公开(公告)号：WO2014037964A3

公开(公告)日：2014-05-01

申请号：PCT/IN2013000542

申请日：2013-09-06

Applicant: COUNCIL SCIENT IND RES

Inventor： RAWAT VARUN ,  DEY SOUMEN ,  SHELKE ANIL MARUTI ,  SURYAVANSHI GURUNATH MALLAPPA ,  SUDALAI ARUMUGAM

IPC: C07D313/00

CPC classification number: C07D313/00 ,  C07B2200/07

Abstract: The present invention discloses organocatalytic process for asymmetric synthesis of highly enantioselective decanolide compounds in high yield with > 99% ee. Further, the present invention disclose cost effective, improved organocatalytic process for asymmetric synthesis of highly enantioselective decanolides compounds from non-chiral, cheap, easily available raw materials.

Abstract translation: 本发明公开了以高达99％ee的高产率非对称合成高对映选择性癸内酯化合物的有机催化方法。 此外，本发明公开了从非手性的，便宜的，容易获得的原料不对称地合成高度对映选择性的癸内酯化合物的成本有效的改进的有机催化方法。