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    PROCESS FOR PREPARING N-SUBSTITUTED HALOGENO ACET ANILIDES
    1.
    发明授权
    PROCESS FOR PREPARING N-SUBSTITUTED HALOGENO ACET ANILIDES 失效

    公开(公告)号：KR820000491B1

    公开(公告)日：1982-04-08

    申请号：KR780000145

    申请日：1978-01-20

    Applicant: BAYER AG

    Inventor： THOMAS RUDOLF ,  SCHMIDT R ,  DRABER W ,  EUE L

    IPC: C07D249/08 ,  C07D257/04

    Abstract: Title compds. I (R = optionally substituted N-contg. heterocycle; X,Y may be same or different, alkyl; Z = halo; n = 0, 1, 2), useful as herbicides, were prepd. by the reaction of N-halogenomethyl-halogenoacetanilide (II, Hal = halo) and heterocyclic compd.(III, M = H, alkali metal). Thus, pyrazole and triethylamine dissolved in anhydrous ethylacetate were mixed with 2,6-diethyl-N-chloromethyl-chloroacetanilide, stirred for 1hr, filtrated, washed, dewatered and recrystallized to give 2,6-diethyl-N-(pyrazol-1-yl-methyl)chloroacetanilide.

    PROCESS FOR PREPARING N-(1,2,4-ARIAZIN-5-ON-4-YL)GLYCIN DERIVATIVES
    2.
    发明授权
    PROCESS FOR PREPARING N-(1,2,4-ARIAZIN-5-ON-4-YL)GLYCIN DERIVATIVES 失效

    公开(公告)号：KR790001310B1

    公开(公告)日：1979-09-24

    申请号：KR760002237

    申请日：1976-09-10

    Applicant: BAYER AG

    Inventor： DRABER W ,  TIMMLER H ,  DICKORE K ,  EUE L ,  SCHMIDT R R

    Abstract: Title compds. (I; R1 = alkyl, alkoxy, alkyl amino ; R2 = alkyl, cycloalkyl, substituted phenyl ; R3 = H, alkyl, alkenyl ; R4 = OH-, alkoxy, alkylthio, amino, alkylamino, dialkylamino), useful as herbicide, were prepd. by reaction of 4-amino-1,2,-4-triazine-5-on(II) with glyoxalic acid or its derivs.(II) and alcohol (IV) (when R3 isn't H in I) in the presence of thickener such as benzene, xylene, toluene, dioxane, THF, and chlorinated hydrocarbone ester.

    N-benzyltriazole compounds and plant growth regulant compositions
    3.
    发明授权
    N-benzyltriazole compounds and plant growth regulant compositions 失效
    N-苄基化合物和植物生长调节剂组合物

    公开(公告)号：US3801590A

    公开(公告)日：1974-04-02

    申请号：US3801590D

    申请日：1970-12-09

    Applicant: BAYER AG

    Inventor： DRABER W ,  EUE L ,  SCHMIDT R ,  REGEL E ,  BUCHEL K

    IPC: C07D249/08 ,  C07D261/08 ,  C07D521/00 ,  C07D85/22

    CPC classification number: C07D233/56 ,  C07D231/12 ,  C07D249/08 ,  C07D261/08

    Abstract: N-BENZYLTRIAZOLES OF THE FORMULA

    (TRIAZOLYL-C(-A)(-B)-),(X)M-BENZENE

    IN WHICH TRIAZOYLY IS 1,2,4 OR 1,2,3 TRIAZOLYL WHICH MAY BE SUBSTITUTED; X IS HALOGN, TRIFLUOROMETHYL, LOWER ALKYL, LOWER ALKOXY, LOWER ALKLTHIO, ARYL, NITRO, CYCANO OR (ALKYLATED) AMINO; M IS 0, 1 OR 2; A IS OPTIONALLY SUBSTITUTED PHENYL, PYRIDYL, ALKYL OR CYCLOALKYL; AND B IS A 5-MEMBERED HETEROCYCLIC RING, E.G., N-HETEROCYCLE; AND HEIR SALT ARE OUTSTANDINGLY EFFECTIVE IN REGULATING PLANT GROWTH, E.G., INHIBITING, STIMULATING OR ALTERING PLANT GROWTH.

    Abstract translation: 新型的N-苄基三唑，其中三唑啉是可以被取代的1,2,4或1,2,3三唑; X为卤素，三氟甲基，低级烷基，低级烷氧基，低级烷硫基，芳基，硝基，氰基或（烷基化）氨基; M IS 0，1或2; A是任选取代的苯基，吡啶基，烷基或环烷基; 并且B是5元杂环，例如N-杂环; 并且它们的销售在调节植物生长，E.G.，抑制，刺激或改变植物生长方面是非常有效的。

    Substituted n-benzylimidazoles
    5.
    发明授权
    Substituted n-benzylimidazoles 失效
    取代的N-苄基咪唑

    公开(公告)号：US3709901A

    公开(公告)日：1973-01-09

    申请号：US3709901D

    申请日：1970-03-04

    Applicant: BAYER AG

    Inventor： DRABER W ,  PLEMPEL M ,  REGEL E ,  BUECHEL K

    IPC: C07D233/54 ,  C07D233/56 ,  C07D233/64 ,  C07D521/00 ,  C07D99/02

    CPC classification number: C07D233/64 ,  C07D231/12 ,  C07D233/56 ,  C07D249/08

    Abstract: SUBSTITUTED N-BENZYLIMIDAZOLES OF THE FORMULA:

    2-R1,3-(((X)M-PHENYL)-C(-A)(-B)-),4-R2,5-R3-IMIDAZOLE

    WHEREIN R1, R2 AND R3 ARE AEACH HYDROGEN, STRAIGHT OR BRANCHED CHAIN LOWER ALKYL OR STRAIGHT OR BRANCHED CHAIN LOWER AKENYL, X IS HYDROGEN, LOWER ALKYL, LOWER ALKOXY, LOWER ALKYLMERCAPTO, LOWER ALKENYLMERCAPTO, TRIFLUOROMETHYL, HALOGEN, NITRO, CYANO, AMINO OR AMINO SUBSTITUTED BY 1 OR 2 ALIPHATIC MOIETIES, M IS 1 OR 2, A IS PHENYL, SUBSTITUTED PHENYL, PYRIDYL, LOWER ALKYL OR CYCLOAKYL, B IS A 5-MEMBERED HETEROAROMATIC RING OF THE FORMULA:

    Y-(DN
    WHEREIN D IS CH OR N, E IS OXYGEN, SULPHUR, N-LOWER ALKYL OR N-ARYL, Y IS HYDROGEN, 1 OR 2 LOWER ALKYLS, 1 OR 2 HALOGENS, ARYL OR SUBSTITUTED ARYL, AND N IS 1 OR 2, ARE PRODUCED BY REACTING A COMPOUND OF THE FORMULA:

    ((X)M-PHENYL)-C(-A)(-B)-Z

    WHEREIN A, B, X AND M ARE AS ABOVE DEFINED AND Z IS CHLORINE OR BROMINE, WITH AT LEAST THE THEORETICALLY NECESSARY AMOUNT OF IMIDAZOLE, OPTIONALLY IN THE PRESENCE OF AN ACID ACCEPTOR, IN A POLAR ORGANIC SOLVENT, AT A TEMPERATURE OF FROM 20* C. TO 150* C. THESE SUBSTITUTED N-BENZYLIMIDAZOLES ARE USEFUL AS ANTIMYCOTICS AND ARE EFFECTIVE AGAINST BOTH YEASTS AND DERMATOPHYTES. THESE COMPOUNDS ARE EFFECTIVE AGAINST A WIDE RANGE OF FUNGI PATHOGENIC TO HUMANS AND ANIMALS.

    Substituted n-benzylimidazoles as antimycotic agents
    8.
    发明授权
    Substituted n-benzylimidazoles as antimycotic agents 失效
    替代N-苄基咪唑作为抗菌剂

    公开(公告)号：US3764690A

    公开(公告)日：1973-10-09

    申请号：US3764690D

    申请日：1972-03-03

    Applicant: BAYER AG

    Inventor： DRABER W ,  REGEL E ,  BUCHEL K ,  PLEMPEL M

    IPC: C07D233/54 ,  A61K27/00

    CPC classification number: C07D233/56

    Abstract: Substituted N-benzylimidazoles of the formula:

    WHEREIN

    WHEREIN A, B, X and m are as above defined and Z is chlorine or bromine, with at least the theoretically necessary amount of imidazole, optionally in the presence of an acid acceptor, in a polar organic solvent, at a temperature of from 20* to 150* C. These substituted N-benzylimidazoles are useful as antimycotics and are effective against both yeasts and dermatophytes. These compounds are effective against a wide range of fungi pathogenic to humans and animals.

    WHEREIN D is CH or N, E is oxygen, sulphur, N-lower alkyl or N-aryl, Y is hydrogen, 1 or 2 lower alkyls, 1 or 2 halogens, aryl or substituted aryl, and N IS 1 OR 2, ARE PRODUCED BY REACTING A COMPOUND OF THE FORMULA:

    WHEREIN R1, R2 and R3 are each hydrogen, straight or branched chain lower alkyl or straight or branched chain lower alkenyl, X is hydrogen, lower alkyl, lower alkoxy, lower alkylmercapto, lower alkenylmercapto, trifluoromethyl, halogen, nitro, cyano, amino or amino substituted by 1 or 2 aliphatic moieties, M IS 1 OR 2, A is phenyl; substituted phenyl, pyridyl, lower alkyl or cycloalkyl, B is a 5-membered heteroaromatic ring of the formula:

    Abstract translation: 下式的取代的N-苄基咪唑：

    Heterocyclic-substituted n-imidazol plant-growth influencing agents
    10.
    发明授权
    Heterocyclic-substituted n-imidazol plant-growth influencing agents 失效
    杂环取代的N-IMIDAZOL植物生长影响因子

    公开(公告)号：US3852056A

    公开(公告)日：1974-12-03

    申请号：US7526470

    申请日：1970-09-24

    Applicant: BAYER AG

    Inventor： SCHMIDT R ,  BUCHEL K ,  EUE L ,  DRABER W ,  REGEL E

    IPC: C07D233/58 ,  A01N43/50 ,  A01N43/80 ,  C07D233/54 ,  C07D521/00 ,  A01N9/20

    CPC classification number: C07D233/56 ,  C07D231/12 ,  C07D233/64 ,  C07D249/08

    Abstract: Compositions containing heterocyclic-substituted Nbenzylimidazoles of the formula

    WHEREIN R, R'' and R'''' are hydrogen, lower alkyl or lower alkenyl, X is hydrogen, halogen, lower alkyl, alkoxy, alkylthio, trifluoromethyl, nitro, cyano, amino or dialkylamino, M IS 0, 1 OR 2, A is unsubstituted or substituted phenyl or pyridyl, alkyl or cycloalkyl, and B is a five-membered heteroaromatic ring of the general formula:

    WHEREIN E is oxygen, sulfur

    Y is hydrogen, lower alkyl, halogen or unsubstituted or substituted aryl; and N IS 0, 1 OR 2 POSSESS MARKED PLANT-GROWTH INFLUENCING, INCLUDING INHIBITING AND PROMOTING, PROPERTIES.

    Abstract translation: 含有式WHEREIN R，R'和R“的杂环取代的N-苄基咪唑的组合物是氢，低级烷基或低级烯基，X是氢，卤素，低级烷基，烷氧基，烷硫基，三氟甲基，硝基，氰基，氨基或 二烷基氨基，M为0,1或2，A为未取代或取代的苯基或吡啶基，烷基或环烷基，B为下列通式的五元杂芳环：其中E为氧，硫为低级烷基， 卤素或未取代或取代的芳基; 和N IS 0，1或2标志性植物生长影响，包括抑制和促进，性质。

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