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公开(公告)号:CA2610800A1
公开(公告)日:2006-12-14
申请号:CA2610800
申请日:2006-05-22
Applicant: UCB PHARMA SA
Inventor: PERRY BENJAMIN
IPC: C07D401/12 , A61K31/4709 , A61P29/00
Abstract: The present invention concerns 2.6-quinolinyl derivatives, processes for preparing them, pharmaceutical compositions containing them and their use as pharmaceu ticals. For example, the compounds according to the invention are useful for the treatment of asthma, allergic rhinitis, sinusitis, conjunctivitis, food allergy, inflammatory skin disorders including dermatitis, psoriasis, urticaria, pruritus and eczema, rheumatoi arthritis, inflammatory bowel diseases including Crohn's disease and ulcerative colitis, multiple sclerosis and other autoimmune disorders, and atherosclerosis.
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公开(公告)号:MX2007014721A
公开(公告)日:2008-02-14
申请号:MX2007014721
申请日:2006-05-22
Applicant: UCB PHARMA SA
Inventor: PERRY BENJAMIN
IPC: C07D401/12 , A61K31/4709 , A61P29/00
Abstract: La presente invencion se refiere a los derivados de 2,6-quinolinilo, los procesos para prepararlos, las composiciones farmaceuticas que los contienen y su uso como farmacos. Por ejemplo, los compuestos de acuerdo con la invencion son utiles para el tratamiento de asma, rinitis alergica, sinusitis, conjuntivitis, alergia a los alimentos, trastornos de la piel inflamatorios, incluyendo dermatitis, soriasis, urticaria, prurito y eczema, artritis reumatoide, enfermedad del intestino inflamatoria incluyendo la enfermedad de Crohn y colitis ulcerativa, esclerosis multiples y otros trastornos autoinmunes, y ateroesclerosis.
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公开(公告)号:NO20080125L
公开(公告)日:2008-01-08
申请号:NO20080125
申请日:2008-01-08
Applicant: UCB PHARMA SA
Inventor: PERRY BENJAMIN
IPC: C07D401/12 , A61K31/4709 , A61P29/00
Abstract: The present invention concerns 2,6-quinolinyl derivatives, processes for preparing them, pharmaceutical compositions containing them and their use as pharmaceuticals.
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公开(公告)号:AU2006254772B2
公开(公告)日:2011-06-02
申请号:AU2006254772
申请日:2006-05-22
Applicant: UCB PHARMA SA
Inventor: PERRY BENJAMIN
IPC: C07D401/12 , A61K31/4709 , A61P29/00
Abstract: The present invention concerns 2,6-quinolinyl derivatives, processes for preparing them, pharmaceutical compositions containing them and their use as pharmaceuticals.
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公开(公告)号:ES2359935T3
公开(公告)日:2011-05-30
申请号:ES06753758
申请日:2006-05-22
Applicant: UCB PHARMA SA
Inventor: PERRY BENJAMIN
IPC: C07D401/12 , A61K31/4709 , A61P29/00
Abstract: Compuesto que tiene la fórmula I, sus enantiómeros, diastereoisómeros o sales de los mismos farmacéuticamente aceptables, en la que: R1 es hidrógeno, hidroxilo o alquilo C 1-6; R2 es hidrógeno o halógeno; n es de 0 a 5; R3 es hidrógeno, o halógeno; n' es de 0 a 4.
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公开(公告)号:DE602006019731D1
公开(公告)日:2011-03-03
申请号:DE602006019731
申请日:2006-05-22
Applicant: UCB PHARMA SA
Inventor: PERRY BENJAMIN
IPC: C07D401/12 , A61K31/4709 , A61P29/00
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公开(公告)号:BRPI0611243A2
公开(公告)日:2010-08-24
申请号:BRPI0611243
申请日:2006-05-22
Applicant: UCB PHARMA SA
Inventor: PERRY BENJAMIN
IPC: C07D401/12 , A61K31/4709 , A61P29/00
Abstract: The present invention concerns 2,6-quinolinyl derivatives, processes for preparing them, pharmaceutical compositions containing them and their use as pharmaceuticals.
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公开(公告)号:UA90319C2
公开(公告)日:2010-04-26
申请号:UAA200714908
申请日:2006-05-22
Applicant: UCB PHARMA SA
Inventor: PERRY BENJAMIN
IPC: C07D401/12 , A61K31/4709 , A61P29/00
Abstract: Данноеизобретениекасаетсясоединений 2,6-хинолинила, процессовихизготовления, фармацевтическихсоставов, которыеихсодержат, иихпримененияв фармацевтическихсоставах.Соединениясогласноизобретениюмогутприменяться, например, влеченииастмы, аллергическогоринита, синусита, конъюнктивита, пищевойаллергии, воспалительныхрасстройствкожи, включаядерматит, псориаз, крапивницу, зуди экзему, ревматоидногоартрита, воспалительныхболезнейкишечника, включаяболезньКронаи язвенныйколит, множественногосклерозаи другихаутоиммунныхрасстройстви атеросклероза.
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公开(公告)号:MY140739A
公开(公告)日:2010-01-15
申请号:MYPI20062356
申请日:2006-05-22
Applicant: UCB PHARMA SA
Inventor: PERRY BENJAMIN
IPC: C07D401/12
Abstract: 1 7 2,6-QUINOLINYL DERIVATIVES, PROCESSES FOR PREPARING THEL AND THEIR USES ABSTPACT THE PRESENT INVENTION CONCERNS 2.6-QLLINOLINYL DERIVATIVES, PROCESSES FOR 5 PREPARING THEM. PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE AS PHARMACEUTICALS.
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公开(公告)号:AU2006254772A1
公开(公告)日:2006-12-14
申请号:AU2006254772
申请日:2006-05-22
Applicant: UCB PHARMA SA
Inventor: PERRY BENJAMIN
IPC: C07D401/12 , A61K31/4709 , A61P29/00
Abstract: The present invention concerns 2,6-quinolinyl derivatives, processes for preparing them, pharmaceutical compositions containing them and their use as pharmaceuticals.
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