公开(公告)号：SE7514094A

公开(公告)日：1976-06-14

申请号：SE7514094

申请日：1975-12-12

Applicant: HOECHST AG

Inventor： SCHORR M ,  SCHRINNER E ,  SCHMITT W

IPC: C07D499/66 ,  C07D499/00 ,  C07D499/64 ,  C07D499/68 ,  C07D499/70

CPC classification number: C07D499/00

公开(公告)号：SE7514094L

公开(公告)日：1976-06-14

申请号：SE7514094

申请日：1975-12-12

Applicant: HOECHST AG

Inventor： SCHORR M ,  SCHRINNER E ,  SCHMITT W

IPC: C07D499/66 ,  C07D499/00 ,  C07D499/64 ,  C07D499/68 ,  C07D499/70

Abstract: Acylaminopenicillanic acids of the general formula in which R1, R2 and R3 represent hydrogen or lower alkyl which may be substituted, and in which the radicals R1 and R2 or R2 and R3 may form together an alkylene radical which may be substituted, R4 and R5 represent hydrogen or lower alkyl, R6 represents phenyl which may be substituted, a monocyclic aromatic heterocycle which may be substituted, or dihydrophenyl, A represents a benzene or thiophene ring which may be substituted, and X represents oxygen or a single bond, a process for preparing them and pharmaceutical compositions active against bacterial infections containing these compounds.

公开(公告)号：NO754232L

公开(公告)日：1976-06-15

申请号：NO754232

申请日：1975-12-12

Applicant: HOECHST AG

Inventor： SCHORR M ,  SCHRINNER E ,  SCHMITT W

IPC: C07D499/66 ,  C07D499/00 ,  C07D499/64 ,  C07D499/68 ,  C07D499/70 ,  C07D

Abstract: Acylaminopenicillanic acids of the general formula in which R1, R2 and R3 represent hydrogen or lower alkyl which may be substituted, and in which the radicals R1 and R2 or R2 and R3 may form together an alkylene radical which may be substituted, R4 and R5 represent hydrogen or lower alkyl, R6 represents phenyl which may be substituted, a monocyclic aromatic heterocycle which may be substituted, or dihydrophenyl, A represents a benzene or thiophene ring which may be substituted, and X represents oxygen or a single bond, a process for preparing them and pharmaceutical compositions active against bacterial infections containing these compounds.

公开(公告)号：NO754232A

公开(公告)日：1976-06-15

申请号：NO754232

申请日：1975-12-12

Applicant: HOECHST AG

Inventor： SCHORR M ,  SCHRINNER E ,  SCHMITT W

IPC: C07D499/66 ,  C07D499/00 ,  C07D499/64 ,  C07D499/68 ,  C07D499/70 ,  C07D

CPC classification number: C07D499/00

公开(公告)号：DK567375A

公开(公告)日：1976-06-14

申请号：DK567375

申请日：1975-12-12

Applicant: HOECHST AG

Inventor： SCHORR M ,  SCHRINNER E ,  SCHMITT W

IPC: C07D499/66 ,  C07D499/00 ,  C07D499/64 ,  C07D499/68 ,  C07D499/70 ,  C07D

Abstract: Acylaminopenicillanic acids of the general formula in which R1, R2 and R3 represent hydrogen or lower alkyl which may be substituted, and in which the radicals R1 and R2 or R2 and R3 may form together an alkylene radical which may be substituted, R4 and R5 represent hydrogen or lower alkyl, R6 represents phenyl which may be substituted, a monocyclic aromatic heterocycle which may be substituted, or dihydrophenyl, A represents a benzene or thiophene ring which may be substituted, and X represents oxygen or a single bond, a process for preparing them and pharmaceutical compositions active against bacterial infections containing these compounds.

公开(公告)号：DK548075A

公开(公告)日：1976-06-06

申请号：DK548075

申请日：1975-12-04

Applicant: HOECHST AG

Inventor： SCHORR M ,  SCHRINNER E ,  SCHMITT W

IPC: C07D499/00 ,  C07D499/46 ,  C07D499/64 ,  C07D

Abstract: Acylaminopenicillanic acids of the general formula in which A represents phenyl which may be substituted, an aromatic monocyclic heterocycle which may be substituted or dihydrophenyl, and X represents one of the groups -SO2-, -CO-, -P(R)- or -P(O)(R)- in which R represents low molecular weight alkyl, alkenyl, alkoxy, aralkyl, aralkoxy, aryl or aryloxy which may be substituted, non-toxic salts of these compounds and pharmaceutical compositions containing these compounds.