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公开(公告)号:PL3313817T3
公开(公告)日:2021-04-06
申请号:PL16730854
申请日:2016-06-22
Applicant: SERVIER LAB , VERNALIS R&D LTD
Inventor: BÁLINT BALÁZS , CSÉKEI MÁRTON , SZABÓ ZOLTÁN , SZLÁVIK ZOLTÁN , KOTSCHY ANDRÁS , CHANRION MAÏA , GENESTE OLIVIER , CHEN I-JEN , DAVIDSON JAMES EDWARD PAUL , MURRAY JAMES BROOKE , SIPOS SZABOLCS , ONDI LEVENTE , PROSZENYÁK ÁGNES
IPC: C07D209/12 , A61K31/381 , A61K31/4355 , A61K31/437 , A61P35/00 , C07D307/80 , C07D307/81 , C07D333/56 , C07D403/12 , C07D405/04 , C07D405/12 , C07D409/12 , C07D471/04 , C07D487/04 , C07D491/04 , C07D495/04
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2.
公开(公告)号:HRP20201782T1
公开(公告)日:2021-01-22
申请号:HRP20201782
申请日:2020-11-05
Applicant: SERVIER LAB , VERNALIS R&D LTD
Inventor: BÁLINT BALÁZS , CSÉKEI MÁRTON , SZABÓ ZOLTÁN , SZLÁVIK ZOLTÁN , KOTSCHY ANDRÁS , CHANRION MAÏA , GENESTE OLIVIER , CHEN I-JEN , DAVIDSON JAMES EDWARD PAUL , MURRAY JAMES BROOKE , SIPOS SZABOLCS , ONDI LEVENTE , PROSZENYÁK ÁGNES
IPC: C07D209/12 , A61K31/381 , A61K31/4355 , A61K31/437 , A61P35/00 , C07D307/80 , C07D307/81 , C07D333/56 , C07D403/12 , C07D405/04 , C07D405/12 , C07D409/12 , C07D471/04 , C07D487/04 , C07D491/04 , C07D495/04
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公开(公告)号:DK3313817T3
公开(公告)日:2020-12-14
申请号:DK16730854
申请日:2016-06-22
Applicant: SERVIER LAB , VERNALIS R&D LTD
Inventor: GENESTE OLIVIER , CHEN I-JEN , DAVIDSON JAMES EDWARD PAUL , MURRAY JAMES BROOKE , SIPOS SZABOLCS , BÁLINT BALÁZS , CSÉKEI MÁRTON , CHANRION MAÏA , KOTSCHY ANDRÁS , ONDI LEVENTE , PROSZENYÁK ÁGNES , SZABÓ ZOLTÁN , SZLÁVIK ZOLTÁN
IPC: C07D209/12 , A61K31/381 , A61K31/4355 , A61K31/437 , A61P35/00 , C07D307/80 , C07D307/81 , C07D333/56 , C07D403/12 , C07D405/04 , C07D405/12 , C07D409/12 , C07D471/04 , C07D487/04 , C07D491/04 , C07D495/04
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公开(公告)号:AU2016282828B2
公开(公告)日:2020-07-16
申请号:AU2016282828
申请日:2016-06-22
Applicant: SERVIER LAB , VERNALIS R&D LTD
Inventor: BÁLINT BALÁZS , CSÉKEI MÁRTON , SZABÓ ZOLTÁN , SZLÁVIK ZOLTÁN , KOTSCHY ANDRÁS , CHANRION MAÏA , GENESTE OLIVIER , CHEN I-JEN , DAVIDSON JAMES EDWARD PAUL , MURRAY JAMES BROOKE , SIPOS SZABOLCS , ONDI LEVENTE , PROSZENYÁK AGNES
IPC: C07D209/12 , A61K31/381 , A61K31/4355 , A61K31/437 , A61P35/00 , C07D307/80 , C07D307/81 , C07D333/56 , C07D403/12 , C07D405/04 , C07D405/12 , C07D409/12 , C07D471/04 , C07D487/04 , C07D491/04 , C07D495/04
Abstract: Compounds of formula (I); wherein R
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5.
公开(公告)号:EA033566B1
公开(公告)日:2019-11-05
申请号:EA201890126
申请日:2016-06-22
Applicant: SERVIER LAB , VERNALIS R&D LTD
Inventor: BALINT BALAZS , CSEKEI MARTON , SZABO ZOLTAN , SZLAVIK ZOLTAN , KOTSCHY ANDRAS , CHANRION MAIA , GENESTE OLIVIER , CHEN I-JEN , DAVIDSON JAMES EDWARD PAUL , MURRAY JAMES BROOKE , SIPOS SZABOLCS , ONDI LEVENTE , PROSZENYAK AGNES
IPC: C07D209/12 , A61K31/381 , A61K31/4355 , A61K31/437 , A61P35/00 , C07D307/80 , C07D307/81 , C07D333/56 , C07D403/12 , C07D405/04 , C07D405/12 , C07D409/12 , C07D471/04 , C07D487/04 , C07D491/04 , C07D495/04
Abstract: Соединенияформулы (I)где R, R, R, R, R, R, R, R, R, A, W и n являютсятакими, какопределенов описании, иприменениесоединенийдляизготовлениялекарственныхсредств.
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公开(公告)号:TN2017000521A1
公开(公告)日:2019-04-12
申请号:TN2017000521
申请日:2016-06-22
Applicant: SERVIER LAB , VERNALIS R&D LTD
Inventor: BALINT BALAZS , BRUNO ALAIN , CHEN I-JEN , CSÉKEI MARTON , DAVIDSON JAMES EDWARD PAUL , GENESTE OLIVIER , KOTSCHY ANDRAS , MURRAY JAMES BROOKE , ONDI LEVENTE , PACZAL ATTILA , PERRON-SIERRA FRANÇOISE , PROSZENYAK AGNES , RADICS GABOR , SIPOS SZABOLCS , SZABÔ ZOLTAN , SZLAVIK ZOLTAN
IPC: A61P35/00 , A61K31/519 , A61P37/00 , C07D495/04
Abstract: Compounds of formula (1): wherein R 1 , R 2 , R 5 , R 6 ,R 7 , R 12 , X, Y, A, E and n are as defined in the description. Medicaments.
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7.
公开(公告)号:SI3313817T1
公开(公告)日:2021-01-29
申请号:SI201631022
申请日:2016-06-22
Applicant: SERVIER LAB , VERNALIS R&D LTD
Inventor: BALINT BALAZS , CSEKEI MARTON , SZABO ZOLTAN , SZLAVIK ZOLTAN , KOTSCHY ANDRAS , CHANRION MAIA , GENESTE OLIVIER , CHEN I-JEN , DAVIDSON JAMES EDWARD PAUL , MURRAY JAMES BROOKE , SIPOS SZABOLCS , ONDI LEVENTE , PROSZENYAK AGNES
IPC: C07D209/00 , A61K31/00 , A61P35/00 , C07D307/00 , C07D333/00 , C07D403/00 , C07D405/00 , C07D409/00 , C07D471/00 , C07D487/00 , C07D491/00 , C07D495/00
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公开(公告)号:UA122498C2
公开(公告)日:2020-11-25
申请号:UAA201800621
申请日:2016-06-22
Applicant: SERVIER LAB , VERNALIS R&D LTD
Inventor: BÁLINT BALÁZS , CSÉKEI MÁRTON , SZABÓ ZOLTÁN , SZLÁVIK ZOLTÁN , KOTSCHY ANDRÁS , CHANRION MAÏA , GENESTE OLIVIER , CHEN I-JEN , DAVIDSON JAMES EDWARD PAUL , MURRAY JAMES BROOKE , SIPOS SZABOLCS , ONDI LEVENTE , PROSZENYÁK ÁGNES
Abstract: Сполукиформули (І): , (І) де R1, R2, R3, R4, R5 R6, R7, R8, R14, W, Аі n єтакими, яквизначенов описі.
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公开(公告)号:LT3313817T
公开(公告)日:2020-11-25
申请号:LT16730854
申请日:2016-06-22
Applicant: SERVIER LAB , VERNALIS R&D LTD
Inventor: BALINT BALAZS , CSÉKEI MARTON , SZABO ZOLTAN , SZLAVIK ZOLTAN , KOTSCHY ANDRAS , CHANRION MAIA , GENESTE OLIVIER , CHEN I-JEN , DAVIDSON JAMES EDWARD PAUL , MURRAY JAMES BROOKE , SIPOS SZABOLCS , ONDI LEVENTE , PROSZENYAK AGNES
IPC: C07D209/12 , A61K31/381 , A61K31/4355 , A61K31/437 , A61P35/00 , C07D307/80 , C07D307/81 , C07D333/56 , C07D403/12 , C07D405/04 , C07D405/12 , C07D409/12 , C07D471/04 , C07D487/04 , C07D491/04 , C07D495/04
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10.
公开(公告)号:AU2016282837B2
公开(公告)日:2020-05-28
申请号:AU2016282837
申请日:2016-06-22
Applicant: SERVIER LAB , VERNALIS R&D LTD
Inventor: SZLÁVIK ZOLTÁN , SZABÓ ZOLTÁN , CSÉKEI MÁRTON , PACZAL ATTILA , KOTSCHY ANDRÁS , BRUNO ALAIN , GENESTE OLIVIER , CHEN I-JEN , DAVIDSON JAMES EDWARD PAUL , MURRAY JAMES BROOKE , ONDI LEVENTE , RADICS GÁBOR , SIPOS SZABOLCS , PROSZENYÁK ÁGNES , PERRON-SIERRA FRANÇOISE , BÁLINT BALÁZS
IPC: C07D495/04 , A61K31/519 , A61P35/00 , A61P37/00
Abstract: Compounds of formula (I): wherein R
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