公开(公告)号：US20110003999A1

公开(公告)日：2011-01-06

申请号：US12919362

申请日：2009-02-17

Applicant: Michael DOCKNER

Inventor： Michael DOCKNER

IPC: C07D213/56 ,  C07D231/10

CPC classification number: G01B11/2441 ,  G01B9/0201 ,  G01B9/02057 ,  G01B9/0209 ,  G01B2290/70 ,  G01N21/95 ,  G01N2021/9513

Abstract: The present invention relates to a process for preparing substituted biphenylanilides of the formula I which comprises reacting a compound of formula II in the presence of a base and of a palladium catalyst selected from the group of: a) palladium-triarylpliosphine or -trialkylphosphine complex with palladium in the zero oxidation state, b) salt of palladium in the presence of triarylphospine or trialkylphosphine as a complex ligand or c) metallic palladium, optionally applied to support, in the presence of triarylphosphine or trialkylphosphine, in a solvent, with a diphenylborinic acid according to formula (III)

Abstract translation: 本发明涉及一种制备式I取代的联苯酰苯胺的方法，其包括在碱存在下与式Ⅱ化合物与钯催化剂反应，所述钯催化剂选自：a）钯 - 三芳基叉膦或三烷基膦配合物与 b）在三芳基膦或三烷基膦作为络合配体的存在下钯的盐，或c）金属钯，任选地在三芳基膦或三烷基膦存在下，在溶剂中与二苯基硼酸 根据式（III）

公开(公告)号：US20110092736A1

公开(公告)日：2011-04-21

申请号：US12991265

申请日：2009-04-24

Applicant: Michael DOCKNER

Inventor： Michael DOCKNER

IPC: C07C231/12

CPC classification number: C07C231/12 ,  C07C233/15

Abstract: The present invention relates to a process for preparing substituted biphenylanilides of the formula I wherein R1 is a protected amino group which comprises reacting a compound of formula II in the presence of a base and of a palladium catalyst in a solvent, with an organoboron compound of formula (III)

Abstract translation: 本发明涉及一种制备式I取代的联苯酰苯胺的方法，其中R 1是被保护的氨基，其包括在碱和Pd催化剂存在下，在溶剂中使式Ⅱ化合物与有机硼化合物反应 式（III）