公开(公告)号：US20160102103A1

公开(公告)日：2016-04-14

申请号：US14892389

申请日：2014-05-14

Applicant: BASF SE

Inventor： Gilbert BESONG ,  Matthias WITSCHEL ,  Ruediger REINGRUBER ,  Helmut KRAUS ,  Thomas SEITZ ,  Liliana PARRA-RAPADO ,  Trevor William NEWTON ,  Gerd KRAEMER ,  Richard Roger EVANS ,  Michael RACK

IPC: C07D495/04 ,  A01N43/90

CPC classification number: C07D495/04 ,  A01N43/90

Abstract: The present invention provides a substituted pyridine compound of the formula I or an agriculturally suitable salt or N-oxide thereof, wherein the variables in the formula I are defined as in the description. Substituted pyridine compounds of formula I are useful as herbicides.

Abstract translation: 本发明提供式I的取代的吡啶化合物或其农业上合适的盐或N-氧化物，其中式I中的变量如说明书所定义。 式I的取代的吡啶化合物可用作除草剂。

公开(公告)号：US20160311747A1

公开(公告)日：2016-10-27

申请号：US15102353

申请日：2014-12-10

Applicant: BASF SE

Inventor： Eric George KLAUBER ,  Michael RACK ,  Thomas ZIERKE ,  Nicole HOLUB ,  David CORTES ,  Gerald SCHMELEBECK ,  Junmin JI

IPC: C07C51/367 ,  C07C51/08

CPC classification number: C07C51/367 ,  C07C45/64 ,  C07C51/08 ,  C07C67/31 ,  C07C253/30 ,  C07C255/54 ,  C07C65/05 ,  C07C69/84 ,  C07C49/825

Abstract: The present invention relates to a process for providing dihalogen substituted salicylic acid derivatives of formula (II):

公开(公告)号：US20160251294A1

公开(公告)日：2016-09-01

申请号：US15026715

申请日：2014-09-25

Applicant: BASF SE

Inventor： Gerald SCHMELEBECK ,  Junmin JI ,  Eric George KLAUBER ,  Michael RACK ,  Thomas ZIERKE ,  Nicole HOLUB ,  David CORTES

IPC: C07C51/09 ,  C07F1/00 ,  C07C67/00 ,  C07C37/02

CPC classification number: C07C51/09 ,  A01N37/40 ,  C07C37/02 ,  C07C51/15 ,  C07C51/367 ,  C07C67/00 ,  C07F1/005 ,  C07C39/30 ,  C07C65/05 ,  C07C65/21

Abstract: The present invention relates to a process for providing a compound of formula (I): wherein Hal is a halogen, the process comprising the step of: reacting a compound of formula (II) wherein Hal is defined as above, with an alkali metal sulfite of the formula X2SO3 and an alkali metal hydroxide of the formula YOH, wherein X and Y are independently selected from an alkali metal.

Abstract translation: 本发明涉及提供式（I）化合物的方法：其中Hal为卤素，该方法包括以下步骤：使其中Hal如上定义的式（II）化合物与碱金属亚硫酸盐反应 的式X 2 SO 3和式YOH的碱金属氢氧化物，其中X和Y独立地选自碱金属。

公开(公告)号：US20160137615A1

公开(公告)日：2016-05-19

申请号：US14899755

申请日：2014-06-17

Applicant: BASF SE

Inventor： Timo FRASSETTO ,  Maximilian DOCHNAHL ,  Michael RACK ,  Volker MAYWALD ,  Bernd WOLF ,  Roland GOETZ ,  Philip MUELHEIMS ,  Rudolf HAEBERLE

IPC: C07D265/36

CPC classification number: C07D265/36 ,  C07C17/16 ,  C07D413/04 ,  C07C21/22

Abstract: The present invention relates to a process for manufacturing 4-propargylated amino-benzoxazinones of formula (I), comprising the following steps: step a) preparing propargyl chloride by reacting propargyl alcohol with thionyl chloride optionally in the presence of a catalyst; and step b) reacting the propargyl chloride prepared in step (a) with a NH-benzoxazinone of formula (II); wherein the variables are defined according to the description.

Abstract translation: 本发明涉及制备式（I）的4-炔丙基化苯并恶嗪酮的方法，包括以下步骤：步骤a）任选地在催化剂存在下，通过炔丙醇与亚硫酰氯反应制备炔丙基氯; 和步骤b）使步骤（a）中制备的炔丙基氯与式（II）的NH-苯并嗪酮反应; 其中根据描述定义变量。

公开(公告)号：US20130041147A1

公开(公告)日：2013-02-14

申请号：US13653615

申请日：2012-10-17

Applicant: BASF SE

Inventor： Thomas ZIERKE ,  Volker MAYWALD ,  Michael RACK ,  Sebastian Peer SMIDT ,  Michael KEIL ,  Bernd WOLF ,  Christopher KORADIN

IPC: C07D231/14 ,  C07D265/30 ,  C07D295/145

CPC classification number: C07D231/14 ,  C07C229/30 ,  C07D295/145

Abstract: The present invention relates to a process for preparing difluoromethyl-substituted pyrazol-4-ylcarboxylic acids and their esters, 2-(aminomethylidene)-4,4-difluoro-3- oxobutteric esters of the formula (I) in which R1, R2 and R3 independently of one another are C1-C6-alkyl, C1-C6-haloalkyl, C2-C6-alkenyl, C3-C10-cycloalkyl or benzyl or NR2R3 is a 5- to 10-membered heterocyclic radical, to a process for preparing compounds of the formula (I) wherein an appropriate 3-aminoacrylic ester is reacted with difluoroacetyl fluoride and to the use of compounds of the formula (I) in the process for preparing difluoromethyl-substituted pyrazol-4-ylcarboxylic acids and their esters.

Abstract translation: 本发明涉及一种制备二氟甲基取代的吡唑-4-基羧酸及其酯的式（I）的2-（氨基亚甲基）-4,4-二氟-3-氧代异丁酯，其中R1，R2和 R 3彼此独立地是C 1 -C 6 - 烷基，C 1 -C 6 - 卤代烷基，C 2 -C 6 - 烯基，C 3 -C 10 - 环烷基或苄基或NR 2 R 3是5-至10-元杂环基， 式（I）的化合物，其中适当的3-氨基丙烯酸酯与二氟乙酰氟反应，以及在制备二氟甲基取代的吡唑-4-基羧酸及其酯的方法中使用式（I）的化合物。

公开(公告)号：US20200055872A1

公开(公告)日：2020-02-20

申请号：US16608290

申请日：2018-04-25

Applicant: BASF SE

Inventor： Harish SHINDE ,  Christopher KORADIN ,  Joachim DICKHAUT ,  Roland GOETZ ,  Michael RACK ,  Eric George KLAUBER ,  Sukunath NARAYANAN ,  Dhanyakumar RAUT

IPC: C07D513/04 ,  C07D417/04 ,  C07D277/32

Abstract: The present invention relates to a process for preparing optically active compounds of formula X and intermediates thereof, wherein the variables of compound of formula X are as defined in the claims or the description.

公开(公告)号：US20170121343A1

公开(公告)日：2017-05-04

申请号：US15304126

申请日：2015-04-07

Applicant: BASF SE

Inventor： Gilbert BESONG ,  Matthias WITSCHEL ,  Ruediger REINGRUBER ,  Helmut KRAUS ,  Thomas SEITZ ,  Liliana PARRA RAPADO ,  Trevor William NEWTON ,  Gerd KRAEMER ,  Richard Roger EVANS ,  Michael RACK

IPC: C07D495/04 ,  A01N43/90

CPC classification number: C07D495/04 ,  A01N43/90

Abstract: The present invention provides a substituted pyridine compound of the formula I or an agriculturally suitable salt or N-oxide thereof, wherein the variables in the formula I are defined as in the description. Substituted pyridine compounds of formula I are useful as herbicides.

公开(公告)号：US20170008824A1

公开(公告)日：2017-01-12

申请号：US15119654

申请日：2015-02-19

Applicant: BASF SE

Inventor： Eric George KLAUBER ,  Michael RACK ,  Thomas ZIERKE ,  Nicole HOLUB ,  Gerald SCHMELEBECK ,  Junmin JI ,  David CORTES

IPC: C07C41/16 ,  C07C51/16 ,  C07C37/62

CPC classification number: C07C41/16 ,  C07C37/02 ,  C07C37/62 ,  C07C51/16 ,  C07C51/285 ,  C07C65/21 ,  C07C43/225 ,  C07C39/30 ,  C07C39/28

Abstract: The present invention relates to a process for providing a compound of formula (IV): wherein R1 and R2 are each independently C1-C4 alkyl, and Hal is independently Cl or Br, the process comprising the steps of: (i) reacting a compound of formula (II) wherein R1 and Hal is defined as above, to obtain a compound of formula (III) wherein R1 and Hal is defined as above, and (ii) reacting the compound of formula (III) to obtain the compound of formula (IV).

Abstract translation: 其中R1和Hal如上定义，和（ii）使式（III）化合物反应得到式（IV）化合物。

公开(公告)号：US20150299148A1

公开(公告)日：2015-10-22

申请号：US14421348

申请日：2013-08-07

Applicant: BASF SE

Inventor： Maximilian DOCHNAHL ,  Roland GÖTZ ,  Joachim GEBHARDT ,  Uwe Josef VOGELBACHER ,  Timo FRASSETTO ,  Michael RACK ,  Volker MAYWALD ,  Bernd WOLF

IPC: C07D265/36 ,  C07D413/04

CPC classification number: C07D265/36 ,  C07D413/04

Abstract: The present invention relates to carbamat-benzoxazinones of formula (I), wherein the variables are defined according to the description, as well as to a process for manufacturing carbamat-benzoxazinones of formula (I), and to the use of carbamat-benzoxazinones of formula (I) in manufacturing benzoxazinones of formula (X).

Abstract translation: 本发明涉及式（I）的氨基甲酰 - 苯并恶嗪酮，其中根据描述定义变量，以及制备式（I）的氨基甲酰 - 苯并恶嗪酮的方法，以及使用式（I）的氨基甲酰 - 苯并恶嗪酮 式（I）在制备式（X）的苯并恶嗪酮时。

公开(公告)号：US20130079513A1

公开(公告)日：2013-03-28

申请号：US13682246

申请日：2012-11-20

Applicant: BASF SE

Inventor： Thomas SCHMIDT ,  Michael PUHL ,  Joachim DICKHAUT ,  Henricus BASTIAANS ,  Michael RACK ,  Deborah L. CULBERTSON ,  Douglas D. ANSPAUGH ,  Franz-Josef BRAUN ,  Toni BUCCI ,  Henry Van Tuyl COTTER ,  David G. KUHN ,  Hassan OLOUMI-SADEGHI

IPC: C07D401/04 ,  C07D413/14 ,  C07D409/14 ,  C07D401/14

CPC classification number: C07D401/04 ,  A01N43/56 ,  A01N43/84 ,  C07D401/14 ,  C07D409/14 ,  C07D413/14

Abstract: N-Thio-anthranilamid compounds of formula (I) wherein A is A1 wherein the variables and the indices are as defined per the description, processes for preparing the compounds I, pesticidal compositions comprising compounds I, use of compounds I for the control of insects, acarids or nematodes, and methods for treating, controlling, preventing or protecting animals against infestation or infection by parasites by use of compounds of formula I.