公开(公告)号：ZA8909722B

公开(公告)日：1990-09-26

申请号：ZA8909722

申请日：1989-12-19

Applicant: HOECHST AG

Inventor： STARK HERBERT ,  HERBERT STARK ,  SALBECK GERHARD ,  GERHARD SALBECK ,  BONIN WERNER ,  WERNER BONIN

IPC: A61K31/415 ,  A61P33/00 ,  C07D233/20 ,  C07D233/22 ,  C07D233/24 ,  C07D ,  A01N

CPC classification number: C07D233/20 ,  C07D233/22 ,  C07D233/24

公开(公告)号：CA2011832A1

公开(公告)日：1990-09-10

申请号：CA2011832

申请日：1990-03-09

Applicant: HOECHST AG

Inventor： SCHNATTERER STEFAN ,  SCHUBERT HANS H ,  SALBECK GERHARD ,  KNAUF WERNER ,  WALTERSDORFER ANNA ,  KERN MANFRED

IPC: C07D233/64 ,  A01N43/08 ,  A01N43/10 ,  A01N43/40 ,  A01N43/50 ,  A01N43/54 ,  A01N43/56 ,  A01N43/74 ,  A01N43/78 ,  A61K31/425 ,  A61K31/426 ,  A61P33/10 ,  C07D213/26 ,  C07D213/30 ,  C07D213/61 ,  C07D213/64 ,  C07D213/643 ,  C07D213/65 ,  C07D239/26 ,  C07D263/32 ,  C07D277/22 ,  C07D277/24 ,  C07D307/12 ,  C07D307/40 ,  C07D307/42 ,  C07D333/12 ,  C07D333/16 ,  C07D333/32 ,  C07D401/06 ,  C07D403/06 ,  C07D407/06 ,  C07D407/12 ,  C07D409/06 ,  C07D409/12 ,  C07D413/06 ,  C07D413/12 ,  C07D417/06 ,  C07D417/12 ,  A01N43/00 ,  C07D401/12

Abstract: of the disclosure Heteroaryl-aryl-butene and -butane derivatives, process for their preparation, agents containing them, and their use as pesticids Compounds of the fonmulae I and II, the stereoisomers thereof, and the mixtures of the latter (I) (II) where R1 is pyridyl, pyrimidyl, thienyl, thiazolyl, furanyl, pyrazolyl, 1,3-oxazolyl or imidazolyl, all of which can be substituted, R2 is H, (C1-C4)alkyl, (C1-C4)haloalkyl, (C1-C4)alkoxy (C3-C6)cycloalkyl, -CH=CH2 or -C=CH, R3 is H or (C1-C4)alkyl, R4 is H, (C1-C4)alkyl, -CN or -C=CH, A is CH2, 0 or S, B is CH, N or C(CH3), R5 is H or halogen and R6 is phenyl, phenoxy or benzyl, all of which can be monosubstituted to pentasubstituted by halogen or (C1-C3)haloalkyl, have advantageous insecticidal or acaricidal properties.

公开(公告)号：CA2005976A1

公开(公告)日：1990-06-20

申请号：CA2005976

申请日：1989-12-19

Applicant: HOECHST AG

Inventor： STARK HERBERT ,  SALBECK GERHARD ,  BONIN WERNER

IPC: A61K31/415 ,  A61P33/00 ,  C07D233/20 ,  C07D233/22 ,  C07D233/24 ,  A01N43/50

Abstract: of the disclosure: Agents containing imidazoline derivatives for systemic combating of ectoparasites in host animals and novel imidazoline derivatives The present invention relates to agents for systemic combating of ectoparasites in host animals, containing a compound of the formula I (I) in which R1 denotes hydrogen, (C1-C5)-alkyl, (C1-C3)-halo- genoalkyl or halogen; R2 and R3 independently of one another denote (C1-C5)- alkyl, (C2-Cs)-alkerLyl, (C2-C5)-alkynyl, (C3-C7)-cycloalkyl, (C3-C7)-cycloalkenyl, (C1-C3)-halo-genoalkyl, halogen, cyano, nitro, (C1-C5)-alkoxy, (C1-C3)-alkoxy-(C1-C3)-alkyl, (C1-C3)-halogenoalkoxy or (C1-C3)-alkylthio, or R2 and R3 together form a polymethylene chain having 2 to 5 carbon atoms; R4 denotes hydrogen, (C1-C10)-alkyl, (C2-C5)-alkenyl or (C3-C7)-cycloalkyl; R5 denotes hydrogen, (C1-C10)-alkyl, (C3-C5)-alk- enyl, (C3-C5)-alkynyl, (C3-C7)-cycloalkyl, (C3C7)-cycloalkenyl, (C1-C3)-halogenoalkyl or (C1C3 )-alkoxy-(C1-C3)-alkyl; X denotes oxygen, sulfur or an -NR6- group; and R6 denoteshydrogen, (C1-C5)-alkyl,(C3-C5)-alkenyl, (C3-C5)-alkynyl, (C3-C7)-cycloalkyl, (C3-C7)-cycloalkenyl, (C1-C3)-halogenoalkyl or (C1-C3)-alkoxy-(C1-C3)-alkyl, or biologically tolerated acid addition salts thereof. The compounds of the formula I are novel in some cases and are likewise included in the invention.

公开(公告)号：PH24101A

公开(公告)日：1990-03-05

申请号：PH35180

申请日：1987-04-24

Applicant: HOECHST AG

Inventor： SCHUBERT HANS HERBERT ,  SALBECK GERHARD ,  LUDERS WALTER ,  KNAUF WERNER ,  WALTERSDORFER ANNA

IPC: A01N55/00 ,  A01N55/10 ,  C07F7/10 ,  A01P7/04 ,  C07F7/08 ,  C07F7/12 ,  C07F7/18 ,  C07F7/02 ,  A01N59/00

Abstract: The compounds of the formula (I) (I) in which X denotes CH2 or O, R1 denotes (subst.) pyridyl or (subst.) pyrimidyl, R2 and R3 denote alkyl or alkenyl or R2 and R3 denote an alkylene chain, R4 denotes -H, -CN, -CCl3, -C 3BOND CH, alkyl, F, or -C(S)-NH2, R5 denotes pyridyl, furyl, thienyl, phthalimidyl, di(C1-C4)alkylmaleimidyl, thiophthalimidyl, dihydrophthalimidyl or tetrahydrophthalimidyl, which may all be substituted, or substituted phenyl, or R4 and R5-together with the carbon atom bridging them-denote an optionally substituted indanyl, cyclopentenoyl or cyclopentenyl radical, have advantageous insecticidal, acaricidal and nematocidal properties.

公开(公告)号：AU3594689A

公开(公告)日：1989-12-07

申请号：AU3594689

申请日：1989-06-01

Applicant: HOECHST AG

Inventor： LUDERS WALTER ,  SALBECK GERHARD ,  BAUER KLAUS ,  BIERINGER HERMANN

IPC: A01N25/32 ,  A01N47/06 ,  C07D237/16 ,  C07D401/04 ,  A01N43/08 ,  A01N43/10

公开(公告)号：DK143989A

公开(公告)日：1989-09-27

申请号：DK143989

申请日：1989-03-22

Applicant: HOECHST AG

Inventor： SCHUBERT HANS HERBERT ,  SALBECK GERHARD ,  KRAUSE HANS-PETER ,  KNAUF WERNER ,  WALTERSDORFER ANNA ,  KERN MANFRED

IPC: C07D253/06 ,  A01N43/40 ,  A01N55/00 ,  A01N55/10 ,  C07D213/32 ,  C07D213/61 ,  C07D213/64 ,  C07D213/643 ,  C07D213/70 ,  C07D237/12 ,  C07D237/14 ,  C07D237/18 ,  C07D239/26 ,  C07D239/32 ,  C07D239/34 ,  C07D241/16 ,  C07D241/18 ,  C07D257/08 ,  C07D401/12 ,  C07D409/12 ,  C07D491/056 ,  C07F7/10

Abstract: Compounds of the formula I, their optical isomers and mixtures thereof … … in which… M represents C or Si,… R represents unsubstituted or substituted pyridyl, unsubstituted or substituted pyrimidyl, and - when M = C - unsubstituted or substituted pyridazinyl, unsubstituted or substituted pyrazinyl, unsubstituted or substituted 1,2,4-triazinyl, unsubstituted or substituted 1,2,4,5-tetrazinyl,… R , R independently of one another represent alkyl, alkenyl, haloalkyl, phenyl, or R and R represent an alkylene chain which - together with the quaternary central atom (M)- forms an unsubstituted or fluorine-substituted ring having four to six ring members (when M = Si) or having three to six ring members (when M = C),… R represents H, F, -CN, -CCl3, -C IDENTICAL CH, (C1-C4)alkyl, - @ -NH2,… R represents pyridyl, furyl, thienyl, all of which can be substituted, phthalimidyl, dialkylmaleimidyl, thiophthalimidyl, dihydrophthalimidyl, tetrahydrophthalimidyl, substituted phenyl,… or R and R - together with the carbon atom linking them - form an optionally substituted indanyl, cyclopentenoyl or cyclopentenyl radical,… and their salts and quaternisation products have advantageous insecticidal, acaricidal or nematocidal properties.

公开(公告)号：DK143989D0

公开(公告)日：1989-03-22

申请号：DK143989

申请日：1989-03-22

Applicant: HOECHST AG

Inventor： SCHUBERT HANS HERBERT ,  SALBECK GERHARD ,  KRAUSE HANS-PETER ,  KNAUF WERNER ,  WALTERSDORFER ANNA ,  KERN MANFRED

IPC: C07D253/06 ,  A01N43/40 ,  A01N55/00 ,  A01N55/10 ,  C07D213/32 ,  C07D213/61 ,  C07D213/64 ,  C07D213/643 ,  C07D213/70 ,  C07D237/12 ,  C07D237/14 ,  C07D237/18 ,  C07D239/26 ,  C07D239/32 ,  C07D239/34 ,  C07D241/16 ,  C07D241/18 ,  C07D257/08 ,  C07D401/12 ,  C07D409/12 ,  C07D491/056 ,  C07F7/10

Abstract: Compounds of the formula I, their optical isomers and mixtures thereof … … in which… M represents C or Si,… R represents unsubstituted or substituted pyridyl, unsubstituted or substituted pyrimidyl, and - when M = C - unsubstituted or substituted pyridazinyl, unsubstituted or substituted pyrazinyl, unsubstituted or substituted 1,2,4-triazinyl, unsubstituted or substituted 1,2,4,5-tetrazinyl,… R , R independently of one another represent alkyl, alkenyl, haloalkyl, phenyl, or R and R represent an alkylene chain which - together with the quaternary central atom (M)- forms an unsubstituted or fluorine-substituted ring having four to six ring members (when M = Si) or having three to six ring members (when M = C),… R represents H, F, -CN, -CCl3, -C IDENTICAL CH, (C1-C4)alkyl, - @ -NH2,… R represents pyridyl, furyl, thienyl, all of which can be substituted, phthalimidyl, dialkylmaleimidyl, thiophthalimidyl, dihydrophthalimidyl, tetrahydrophthalimidyl, substituted phenyl,… or R and R - together with the carbon atom linking them - form an optionally substituted indanyl, cyclopentenoyl or cyclopentenyl radical,… and their salts and quaternisation products have advantageous insecticidal, acaricidal or nematocidal properties.

公开(公告)号：DK204988A

公开(公告)日：1988-10-16

申请号：DK204988

申请日：1988-04-14

Applicant: HOECHST AG

Inventor： SCHUBERT HANS HERBERT ,  SALBECK GERHARD ,  KRAUSE HANS-PETER ,  LUEDERS WALTER ,  KNAUF WERNER ,  WALTERSDORFER ANNA ,  KERN MANFRED

IPC: A01N43/40 ,  A01N43/54 ,  A01N43/58 ,  A01N43/60 ,  A01N55/10 ,  A01P7/02 ,  A01P7/04 ,  C07D213/61 ,  C07D253/06 ,  C07D213/63 ,  C07D213/64 ,  C07D213/643 ,  C07D213/65 ,  C07D213/70 ,  C07D237/12 ,  C07D237/14 ,  C07D237/18 ,  C07D239/26 ,  C07D239/30 ,  C07D239/34 ,  C07D239/38 ,  C07D241/16 ,  C07D241/18 ,  C07D253/07 ,  C07D253/08 ,  C07D257/08 ,  C07D401/06 ,  C07D401/08 ,  C07D401/12 ,  C07D409/06 ,  C07D409/08 ,  C07D491/04 ,  C07D491/056 ,  C07D213/60 ,  A01N43/48

Abstract: Compounds of the formula (I) and their stereoisomers (I) wherein A, B, C' and D independently of one another denote CH or N, in which at least one of the symbols A, B, C' or D must correspond to a nitrogen atom, X denotes CH2 or oxygen, R1 denotes a radical bonded to a carbon atom from the series comprising H, trialkylsilyl, halogen, nitro, cyano, alkenyl, alkynyl, amino, cycloalkyl, phenyl, phenxy, alkoxy, alkenyloxy, alkynyloxy, hydroxycarbonyl, alkylthio, cycloalkyloxy, alkylcarbonyl, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, halogenoalkyl, alkoxyalkyl, halogenoalkoxy, halogenoalkylthio, halogenoalkoxyalkyl, alkylthioalkyl, alkoxyalkoxy, halogenoalkoxyalkoxy, alkenyloxyalkoxy, halogenoalkenyloxy, alkoxyalkylthio, alkylthioalkoxy, alkylthioalkylthio, halogenoalkoxycarbonyl, halogenoalkenyloxycarbonyl or dialkylamino or two radicals R1 when they are positioned ortho to one another together denote a methylenedioxy, ethylenedioxy or alkylene radical, R2 and R3 independently of one another denote alkyl, alkenyl or phenyl, or R2 and R3 denote an alkylene chain which-together with the quaternary carbon atom-forms an unsubstituted or fluorinesubstituted ring having three to six ring members, R4 denotes -H, F, -CN, -CCl3, -C 3BOND CH, (C1-C4)alkyl, -C-NH2, S R5 denotes pyridyl, furyl or thienyl which can all be substituted, phthalimidyl, dialkylmaleimidyl, thiophthalimidyl, dihydrophthalimidyl, tetrahydrophthalimidyl or substituted phenyl, or R4 and R5-together with the carbon atom bridging them-denote an optionally substituted indanyl, cyclopentenoyl or cyclopentenyl radical and n denotes 0, 1 or 2, possess advantageous properties for combating pests, in particular insects and acarids. Furthermore, processes for the preparation of compounds of the formula I are described.

公开(公告)号：DK204988D0

公开(公告)日：1988-04-14

申请号：DK204988

申请日：1988-04-14

Applicant: HOECHST AG

Inventor： SCHUBERT HANS HERBERT ,  SALBECK GERHARD ,  KRAUSE HANS-PETER ,  LUEDERS WALTER ,  KNAUF WERNER ,  WALTERSDORFER ANNA ,  KERN MANFRED

IPC: A01N43/40 ,  A01N43/54 ,  A01N43/58 ,  A01N43/60 ,  A01N55/10 ,  A01P7/02 ,  A01P7/04 ,  C07D213/61 ,  C07D253/06 ,  C07D213/63 ,  C07D213/64 ,  C07D213/643 ,  C07D213/65 ,  C07D213/70 ,  C07D237/12 ,  C07D237/14 ,  C07D237/18 ,  C07D239/26 ,  C07D239/30 ,  C07D239/34 ,  C07D239/38 ,  C07D241/16 ,  C07D241/18 ,  C07D253/07 ,  C07D253/08 ,  C07D257/08 ,  C07D401/06 ,  C07D401/08 ,  C07D401/12 ,  C07D409/06 ,  C07D409/08 ,  C07D491/04 ,  C07D491/056 ,  C07D213/60 ,  A01N43/48

Abstract: Compounds of the formula (I) and their stereoisomers (I) wherein A, B, C' and D independently of one another denote CH or N, in which at least one of the symbols A, B, C' or D must correspond to a nitrogen atom, X denotes CH2 or oxygen, R1 denotes a radical bonded to a carbon atom from the series comprising H, trialkylsilyl, halogen, nitro, cyano, alkenyl, alkynyl, amino, cycloalkyl, phenyl, phenxy, alkoxy, alkenyloxy, alkynyloxy, hydroxycarbonyl, alkylthio, cycloalkyloxy, alkylcarbonyl, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, halogenoalkyl, alkoxyalkyl, halogenoalkoxy, halogenoalkylthio, halogenoalkoxyalkyl, alkylthioalkyl, alkoxyalkoxy, halogenoalkoxyalkoxy, alkenyloxyalkoxy, halogenoalkenyloxy, alkoxyalkylthio, alkylthioalkoxy, alkylthioalkylthio, halogenoalkoxycarbonyl, halogenoalkenyloxycarbonyl or dialkylamino or two radicals R1 when they are positioned ortho to one another together denote a methylenedioxy, ethylenedioxy or alkylene radical, R2 and R3 independently of one another denote alkyl, alkenyl or phenyl, or R2 and R3 denote an alkylene chain which-together with the quaternary carbon atom-forms an unsubstituted or fluorinesubstituted ring having three to six ring members, R4 denotes -H, F, -CN, -CCl3, -C 3BOND CH, (C1-C4)alkyl, -C-NH2, S R5 denotes pyridyl, furyl or thienyl which can all be substituted, phthalimidyl, dialkylmaleimidyl, thiophthalimidyl, dihydrophthalimidyl, tetrahydrophthalimidyl or substituted phenyl, or R4 and R5-together with the carbon atom bridging them-denote an optionally substituted indanyl, cyclopentenoyl or cyclopentenyl radical and n denotes 0, 1 or 2, possess advantageous properties for combating pests, in particular insects and acarids. Furthermore, processes for the preparation of compounds of the formula I are described.

公开(公告)号：BR8701971A

公开(公告)日：1988-02-02

申请号：BR8701971

申请日：1987-04-24

Applicant: HOECHST AG

Inventor： SCHUBERT HANS HERBERT ,  SALBECK GERHARD ,  LUEDERS WALTER ,  KNAUF WERNER ,  WALTERSDORFER ANNA

IPC: C07F7/10 ,  A01N55/00 ,  A01N55/10 ,  A01P7/04 ,  C07F7/08 ,  C07F7/12 ,  C07F7/18 ,  A01N59/00

Abstract: The compounds of the formula (I) (I) in which X denotes CH2 or O, R1 denotes (subst.) pyridyl or (subst.) pyrimidyl, R2 and R3 denote alkyl or alkenyl or R2 and R3 denote an alkylene chain, R4 denotes -H, -CN, -CCl3, -C 3BOND CH, alkyl, F, or -C(S)-NH2, R5 denotes pyridyl, furyl, thienyl, phthalimidyl, di(C1-C4)alkylmaleimidyl, thiophthalimidyl, dihydrophthalimidyl or tetrahydrophthalimidyl, which may all be substituted, or substituted phenyl, or R4 and R5-together with the carbon atom bridging them-denote an optionally substituted indanyl, cyclopentenoyl or cyclopentenyl radical, have advantageous insecticidal, acaricidal and nematocidal properties.