)羰基,NR 17 R 18,CO-NR 17 R 18或苯氧基,其中 可以是未取代的或可以携带1,2,3,4或5个取代基R e; 或者如果Cy是苯基,R 2和R 4一起也可以形成二价基团Z,其特别是从-O - , - S - , - N (R b1) - , - OC(O) - , - O-CH(R b2) - , - (O)-N(R b) ) - , - (R b5)= N-; R 5a尤其是氢,卤素,氰基,硝基,C 1 -C 10 - 烷基,C 1〜 C 1 -C 10 - 卤代烷基,(C 1 -C 4 -C 4 - 烷氧基)-C 1 -C C 1-4烷基,C 3 -C 10 - C 1 -C 10烷基,C 2 -C 10 - 烷基,C 3 -C 10 - → - 烯基,C 1 -C 10 - 烷氧基,吡啶基,苯基,苄基和苯氧基,其中最后提到的6个基团的芳环可以是未取代的或可以携带 1,2,3或4或取代基R f; R 5b是氢,卤素,C 1 -C 4 - 烷基或C 1 -C 3 - 4 - 烷氧基; 或R 5a和R 5b一起也可以形成二价基团Y; R 6尤其是氢,C 1 -C 10 - 烷基,C 1 -C 3 - 10个 - 卤代烷基,C 3 -C 10 - 环烷基,C 1 -C 4 - 烷氧基-C 1 -C 10 - 烷基,苄基和杂芳基-C 1 -C 4 - 烷基,其中 最后提到的2个基团的芳环可以是未取代的或可以携带1,2,3,4或取代基R h。

    THE USE OF N-ARYLHYDRAZINE DERIVATIVES FOR COMBATING PESTS IN AND ON ANIMALS
    9.
    发明申请
    THE USE OF N-ARYLHYDRAZINE DERIVATIVES FOR COMBATING PESTS IN AND ON ANIMALS 审中-公开
    N-芳基肼衍生物在动物中和动物中的应用

    公开(公告)号:WO2005053402A2

    公开(公告)日:2005-06-16

    申请号:PCT/EP2004/013685

    申请日:2004-12-02

    CPC classification number: A01N37/52

    Abstract: Use of compounds of formula (I) wherein Q is (II), (III), or (IV) ; X 1 is chlorine, bromine, or fluorine; R 1 , R 2 are each independently H, alkyl, alkenyl, alkynyl, or cycloalkyl, alkylamino, dialkylamino, alkylcarbonylamino, alkylsulfonyl, or alkylsulfinyl, wherein the carbon atoms in these groups may be substituted, or R 1 and R 2 may be taken together to form a ring represented by the structure (V); p,m are 1, 2 or 3; X' is oxygen, sulfur, amino, alkylamino, phenylamino, or methylene; Z is alkyl or phenyl; R 3 is H, alkyl, alkenyl, alkynyl, cycloalkyl, wherein the carbon atoms in these groups may be substituted; R, R 4 are H or alkyl, alkoxycarbonyl, alkylaminocarbonyl, or dialkylaminocarbonyl, wherein the carbon atoms in the these groups may be substituted; A is C-R 5 or N; B is C-R 6 or N; W is C-R 7 or N; with the proviso that one of A, B and W is other than N; R 5 , R 6 , R 7 are H, halogen, nitro, cyano, amino, mercapto, hydroxy, alkyl, alkenyl, alkynyl, cycloalkyl, alkoxy, alkylamino, dialkylamino, alkylthio, alkylsulfonyl, or alkylsulfinyl, wherein the carbon atoms in these groups may be substituted, a 5- to 6-membered aromatic ringsystem which may contain 1 to 4 heteroatoms selected from oxygen, sulfur and nitrogen and which may be substituted; Y is hydrogen, halogen, cyano, nitro, amino, hydroxy, mercapto, alkyl, alkenyl, alkynyl, cycloalkyl, alkoxy, alkylamino, dialkylamino, alkylthio, alkylsulfonyl, or alkylsulfinyl, wherein the carbon atoms in these groups may be substituted; n is 0, 1, or 2; for combating parasites in and on animals.

    Abstract translation: 其中Q是(II),(III)或(IV)的式(I)化合物的用途; X 1是氯,溴或氟; R 1,R 2各自独立地为H,烷基,烯基,炔基或环烷基,烷基氨基,二烷基氨基,烷基羰基氨基,烷基磺酰基或烷基亚磺酰基,其中这些中的碳原子 基团可以被取代,或者R 1和R 2可以一起形成由结构(V)表示的环; p,m是1,2或3; X'是氧,硫,氨基,烷基氨基,苯基氨基或亚甲基; Z是烷基或苯基; R 3是H,烷基,烯基,炔基,环烷基,其中这些基团中的碳原子可以被取代; R,R 4为H或烷基,烷氧基羰基,烷基氨基羰基或二烷基氨基羰基,其中这些基团中的碳原子可以被取代; A是C-R 5或N; B是C-R 6或N; W是C-R 7或N; 条件是A,B和W中的一个不是N; R 5,R 6,R 7为H,卤素,硝基,氰基,氨基,巯基,羟基,烷基,链烯基,炔基, 环烷基,烷氧基,烷基氨基,二烷基氨基,烷硫基,烷基磺酰基或烷基亚磺酰基,其中这些基团中的碳原子可被取代,可含有1-4个选自氧,硫和氮的杂原子的5-6元芳族环体系和 它可以被替代; Y是氢,卤素,氰基,硝基,氨基,羟基,巯基,烷基,烯基,炔基,环烷基,烷氧基,烷基氨基,二烷基氨基,烷硫基,烷基磺酰基或烷基亚磺酰基,其中这些基团中的碳原子可以被取代; n是0,1或2; 打击动物体内和体内的寄生虫。

    1-(1,2-DIPHENYL-ETHYL)-3-(2-HYDROXYETHYL)-THIOUREA COMPOUNDS FOR COMBATING ANIMAL PESTS
    10.
    发明公开
    1-(1,2-DIPHENYL-ETHYL)-3-(2-HYDROXYETHYL)-THIOUREA COMPOUNDS FOR COMBATING ANIMAL PESTS 审中-公开
    1-(1,2-二苯基乙基)-3-(2-羟乙基),用于控制动物害虫 - 硫脲化合物

    公开(公告)号:EP1890541A2

    公开(公告)日:2008-02-27

    申请号:EP06755247.1

    申请日:2006-05-18

    CPC classification number: C07C335/12 A01N47/28

    Abstract: The present invention relates to a method of combating animal pests which comprises contacting the animal pest, their habit, breeding ground, food supply, plant, seed, soil, area, material or environment in which the animal pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from animal at- tack or infestation, with a pesticidally effective amount of at least one 1-(1 ,2-diphenyl- ethyl)-3-(2-hydroxyethyl)-thiourea compound I or an agriculturally acceptable salt thereof, wherein m is 0 to 5, n is 0 to 5, R3 and R4 are H or optionally substituted alkyl, haloalkyl, cycloalkyl, phenyl or benzyl, R7, R8, R9 and R10 are H or optionally substituted C1-C6-alkyl, C1-C6-haloalkyl, C1-C6- alkylamino, C1-C6-alkoxy, C3-C6-cycloalkyl, phenyl or benzyl and the variables R1, R2, R5 and R6 are as defined in the claims. The invention relates also to a method for protecting crops from attack or infestation by animal pests, a method for protecting non-living materials from attack or infestation by animal pests, novel 1-(1 ,2-diphenyl-ethyl)-3-(2-hydroxyethyl)-thiourea compounds I and their agriculturally acceptable salts as well as to an agricultural composition comprising a 1-(1 ,2-diphenyl-ethyl)-3-(2-hydroxyethyl)-thiourea compound I or a salt thereof.

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