公开(公告)号：UA125542C2

公开(公告)日：2022-04-13

申请号：UAA202002882

申请日：2018-10-16

Applicant: SYNGENTA PARTICIPATIONS AG

Inventor： SMITS HELMARS ,  GRIBKOV DENIS ,  GODINEAU EDOUARD ,  SCARBOROUGH CHRISTOPHER CHARLES ,  ROBINSON ALAN JAMES ,  DIECKMANN MICHAEL CHRISTIAN

Abstract: Cпосібодержаннясполукиформули (I), де A1, R1, R2, R3, R4, R5 і R6 визначенів даномудокументі; такожу винаходідодатковопередбаченіпроміжнісполуки, застосовуваніу вказаномуспособі, іспособиодержаннявказанихпроміжнихсполук. (I)

公开(公告)号：BR122021004312B1

公开(公告)日：2022-02-08

申请号：BR122021004312

申请日：2015-04-30

Applicant: SYNGENTA PARTICIPATIONS AG

Inventor： LOTHSCHUETZ CHRISTIAN ,  SMITS HELMARS ,  TERINEK MIROSLAV ,  SMEJKAL TOMAS

IPC: C07C259/06 ,  C07D261/04

Abstract: processo para a preparação de ciclosserinas substituídas e seus compostos. a presente invenção refere-se a processos para a preparação de compostos de ciclosserina substituída da fórmula (i) em que r1 é alquila c1-c8, haloalquila c1-c8, cicloalquila c3-c6, arila ou arila substituída com um a cinco r11, ou aril-alquileno(c1-c4) ou aril-alquileno(c1-c4) substituído com um a cinco r11; e cada r11 é independentemente alquila c1-c4, haloalquila c1-c4, alcoxi c1-c4, haloalcoxi c1-c4, ciano ou halogênio. a invenção também se refere a intermediários produzidos pelos processos. os compostos da fórmula (i) são intermediários úteis para a produção de compostos nas áreas agrícola e farmacêutica.

公开(公告)号：HUE050000T2

公开(公告)日：2020-11-30

申请号：HUE15787482

申请日：2015-10-08

Applicant: SYNGENTA PARTICIPATIONS AG

Inventor： SMITS HELMARS ,  KNOCHEL PAUL ,  KLATT THOMAS ,  BECKER MATTHIAS

IPC: C07C17/12 ,  C07C25/13

公开(公告)号：HUE049170T2

公开(公告)日：2020-09-28

申请号：HUE15722685

申请日：2015-04-30

Applicant: SYNGENTA PARTICIPATIONS AG

Inventor： SMEJKAL TOMAS ,  SMITS HELMARS ,  LOTHSCHUETZ CHRISTIAN ,  TERINEK MIROSLAV

IPC: A01N43/80

公开(公告)号：SI3137449T1

公开(公告)日：2020-04-30

申请号：SI201531115

申请日：2015-04-30

Applicant: SYNGENTA PARTICIPATIONS AG

Inventor： SMEJKAL TOMAS ,  SMITS HELMARS ,  LOTHSCHUETZ CHRISTIAN ,  TERINEK MIROSLAV

IPC: C07D261/00 ,  A01N43/00

公开(公告)号：CA3079498A1

公开(公告)日：2019-04-25

申请号：CA3079498

申请日：2018-10-16

Applicant: SYNGENTA PARTICIPATIONS AG

Inventor： SMITS HELMARS ,  GRIBKOV DENIS ,  GODINEAU EDOUARD ,  SCARBOROUGH CHRISTOPHER CHARLES ,  ROBINSON ALAN JAMES ,  DIECKMANN MICHAEL CHRISTIAN

IPC: C07D237/14

Abstract: The present invention provides, inter alia, a process for producing a compound of Formula (I): wherein A1, R1, R2, R3, R4, R5 and R6 are as defined herein. The present invention further provides intermediate compounds utilised in said process, and methods for producing said intermediate compounds.

公开(公告)号：MX2016000551A

公开(公告)日：2016-04-20

申请号：MX2016000551

申请日：2014-07-11

Applicant: SYNGENTA PARTICIPATIONS AG

Inventor： MUEHLEBACH MICHEL ,  SMITS HELMARS ,  MONDIERE REGIS JEAN GEORGES ,  GODINEAU EDOUARD ,  SMEJKAL TOMAS ,  PELLETIER SOPHIE ,  WECKESSER JOCHEN ,  ROBINSON ALAN JAMES

IPC: C07D409/12 ,  A01N43/38 ,  C07D471/10

Abstract: Un proceso para preparar ciertos derivados de pirrolidina-diona espiroheterocíclica.

公开(公告)号：CA2888041A1

公开(公告)日：2014-05-08

申请号：CA2888041

申请日：2013-10-24

Applicant: SYNGENTA PARTICIPATIONS AG

Inventor： HUETER OTTMAR FRANZ ,  JUNG PIERRE JOSEPH MARCEL ,  PITTERNA THOMAS ,  SMITS HELMARS ,  STOLLER ANDRE

IPC: C07C235/64

Abstract: The present invention relates to novel triazole derivatives of formula (I) having insecticidal activity, to processes and intermediates for preparing them, to insecticidal, acaricidal, nematicidal or molluscicidal compositions comprising them and to methods of using them to combat and control insect, acarine, nematode or mollusc pests; wherein R1, R2, G1, G2, Q1 and Q2 are as defined in claim 1; or salts thereof.

公开(公告)号：CL2012003491A1

公开(公告)日：2013-05-24

申请号：CL2012003491

申请日：2012-12-10

Applicant: SYNGENTA PARTICIPATIONS AG ,  SYNGENTA LTD

Inventor： EL QACEMI MYRIEM ,  CASSAYRE JEROME YVES ,  RENOLD PETER ,  PITTERNA THOMAS ,  GODINEAU EDOUARD ,  SMITS HELMARS ,  MULHOLLAND NICHOLAS PHILLIP

IPC: C07D413/12

Abstract: Compuesto derivado de dihidropirrol sustituidos; proceso para preparar dichos derivados.

公开(公告)号：CA2800114A1

公开(公告)日：2011-12-15

申请号：CA2800114

申请日：2011-06-14

Applicant: SYNGENTA PARTICIPATIONS AG ,  SYNGENTA LTD

Inventor： EL QACEMI MYRIEM ,  SMITS HELMARS ,  CASSAYRE JEROME YVES ,  MULHOLLAND NICHOLAS PHILLIP ,  RENOLD PETER ,  GODINEAU EDOUARD ,  PITTERNA THOMAS

IPC: C07D413/12 ,  A01N43/36 ,  A01N43/40 ,  A01N43/80 ,  C07C1/32 ,  C07D207/20 ,  C07D401/04 ,  C07D403/04 ,  C07D409/12 ,  C07D409/14 ,  C07D413/14 ,  C07D417/14

Abstract: The present invention provides stereoselective processes for the preparation of compounds of formula (I) wherein P is phenyl, naphthyl, a 6-membered heteroaryl group containing one or two nitrogen atoms as ring members, or a 10-membered bicyclic heteroaryl group containing one or two nitrogen atoms as ring members, and wherein the phenyl, naphthyl and heteroaryl groups are optionally substituted; R1 is chlorodifluoromethyl or trifluoromethyl; R2 is optionally substituted aryl or optionally substituted heteroaryl; n is 0 or 1; including the process comprising (a-i) reacting a compound of formula II wherein P, R1 and R2 are as defined for the compound of formula I; with nitromethane in the presence a chiral catalyst to give a compound of formula III Wherein P, R1 and R2 are as defined for the compound of formula I; and (a-ii) reductively cyclising the compound of formula III to give the compound of formula I. The invention also provides intermediates useful for processes for the synthesis of compounds of formula (I).