公开(公告)号：HU202837B

公开(公告)日：1991-04-29

申请号：HU192088

申请日：1988-04-14

Applicant: HOECHST AG

Inventor： SCHUBERT HANS HERBERT ,  SALBECK GERHARD ,  LUEDERS WALTER ,  KNAUF WERNER ,  WALTERSDORFER ANNA ,  KERN MANFRED

IPC: A01N43/40 ,  A01N43/54 ,  A01N43/58 ,  A01N43/60 ,  C07D253/06 ,  A01N55/10 ,  A01P7/02 ,  A01P7/04 ,  C07D213/61 ,  C07D213/63 ,  C07D213/64 ,  C07D213/643 ,  C07D213/65 ,  C07D213/70 ,  C07D237/12 ,  C07D237/14 ,  C07D237/18 ,  C07D239/26 ,  C07D239/30 ,  C07D239/34 ,  C07D239/38 ,  C07D241/16 ,  C07D241/18 ,  C07D253/07 ,  C07D253/08 ,  C07D257/08 ,  C07D401/06 ,  C07D401/08 ,  C07D401/12 ,  C07D409/06 ,  C07D409/08 ,  C07D491/04 ,  C07D491/056 ,  C07D213/60 ,  C07D247/00 ,  A01N43/48

Abstract: Compounds of the formula (I) and their stereoisomers (I) wherein A, B, C' and D independently of one another denote CH or N, in which at least one of the symbols A, B, C' or D must correspond to a nitrogen atom, X denotes CH2 or oxygen, R1 denotes a radical bonded to a carbon atom from the series comprising H, trialkylsilyl, halogen, nitro, cyano, alkenyl, alkynyl, amino, cycloalkyl, phenyl, phenxy, alkoxy, alkenyloxy, alkynyloxy, hydroxycarbonyl, alkylthio, cycloalkyloxy, alkylcarbonyl, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, halogenoalkyl, alkoxyalkyl, halogenoalkoxy, halogenoalkylthio, halogenoalkoxyalkyl, alkylthioalkyl, alkoxyalkoxy, halogenoalkoxyalkoxy, alkenyloxyalkoxy, halogenoalkenyloxy, alkoxyalkylthio, alkylthioalkoxy, alkylthioalkylthio, halogenoalkoxycarbonyl, halogenoalkenyloxycarbonyl or dialkylamino or two radicals R1 when they are positioned ortho to one another together denote a methylenedioxy, ethylenedioxy or alkylene radical, R2 and R3 independently of one another denote alkyl, alkenyl or phenyl, or R2 and R3 denote an alkylene chain which-together with the quaternary carbon atom-forms an unsubstituted or fluorinesubstituted ring having three to six ring members, R4 denotes -H, F, -CN, -CCl3, -C 3BOND CH, (C1-C4)alkyl, -C-NH2, S R5 denotes pyridyl, furyl or thienyl which can all be substituted, phthalimidyl, dialkylmaleimidyl, thiophthalimidyl, dihydrophthalimidyl, tetrahydrophthalimidyl or substituted phenyl, or R4 and R5-together with the carbon atom bridging them-denote an optionally substituted indanyl, cyclopentenoyl or cyclopentenyl radical and n denotes 0, 1 or 2, possess advantageous properties for combating pests, in particular insects and acarids. Furthermore, processes for the preparation of compounds of the formula I are described.

公开(公告)号：PH25134A

公开(公告)日：1991-02-19

申请号：PH34413

申请日：1986-10-24

Applicant: HOECHST AG

Inventor： SCHUBERT HANS HERBERT ,  WALTERSDORFER ANNA ,  SALBECK GERHARD ,  LUDERS WALTER ,  KNAUF WERNER

IPC: A01N20060101 ,  A01N43/40 ,  A01N55/00 ,  A01N55/02 ,  A01N55/10 ,  A01P7/04 ,  A23K20060101 ,  A61K20060101 ,  C07C20060101 ,  C07C7/08 ,  C07C25/13 ,  C07C43/215 ,  C07C43/225 ,  C07D213/64 ,  C07F20060101 ,  C07F7/08 ,  C07F7/10 ,  C07F7/14

Abstract: The compounds of the formula (I) (I) in which X denotes CH2, O, S or NR6, R1 denotes alkyl, cycloalkyl, alkenyl, (substituted) phenyl, or (substituted) naphthyl, R2 and R3 denote alkyl, alkenyl or phenyl, or R2 and R3 together denote an alkylene chain, R4 denotes -H, -CN, -CCl3, -C 3BOND CH, alkyl, F, or -C(S)-NH2, R5 denotes pyridyl, furyl, thienyl, phthalimidyl, di(C1-C4)alkylmaleinimidyl, thiophthalimidyl, dihydrophthalimidyl or tetrahydrophthalimidyl, which may all be substituted, or substituted phenyl, or R4 and R5-together with the carbon atom bridging them-denote an optionally substituted indanyl, cyclopentenoyl or cyclopentenyl radical, with the proviso that compounds of the formula I in which R1 denotes phenyl which is substituted in the para-position by (C1-C4)alkoxy, halogen or (C1-C4)alkyl; R2 and R3 denote CH3; X denotes O; R4 denotes H and R5 denotes 3-phenoxyphenyl or (4-fluoro-3-phenoxy)phenyl being excepted, have advantageous insecticidal, acaricidal and nematocidal properties.

公开(公告)号：ES2016793B3

公开(公告)日：1990-12-01

申请号：ES86114578

申请日：1986-10-21

Applicant: HOECHST AG

Inventor： SCHUBERT HANS HERBERT ,  SALBECK GERHARD ,  LUDERS WALTER ,  KNAUF WERNER ,  WALTERSDORFER ANNA

IPC: A01N20060101 ,  A01N43/40 ,  A01N55/00 ,  A01N55/02 ,  A01N55/10 ,  A01P7/04 ,  A23K20060101 ,  A61K20060101 ,  C07C20060101 ,  C07C7/08 ,  C07C25/13 ,  C07C43/215 ,  C07C43/225 ,  C07D213/64 ,  C07F20060101 ,  C07F7/08 ,  C07F7/10

公开(公告)号：ZA9001846B

公开(公告)日：1990-11-28

申请号：ZA9001846

申请日：1990-03-09

Applicant: HOECHST AG

Inventor： SCHNATTERER STEFAN ,  STEFAN SCHNATTERER ,  KERN MANFRED ,  MANFRED KERN ,  KNAUF WERNER ,  WERNER KNAUF ,  SCHUBERT HANS HERBERT ,  HANS HERBERT SCHUBERT ,  SALBECK GERHARD ,  GERHARD SALBECK ,  WALTERSDORFER ANNA ,  ANNA WALTERSDORFER

IPC: C07D233/64 ,  A01N43/08 ,  A01N43/10 ,  A01N43/40 ,  A01N43/50 ,  A01N43/54 ,  A01N43/56 ,  A01N43/74 ,  A01N43/78 ,  A61K31/425 ,  A61K31/426 ,  A61P33/10 ,  C07D213/26 ,  C07D213/30 ,  C07D213/61 ,  C07D213/64 ,  C07D213/65 ,  C07D239/26 ,  C07D263/32 ,  C07D277/22 ,  C07D277/24 ,  C07D307/40 ,  C07D307/42 ,  C07D333/12 ,  C07D333/16 ,  C07D333/32 ,  C07D401/06 ,  C07D403/06 ,  C07D407/06 ,  C07D407/12 ,  C07D409/06 ,  C07D409/12 ,  C07D413/06 ,  C07D413/12 ,  C07D417/06 ,  C07D417/12 ,  C07D ,  A01N

CPC classification number: C07D213/30 ,  A01N43/08 ,  A01N43/10 ,  A01N43/40 ,  A01N43/50 ,  A01N43/54 ,  A01N43/56 ,  A01N43/74 ,  C07D213/26 ,  C07D213/61 ,  C07D213/64 ,  C07D239/26 ,  C07D277/22 ,  C07D307/42 ,  C07D333/12 ,  C07D333/16 ,  C07D333/32

公开(公告)号：AU5118090A

公开(公告)日：1990-09-13

申请号：AU5118090

申请日：1990-03-09

Applicant: HOECHST AG

Inventor： SCHNATTERER STEFAN ,  SCHUBERT HANS HERBERT ,  SALBECK GERHARD ,  KNAUF WERNER ,  WALTERSDORFER ANNA ,  KERN MANFRED

IPC: C07D233/64 ,  A01N43/08 ,  A01N43/10 ,  A01N43/40 ,  A01N43/50 ,  A01N43/54 ,  A01N43/56 ,  A01N43/74 ,  A01N43/78 ,  A61K31/425 ,  A61K31/426 ,  A61P33/10 ,  C07D213/26 ,  C07D213/30 ,  C07D213/61 ,  C07D213/64 ,  C07D213/643 ,  C07D213/65 ,  C07D239/26 ,  C07D263/32 ,  C07D277/22 ,  C07D277/24 ,  C07D307/12 ,  C07D307/40 ,  C07D307/42 ,  C07D333/12 ,  C07D333/16 ,  C07D333/32 ,  C07D401/06 ,  C07D403/06 ,  C07D407/06 ,  C07D407/12 ,  C07D409/06 ,  C07D409/12 ,  C07D413/06 ,  C07D413/12 ,  C07D417/06 ,  C07D417/12 ,  C07D401/12 ,  C07D405/06 ,  C07D405/12 ,  A01N43/76

Abstract: The compounds of the formulae I and II, their stereoisomers and the mixtures of these in which R represents pyridyl, pyrimidyl, thienyl, thiazolyl, furanyl, pyrazolyl, 1,3-oxazolyl or imidazolyl, each of which can be substituted, R represents H, (C1-C4)alkyl, (C1-C4)haloalkyl, (C1-C4)alkoxy, (C3-C6)cycloalkyl, -CH=CH2 or -C IDENTICAL CH, R represents H or (C1-C4)alkyl, R represents H, (C1-C4)alkyl, -CN or -C IDENTICAL CH, A represents CH2, O or S, B represents CH, N or C(CH3), R represents H or halogen and R represents phenyl, phenoxy or benzyl, each of which can be monosubstituted to pentasubstituted by halogen or (C1-C3)haloalkyl, have advantageous insecticidal or acaricidal properties.

公开(公告)号：AU599932B2

公开(公告)日：1990-08-02

申请号：AU6437686

申请日：1986-10-24

Applicant: HOECHST AG

Inventor： SCHUBERT HANS HERBERT ,  SALBECK GERHARD ,  LUDERS WALTER ,  KNAUF WERNER ,  WALTERSDORFER ANNA

IPC: A01N20060101 ,  A01N43/40 ,  A01N55/00 ,  A01N55/02 ,  A01N55/10 ,  A01P7/04 ,  A23K20060101 ,  A61K20060101 ,  C07C20060101 ,  C07C7/08 ,  C07C25/13 ,  C07C43/215 ,  C07C43/225 ,  C07D213/64 ,  C07F20060101 ,  C07F7/08 ,  C07F7/10

Abstract: The compounds of the formula (I) (I) in which X denotes CH2, O, S or NR6, R1 denotes alkyl, cycloalkyl, alkenyl, (substituted) phenyl, or (substituted) naphthyl, R2 and R3 denote alkyl, alkenyl or phenyl, or R2 and R3 together denote an alkylene chain, R4 denotes -H, -CN, -CCl3, -C 3BOND CH, alkyl, F, or -C(S)-NH2, R5 denotes pyridyl, furyl, thienyl, phthalimidyl, di(C1-C4)alkylmaleinimidyl, thiophthalimidyl, dihydrophthalimidyl or tetrahydrophthalimidyl, which may all be substituted, or substituted phenyl, or R4 and R5-together with the carbon atom bridging them-denote an optionally substituted indanyl, cyclopentenoyl or cyclopentenyl radical, with the proviso that compounds of the formula I in which R1 denotes phenyl which is substituted in the para-position by (C1-C4)alkoxy, halogen or (C1-C4)alkyl; R2 and R3 denote CH3; X denotes O; R4 denotes H and R5 denotes 3-phenoxyphenyl or (4-fluoro-3-phenoxy)phenyl being excepted, have advantageous insecticidal, acaricidal and nematocidal properties.

公开(公告)号：AU4685689A

公开(公告)日：1990-06-28

申请号：AU4685689

申请日：1989-12-19

Applicant: HOECHST AG

Inventor： STARK HERBERT ,  SALBECK GERHARD ,  BONIN WERNER

IPC: A61K31/415 ,  A61P33/00 ,  C07D233/20 ,  C07D233/22 ,  C07D233/24

Abstract: The present invention relates to agents for systemic combating of ectoperasites in host animals, containing a compound of the formul I (I) in which R1 denotes hydrogen, (C1-C5)-alkyl, (C1-C3)-halogenoalkyl or halogen; R2 and R3 independently of one another denote (c1-C5)-alkyl, (C2-C5)-alkenyl, (C2-C5)-alkynyl, (C3-C7)-cycloalkyl, (C3-C7)-cycloalkenyl, (C1-C3)-halogenoalkyl, halogen, cyano, nitro, (C1-C5)-alkoxy, (C1 -C3)-alkoxy-C1-C3)-alkyl, (C1-C3)-halogenoalkoxy or (C1-C3)-alkylthio, or R2 and R3 together form a polymethylene chain having 2 to 5 carbon atoms: R4 denotes hydrogen, (c1-C10)-alkyl, (C2-C5)-alkenyl or (C3-C7)-cycloalkyl; R5 denotes hydrogen, (C1-C10)-alkyl, (C3-C5)-alkenyl, C3-C5)-alkynyl, (C3-C7)- cycloalkyl, (C3-C7)-cycloalkenyl, (C1-C3)-halogenoalkyl or (C1-C3)-alkoxy-(C hd 1-C3)-alkyl; X denotes oxygen, sulfur or an -NR6-group; and R6 denotes hydrogen, (C1-C5)-alkyl, (C3-C5)-alkenyl, C3-C5)-alkynyl, (C3-C7)-cycloalkyl, C3-C7)-cycloalkenyl, (C1-C3)-halogenoalkyl or (C1-C3)-alkoxy-(C1 -C3)-alkyl, or biologically tolerated acid addition salts thereof. The compounds of the formulas I are novel in some cases and are likewise included in the invention.

公开(公告)号：HU901378D0

公开(公告)日：1990-05-28

申请号：HU137890

申请日：1990-03-09

Applicant: HOECHST AG

Inventor： SCHNATTERER STEFAN ,  SCHUBERT HANS HERBERT ,  SALBECK GERHARD ,  KNAUF WERNER ,  WALTERSDORFER ANNA ,  KERN MANFRED

IPC: C07D233/64 ,  A01N43/08 ,  A01N43/10 ,  A01N43/40 ,  A01N43/50 ,  A01N43/54 ,  A01N43/56 ,  A01N43/74 ,  A01N43/78 ,  A61K31/425 ,  A61K31/426 ,  A61P33/10 ,  C07D213/26 ,  C07D213/30 ,  C07D213/61 ,  C07D213/64 ,  C07D213/643 ,  C07D213/65 ,  C07D239/26 ,  C07D263/32 ,  C07D277/22 ,  C07D277/24 ,  C07D307/12 ,  C07D307/40 ,  C07D307/42 ,  C07D333/12 ,  C07D333/16 ,  C07D333/32 ,  C07D401/06 ,  C07D403/06 ,  C07D407/06 ,  C07D407/12 ,  C07D409/06 ,  C07D409/12 ,  C07D413/06 ,  C07D413/12 ,  C07D417/06 ,  C07D417/12

Abstract: The compounds of the formulae I and II, their stereoisomers and the mixtures of these in which R represents pyridyl, pyrimidyl, thienyl, thiazolyl, furanyl, pyrazolyl, 1,3-oxazolyl or imidazolyl, each of which can be substituted, R represents H, (C1-C4)alkyl, (C1-C4)haloalkyl, (C1-C4)alkoxy, (C3-C6)cycloalkyl, -CH=CH2 or -C IDENTICAL CH, R represents H or (C1-C4)alkyl, R represents H, (C1-C4)alkyl, -CN or -C IDENTICAL CH, A represents CH2, O or S, B represents CH, N or C(CH3), R represents H or halogen and R represents phenyl, phenoxy or benzyl, each of which can be monosubstituted to pentasubstituted by halogen or (C1-C3)haloalkyl, have advantageous insecticidal or acaricidal properties.

公开(公告)号：DK648489D0

公开(公告)日：1989-12-19

申请号：DK648489

申请日：1989-12-19

Applicant: HOECHST AG

Inventor： STARK HERBERT ,  SALBECK GERHARD ,  BONIN WERNER

IPC: A61K31/415 ,  A61P33/00 ,  C07D233/20 ,  C07D233/22 ,  C07D233/24 ,  A01N43/50

Abstract: The present invention relates to agents for systemic combating of ectoperasites in host animals, containing a compound of the formul I (I) in which R1 denotes hydrogen, (C1-C5)-alkyl, (C1-C3)-halogenoalkyl or halogen; R2 and R3 independently of one another denote (c1-C5)-alkyl, (C2-C5)-alkenyl, (C2-C5)-alkynyl, (C3-C7)-cycloalkyl, (C3-C7)-cycloalkenyl, (C1-C3)-halogenoalkyl, halogen, cyano, nitro, (C1-C5)-alkoxy, (C1 -C3)-alkoxy-C1-C3)-alkyl, (C1-C3)-halogenoalkoxy or (C1-C3)-alkylthio, or R2 and R3 together form a polymethylene chain having 2 to 5 carbon atoms: R4 denotes hydrogen, (c1-C10)-alkyl, (C2-C5)-alkenyl or (C3-C7)-cycloalkyl; R5 denotes hydrogen, (C1-C10)-alkyl, (C3-C5)-alkenyl, C3-C5)-alkynyl, (C3-C7)- cycloalkyl, (C3-C7)-cycloalkenyl, (C1-C3)-halogenoalkyl or (C1-C3)-alkoxy-(C hd 1-C3)-alkyl; X denotes oxygen, sulfur or an -NR6-group; and R6 denotes hydrogen, (C1-C5)-alkyl, (C3-C5)-alkenyl, C3-C5)-alkynyl, (C3-C7)-cycloalkyl, C3-C7)-cycloalkenyl, (C1-C3)-halogenoalkyl or (C1-C3)-alkoxy-(C1 -C3)-alkyl, or biologically tolerated acid addition salts thereof. The compounds of the formulas I are novel in some cases and are likewise included in the invention.

公开(公告)号：DD273968A5

公开(公告)日：1989-12-06

申请号：DD31470388

申请日：1988-04-13

Applicant: HOECHST AG

Inventor： SCHUBERT HANS H ,  SALBECK GERHARD ,  KRAUSE HANS-PETER ,  LUEDERS WALTER ,  KNAUF WERNER ,  WALTERSDORFER ANNA ,  KERN MANFRED

IPC: C07D253/06 ,  A01N43/40 ,  A01N43/54 ,  A01N43/58 ,  A01N43/60 ,  A01N55/10 ,  A01P7/02 ,  A01P7/04 ,  C07D213/61 ,  C07D213/63 ,  C07D213/64 ,  C07D213/643 ,  C07D213/65 ,  C07D213/70 ,  C07D237/12 ,  C07D237/14 ,  C07D237/18 ,  C07D239/26 ,  C07D239/30 ,  C07D239/34 ,  C07D239/38 ,  C07D241/16 ,  C07D241/18 ,  C07D253/07 ,  C07D253/08 ,  C07D257/08 ,  C07D401/06 ,  C07D401/08 ,  C07D401/12 ,  C07D409/06 ,  C07D409/08 ,  C07D491/04 ,  C07D491/056 ,  A01N43/48 ,  A01N43/64 ,  A01N43/713 ,  A01N39/00 ,  A01N37/34

Abstract: Compounds of the formula (I) and their stereoisomers (I) wherein A, B, C' and D independently of one another denote CH or N, in which at least one of the symbols A, B, C' or D must correspond to a nitrogen atom, X denotes CH2 or oxygen, R1 denotes a radical bonded to a carbon atom from the series comprising H, trialkylsilyl, halogen, nitro, cyano, alkenyl, alkynyl, amino, cycloalkyl, phenyl, phenxy, alkoxy, alkenyloxy, alkynyloxy, hydroxycarbonyl, alkylthio, cycloalkyloxy, alkylcarbonyl, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, halogenoalkyl, alkoxyalkyl, halogenoalkoxy, halogenoalkylthio, halogenoalkoxyalkyl, alkylthioalkyl, alkoxyalkoxy, halogenoalkoxyalkoxy, alkenyloxyalkoxy, halogenoalkenyloxy, alkoxyalkylthio, alkylthioalkoxy, alkylthioalkylthio, halogenoalkoxycarbonyl, halogenoalkenyloxycarbonyl or dialkylamino or two radicals R1 when they are positioned ortho to one another together denote a methylenedioxy, ethylenedioxy or alkylene radical, R2 and R3 independently of one another denote alkyl, alkenyl or phenyl, or R2 and R3 denote an alkylene chain which-together with the quaternary carbon atom-forms an unsubstituted or fluorinesubstituted ring having three to six ring members, R4 denotes -H, F, -CN, -CCl3, -C 3BOND CH, (C1-C4)alkyl, -C-NH2, S R5 denotes pyridyl, furyl or thienyl which can all be substituted, phthalimidyl, dialkylmaleimidyl, thiophthalimidyl, dihydrophthalimidyl, tetrahydrophthalimidyl or substituted phenyl, or R4 and R5-together with the carbon atom bridging them-denote an optionally substituted indanyl, cyclopentenoyl or cyclopentenyl radical and n denotes 0, 1 or 2, possess advantageous properties for combating pests, in particular insects and acarids. Furthermore, processes for the preparation of compounds of the formula I are described.