公开(公告)号：DD147194A5

公开(公告)日：1981-03-25

申请号：DD21664679

申请日：1979-11-02

Applicant: CIBA GEIGY AG

Inventor： STURM ELMAR ,  NYFELER ROBERT

IPC: A01N35/04 ,  A01N35/06 ,  A01N37/00 ,  A01N37/02 ,  A01N37/06 ,  A01N37/08 ,  A01N37/10 ,  A01N37/34 ,  A01N37/40 ,  A01N37/48 ,  A01N47/06 ,  A01N47/22 ,  A01N53/00 ,  B01J27/00 ,  B01J27/125 ,  C07C45/00 ,  C07C45/45 ,  C07C45/46 ,  C07C49/733 ,  C07C49/747 ,  C07C49/825 ,  C07C49/835 ,  C07C67/00 ,  C07C68/00 ,  C07C69/017 ,  C07C69/157 ,  C07C69/54 ,  C07C69/63 ,  C07C69/653 ,  C07C69/96 ,  C07C201/00 ,  C07C205/45 ,  C07C205/57 ,  C07C239/00 ,  C07C255/57 ,  C07C271/06 ,  C07C271/08 ,  C07C271/44 ,  C07C325/00 ,  C07C329/06 ,  C07C329/08

Abstract: 2,3-Dichloro-7-hydroxy-1H-inden-1-one derivatives of the formula I (I) wherein R1 is hydrogen or one of the groups R2 and R3 independently of one another are each hydrogen, fluorine, chlorine, bromine, C1-C4-alkyl, trifluoromethyl or nitro, R4 is hydrogen, C1-C6-alkyl or C2-C4-alkenyl, each of which is unsubstituted or substituted by halogen, or R4 is phenyl which is unsubstituted or is substituted by C1-C4-alkyl, C1-C4-alkoxy, halogen, trifluoromethyl, cyano or nitro, or it is a C3-C6-cycloalkyl group, and R5 is C1-C6-alkyl, C3-C6-cycloalkyl or C2-C4-alkenyl. These compounds exhibit a microbicidal action against in particular phytopathogenic fungi and bacteria.

公开(公告)号：CA989409A

公开(公告)日：1976-05-18

申请号：CA161679

申请日：1973-01-19

Applicant: CIBA GEIGY AG

Inventor： CELLARIUS HANS JORG ,  CELLARIUS HERTHA M T HEIR ,  KUENG-MEYER HEINI GUARDIAN ,  STURM ELMAR

IPC: A01N57/08 ,  A01N57/16 ,  C07D209/08 ,  C07D215/08 ,  C07D221/04 ,  C07F9/165 ,  C07F9/572 ,  C07F9/576 ,  C07F9/60

公开(公告)号：DK161199C

公开(公告)日：1991-11-25

申请号：DK573883

申请日：1983-12-13

Applicant: CIBA GEIGY AG

Inventor： STURM ELMAR ,  MEYER ALFRED

IPC: A01N43/50 ,  A01N43/653 ,  A01P3/00 ,  C07C39/00 ,  C07C45/63 ,  C07C45/71 ,  C07D233/60 ,  C07D233/64 ,  C07D249/08 ,  C07D303/08 ,  C07D303/22 ,  C07D303/34 ,  C07D521/00

Abstract: 1-Azolyl-2-aryl-3-fluoro-alkan-2- ols of the general formula I in which Az is 1H-1,2,4-triazole, 4H-1,2,4-triazole or 1H-imidazole; Ar is an unsubstituted or substituted aromatic radical from the series comprising phenyl, biphenyl, phenoxyphenyl and naphthyl; R1 is hydrogen, C1-C4-alkyl, C3-C5-alkenyl or benzyl; R2 is hydrogen, fluorine or C1-C6-alkyl and R3 is hydrogen, fluorine, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy, C1-C6-alkylthio, phenyl, phenoxy, phenylthio or C3-C7-cycloalkyl, and each aromatic substituent or aromatic moiety of a substituent is unsubstituted or mono- or poly-substituted by halogen, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, nitro and/or cyano; including the acid addition salts, quaternary azolium salts and metal complexes, are useful for controlling phytopathogenic microorganisms.

公开(公告)号：DK159093B

公开(公告)日：1990-09-03

申请号：DK380682

申请日：1982-08-25

Applicant: CIBA GEIGY AG

Inventor： FANKHAUSER ERNST ,  STURM ELMAR

IPC: A01N20060101 ,  A01N41/10 ,  A01N53/00 ,  C07C20060101 ,  C07C317/22

公开(公告)号：AU599014B2

公开(公告)日：1990-07-12

申请号：AU5349286

申请日：1986-02-14

Applicant: CIBA GEIGY AG

Inventor： STURM ELMAR ,  GALLAY JEAN JACQUES ,  KRISTINSSON HAUKUR ,  PISSIOTAS GEORG

IPC: C07D263/58 ,  A61K31/496 ,  A61K31/515 ,  A61P33/10 ,  C07D233/70 ,  C07D235/26 ,  C07D239/62 ,  C07D239/66 ,  C07D249/08 ,  C07D249/12 ,  C07D263/34 ,  C07D271/06 ,  C07D271/10 ,  C07D271/113 ,  C07D277/24 ,  C07D277/34 ,  C07D277/58 ,  C07D277/68 ,  C07D285/08 ,  C07D285/12 ,  C07D285/13 ,  C07D403/12 ,  C07D413/12 ,  C07D417/12 ,  A61K31/505

Abstract: The invention relates to novel 5-(azolyloxyphenylcarbamoyl)barbituric acid derivatives of the general formula I (I) wherein X is oxygen or sulfur; R1 is C1-C6alkyl, C1-C6alkoxy, C3-C6cycloalkyl or allyl; R2 is C1-C6alkyl or allyl; R3 is an unsubstituted or substituted five-membered azole ring which is bound through carbon and is selected from the group consisting of benzimadazole, benzoxazole, benzothiazole, imidazole, oxazole, thiazole, oxadiazole, thiadiazole and triazole; and R4 and R5 are each independently of the other hydrogen, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkoxy or C1-C6haloalkoxy; and to the tautomers and salts thereof, as anthelmintic compounds. Together with suitable carriers and further assistants, these compounds may be used in particular for controlling helminths which are parasites of animals.

公开(公告)号：PH24447A

公开(公告)日：1990-06-25

申请号：PH37183

申请日：1988-07-06

Applicant: CIBA GEIGY AG

Inventor： STURM ELMAR ,  GALLAY JEAN JAQUES ,  KRISTINSSON HAUKUR ,  PISSIOTAS GEORG

IPC: C07D263/58 ,  A61K31/496 ,  A61K31/515 ,  A61P33/10 ,  C07D233/70 ,  C07D235/26 ,  C07D239/62 ,  C07D239/66 ,  C07D249/08 ,  C07D249/12 ,  C07D263/34 ,  C07D271/06 ,  C07D271/10 ,  C07D271/113 ,  C07D277/24 ,  C07D277/34 ,  C07D277/58 ,  C07D277/68 ,  C07D285/08 ,  C07D285/12 ,  C07D285/13 ,  C07D403/12 ,  C07D413/12 ,  C07D417/12

Abstract: The invention relates to novel 5-(azolyloxyphenylcarbamoyl)barbituric acid derivatives of the general formula I (I) wherein X is oxygen or sulfur; R1 is C1-C6alkyl, C1-C6alkoxy, C3-C6cycloalkyl or allyl; R2 is C1-C6alkyl or allyl; R3 is an unsubstituted or substituted five-membered azole ring which is bound through carbon and is selected from the group consisting of benzimadazole, benzoxazole, benzothiazole, imidazole, oxazole, thiazole, oxadiazole, thiadiazole and triazole; and R4 and R5 are each independently of the other hydrogen, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkoxy or C1-C6haloalkoxy; and to the tautomers and salts thereof, as anthelmintic compounds. Together with suitable carriers and further assistants, these compounds may be used in particular for controlling helminths which are parasites of animals.

公开(公告)号：NO161256C

公开(公告)日：1989-07-26

申请号：NO834592

申请日：1983-12-13

Applicant: CIBA GEIGY AG

Inventor： STURM ELMAR ,  MEYER ALFRED

IPC: A01N43/50 ,  A01N43/653 ,  A01P3/00 ,  C07C39/00 ,  C07C45/63 ,  C07C45/71 ,  C07D233/60 ,  C07D233/64 ,  C07D249/08 ,  C07D303/08 ,  C07D303/22 ,  C07D303/34 ,  C07D521/00

Abstract: 1-Azolyl-2-aryl-3-fluoro-alkan-2- ols of the general formula I in which Az is 1H-1,2,4-triazole, 4H-1,2,4-triazole or 1H-imidazole; Ar is an unsubstituted or substituted aromatic radical from the series comprising phenyl, biphenyl, phenoxyphenyl and naphthyl; R1 is hydrogen, C1-C4-alkyl, C3-C5-alkenyl or benzyl; R2 is hydrogen, fluorine or C1-C6-alkyl and R3 is hydrogen, fluorine, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy, C1-C6-alkylthio, phenyl, phenoxy, phenylthio or C3-C7-cycloalkyl, and each aromatic substituent or aromatic moiety of a substituent is unsubstituted or mono- or poly-substituted by halogen, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, nitro and/or cyano; including the acid addition salts, quaternary azolium salts and metal complexes, are useful for controlling phytopathogenic microorganisms.

公开(公告)号：AU584861B2

公开(公告)日：1989-06-08

申请号：AU3245084

申请日：1984-08-28

Applicant: CIBA GEIGY

Inventor： HUBELE ADOLF ,  ECKHARDT WOLFGANG ,  STURM ELMAR ,  ZONDLER HELMUT

IPC: A01N43/54 ,  C07D239/42 ,  C07D239/46 ,  C07D239/47 ,  C07D239/48 ,  C07D239/50 ,  C07D239/52 ,  C07D239/56 ,  C07D401/12 ,  C07D405/12 ,  A61K31/505 ,  C07D239/58

公开(公告)号：HU196891B

公开(公告)日：1989-02-28

申请号：HU424683

申请日：1983-12-13

Applicant: CIBA GEIGY AG

Inventor： STURM ELMAR ,  MEYER ALFRED

IPC: A01N43/50 ,  A01N43/653 ,  A01P3/00 ,  C07C39/00 ,  C07C45/63 ,  C07C45/71 ,  C07D233/60 ,  C07D233/64 ,  C07D249/08 ,  C07D303/08 ,  C07D303/22 ,  C07D303/34 ,  C07D521/00

Abstract: 1-Azolyl-2-aryl-3-fluoro-alkan-2- ols of the general formula I in which Az is 1H-1,2,4-triazole, 4H-1,2,4-triazole or 1H-imidazole; Ar is an unsubstituted or substituted aromatic radical from the series comprising phenyl, biphenyl, phenoxyphenyl and naphthyl; R1 is hydrogen, C1-C4-alkyl, C3-C5-alkenyl or benzyl; R2 is hydrogen, fluorine or C1-C6-alkyl and R3 is hydrogen, fluorine, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy, C1-C6-alkylthio, phenyl, phenoxy, phenylthio or C3-C7-cycloalkyl, and each aromatic substituent or aromatic moiety of a substituent is unsubstituted or mono- or poly-substituted by halogen, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, nitro and/or cyano; including the acid addition salts, quaternary azolium salts and metal complexes, are useful for controlling phytopathogenic microorganisms.

公开(公告)号：GB2171099B

公开(公告)日：1988-10-19

申请号：GB8603352

申请日：1986-02-11

Applicant: CIBA GEIGY AG

Inventor： STURM ELMAR ,  GALLAY JEAN JACQUES ,  KRISTINSSON HAUKUR ,  PISSIOTAS GEORG

IPC: C07D263/58 ,  A61K31/496 ,  A61K31/515 ,  A61P33/10 ,  C07D233/70 ,  C07D235/26 ,  C07D239/62 ,  C07D239/66 ,  C07D249/08 ,  C07D249/12 ,  C07D263/34 ,  C07D271/06 ,  C07D271/10 ,  C07D271/113 ,  C07D277/24 ,  C07D277/34 ,  C07D277/58 ,  C07D277/68 ,  C07D285/08 ,  C07D285/12 ,  C07D285/13 ,  C07D403/12 ,  C07D413/12 ,  C07D417/12

Abstract: The invention relates to novel 5-(azolyloxyphenylcarbamoyl)barbituric acid derivatives of the general formula I (I) wherein X is oxygen or sulfur; R1 is C1-C6alkyl, C1-C6alkoxy, C3-C6cycloalkyl or allyl; R2 is C1-C6alkyl or allyl; R3 is an unsubstituted or substituted five-membered azole ring which is bound through carbon and is selected from the group consisting of benzimadazole, benzoxazole, benzothiazole, imidazole, oxazole, thiazole, oxadiazole, thiadiazole and triazole; and R4 and R5 are each independently of the other hydrogen, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkoxy or C1-C6haloalkoxy; and to the tautomers and salts thereof, as anthelmintic compounds. Together with suitable carriers and further assistants, these compounds may be used in particular for controlling helminths which are parasites of animals.