PROCESS FOR PREPARING N-SUBSTITUTED 1H-PYRAZOLE-5-CARBONYLCHLORIDE COMPOUNDS
    95.
    发明公开
    PROCESS FOR PREPARING N-SUBSTITUTED 1H-PYRAZOLE-5-CARBONYLCHLORIDE COMPOUNDS 审中-公开
    制备N-取代的1H-吡唑-5-碳酰氯化合物的方法

    公开(公告)号:EP2742035A1

    公开(公告)日:2014-06-18

    申请号:EP12744006.3

    申请日:2012-08-10

    Applicant: BASF SE

    CPC classification number: C07D401/04

    Abstract: The present invention relates to a process for preparing an N-substi- tuted 1 H-pyrazole-5-carbonylchloride compound of the formula (I) comprising the steps of i) deprotonating a compound of the formula (II) with a base selected from lithium-organic base having a carbon or nitrogen bound lithium or with a magnesium-organic base having a carbon bound magnesium; and ii) subjecting the product obtained in step (i) to a chlorocarbonylation by reacting it with a reagent selected from the group consisting of phosgene or a phosgene equivalent, to obtain a compound of formula (I).

    Abstract translation: 本发明涉及一种制备式(I)的N-取代的1H-吡唑-5-碳酰氯化合物的方法,该方法包括以下步骤:i)用选自以下的碱进行式(II)的化合物的去质子化: 具有碳或氮结合锂的锂 - 有机碱或具有碳结合镁的镁 - 有机碱; 和ii)使步骤(i)中获得的产物通过使其与选自光气或光气等价物的试剂反应而进行氯羰基化,得到式(I)化合物。

    SUBSTITUTED AZOLIN-2-YL-AMINO COMPOUNDS
    99.
    发明公开
    SUBSTITUTED AZOLIN-2-YL-AMINO COMPOUNDS 审中-公开
    取代喹唑啉-2-基阿明CONNECTIONS

    公开(公告)号:EP2051970A1

    公开(公告)日:2009-04-29

    申请号:EP07802500.4

    申请日:2007-08-06

    Applicant: BASF SE

    CPC classification number: C07D417/12 A01N43/50 A01N43/76 A01N43/78 C07D277/18

    Abstract: The present invention relates to azolin-2-yl-amino compounds of formulae (I. a) and (l.b) and their salts which are useful for combating animal pest, in particular arthropod and nematodes. The present invention also relates to a method for combating such pests and for protecting crops against infestation or infection by such pests. Furthermore, the present invention relates to veterinary compositions for combating animal pests. Formula (I.a), formula (I.b) wherein n is 0 to 4; X is S, O or NR5; A is -C(R6a)(R6b)-, O, NR7, S, S(O) or S(O)2; B is a bond Or CH2; R1 is H, CN, C1-C6-alkyl, C2-C6-alkenyl, C1-C6-alkylcarbonyl, C3-C6-cycloalkyl, phenyl, benzyl, etc.; R2a, R2b are H, CN, C1-C6-alkyl, C2-C6-alkenyl, C1-C6-alkylcarbonyl, C1-C6-alkoxycarbonyl, (C1-C6-alkyl)thiocarbonyl, C(O)NRaRb, C(S)NRaRb, (SO2)NRaRb, phenyl, benzyl, 5 or 6 membered heterocyclic ring etc.; or R1 together with R2a is C3-C5-alkandiyl; or R1 together with R2b are C(O); R3a, R3b, R3c, R3d are H, halogen, CN, C1-C6-alkyl, C1-C6-alkylamino, C3-C6-cycloalkyl, phenyl, benzyl, etc.; R4a, R4b are H, halogen, C1-C6-alkyl, C2-C6-alkenyl, phenyl, benzyl, 5 or 6 membered hetaryl; or R4a together with R4b may also be =0, =NRC or =CRdRe; or R2a together with R4a may form a bridging bivalent radical.

    PESTCIDAL COMPOSITIONS
    100.
    发明公开
    PESTCIDAL COMPOSITIONS 审中-公开
    农药组合物

    公开(公告)号:EP1968974A1

    公开(公告)日:2008-09-17

    申请号:EP06830499.7

    申请日:2006-12-11

    Applicant: BASF SE

    CPC classification number: C07D417/12

    Abstract: The present invention relates to 1-(Azolin-2-yl)-amino-alkane compounds, which are useful for combating insects, arachnids and nematodes. The present invention also relates to a method for combating animal pests selected from insects, arachnids and nematodes, and to agricultural compositions for combating animal pests. It has been found that animal pests can be combated by 1-(Azolin-2-yl)-amino-alkane compounds of the general formula (I) wherein A is a radical of the formulae (A1) or (A2): and wherein X is sulfur or oxygen and W, B and R1 to R6 are defined as in the description.

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