Diazacyclobutene derivatives as anti-parasitic drug substances

    公开(公告)号:US11510906B1

    公开(公告)日:2022-11-29

    申请号:US16811135

    申请日:2020-03-06

    Abstract: A drug product and method for treating a parasitic disease in a host is described. The drug product comprises:
    a carrier matrix; and
    a drug substance having the formula: wherein:
    R1 is selected from the group consisting of H, aliphatic of 1 to 100 carbons and arene comprising up to 100 carbons;
    each R3 is independently selected from the group consisting of H, aliphatic of 1 to 100 carbons and arene comprising up to 100 carbons;
    Y represents those elements necessary to form a 5 or 6 membered ring;
    X is selected from the group consisting of B, O, N, S, Se and P; and
    n is 1-4 as necessary to complete the valence of X.

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