公开(公告)号：WO2015102024A3

公开(公告)日：2015-10-08

申请号：PCT/IN2015000004

申请日：2015-01-05

Applicant: COUNCIL SCIENT IND RES

Inventor： AHER RAVINDRA DATTATRAY ,  KUMAR BOOPATHI SENTHIL ,  SUDALAI ARUMUGAM ,  LALWANI KOMAL GIRDHARI

IPC: C07D231/04 ,  A61K31/40 ,  A61K31/401 ,  A61K31/4025 ,  A61K31/415 ,  A61K31/4155 ,  A61P31/06 ,  C07D207/48 ,  C07D405/06 ,  C07D409/06

CPC classification number: C07D207/48 ,  C07D231/04 ,  C07D405/06 ,  C07D409/06 ,  C07D498/04

Abstract: Novel substituted 5 membered heterocyclic compounds of Formula I are disclosed. The invention further discloses a process for the preparation of compounds of Formula I. The compounds find use as anti mycobacterial agents.

Abstract translation: 公开了新的式I的5元杂环化合物。 本发明还公开了制备式I化合物的方法。该化合物可用作抗分枝杆菌剂。

公开(公告)号：WO2013110998A8

公开(公告)日：2014-06-12

申请号：PCT/IB2013000083

申请日：2013-01-25

Applicant: COUNCIL SCIENT IND RES ,  AHER RAVINDRA DATTATRAY ,  GADE MADHURI HANUMANT ,  REKULA REDDY SANTHOSH ,  KARABAL PRATIBHA UTTAM ,  SURYAVANSHI GURUNATH MALLAPPA ,  SUDALAI ARUMUGAM

Inventor： AHER RAVINDRA DATTATRAY ,  GADE MADHURI HANUMANT ,  REKULA REDDY SANTHOSH ,  KARABAL PRATIBHA UTTAM ,  SURYAVANSHI GURUNATH MALLAPPA ,  SUDALAI ARUMUGAM

IPC: C07C51/15 ,  C07C57/18 ,  C07C57/42 ,  C07C59/64

CPC classification number: C07C51/15 ,  C07C57/18 ,  C07C57/42 ,  C07C59/64

Abstract: The invention provides a simple, efficient, environmental friendly catalytic system for the direct carboxylation reaction using C02 under mild condition. A single step heterogeneous catalytic process for preparation of alkynyl carboxylic acids of formula I is disclosed.

Abstract translation: 本发明提供了在温和条件下使用CO 2的直接羧化反应的简单，有效的环境友好的催化体系。 公开了用于制备式I的炔基羧酸的单步非均相催化方法。