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21.
公开(公告)号:AU2016282837A1
公开(公告)日:2018-01-18
申请号:AU2016282837
申请日:2016-06-22
Applicant: SERVIER LAB , VERNALIS R&D LTD
Inventor: PACZAL ATTILA , KOTSCHY ANDRÁS , BRUNO ALAIN , GENESTE OLIVIER , CHEN I-JEN , DAVIDSON JAMES EDWARD PAUL , MURRAY JAMES BROOKE , ONDI LEVENTE , RADICS GÁBOR , SIPOS SZABOLCS , PROSZENYÁK ÁGNES , PERRON-SIERRA FRANÇOISE , BÁLINT BALÁZS , SZLÁVIK ZOLTÁN , SZABÓ ZOLTÁN , CSÉKEI MÁRTON
IPC: C07D495/04 , A61K31/519 , A61P35/00 , A61P37/00
Abstract: Compounds of formula (I): wherein R
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22.
公开(公告)号:AU2016282828A1
公开(公告)日:2018-01-18
申请号:AU2016282828
申请日:2016-06-22
Applicant: SERVIER LAB , VERNALIS R&D LTD
Inventor: BÁLINT BALÁZS , CSÉKEI MÁRTON , SZABÓ ZOLTÁN , SZLÁVIK ZOLTÁN , KOTSCHY ANDRÁS , CHANRION MAÏA , GENESTE OLIVIER , CHEN I-JEN , DAVIDSON JAMES EDWARD PAUL , MURRAY JAMES BROOKE , SIPOS SZABOLCS , ONDI LEVENTE , PROSZENYÁK AGNES
IPC: C07D209/12 , A61K31/381 , A61K31/4355 , A61K31/437 , A61P35/00 , C07D307/80 , C07D307/81 , C07D333/56 , C07D403/12 , C07D405/04 , C07D405/12 , C07D409/12 , C07D471/04 , C07D487/04 , C07D491/04 , C07D495/04
Abstract: Compounds of formula (I); wherein R
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23.
公开(公告)号:CA2990089A1
公开(公告)日:2016-12-29
申请号:CA2990089
申请日:2016-06-22
Applicant: VERNALIS (R&D) LTD , SERVIER LAB
Inventor: SZLAVIK ZOLTAN , SZABO ZOLTAN , CSEKEI MARTON , PACZAL ATTILA , KOTSCHY ANDRAS , BRUNO ALAIN , GENESTE OLIVIER , CHEN I-JEN , DAVIDSON JAMES EDWARD PAUL , MURRAY JAMES BROOKE , ONDI LEVENTE , RADICS GABOR , SIPOS SZABOLCS , PROSZENYAK AGNES , PERRON-SIERRA FRANCOISE , BALINT BALAZS
IPC: C07D495/04 , A61K31/519 , A61P35/00 , A61P37/00
Abstract: Compounds of formula (I): wherein R1, R2, R5, R6, R7, R12, X, Y, A, E and n are as defined in the description. Medicaments.
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公开(公告)号:CA2990088A1
公开(公告)日:2016-12-29
申请号:CA2990088
申请日:2016-06-22
Applicant: VERNALIS (R&D) LTD , SERVIER LAB
Inventor: SZLAVIK ZOLTAN , KOTSCHY ANDRAS , CHANRION MAIA , DEMARLES DIDIER , GENESTE OLIVIER , DAVIDSON JAMES EDWARD PAUL , MURRAY JAMES BROOKE , SIPOS SZABOLCS , PACZAL ATTILA , BALINT BALAZS
IPC: C07D495/04 , A61K31/519 , A61P35/00 , A61P37/00
Abstract: Compounds of formula (1) wherein R1, R2, R3, R4, R5, R6, R7, R13, Ra, Rb, A and n are as defined in the description. Medicaments containing them for use in the treatment of cancers.
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25.
公开(公告)号:CA2990084A1
公开(公告)日:2016-12-29
申请号:CA2990084
申请日:2016-06-22
Applicant: SERVIER LAB , VERNALIS (R&D) LTD
Inventor: BALINT BALAZS , CSEKEI MARTON , SZABO ZOLTAN , SZLAVIK ZOLTAN , KOTSCHY ANDRAS , CHANRION MAIA , GENESTE OLIVIER , CHEN I-JEN , DAVIDSON JAMES EDWARD PAUL , MURRAY JAMES BROOKE , SIPOS SZABOLCS , ONDI LEVENTE , PROSZENYAK AGNES
IPC: C07D209/12 , A61K31/381 , A61K31/4355 , A61K31/437 , A61P35/00 , C07D307/80 , C07D307/81 , C07D333/56 , C07D403/12 , C07D405/04 , C07D405/12 , C07D409/12 , C07D471/04 , C07D487/04 , C07D491/04 , C07D495/04
Abstract: Compounds of formula (I); wherein R1, R2, R3, R4, R5, R6, R7, R8, R14, W, A and n are as defined in the description. Medicaments.
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26.
公开(公告)号:HRP20161203T1
公开(公告)日:2016-11-04
申请号:HRP20161203
申请日:2016-09-20
Applicant: SERVIER LAB , VERNALIS (R&D) LTD
Inventor: KOTSCHY ANDRAS , SZLÁVIK ZOLTÁN , CSÉKEI MÁRTON , PACZAL ATTILA , SZABÓ ZOLTÁN , SIPOS SZABOLCS , RADICS GÁBOR , PROSZENYÁK ÁGNES , BÁLINT BALÁZS , BRUNO ALAIN , GENESTE OLIVIER , DAVIDSON JAMES EDWARD PAUL , MURRAY JAMES BROOKE , CHEN I-JEN , PERRON-SIERRA FRANÇOISE
IPC: C07D495/04 , A61K31/519 , A61P35/00 , A61P37/00
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公开(公告)号:DOP2014000282A
公开(公告)日:2016-06-30
申请号:DO2014000282
申请日:2014-12-15
Applicant: SERVIER LAB , VERNALIS R&D LTD
Inventor: MURRAY JAMES BROOKE , GENESTE OLIVIER , KOTSCHY ANDRAS , SZLAVIK ZOLTAN , CSEKEI MARTON , PACZAL ATTILA , SZABO ZOLTAN , SIPOS SZABOLCS , RADICS GABOR , PROSZENYAK AGNES , BELINT BALAZS , BRUNO ALAIN , DAVIDSON JAMES EDWARD PAUL , CHEN I-JEN , PERRON-SIERRA FRANCOISE
IPC: A61K31/505 , A61K31/513 , A61P35/00
Abstract: Compuestos de fórmula (I): en la que R1, R2, R3, R4, R5, R6, R7, R12, X, A y n son como se definen en la descripción. Medicamentos.
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28.
公开(公告)号:BR102014032336A2
公开(公告)日:2016-06-07
申请号:BR102014032336
申请日:2014-12-22
Applicant: SERVIER LAB , VERNALIS R&D LTD
Inventor: BRUNO ALAIN , KOTSCHY ANDRÁS , PACZAL ATTILA , BÁLINT BALÁZS , PERRON-SIERRA FRANÇOISE , RADICS GÁBOR , CHEN I-JEN , MURRAY JAMES BROOKE , DAVIDSON JAMES EDWARD PAUL , CSÉKEI MÁRTON , GENESTE OLIVIER , SIPOS SZABOLCS , SZABÓ ZOLTÁN , SZLÁVIK ZOLTÁN , PROSZENYÁK ÁGNES
IPC: C07D285/15 , A61K31/4365 , A61P35/00
Abstract: derivados de tienopirimidina, respectivo processo de preparo e composições farmacêuticas que os contêm. compostos de fórmula (i):nos quais r1, r2, r3, r4, r5, r6, r7, r12, x, a e n são tais como definidos na descrição. medicamentos.
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29.
公开(公告)号:MX376028B
公开(公告)日:2025-03-07
申请号:MX2018008808
申请日:2018-07-18
Applicant: SERVIER LAB , VERNALIS R&D LTD
Inventor: MARAGNO ANA LETICIA , KOTSCHY ANDRÁS , PACZAL ATTILA , BÁLINT BALÁZS , DEMARLES DIDIER , CHANRION MAÏA , GENESTE OLIVIER , SIPOS SZABOLCS , SZLÁVIK ZOLTÁN
IPC: C07F9/6561 , A61K31/519 , A61K31/661 , A61K45/06 , A61P35/00 , A61P35/02 , C07D495/04
Abstract: Compuestos de fórmula (I): (ver Fórmula) en la que R1, R2, R3, R4, R5, R6 e Y son como se han definido en la descripción. Medicamentos.
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公开(公告)号:AU2023302094A1
公开(公告)日:2025-01-23
申请号:AU2023302094
申请日:2023-07-07
Applicant: SERVIER LAB , VERNALIS R&D LTD
Inventor: BALASSA ANNAMÁRIA , CSÉKEI MÁRTON , ECKER ÁGOTA , GARAMVÖLGYI RITA , KOTSCHY ANDRÁS , LE TOUMELIN-BRAIZAT GAËTANE , MADARÁSZ ZOLTÁN , PROSZENYÁK ÁGNES , SIPOS SZABOLCS , SZABÓ ZOLTÁN , ZWILLINGER MÁRTON , BEDFORD SIMON , CHEN I-JEN , DAVIDSON JAMES EDWARD PAUL , MADDOX DANIEL , MCKENNA SEAN MARTIN , MURRAY JAMES BROOKE , PARSONS RACHEL JANE , STOKES STEPHEN , WALMSLEY CLAIRE LOUISE
IPC: C07D401/12 , A61K31/4709 , A61K31/506 , A61P35/00 , C07D215/233 , C07D403/12 , C07D403/14 , C07D405/12 , C07D417/14
Abstract: Compounds of Formula (I): wherein R
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