公开(公告)号：JP2003313161A

公开(公告)日：2003-11-06

申请号：JP2003104164

申请日：2003-04-08

Applicant: Syngenta Participations Ag ,  シンジェンタ パーティシペーションズ アクチェンゲゼルシャフト

Inventor： SCHNEIDER HERMANN ,  LUETHY CHRISTOPH ,  EDMUNDS ANDREW

IPC: C07B61/00 ,  C07C45/45 ,  C07C45/54 ,  C07C45/57 ,  C07C45/60 ,  C07C49/733 ,  C07C315/04 ,  C07C317/24 ,  C07C317/44 ,  C07C319/20 ,  C07C323/22 ,  C07C323/62 ,  C07D213/50 ,  C07D307/79

CPC classification number: C07D307/79 ,  C07C45/455 ,  C07C45/54 ,  C07C45/57 ,  C07C45/60 ,  C07C49/733 ,  C07C315/04 ,  C07C319/20 ,  C07C323/22 ,  C07C2602/44 ,  C07D213/50 ,  C07C323/62 ,  C07C317/44

Abstract: PROBLEM TO BE SOLVED: To provide a new method for producing a cyclic 1,3-diketone derivative carbonylated at 2 position.
SOLUTION: This method for producing the cyclic 1,3-diketone derivative represented by formula (I) (wherein substituent groups are defined in a claim 1) comprises converting a compound represented by formula (II) to a salt represented by formula (III), reacting the compound (III) with a compound represented by the formula (IV): X-C(O)-Q (wherein X is an eliminable group) to obtain a compound represented by formula (V) and treating the compound (V) with a catalytic amount of a cyanide ion in the presence of a base.
COPYRIGHT: (C)2004,JPO

Abstract translation: 待解决的问题：提供一种制备在2位羰基化的环状1,3-二酮衍生物的新方法。 解决方案：用于制备由式（I）表示的环状1,3-二酮衍生物（其中取代基如权利要求1所定义）的方法包括将由式（II）表示的化合物转化成式 （III）表示的化合物与式（IV）表示的化合物反应：XC（O）-Q（其中X为可消除基团），得到式（V）表示的化合物，并处理化合物 V）与催化量的氰化物离子在碱的存在下反应。 版权所有（C）2004，JPO

公开(公告)号：WO2004058712A3

公开(公告)日：2004-09-16

申请号：PCT/EP0314949

申请日：2003-12-29

Applicant: SYNGENTA PARTICIPATIONS AG ,  BEAUDEGNIES RENAUD ,  EDMUNDS ANDREW ,  LUETHY CHRISTOPH ,  HALL ROGER GRAHAM ,  WENDEBORN SEBASTIAN ,  SCHAETZER JUERGEN

Inventor： BEAUDEGNIES RENAUD ,  EDMUNDS ANDREW ,  LUETHY CHRISTOPH ,  HALL ROGER GRAHAM ,  WENDEBORN SEBASTIAN ,  SCHAETZER JUERGEN

IPC: C07D213/50 ,  C07D213/89 ,  C07D451/02 ,  C07D493/08

CPC classification number: C07D213/89 ,  C07D213/50 ,  C07D451/02 ,  C07D493/08

Abstract: Compounds of formula (I), wherein the substituents are as defined in claim 1, and the agrochemically acceptable salts and all stereoisomers and tautomeric forms of the compounds of formula I are suitable for use as herbicides.

Abstract translation: 式（I）化合物，其中取代基如权利要求1所定义，并且式I化合物的农业化学可接受的盐和所有立体异构体和互变异构体形式适合用作除草剂。

公开(公告)号：WO2016023954A3

公开(公告)日：2016-04-07

申请号：PCT/EP2015068577

申请日：2015-08-12

Applicant: SYNGENTA PARTICIPATIONS AG

Inventor： JUNG PIERRE JOSEPH MARCEL ,  EDMUNDS ANDREW ,  JEANGUENAT ANDRÉ ,  MUEHLEBACH MICHEL ,  STOLLER ANDRÉ ,  EMERY DANIEL ,  HALL ROGER GRAHAM

IPC: C07D471/04 ,  A01N31/08 ,  A61K31/4188 ,  A61K31/437

CPC classification number: C07D471/04 ,  A01N25/08 ,  A01N43/90 ,  A01N25/00 ,  A01N2300/00

Abstract: Compounds of formula (I), wherein the substituents are as defined in claim 1, and the agrochemically acceptable salts, stereoisomers, enantiomers, tautomers and N-oxides of those compounds, can be used as insecticides and can be prepared in a manner known per se.

Abstract translation: 其中取代基如权利要求1所定义的式（I）化合物以及这些化合物的农业化学上可接受的盐，立体异构体，对映异构体，互变异构体和N-氧化物可以用作杀虫剂并且可以以已知方式制备 SE。

公开(公告)号：WO2012069652A3

公开(公告)日：2012-07-19

申请号：PCT/EP2011071073

申请日：2011-11-25

Applicant: SYNGENTA PARTICIPATIONS AG ,  QUARANTA LAURA ,  LAMBERTH CLEMENS ,  LEFRANC DAVID GUILLAUME CLAUDE FRANCOIS ,  UMARYE JAYANT ,  RENOLD PETER ,  EDMUNDS ANDREW

Inventor： QUARANTA LAURA ,  LAMBERTH CLEMENS ,  LEFRANC DAVID GUILLAUME CLAUDE FRANCOIS ,  UMARYE JAYANT ,  RENOLD PETER ,  EDMUNDS ANDREW

IPC: A01N43/54 ,  A01P3/00

CPC classification number: A01N43/54 ,  A01N2300/00 ,  A01N37/36 ,  A01N43/40 ,  A01N43/653 ,  A01N45/02

Abstract: A composition suitable for control of diseases caused by phytopathogens comprising (A) a compound of formula (I) wherein wherein the substituents have the definitions as defined in claim 1 or a salt or a N-oxide thereof and (B) at least one compound selected from compounds known for their fungicidal activity; and a method of controlling diseases on useful plants.

Abstract translation: （A）其中取代基具有如权利要求1中定义的取代基或其盐或N-氧化物的式（I）化合物和（B）至少一种化合物 选自已知具有杀真菌活性的化合物; 以及控制有用植物疾病的方法。

公开(公告)号：WO2009024341A8

公开(公告)日：2010-04-15

申请号：PCT/EP2008006868

申请日：2008-08-21

Applicant: SYNGENTA PARTICIPATIONS AG ,  LOISELEUR OLIVIER ,  HALL ROGER GRAHAM ,  STOLLER ANDRE DENIS ,  CRAIG GERALD WAYNE ,  JEANGUENAT ANDRE ,  EDMUNDS ANDREW

Inventor： LOISELEUR OLIVIER ,  HALL ROGER GRAHAM ,  STOLLER ANDRE DENIS ,  CRAIG GERALD WAYNE ,  JEANGUENAT ANDRE ,  EDMUNDS ANDREW

IPC: C07D401/14 ,  A01N43/56 ,  C07D405/14 ,  C07D409/14 ,  C07D417/14

CPC classification number: C07D401/14 ,  C07D405/14 ,  C07D409/14 ,  C07D417/14

Abstract: Compounds of Formula I wherein the substituents are as defined in claim 1, and the agrochemically acceptable salts and all stereoisomers and tautomeric forms of the compounds of formula I can be used as agrochemical active ingredients and can be prepared in a manner known per se.

Abstract translation: 其中取代基如权利要求1所定义的式I化合物，以及式I化合物的农业化学上可接受的盐和所有立体异构体和互变异构形式可用作农业化学活性成分，并且可以以本身已知的方式制备。

公开(公告)号：WO2009024341A2

公开(公告)日：2009-02-26

申请号：PCT/EP2008006868

申请日：2008-08-21

Applicant: SYNGENTA PARTICIPATIONS AG ,  LOISELEUR OLIVIER ,  HALL ROGER GRAHAM ,  STOLLER ANDRE DENIS ,  GRAIG GERALD WAYNE ,  JEANGUENAT ANDRE ,  EDMUNDS ANDREW

Inventor： LOISELEUR OLIVIER ,  HALL ROGER GRAHAM ,  STOLLER ANDRE DENIS ,  CRAIG GERALD WAYNE ,  JEANGUENAT ANDRE ,  EDMUNDS ANDREW

IPC: C07D401/14 ,  A01N43/56 ,  C07D405/14 ,  C07D409/14 ,  C07D417/14

CPC classification number: C07D401/14 ,  C07D405/14 ,  C07D409/14 ,  C07D417/14

Abstract: Compounds of Formula I wherein the substituents are as defined in claim 1, and the agrochemically acceptable salts and all stereoisomers and tautomeric forms of the compounds of formula I can be used as agrochemical active ingredients and can be prepared in a manner known per se.

Abstract translation: 其中取代基如权利要求1所定义的式I化合物，以及式I化合物的农业化学上可接受的盐和所有立体异构体和互变异构形式可用作农业化学活性成分，并且可以以本身已知的方式制备。

公开(公告)号：WO2005077178A3

公开(公告)日：2006-01-26

申请号：PCT/EP2005001518

申请日：2005-02-15

Applicant: SYNGENTA PARTICIPATIONS AG ,  HOLE STEPHEN JOHN ,  LUETHY CHRISTOPH ,  BEAUDEGNIES RENAUD ,  EDMUNDS ANDREW ,  SCHAETZER JUERGEN ,  WENDEBORN SEBASTIAN

Inventor： HOLE STEPHEN JOHN ,  LUETHY CHRISTOPH ,  BEAUDEGNIES RENAUD ,  EDMUNDS ANDREW ,  SCHAETZER JUERGEN ,  WENDEBORN SEBASTIAN

IPC: A01N25/32 ,  A01N43/40 ,  A01N43/44 ,  A01N43/50 ,  A01N43/54 ,  A01N43/56 ,  A01N43/653 ,  A01N43/713 ,  A01N43/76 ,  A01N43/80 ,  A01N43/82

CPC classification number: A01N43/76 ,  A01N25/32 ,  A01N43/40 ,  A01N43/44 ,  A01N43/50 ,  A01N43/54 ,  A01N43/56 ,  A01N43/653 ,  A01N43/713 ,  A01N43/80 ,  A01N43/82 ,  A01N61/00 ,  A01N2300/00

Abstract: A herbicidal composition comprising a) a compound of formula (I) wherein the substituents are as defined in claim 1, or an agronomically acceptable salt of such a compound, and b) a synergistically effective amount of one or more compounds selected from pyridafol, dicamba and its salts, procarbazone, benflubutamid, tralkoxydim, mesosulfuron, chlorsulfuron, triasulfuron, flamprop-M, metoxuron, glufosinate, L-glufosinate, fluthiacet, imazamox, imazethapyr, nicosulfuron, primisulfuron-methyl, rimsulfuron, halosulfuron, cloransulam, clomazone, diclosulam, 2,4-D and its salts, florasulam, flumiclorac, bromoxynil, sethoxydim, ioxynil, tepraloxydim, carfentrazone, clethodim, sulfentrazone, imazaquin, sulcotrione, imazapyr, mesotrione, thifensulfuron, isoxaflutole, prosulfuron, isoxachlortole, bentazone, iodosulfuron, prohexadione, diflufenzopyr, flurtamone, butylate, flumioxazin, fentrazamide, benzfendizone, isopropazole, fluazolate, aclonifen, tritosulfuron, cinidon-ethyl, glyphosate and its potassium, isopropylammonium, sodium, trimesium, ammonium and diammonium salts, terbuthylazine, mesotrione + terbuthylazine, paraquat, ketospiradox, aminopyralid, amicarbazone, azafenidin, flufenpyr-ethyl, the compound of formula (II) and the compounds clodinafop-propargyl, prosulfocarb, picolinafen, pyrafIufan-ethyl, beflubutamid, fenoxaprop-P-ethyl, diclofop-methyl, amidosulfuron, flupyrsulfuron, flupyrsulfuron-methyl-sodium, metsulfuron-methyl, sulfosulfuron, tribenuron-methyl, imazamethabenz-methyl, flucarbazone, chiortoluron, isoproturon, methabenzthiazuron, bifenox, fluoroglycofen-ethyl, imazosuifuron, diflufenican, bilanafos, ethaifluralin, fluthiamide, isoxaben, trialiate, 2,4-DB, dichiorprop, MCPA, MCPB, mecoprop, MCPP, mecoprop-P, clopyralid, fluroxypyr, quinmerac, benazolin-ethyl, difenzoqual, cyhalofop-butyl, dithiopyr, quinclorac, prodiamine, benefin and trifluralin. The compositions according to the invention may also comprise a safener.

Abstract translation: 一种除草组合物，其包含a）式（I）化合物，其中取代基如权利要求1所定义，或该化合物的农学上可接受的盐，和b）协同有效量的一种或多种选自吡哆醛，麦草畏 吡磺隆，氯磺隆，氯磺隆，氯磺隆，氯磺隆，氯磺隆，氯磺隆，氯磺隆，氯磺隆，氯磺隆，氯磺隆，氯磺隆，氯磺隆，氯磺隆， 2,4-D及其盐，氟妥拉苏，氟氯尼，溴苯腈，卡非那唑，烯草酮，磺扎酮，咪唑啉酮，磺草酮，咪草烟，甲基磺草酮，噻吩磺隆，异山梨醇，次磺草胺，异恶草酮，苯达唑，碘磺隆， ，氟酸酯，丁酸酯，氟咪嗪，氟哌嗪，苯并芬那唑，异丙唑，氟酸酯，aclonifen，三氯嘧磺隆，cinidon-乙基，草甘膦及其 钾，异丙基铵，钠，三甲基铵，铵和二铵盐，特丁津，甲基磺草酮+特丁津，百草枯，酮基吡唑，氨基吡啶，氨基吡嗪，azafenidin，氟吡啶 - 乙基，式（II）化合物和化合物clodinafop-炔丙基， ，吡咯布酮，异丙肾上腺素，二氟甲磺酸，氨磺嘧磺隆，氟吡磺隆，氟吡磺隆 - 甲基钠，甲磺隆，磺嘧磺隆，三甲苯隆 - 甲基，咪草丁溴甲基，氟卡沙赞，氯耳普隆，异丙隆，甲苯噻嗪， 氟替芬，乙酰，咪唑苏氟脲，氟苯丙胺，双胍，乙酸菌素，氟尿嘧啶，异山梨醇，三钠，2,4-DB，二氯丙酸，MCPA，MCPB，mecoprop，MCPP，mecoprop-P，clopyralid，氟草吡啶，quinmerac，benazolin- ，三氟氯丙基，二硫代吡啶，喹氯林，丙二胺，益氟酸和氟乐灵。 根据本发明的组合物还可以包含安全剂。

公开(公告)号：WO2009010260A3

公开(公告)日：2009-05-22

申请号：PCT/EP2008005732

申请日：2008-07-14

Applicant: SYNGENTA PARTICIPATIONS AG ,  HALL ROGER GRAHAM ,  LOISELEUR OLIVIER ,  PABBA JAGADISH ,  PAL SITARAM ,  JEANGUENAT ANDRE ,  EDMUNDS ANDREW ,  STOLLER ANDRE

Inventor： HALL ROGER GRAHAM ,  LOISELEUR OLIVIER ,  PABBA JAGADISH ,  PAL SITARAM ,  JEANGUENAT ANDRE ,  EDMUNDS ANDREW ,  STOLLER ANDRE

IPC: C07D317/68 ,  A01N43/56 ,  C07D401/04 ,  C07D401/14 ,  C07D405/14 ,  C07D409/14 ,  C07D411/14 ,  C07D413/14 ,  C07D417/14 ,  C07D498/12

CPC classification number: C07D317/68 ,  C07D401/04 ,  C07D401/14 ,  C07D405/14 ,  C07D409/14 ,  C07D411/14 ,  C07D413/14 ,  C07D417/14 ,  C07D498/12

Abstract: An insecticidal compound of formula (I) in which G1, G2, and G3 together with the two carbon atoms to which G1 and G3 are attached, form a non-aromatic 4- or 5-membered ring system; wherein G1 is sulfur, SO, SO2, oxygen, a direct bond, NRa or CR5aR5b; G2 is sulfur, SO, SO2, oxygen, a direct bond, NRb or CR5cR5d; G3 is sulfur, SO, SO2, oxygen, a direct bond, NRc or CR5eR5f; with the provisos that a) not more than 1 group G can be a direct bond, b) not more than 2 G groups can be oxygen, sulfur, SO or SO2 and c) when 2 G groups are oxygen, SO, SO2 and/or sulfur the two groups are separated by a carbon atom; each of Z1 and Z2, which may be the same or different, represents oxygen or sulfur; D is phenyl or a 5- or 6-membered heteroaromatic ring and R1a, R1b, R5a, R5b, R5c, R5d, R5e, R5f, Ra, Rb Rc, R2, R3 and R20 are specified organic groups and agronomically acceptable salts/isomers/enantiomers/tautomers/N-oxides of those compounds.

Abstract translation: 其中G1，G2和G3与G1和G3所连接的两个碳原子连接的式（I）杀虫化合物形成非芳族4-或5-元环系; 其中G1是硫，SO，SO2，氧，直接键，NRa或CR5aR5b; G2是硫，SO，SO2，氧，直接键，NRb或CR5cR5d; G3是硫，SO，SO2，氧，直接键，NRc或CR5eR5f; 条件是a）不超过1组G可以是直接键，b）不超过2G基团可以是氧，硫，SO或SO 2，以及c）当2G基团是氧，SO，SO 2和/ 或硫，两个基团被碳原子隔开; Z1和Z2中的每一个可以相同或不同，表示氧或硫; D是苯基或5-或6-元杂芳环，R1a，R1b，R5a，R5b，R5c，R5d，R5e，R5f，Ra，RbRc，R2，R3和R20是指定的有机基团和农艺学上可接受的盐/异构体 /对映异构体/互变异构体/ N-氧化物。

公开(公告)号：WO2007020050A3

公开(公告)日：2007-04-19

申请号：PCT/EP2006008040

申请日：2006-08-14

Applicant: SYNGENTA PARTICIPATIONS AG ,  JEANGUENAT ANDRE ,  HALL ROGER GRAHAM ,  LOISELEUR OLIVIER ,  TRAH STEPHAN ,  DURIEUX PATRICIA ,  EDMUNDS ANDREW ,  STOLLER ANDRE

Inventor： JEANGUENAT ANDRE ,  HALL ROGER GRAHAM ,  LOISELEUR OLIVIER ,  TRAH STEPHAN ,  DURIEUX PATRICIA ,  EDMUNDS ANDREW ,  STOLLER ANDRE

IPC: C07D401/14 ,  A01N43/52 ,  A01N43/56 ,  A01N43/60 ,  A01N43/78 ,  A01N43/832 ,  C07D413/14 ,  C07D417/14

CPC classification number: C07D413/14 ,  A01N43/56 ,  A01N43/60 ,  A01N43/64 ,  A01N43/707 ,  A01N43/76 ,  A01N43/78 ,  A01N43/82 ,  C07D401/14 ,  C07D417/14

Abstract: Compounds of formula (I), wherein the substituents are as defined in claim (1), and the agrochemically acceptable salts and all stereoisomers and tautomeric forms of the compounds of formula (I) can be used as agrochemical active ingredients and can be prepared in a manner known per se.

Abstract translation: 式（I）化合物，其中取代基如权利要求（1）中所定义，以及式（I）化合物的农业化学上可接受的盐和所有立体异构体和互变异构形式可用作农业化学活性成分，并且可以制备为 本身已知的方式。

公开(公告)号：WO2005105718A3

公开(公告)日：2006-05-04

申请号：PCT/EP2005004680

申请日：2005-04-29

Applicant: SYNGENTA PARTICIPATIONS AG ,  SYNGENTA LTD ,  JACKSON DAVID ANTHONY ,  EDMUNDS ANDREW ,  BOWDEN MARTIN CHARLES ,  BROCKBANK BEN

Inventor： JACKSON DAVID ANTHONY ,  EDMUNDS ANDREW ,  BOWDEN MARTIN CHARLES ,  BROCKBANK BEN

IPC: C07C17/10 ,  C07C17/23 ,  C07C23/32 ,  C07C45/45 ,  C07C45/71 ,  C07C67/11 ,  C07C315/04 ,  C07C317/44 ,  C07D213/50 ,  C07D213/80 ,  C07C49/403 ,  C07C49/603 ,  C07C49/733

CPC classification number: C07D213/80 ,  C07C17/10 ,  C07C17/23 ,  C07C23/32 ,  C07C67/11 ,  C07C315/04 ,  C07D213/50 ,  C07C69/78 ,  C07C69/76 ,  C07C317/44

Abstract: The present invention relates to a process for the preparation of compounds of formula (I), wherein the substituents are as defined in claim 1, by reacting a compound of formula (II), with a bromine or chlorine source to form a compound of formula (III), wherein X is chlorine or bromine; reacting that compound with water to form the compound of formula (IV), converting that compound, using a compound of formula (V), wherein M + is the hydrogen cation or an alkali metal ion, alkaline earth metal ion or ammonium ion, into the compound of formula (VI), and treating that compound with a cyanide source in the presence of a base.

Abstract translation: 本发明涉及制备式（I）化合物的方法，其中取代基如权利要求1所定义，通过使式（II）化合物与溴或氯源反应形成式 （III），其中X为氯或溴; 使该化合物与水反应以形成式（IV）化合物，使用其中M +为氢阳离子或碱金属离子，碱土金属的式（Ⅴ）化合物转化该化合物 金属离子或铵离子转化成式（VI）的化合物，并在碱的存在下用氰化物源处理该化合物。