AGENTS CONTAINING IMIDAZOLINE DERIVATIVES FOR SYSTEMIC COMBATING OF ECTO-PARASITES IN HOST ANIMALS AND NOVEL IMIDAZOLINE DERIVATIVES

    公开(公告)号:CA2005976A1

    公开(公告)日:1990-06-20

    申请号:CA2005976

    申请日:1989-12-19

    Applicant: HOECHST AG

    Abstract: of the disclosure: Agents containing imidazoline derivatives for systemic combating of ectoparasites in host animals and novel imidazoline derivatives The present invention relates to agents for systemic combating of ectoparasites in host animals, containing a compound of the formula I (I) in which R1 denotes hydrogen, (C1-C5)-alkyl, (C1-C3)-halo- genoalkyl or halogen; R2 and R3 independently of one another denote (C1-C5)- alkyl, (C2-Cs)-alkerLyl, (C2-C5)-alkynyl, (C3-C7)-cycloalkyl, (C3-C7)-cycloalkenyl, (C1-C3)-halo-genoalkyl, halogen, cyano, nitro, (C1-C5)-alkoxy, (C1-C3)-alkoxy-(C1-C3)-alkyl, (C1-C3)-halogenoalkoxy or (C1-C3)-alkylthio, or R2 and R3 together form a polymethylene chain having 2 to 5 carbon atoms; R4 denotes hydrogen, (C1-C10)-alkyl, (C2-C5)-alkenyl or (C3-C7)-cycloalkyl; R5 denotes hydrogen, (C1-C10)-alkyl, (C3-C5)-alk- enyl, (C3-C5)-alkynyl, (C3-C7)-cycloalkyl, (C3C7)-cycloalkenyl, (C1-C3)-halogenoalkyl or (C1C3 )-alkoxy-(C1-C3)-alkyl; X denotes oxygen, sulfur or an -NR6- group; and R6 denoteshydrogen, (C1-C5)-alkyl,(C3-C5)-alkenyl, (C3-C5)-alkynyl, (C3-C7)-cycloalkyl, (C3-C7)-cycloalkenyl, (C1-C3)-halogenoalkyl or (C1-C3)-alkoxy-(C1-C3)-alkyl, or biologically tolerated acid addition salts thereof. The compounds of the formula I are novel in some cases and are likewise included in the invention.

    AGENTS CONTAINING IMIDAZOLINE DERIVATIVES FOR SYSTEMIC COMBATING OF ECTOPARASITES IN HOST ANIMALS AND NOVEL IMIDAZOLINE DERIVATIVES

    公开(公告)号:AU4685689A

    公开(公告)日:1990-06-28

    申请号:AU4685689

    申请日:1989-12-19

    Applicant: HOECHST AG

    Abstract: The present invention relates to agents for systemic combating of ectoperasites in host animals, containing a compound of the formul I (I) in which R1 denotes hydrogen, (C1-C5)-alkyl, (C1-C3)-halogenoalkyl or halogen; R2 and R3 independently of one another denote (c1-C5)-alkyl, (C2-C5)-alkenyl, (C2-C5)-alkynyl, (C3-C7)-cycloalkyl, (C3-C7)-cycloalkenyl, (C1-C3)-halogenoalkyl, halogen, cyano, nitro, (C1-C5)-alkoxy, (C1 -C3)-alkoxy-C1-C3)-alkyl, (C1-C3)-halogenoalkoxy or (C1-C3)-alkylthio, or R2 and R3 together form a polymethylene chain having 2 to 5 carbon atoms: R4 denotes hydrogen, (c1-C10)-alkyl, (C2-C5)-alkenyl or (C3-C7)-cycloalkyl; R5 denotes hydrogen, (C1-C10)-alkyl, (C3-C5)-alkenyl, C3-C5)-alkynyl, (C3-C7)- cycloalkyl, (C3-C7)-cycloalkenyl, (C1-C3)-halogenoalkyl or (C1-C3)-alkoxy-(C hd 1-C3)-alkyl; X denotes oxygen, sulfur or an -NR6-group; and R6 denotes hydrogen, (C1-C5)-alkyl, (C3-C5)-alkenyl, C3-C5)-alkynyl, (C3-C7)-cycloalkyl, C3-C7)-cycloalkenyl, (C1-C3)-halogenoalkyl or (C1-C3)-alkoxy-(C1 -C3)-alkyl, or biologically tolerated acid addition salts thereof. The compounds of the formulas I are novel in some cases and are likewise included in the invention.

    6.
    发明专利
    未知

    公开(公告)号:DK648489D0

    公开(公告)日:1989-12-19

    申请号:DK648489

    申请日:1989-12-19

    Applicant: HOECHST AG

    Abstract: The present invention relates to agents for systemic combating of ectoperasites in host animals, containing a compound of the formul I (I) in which R1 denotes hydrogen, (C1-C5)-alkyl, (C1-C3)-halogenoalkyl or halogen; R2 and R3 independently of one another denote (c1-C5)-alkyl, (C2-C5)-alkenyl, (C2-C5)-alkynyl, (C3-C7)-cycloalkyl, (C3-C7)-cycloalkenyl, (C1-C3)-halogenoalkyl, halogen, cyano, nitro, (C1-C5)-alkoxy, (C1 -C3)-alkoxy-C1-C3)-alkyl, (C1-C3)-halogenoalkoxy or (C1-C3)-alkylthio, or R2 and R3 together form a polymethylene chain having 2 to 5 carbon atoms: R4 denotes hydrogen, (c1-C10)-alkyl, (C2-C5)-alkenyl or (C3-C7)-cycloalkyl; R5 denotes hydrogen, (C1-C10)-alkyl, (C3-C5)-alkenyl, C3-C5)-alkynyl, (C3-C7)- cycloalkyl, (C3-C7)-cycloalkenyl, (C1-C3)-halogenoalkyl or (C1-C3)-alkoxy-(C hd 1-C3)-alkyl; X denotes oxygen, sulfur or an -NR6-group; and R6 denotes hydrogen, (C1-C5)-alkyl, (C3-C5)-alkenyl, C3-C5)-alkynyl, (C3-C7)-cycloalkyl, C3-C7)-cycloalkenyl, (C1-C3)-halogenoalkyl or (C1-C3)-alkoxy-(C1 -C3)-alkyl, or biologically tolerated acid addition salts thereof. The compounds of the formulas I are novel in some cases and are likewise included in the invention.

    7.
    发明专利
    未知

    公开(公告)号:DE59209757D1

    公开(公告)日:1999-11-18

    申请号:DE59209757

    申请日:1992-12-24

    Applicant: HOECHST AG

    Abstract: A herbicide-safener combination comprises a cyclic 2-acyl-1,3-dicarbonyl compound herbicide (I) and an 8-quinolinyloxyalkanoic acid derivative safener (II). A herbicidal composition contains at least one 2-acyl-1,3-dicarbonyl compound herbicide of formula (I) (or its salt) and at least one quinoline derivative safener of formula (II). R1, R3 = H, halo, alkyl, haloalkyl, haloalkoxy, CN, NO2, S(O)mR11, NR12R13, NR14COR15, COR16 or OCH2CH2OR21; R2 = halo, CN, NO2, alkyl, alkoxy, haloalkyl, haloalkoxy, S(O)pR10, OSO2R10 or N(R20)SO2R19; W = N or CH; R10 = alkyl, haloalkyl or alkoxy; R11 = alkyl, haloalkyl or NR17R16; or phenyl or benzyl (both optionally ring-substituted); R12-R15, R17, R18, R21 = H or alkyl; R16 = H, alkyl, haloalkyl or alkoxy; R19, R20 = alkyl or haloalkyl; m, p = 0-2; U = group completing an optionally further substituted 5- or 6-membered carbocyclic or heterocyclic ring; Y = halo, A', NO2 or OA; A = 1-4C alkyl; A' = 1-4C alkyl or 1-4C haloalkyl; n = 1-5; Q = 1-2C alkylene (optionally substituted by 1 or 2 A); Z' = ORa, SRa or NRRa; R = H, 1-6C alkyl, 1-6C alkoxy or optionally substituted phenyl; Ra = H; or 1-18C alkyl, 3-12C cycloalkyl, 2-8C alkenyl or 2-8C alkynyl (all optionally substituted by one or more of halo, OH, OB, SB, 3-7C cycloalkyl, 3-7C cycloalkoxy, CN, NHA, N(A)2, BOCO, 1-8C alkylthiocarbonyl, BCO, 1-(=NOH, =NA or =NOA)-1-6C alkyl, BCONH, CONH2, mono- or di-(1-6C alkyl)-aminocarbonyl, (2-6C alkenyl, 2-6C alkynyl or 1-8C alkoxy)-aminocarbonyl, 1-8C alkylaminocarbonylamino, 1-6C alkylcarbonyloxy (optionally substituted by halo, NO2, OA or optionally substituted phenyl), (2-6C alkenyl or 2-6C alkynyl)carbonyloxy, 1-8C alkylsulfonyl, Ar, Ar-(1-6C) alkoxy, Ar-(1-6C) alkoxycarbonyl, OAr, ArCOO, ArCONH, Ar-(1-6C) alkylcarbonylamino, Si(R')3, OSi(R')3, (R')3-(1-6C) alkoxy, COON(R')2, ON=C(R')2, N=C(R')2, ON(R')2, CH(OR')2, O(CH2)qCH(OR')2 or R''OCR'''(OR'')-(1-6C) alkoxy); or NRRa = optionally unsaturated 3-7 membered heterocycle containing 1-3 heteroatoms (optionally substituted by A, OA or optionally substituted phenyl); B = 1-8C alkyl, 2-8C alkenyl or 2-8C alkynyl; Ar = phenyl (optionally substituted by one or more of halo, A', OA' and NO2); R' = H, A or phenyl (optionally substituted by one or more of halo, A', OA; and NO2); or (R')2 = 2-6C alkylene; q = 0-6; R'' = A; or (R'')2 = 1-6C alkylene; R''' = H or A. Independent claims are included for: (1) a method for protecting crop plants against the phytotoxic side-effects of (I), involving applying (II) to the plants (or their seeds or growth area) before, after or simultaneously with application of (I); and (2) the use of (II) for protecting crop plants against the phytotoxic side-effects of herbicides (I).

    9.
    发明专利
    未知

    公开(公告)号:BR8906608A

    公开(公告)日:1990-09-04

    申请号:BR8906608

    申请日:1989-12-20

    Applicant: HOECHST AG

    Abstract: The present invention relates to agents for systemic combating of ectoperasites in host animals, containing a compound of the formul I (I) in which R1 denotes hydrogen, (C1-C5)-alkyl, (C1-C3)-halogenoalkyl or halogen; R2 and R3 independently of one another denote (c1-C5)-alkyl, (C2-C5)-alkenyl, (C2-C5)-alkynyl, (C3-C7)-cycloalkyl, (C3-C7)-cycloalkenyl, (C1-C3)-halogenoalkyl, halogen, cyano, nitro, (C1-C5)-alkoxy, (C1 -C3)-alkoxy-C1-C3)-alkyl, (C1-C3)-halogenoalkoxy or (C1-C3)-alkylthio, or R2 and R3 together form a polymethylene chain having 2 to 5 carbon atoms: R4 denotes hydrogen, (c1-C10)-alkyl, (C2-C5)-alkenyl or (C3-C7)-cycloalkyl; R5 denotes hydrogen, (C1-C10)-alkyl, (C3-C5)-alkenyl, C3-C5)-alkynyl, (C3-C7)- cycloalkyl, (C3-C7)-cycloalkenyl, (C1-C3)-halogenoalkyl or (C1-C3)-alkoxy-(C hd 1-C3)-alkyl; X denotes oxygen, sulfur or an -NR6-group; and R6 denotes hydrogen, (C1-C5)-alkyl, (C3-C5)-alkenyl, C3-C5)-alkynyl, (C3-C7)-cycloalkyl, C3-C7)-cycloalkenyl, (C1-C3)-halogenoalkyl or (C1-C3)-alkoxy-(C1 -C3)-alkyl, or biologically tolerated acid addition salts thereof. The compounds of the formulas I are novel in some cases and are likewise included in the invention.

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