公开(公告)号：WO2004056177A2

公开(公告)日：2004-07-08

申请号：PCT/IB0306501

申请日：2003-10-23

Applicant: NIPPON SODA CO

Inventor： IWATAKI ISAO ,  IWASA TAKAO ,  HATANO RENPEI ,  MOYANO ELIZABETH LAURA

IPC: C07D277/20 ,  A01N43/78 ,  C07D277/32 ,  C07D277/46 ,  C07D277/54 ,  C07D277/56 ,  A01N

CPC classification number: A01N43/78

Abstract: Insecticidal aminothiazole derivatives and the use as an insecticide and acaricide of the compounds of formula (1): wherein R is cyano or fluoroalkyl, R is halogen, SCN or aryl, R is H, C1-C6 alkyl, S02R or C(O)R , R and R are, independently, aryl, phenylalkyl, alkyl, cycloalkyl groups, being optionally substituted by one or more of halogen, cyano, alkyl, alkenyl, alkynyl, haloalkyl, alkoxy, nitro, alkoxycarbonyl, alkylcarbonyloxy, alkylenedioxy, alkylcarbonyl, amino, alkylamino, haloalkoxy, alkylthio, alkylsulfonyl, haloalkenyl, alkoxycarbonylalkyl or alkoxycarbonylalkoxy; said aryl, phenylalkyl groups may additionally be fused to a cycloalkyl ring, R is C1-C 6alkyl, haloalkyl, X is 0, S, NR , R is alkyl, cycloalkyl, alkoxy, alkenylalkyloxy, alkynylalkyloxy, alkoxycarbonylalkyloxy.

Abstract translation: 杀虫氨基噻唑衍生物和式（1）化合物的杀虫剂和杀螨剂的用途：其中R 1是氰基或氟代烷基，R 2是卤素，SCN或芳基，R 3是H，C1- C 6烷基，SO 2 R 5或C（O）R 6，R 4和R 6独立地是芳基，苯基烷基，烷基，环烷基，任选地被一个或多个卤素，氰基 烷基，烯基，炔基，卤代烷基，烷氧基，硝基，烷氧基羰基，烷基羰基氧基，亚烷基二氧基，烷基羰基，氨基，烷基氨基，卤代烷氧基，烷硫基，烷基磺酰基，卤代烯基，烷氧基羰基烷基或烷氧羰基烷氧基。 所述芳基苯基烷基可另外与环烷基稠合，R 5为C 1 -C 6烷基，卤代烷基，X为0，S，NR 7，R 7为烷基，环烷基，烷氧基，烯基烷氧基， 炔基烷氧基，烷氧羰基烷氧基。

公开(公告)号：KR20200130263A

公开(公告)日：2020-11-18

申请号：KR20207024762

申请日：2019-03-08

Applicant: NIPPON SODA CO

Inventor： SAKANISHI KEITA ,  AOYAMA HIKARU ,  SAKIYAMA NORIFUMI ,  IWASA TAKAO ,  MATSUI MAKI ,  KOBAYASHI TOMOMI ,  KITAYAMA TAKASHI

IPC: C07D471/04 ,  A01N43/76 ,  A01N43/90 ,  A01N47/02 ,  A61K31/437 ,  A61K31/506 ,  A61P33/00 ,  A61P33/14 ,  C07D413/14

Abstract: 본발명은, 우수한살충활성, 살진드기, 및/또는살선충활성을갖고, 안전성이우수하며, 또한공업적으로유리하게합성할수 있는식 (I) 로나타내는화합물또는그 염, 그리고이것을유효성분으로서함유하는유해생물방제제에관한것이다. 식 (I) 중, X 는, 할로게노기, 치환혹은무치환의 C1 ∼ 6 알킬기등이며, n 은, 1 ∼ 3 중어느정수이며, Z 는, 산소원자, 황원자, 또는 NR 이며, R 은, 수소원자또는치환혹은무치환의 C1 ∼ 6 알킬기이며, A 는, 벤젠고리또는 6 원헤테로아릴고리이며, Ra 는, 치환혹은무치환의 C1 ∼ 6 알킬술포닐기이며, Rb 는, 치환혹은무치환의 C1 ∼ 6 알킬기등이다. JPEGpct00054.jpg3670

公开(公告)号：KR20200140261A

公开(公告)日：2020-12-15

申请号：KR20207027839

申请日：2019-04-03

Applicant: NIPPON SODA CO

Inventor： KATO TETSURO ,  TAKAHASHI JUN ,  SAIKI YUTO ,  IWASA TAKAO ,  SUGAHARA ERIKA

IPC: C07D401/04 ,  A01N43/56 ,  A01N43/653 ,  A01N43/90 ,  A01N47/04 ,  C07D403/04 ,  C07D403/14 ,  C07D409/04

Abstract: 식 (I) 로나타내는화합물또는그 염, 그리고그 화합물및 그염으로이루어지는군에서선택되는적어도 1 개를유효성분으로서함유하는유해생물방제제, 살충혹은살진드기제, 살선충제, 또는내부기생충방제혹은구제제. JPEGpct00031.jpg4156 (식 (I) 중, Ar1 은벤젠고리또는피리딘고리이고, R1 은 C1 ∼ 6 알킬기, 할로게노기등이고, n 은 R1 의수를나타내고또한 1, 2 또는 3 이고, n 이 2 이상일때 복수의 R1 은서로동일해도되고상이해도되고, R2 는 C1 ∼ 6 알킬기, C1 ∼ 6 할로알킬기등이고, R3 은수소원자, C1 ∼ 6 알킬기, C1 ∼ 6 알킬카르보닐기등이고, 또한 Ar2 는, 치환혹은무치환헤테로아릴기이다.)

公开(公告)号：EP1932844A4

公开(公告)日：2010-08-25

申请号：EP06811460

申请日：2006-10-06

Applicant: NIPPON SODA CO

Inventor： HAMAMOTO ISAMI ,  TAKAHASHI JUN ,  YANO MAKIO ,  KAWAGUCHI MASAHIRO ,  HANAI DAISUKE ,  IWASA TAKAO

IPC: C07D451/14 ,  A01N43/42 ,  A01N43/56 ,  A01N43/58 ,  A01N43/78 ,  A01N43/824 ,  A01N43/90 ,  A01P7/02 ,  A01P7/04 ,  C07D471/04 ,  C07D491/08

CPC classification number: C07D221/22 ,  A01N43/40 ,  A01N43/42 ,  A01N43/54 ,  A01N43/56 ,  A01N43/58 ,  A01N43/60 ,  A01N43/76 ,  A01N43/78 ,  A01N43/80 ,  A01N43/82 ,  A01N43/90 ,  C07D211/54 ,  C07D211/58 ,  C07D221/24 ,  C07D237/08 ,  C07D241/16 ,  C07D401/04 ,  C07D401/12 ,  C07D417/04

公开(公告)号：EP3135277A4

公开(公告)日：2017-11-22

申请号：EP15783087

申请日：2015-04-20

Applicant: NIPPON SODA CO

Inventor： IWASA TAKAO

IPC: A61K31/17 ,  A61K31/41 ,  A61K31/4196 ,  A61K31/426 ,  A61K31/44 ,  A61K31/4402 ,  A61K31/444 ,  A61K31/47 ,  A61K31/4709 ,  A61K31/505 ,  A61K31/506 ,  A61P33/00 ,  A61P33/10

CPC classification number: A61K31/17 ,  A61K31/41 ,  A61K31/4196 ,  A61K31/426 ,  A61K31/44 ,  A61K31/4402 ,  A61K31/444 ,  A61K31/47 ,  A61K31/4709 ,  A61K31/4965 ,  A61K31/505 ,  A61K31/506 ,  A61K31/53

Abstract: A parasite-control or parasiticide agent that exhibis excellent effects of controlling or expelling parasites, particularly endoparasites and that can be used safely contains at least one selected from the group consisting of compounds represented by formula (I) and salts thereof as an active ingredient thereof. (In the formula (I), Cy represents a heteroaryl group or the like, X represents a halogeno group or the like, n is an integer of 0 to 5, in the case where n is 2 or more, X is identical or different, R 1 represents an unsubstituted or substituted C1-6 alkyl group or the like, A represents a nitrogen atom or the like, R 2 , R 3 , and R 4 each independently represents a hydrogen atom, an unsubstituted or substituted C1-6 alkyl group, or the like, and R 5 represents an unsubstituted or substituted C6-10 aryl group, unsubstituted or substituted heteroaryl group, or the like.)

公开(公告)号：EP1731518A4

公开(公告)日：2010-04-28

申请号：EP05728646

申请日：2005-03-30

Applicant: NIPPON SODA CO

Inventor： HAMAMOTO ISAMI ,  TAKAHASHI JUN ,  YANO MAKIO ,  HANAI DAISUKE ,  IWASA TAKAO

IPC: C07D401/04 ,  A01N43/40 ,  A01N43/42 ,  A01N43/46 ,  C07D405/14 ,  C07D413/14 ,  C07D451/06

CPC classification number: A01N43/40 ,  A01N43/42 ,  C07D401/04 ,  C07D405/14 ,  C07D413/14 ,  C07D451/06

公开(公告)号：EP3181552A4

公开(公告)日：2018-01-31

申请号：EP15831879

申请日：2015-08-11

Applicant: NIPPON SODA CO

Inventor： AOYAMA HIKARU ,  MATSUI MAKI ,  IWASA TAKAO ,  FUJII KAZUSHIGE ,  KOBAYASHI TOMOMI ,  SAKANISHI KEITA

IPC: C07D233/64 ,  A01N43/50 ,  A01P7/02 ,  A01P7/04 ,  A61K31/4164 ,  A61K31/4439 ,  A61P31/00 ,  A61P33/00 ,  A61P33/10 ,  A61P33/14 ,  C07D401/04

CPC classification number: A01N43/50 ,  A01N43/54 ,  A01N43/56 ,  A01N43/58 ,  A01N43/74 ,  A61K31/4164 ,  A61K31/4439 ,  C07D233/64 ,  C07D401/04 ,  C07D401/14 ,  C07D403/04 ,  C07D405/04 ,  C07D409/04 ,  C07D417/14

Abstract: The present invention provides a compound represented by formula (I) or salt thereof (in the formula, A 1 and A 2 each independently represents a nitrogen atom or the like, B 1 , B 2 , B 3 and B 4 each independently represents a carbon atom or nitrogen atom, X 1 represents an unsubstituted or substituted C1-6 alkyl group or the like, n represents a number of X 1 and represents an integer of 0-4, R 1 represents a halogeno group or the like, R 2 represents an unsubstituted or substituted C1-6 alkyl group or the like, m represents a number of the oxide group bonding with the nitrogen atom which does not bond with R 2 on the imidazole ring, and represents 0 or 1, R 3 represents a hydrogen atom or the like, Ar represents an unsubstituted or substituted C6-10 aryl group.

公开(公告)号：EP2965627A4

公开(公告)日：2016-09-28

申请号：EP14759592

申请日：2014-02-28

Applicant: NIPPON SODA CO

Inventor： IWASA TAKAO ,  HIRATA KOICHI

IPC: A01N43/18 ,  A01N43/10 ,  A01N43/16 ,  A61K31/351 ,  A61K31/381 ,  A61K31/382 ,  A61P33/14 ,  A61P43/00 ,  C07D333/36 ,  C07D335/02

CPC classification number: A61K31/382 ,  A01N43/10 ,  A01N43/16 ,  A01N43/18 ,  A61K31/351 ,  A61K31/381 ,  C07D333/36 ,  C07D335/02

Abstract: wherein, in formula (III), X 1 represents a C1-6 alkyl group which is unsubstituted or has a substituent, or other groups; ml represents any integer of 0 to 5; A represents an oxygen atom or a sulfur atom; each of R 1 and R 2 independently represents a hydrogen atom, a C1-6 alkyl group which is unsubstituted or has a substituent, or other groups; R 5 represents a hydrogen atom or a C1-6 alkyl group which is unsubstituted or has a substituent; B represents an oxygen atom or a sulfur atom; Q 2 represents a C7-11 aralkyl group which is unsubstituted or has a substituent X 2 , or other groups; and each of R 3a , R 3b , R 4a , and R 4b independently represents a hydrogen atom, a C1-6 alkyl group which is unsubstituted or has a substituent, or other groups.

公开(公告)号：EP2322037A4

公开(公告)日：2013-07-10

申请号：EP09812840

申请日：2009-08-24

Applicant: NIPPON SODA CO

Inventor： NISHIMURA KAORU ,  IWASA TAKAO

IPC: A01N25/30 ,  A01G13/00 ,  A01N25/08 ,  A01N25/34 ,  A01N43/40 ,  A01N47/40 ,  A01N47/44 ,  A01N51/00 ,  A01P3/00 ,  A01P7/04

CPC classification number: A01G13/0237 ,  A01N25/08 ,  A01N25/30 ,  A01N25/34 ,  A01N33/04 ,  A01N47/44 ,  Y10T428/1334 ,  Y10T428/31801 ,  A01N43/40 ,  A01N47/40 ,  A01N51/00 ,  A01N2300/00 ,  A01N41/04

公开(公告)号：EP3181552A1

公开(公告)日：2017-06-21

申请号：EP15831879

申请日：2015-08-11

Applicant: NIPPON SODA CO

Inventor： AOYAMA HIKARU ,  MATSUI MAKI ,  IWASA TAKAO ,  FUJII KAZUSHIGE ,  KOBAYASHI TOMOMI ,  SAKANISHI KEITA

IPC: C07D233/64 ,  A01N43/50 ,  A01P7/02 ,  A01P7/04 ,  A61K31/4164 ,  A61K31/4439 ,  A61P31/00 ,  A61P33/00 ,  A61P33/10 ,  A61P33/14 ,  C07D401/04

CPC classification number: A01N43/50 ,  A01N43/54 ,  A01N43/56 ,  A01N43/58 ,  A01N43/74 ,  A61K31/4164 ,  A61K31/4439 ,  C07D233/64 ,  C07D401/04 ,  C07D401/14 ,  C07D403/04 ,  C07D405/04 ,  C07D409/04 ,  C07D417/14

Abstract: The present invention provides a compound represented by formula (I) or salt thereof (in the formula, A 1 and A 2 each independently represents a nitrogen atom or the like, B 1 , B 2 , B 3 and B 4 each independently represents a carbon atom or nitrogen atom, X 1 represents an unsubstituted or substituted C1-6 alkyl group or the like, n represents a number of X 1 and represents an integer of 0-4, R 1 represents a halogeno group or the like, R 2 represents an unsubstituted or substituted C1-6 alkyl group or the like, m represents a number of the oxide group bonding with the nitrogen atom which does not bond with R 2 on the imidazole ring, and represents 0 or 1, R 3 represents a hydrogen atom or the like, Ar represents an unsubstituted or substituted C6-10 aryl group.

Abstract translation: 本发明提供由式（I）表示的化合物或其盐（式中，A 1和A 2各自独立地表示氮原子等，B 1，B 2，B 3和B 4各自独立地表示 碳原子或氮原子，X 1表示未取代或取代的C 1-6烷基等，n表示X 1的数且表示0-4的整数，R 1表示卤代基等，R 2 表示未取代或取代的C 1-6烷基等，m表示与咪唑环上不与R 2键合的氮原子键合的氧化物基团的数目，并且表示0或1，R 3表示氢 原子等，Ar表示未取代或取代的C 6-10芳基。