中科微点-全球专利检索

  1. Login
  2. Sign Up

Search Results

103 records (took 0.03 seconds)

    CRYSTALLINE FORM B OF AN ANTHRANILAMIDE INSECTICIDE AND CONVERSION OF FORM B INTO FORM A
    1.
    发明申请
    CRYSTALLINE FORM B OF AN ANTHRANILAMIDE INSECTICIDE AND CONVERSION OF FORM B INTO FORM A 审中-公开
    ANTHRANILAMIDE INSECTICIDE的晶体形式B和形式B的转化形式A

    公开(公告)号：WO2015169883A1

    公开(公告)日：2015-11-12

    申请号：PCT/EP2015/060018

    申请日：2015-05-07

    Applicant: BASF SE

    Inventor： KÖRBER, Karsten ,  KORADIN, Christopher ,  ZIERKE, Thomas ,  CHIODO, Tiziana ,  VIERTELHAUS, Martin

    IPC: A01N43/56 ,  A01P7/04

    CPC classification number: A01N43/56 ,  A01N25/12

    Abstract: The present invention relates to a crystalline form B of the anthranilamide insecticide 2-(3- chloro-2-pyridyl)-N-[2-methyl-4-chloro-6-[(diethyl-A4-sulfanylidene)carbamoyl]phenyl]-5- (trifluoromethyl)pyrazole-3-carboxamide (compound I) and to different processes for converting said crystalline form B into a crystalline form A of compound I.

    Abstract translation: 本发明涉及邻氨基苯甲酰胺杀虫剂2-（3-氯-2-吡啶基）-N- [2-甲基-4-氯-6 - [（二乙基亚苄基）氨基甲酰基]苯基] -5-（三氟甲基）吡唑-3-甲酰胺（化合物I），以及将所述结晶B转化为化合物I的结晶形式A的不同方法。

    VERFAHREN ZUR HERSTELLUNG VON 2-(AMINOMETHYLIDEN)-4,4-DIFLUOR-3-OXOBUTTERSÄUREESTERN
    2.
    发明申请
    VERFAHREN ZUR HERSTELLUNG VON 2-(AMINOMETHYLIDEN)-4,4-DIFLUOR-3-OXOBUTTERSÄUREESTERN 审中-公开
    用于生产2-（氨基亚甲基）-4,4-二氟-3-氧代丁酸酯

    公开(公告)号：WO2009133178A1

    公开(公告)日：2009-11-05

    申请号：PCT/EP2009/055283

    申请日：2009-04-30

    Applicant: BASF SE ,  ZIERKE, Thomas ,  MAYWALD, Volker ,  RACK, Michael ,  SMIDT, Sebastian Peer ,  KEIL, Michael ,  WOLF, Bernd ,  KORADIN, Christopher

    Inventor： ZIERKE, Thomas ,  MAYWALD, Volker ,  RACK, Michael ,  SMIDT, Sebastian Peer ,  KEIL, Michael ,  WOLF, Bernd ,  KORADIN, Christopher

    IPC: C07C227/16 ,  C07C229/30 ,  C07D231/14

    CPC classification number: C07D231/14 ,  C07C229/30 ,  C07D295/145

    Abstract: Die vorliegende Erfindung betrifft ein Verfahren zur Herstellung von difluormethylsubsti- tuierten Pyrazol4-ylcarbonsäuren und deren Ester, 2-(Aminomethyliden)-4,4-difluor-3- oxobuttersäureester der Formel (I), worin R 1 , R 2 und R 3 unabhängig voneinander für C 1 -C 6 -Alkyl, C 1 -C 6 -Haloalkyl, C 2 -C 6 -Alkenyl, C 3 -C 10 -Cycloalkyl oder Benzyl steht oder NR 2 R 3 für einen 5- bis 10-gliedrigen heterocyclischen Rest steht, ein Verfahren zur Herstellung von Verbindungen der Formel (I), bei dem man einen entsprechenden 3-Aminoacrylsäureester mit Difluoracetylfluorid umsetzt sowie die Verwendung von Verbindungen der Formel (I) in dem Verfahren zur Herstellung von difluormethylsubstituierten Pyrazol- 4-ylcarbonsäuren und deren Ester.

    Abstract translation: 本发明涉及一种用于difluormethylsubsti的制备 - 取代的吡唑基甲酸及其酯，2-（氨基亚甲基）的式（I）的-4,4-二氟-3-氧代丁酸乙酯，其特征在于R1，R2和R3各自独立地为C1 C6烷基，C1-C6卤代烷基，C2-C6链烯基，C3-C10环烷基或苄基或NR2R3表示5至10元杂环基团，为式I化合物的制备方法（I） ，该方法包括用二氟乙酰氟一个相应的3-氨基丙烯酸酯，以及用于制备吡唑difluormethylsubstituierten唑-4-基甲酸和它们的酯的使用过程中的式（I）的化合物的反应。

    1-(AZOLIN-2-YL)AMINO-1,2-DIPHENYLETHANE COMPOUNDS FOR COMBATING ANIMAL PESTS
    3.
    发明申请
    1-(AZOLIN-2-YL)AMINO-1,2-DIPHENYLETHANE COMPOUNDS FOR COMBATING ANIMAL PESTS 审中-公开
    1-（AZOLIN-2-YL）氨基-1,2-二苯醚化合物，用于组合动物饲料

    公开(公告)号：WO2009004032A1

    公开(公告)日：2009-01-08

    申请号：PCT/EP2008/058517

    申请日：2008-07-02

    Applicant: BASF SE ,  KORDES, Markus ,  KORADIN, Christopher ,  LE VEZOUET, Ronan ,  BAUMANN, Ernst ,  CULBERTSON, Deborah L. ,  ANSPAUGH, Douglas D. ,  OLOUMI-SADEGHI, Hassan ,  EBUENGA, Cecile

    Inventor： KORDES, Markus ,  KORADIN, Christopher ,  LE VEZOUET, Ronan ,  BAUMANN, Ernst ,  CULBERTSON, Deborah L. ,  ANSPAUGH, Douglas D. ,  OLOUMI-SADEGHI, Hassan ,  EBUENGA, Cecile

    IPC: C07D233/48 ,  C07D263/28 ,  C07D277/18 ,  C07D417/12 ,  C07D417/06 ,  A01N43/50 ,  A01N43/76 ,  A01N43/78

    CPC classification number: C07D263/28 ,  A01N43/50 ,  A01N43/76 ,  A01N43/78 ,  A01N47/12 ,  A01N47/16 ,  C07D233/48 ,  C07D277/18 ,  C07D417/06 ,  C07D417/12

    Abstract: The present invention relates to 1-(azolin-2-yl)amino-1,2-diphenylethane compounds of the formula I and to their salts which are useful for combating animal pests. The invention also relates to a method for controlling animal pests by using these compounds, to seed and to an agricultural and veterinary composition comprising said compounds, wherein A is a radical of formulae A.1 or A.2 wherein # denotes the bond to the remaining compound of formula I, X is selected from O, S and NR x , R 1 is selected from the group consisting of -OR A , -NR B1 R B2 , -C(=O)-R C , -C(=O)-OR D , -C(=O)-SR E , -C(=O)-NR B1 R B2' , -C(=S)-R C' , -C(=S)-OR D' , -C(=S)-SR E' , -C(=S)-NR B1 R B2 , -C(=NR 1a )-R C' , -C(=NR 1b )-OR D' , -C(=NR 1c )-SR E' , -C(=NR 1d )-NR B1 R B2 , -S(=O)-R F , -S(=O) 2 -R G , -S(=O) 2 -NR B1 R B2' , -P(=O)R H1 R H2 , -P(=S)R H1 R H2 , -B-C(=O)-R I , -B-O-C(=O)-R I , -B-S-C(=O)-R I , -B-N(R J )-C(=O)-R K , -B-C(=S)-R K , -B-O-C(=S)-R K , -B-S-C(=S)-R K , -B-N(R J )-C(=S)-R K , C 1 -C 8 -alkenyl, C 1 -C 8 -alkynyl, C 3 -C 8 -cycloalkyl, which is unsubstituted or may carry 1 to 4 substituents R 1e , naphthyl, which is unsubstituted or may carry 1 to 4 substituents R 1f , a saturated or partially unsaturated heterocycle, which is unsubstituted or may carry 1 to 4 substituents R 1g , hetaryl, which is unsubstituted or may carry 1 to 4 substituents R 1h , and C 1 -C 6 -alkyl, which carries a radical selected from the group consisting of -NR 1i R 1j , C 1 -C 4 -alkoxycarbonyl, C 3 -C 8 -cycloalkyl, aryl, aryloxy, arylthio, heterocyclyl, heterocyclyloxy and heterocyclylthio, R 2 , R 3 , R 4 , R 5 , R 6 and R 7 are each independently hydrogen, halogen, OH, SH, NH 2 , SO 3 H, COOH, cyano, nitro, C 1 -C 6 -alkyl, C 1 -C 6 -alkoxy, C 1 -C 6 -alkylamino etc.

    Abstract translation: 本发明涉及式I的1-（吡唑-2-基）氨基-1,2-二苯基乙烷化合物及其盐，其可用于防治动物害虫。 本发明还涉及通过使用这些化合物，种子和包含所述化合物的农业和兽医组合物来控制动物害虫的方法，其中A是式A.1或A.2的基团，其中＃表示与 剩余的式I化合物，X选自O，S和NR x，R1选自-ORA，-NRB1RB2，-C（= O）-RC，-C（= O）-OR，-C （= O）-SRE，-C（= O）-NRB1RB2'，-C（= S）-RC'，-C（= S）-OR'，-C（= S）-SRE' =（NR1c）-SR'，-C（= NR1d）-NRB1RB2，-S（= O） ）-RF，-S（= O）2 -RG，-S（= O）2 -NRB 1 R B 2'，-P（= O）RH1RH 2，-P（= S）RH1RH 2，-BC（= O） -BOC（= O）-RI，-BSC（= O）-RI，-BN（RJ）-C（= O）-RK，-BC（= S）-RK，-BOC（= S）-RK， -BSC（= S）-RK，-BN（RJ）-C（= S）-RK，C1-C8-烯基，C1-C8-炔基，C3-C8-环烷基，其未被取代或可携带1至4 取代基R 1e，萘基，其是未取代的或可以携带1至4个取代基R 1f，饱和或部分不饱和的杂环，其为未制备的 或可以携带1至4个未取代的或可以携带1至4个取代基R 1h的取代基R 1g，杂芳基，其中C 1 -C 6 - 烷基带有选自以下的基团：-NR 1 1 R 1，C 1 -C 4 - 烷氧基羰基， C 3 -C 8 - 环烷基，芳基，芳氧基，芳硫基，杂环基，杂环基氧基和杂环硫基，R 2，R 3，R 4，R 5，R 6和R 7各自独立地为氢，卤素，OH，SH，NH 2，SO 3 H，COOH，氰基，硝基， C 1 -C 6 - 烷基，C 1 -C 6 - 烷氧基，C 1 -C 6烷基氨基等

    PROCESS FOR PREPARING SULFIMINES AND THEIR IN-SITU CONVERSION INTO N-(2-AMINO-BENZOYL)-SULFIMINES
    7.
    发明申请
    PROCESS FOR PREPARING SULFIMINES AND THEIR IN-SITU CONVERSION INTO N-(2-AMINO-BENZOYL)-SULFIMINES 审中-公开
    制备硫化物的方法及其在N-（2-氨基苯甲酰基） - 硫脲中的原位转化

    公开(公告)号：WO2014154807A1

    公开(公告)日：2014-10-02

    申请号：PCT/EP2014/056164

    申请日：2014-03-27

    Applicant: BASF SE

    Inventor： FRASSETTO, Timo ,  JOCKERS, Harald ,  KORADIN, Christopher ,  ZIERKE, Thomas ,  KÖRBER, Karsten

    IPC: A01N43/56 ,  C07D401/04

    CPC classification number: C07C381/10 ,  A01N37/28 ,  A01N43/56 ,  C07C2601/02 ,  C07D401/04 ,  C07D409/14

    Abstract: The present invention relates to a process for preparing a compound of the formulae (la) or (lb), or a mixture thereof, wherein R 1 and R 2 independently of one another are hydrogen, C 1 -C 10 -alkyl, C 1 -C 10 -haloalkyl, C 3 -C 10 -cycloalkyl, C 3 -C 10 -halocycloalkyl, C 2 -C 10 -alkenyl, C 2 -C 10 -haloalkenyl or together represent an aliphatic chain, or the like; A- is HSO 4 - or 1/2 SO4 2- ; the process comprising the reaction of a sulfide of formula SR 1 R 2 with hydroxylamine- O-sulfonic acid of formula; wherein the reaction is carried out in an aqueous medium in the presence of a base. The present invention also relates to a process for preparing a compound of the formula (IV), wherein R 3 is halogen, cyano, C 1 -C 8 -alkyl, C 1 -C 8 -haloalkyl, C 3 -C 8 -cycloalkyl, C 3 -C 8 - halocycloalkyl, C 2 -C 8 -alkenyl, C 2 -C 8 -haloalkenyl, C 1 -C 8 -alkoxy, phenyl, or the like; R 4 is hydrogen, C 1 -C 10 -alkyl, C 1 -C 10 -haloalkyl, C 3 -C 8 -cycloalkyl, C 3 -C 8 -halocycloalkyl, C 2 -C 10 -alkenyl, C 2 -C 10 -haloalkenyl, phenyl, or the like; p is 0, 1, 2, 3 or 4; the process comprising: (i) providing the compound of the formulae (la) or (lb), or a mixture thereof, (ii) reacting a compound of the formulae (la) or (lb), or a mixture thereof, obtained in step (i) with a compound of the formula (V) in the presence of a base,

    Abstract translation: 本发明涉及制备式（Ia）或（Ib）化合物或其混合物的方法，其中R 1和R 2彼此独立地是氢，C 1 -C 10 - 烷基，C 1 -C 10 - 卤代烷基， C 3 -C 10 - 环烷基，C 3 -C 10 - 卤代环烷基，C 2 -C 10 - 烯基，C 2 -C 10 - 卤代烯基或一起代表脂族链等; A-是HSO4-或1/2 SO42-; 该方法包括式SR 1 R 2的硫化物与式的羟胺-O-磺酸的反应; 其中反应在碱的存在下在水性介质中进行。 本发明还涉及制备式（Ⅳ）化合物的方法，其中R 3为卤素，氰基，C 1 -C 8 - 烷基，C 1 -C 8 - 卤代烷基，C 3 -C 8 - 环烷基，C 3 -C 8 - 卤代环烷基， C 2 -C 8 - 烯基，C 2 -C 8 - 卤代烯基，C 1 -C 8 - 烷氧基，苯基等; R4是氢，C1-C10-烷基，C1-C10-卤代烷基，C3-C8-环烷基，C3-C8-卤代环烷基，C2-C10-烯基，C2-C10-卤代烯基，苯基等; p是0，1，2，3或4; 所述方法包括：（i）提供式（Ia）或（Ib）化合物或其混合物，（ii）使式（Ia）或（Ib）的化合物或其混合物与 步骤（i）与式（Ⅴ）化合物在碱的存在下反应，

    PESTICIDAL COMPOSITIONS COMPRISING 3 -ACETYL-I- PHENYLPYRAZOLE COMPOUNDS
    8.
    发明申请
    PESTICIDAL COMPOSITIONS COMPRISING 3 -ACETYL-I- PHENYLPYRAZOLE COMPOUNDS 审中-公开

    公开(公告)号：WO2008092851A3

    公开(公告)日：2008-08-07

    申请号：PCT/EP2008/051026

    申请日：2008-01-29

    Applicant: BASF SE ,  KORADIN, Christopher ,  LANGEWALD, Jürgen ,  ANSPAUGH, Douglas D. ,  COTTER, Henry Van Tuyl

    Inventor： KORADIN, Christopher ,  LANGEWALD, Jürgen ,  ANSPAUGH, Douglas D. ,  COTTER, Henry Van Tuyl

    IPC: A01N43/56 ,  A01N47/02 ,  A01P7/04

    Abstract: The present invention relates to pesticidal compositionscomprising as active componentsat least one 3-acetyl-1-phenylpyrazole compound of the formula (I) or a salt thereof: wherein X is N or C-R 5 ; R 1 is C 1 -C 4 -alkyl or C 1 -C 4 -haloalkyl; R 2 is NR 6 R 7 or S(O) n R 8 ; R 3 is halogen, C 1 -C 4 -haloalkyl, C 1 -C 4 -haloalkoxy, SF 5 or S(O) p R 9 ; R 4 is hydrogen or halogen; R 5 is halogen; R 6 is hydrogen, C 1 -C 4 -alkyl, C 1 -C 4 -haloalkyl,C(O)R 10 , S(O) q CF 3 ; R 7 is hydrogen or C 1 -C 4 -alkyl, or R 6 and R 7 are joined so as together form a C 4 - C 6 -alkylene moiety, wherein one CH 2 -group may be replaced by oxygen or a radical N-R 11 ; R 8 , R 9 , R 10 , R 11 are each independently hydrogen, C 1 -C 4 -alkylorC 1 -C 4 -haloalkyl; m, n, p and q are each independently 0, 1 or 2; and at least one further pesticidally active compound II, selected from A.1GABA-gated chloride channel antagonists; A.2Nicotinic acetylcholine receptor agonists/antagonists A.3Juvenile hormone mimics; A.4Compounds affecting the oxidative phosphorylation; A.5Inhibitors of the chitin biosynthesis; A.6Moulting disruptors; A.7Mitochondrial electron transport inhibitors;. A.8Voltage-dependent sodium channel blockers; A.9Inhibitors of the lipid synthesis; and A.10group of various compounds.

Patent Agency Ranking