公开(公告)号：WO2005087771A3

公开(公告)日：2005-12-01

申请号：PCT/EP2005002425

申请日：2005-03-08

Applicant: BASF AG ,  TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  NIEDENBRUECK MATTHIAS ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

Inventor： TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  NIEDENBRUECK MATTHIAS ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

IPC: C07D487/04

CPC classification number: C07D487/04

Abstract: The invention relates to 5,6-dialkyl-7-amino-triazolopyrimidines of formula (I), in which the substituents are defined as follows: R represents alkyl or alkoxyalkyl; R represents alkyl, R and/or R being substituted according to the description. The invention also relates to a method for producing said compounds, to agents containing the latter and to their use for controlling plant-pathogenic fungi.

Abstract translation: 式（I）的5,6-二烷基 - 7-氨基 - 三唑并嘧啶，其中取代基具有以下含义：R t <1>是烷基或烷氧基烷基，R <2>是烷基，其中R <1>和/或R <2> 可以如上所述被替换; 这些化合物的制备方法，含有它们的试剂及其用于防治植物病原性有害真菌的用途。

公开(公告)号：WO2005080396A2

公开(公告)日：2005-09-01

申请号：PCT/EP2005001965

申请日：2005-02-24

Applicant: BASF AG ,  SCHWOEGLER ANJA ,  GEWEHR MARKUS ,  MUELLER BERND ,  GROTE THOMAS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  RHEINHEIMER JOACHIM ,  BLETTNER CARSTEN ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  WAGNER OLIVER ,  STIERL REINHARD ,  SCHOEFL ULRICH ,  STRATHMANN SIEGFRIED ,  SCHERER MARIA

Inventor： SCHWOEGLER ANJA ,  GEWEHR MARKUS ,  MUELLER BERND ,  GROTE THOMAS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  RHEINHEIMER JOACHIM ,  BLETTNER CARSTEN ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  WAGNER OLIVER ,  STIERL REINHARD ,  SCHOEFL ULRICH ,  STRATHMANN SIEGFRIED ,  SCHERER MARIA

IPC: A01N43/90 ,  C07D487/04 ,  C07D487/00

CPC classification number: C07D487/04

Abstract: The invention relates to azolopyrimidine compounds of general formula (I), wherein A represents N or C-R ; X and Y, independent of one another, represent a chemical compound or oxygen, sulphur or a group N-R ; the variables R , R , R , R , R , R and R have the meanings cited in the claims and the description. The invention also relates to tautomers of compounds of formula (I) and to the agriculturally compatible salts of compounds (I) and of the tautomers thereof. The invention further relates to the use of azolopyrimidine compounds of general formula (I), to the tautomers thereof and to the agriculturally compatible salts thereof which are used to combat phytopathogenic fungi, and to a method for combating phytopathogenic fungi and means for combating fungi, said means containing at least one compound of general formula (I), a tautomer of formula (I) and/or an agriculturally compatible salt thereof or the tautomer thereof and at least one liquid or solid carrier medium.

Abstract translation: 本发明涉及通式（I）的唑基嘧啶化合物，其中A是N或C-R 6; X，Y彼此独立地代表化学键或氧，硫或基团N-R 7; 其中变量R <1>，R <2>，R <3>，R <4>，R <5> - [R <6>和R <7>具有权利要求书所给出的含义和描述中，互变异构体 式（I）化合物和化合物I及其互变异构体的农业上可接受的盐。 本发明还涉及使用通式（I）的唑并嘧啶化合物，它们的互变异构体以及它们用于防治植物致病真菌（=有害真菌），以及用于防治植物病原性有害真菌的方法和用于防治有害真菌的手段农业上可接受的盐，含 至少一种通式（I）的化合物，（I）的互变异构体和/或其农业上可接受的盐或其互变异构体以及至少一种液体或固体载体。

公开(公告)号：WO2005036960A3

公开(公告)日：2005-07-07

申请号：PCT/EP2004011257

申请日：2004-10-08

Applicant: BASF AG ,  TORMO I BLASCO JORDI ,  GROTE THOMAS ,  SCHERER MARIA ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH

Inventor： TORMO I BLASCO JORDI ,  GROTE THOMAS ,  SCHERER MARIA ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH

IPC: A01N43/90

CPC classification number: A01N43/90 ,  A01N59/02 ,  A01N2300/00

Abstract: The invention relates to fungicidal mixtures for controlling rice pathogens. Said mixtures comprise as the active components 1) the triazolopyrimidine derivative of formula (I), and 2) sulfur (II), in a synergistically effective amount. The invention also relates to a method for controlling rice pathogens using mixtures of compound (I) with sulfur (II) and to the use of compound (I) together with sulfur (II) for producing said mixtures, and to agents containing said mixtures.

Abstract translation: 用于控制水稻病原体，其包含作为活性组分1）式（I）的三唑并嘧啶衍生物，和杀真菌混合物2）硫（II），（协同有效量，用于控制使用I化合物的混合物与硫II稻病原体的方法） 及使用化合物I与硫（II）的用于生产这样的混合物和包含这些混合物的组合物。

公开(公告)号：WO2004006666A2

公开(公告)日：2004-01-22

申请号：PCT/EP0306888

申请日：2003-06-30

Applicant: BASF AG ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  SCHOEFL ULRICH ,  SCHELBERGER KLAUS ,  SCHERER MARIA ,  HENNINGSEN MICHAEL ,  GOLD RANDALL EVEN

Inventor： AMMERMANN EBERHARD ,  STIERL REINHARD ,  SCHOEFL ULRICH ,  SCHELBERGER KLAUS ,  SCHERER MARIA ,  HENNINGSEN MICHAEL ,  GOLD RANDALL EVEN

IPC: A01N25/04 ,  A01N43/32 ,  A01N43/653 ,  A01N

CPC classification number: A01N43/32 ,  A01N43/653 ,  A01N2300/00

Abstract: The invention relates to fungicidal mixtures containing, in a synergistically effective amount: A) the compound of formula (I) and; B) at least one azole derivative II selected from the group consisting of compounds (II-1) to (II-7). The invention also relates to methods for controlling harmful fungi by using mixtures of compounds (I) and (II), and to the use of compounds (I) and (II) for producing mixtures of this type.

Abstract translation: 一种杀真菌混合物，包含：A）通式（I）和B）至少一种唑类衍生物选自化合物（II-1的IIausgewäht）至（II-7）的化合物在协同有效量，方法用于控制使用混合物防治有害真菌的 化合物（I）和（II）以及化合物（I）和（II）在制备这种混合物中的用途。

公开(公告)号：WO03008417A9

公开(公告)日：2003-10-30

申请号：PCT/EP0207578

申请日：2002-07-08

Applicant: BASF AG ,  TORMO I BLASCO JORDI ,  SAUTER HUBERT ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  RACK MICHAEL ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

Inventor： TORMO I BLASCO JORDI ,  SAUTER HUBERT ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  RACK MICHAEL ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N43/90 ,  C07D487/04

CPC classification number: C07D487/04 ,  A01N43/90

Abstract: Substituted 6-(2-tolyl)-triazolopyrimidines of formula (I) in which R and R independently denote hydrogen or alkyl, alkenyl, alkynyl, or alkadienyl, haloalkyl, haloalkenyl, cycloalkyl, phenyl, naphthyl, or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or where R and R radicals may be unsubstituted or substituted as defined in the description, or R and R together with the interjacent nitrogen atom represent a 5- or 6-membered heterocyclic ring, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which may be substituted; R is halogen, cyano, alkyl, alkoxy, haloalkyl, or C(=O)A, wherein A is hydrogen, hydroxy, alkyl, amino, or mono- or dialkyl-amino; n is an integer from 1 to 4; and X is halogen, cyano, alkyl, alkoxy, haloalkoxy or alkenyloxy; processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi.

Abstract translation: 式（I）的取代的6-（2-甲苯基） - 三唑并嘧啶，其中R 1和R 2独立地表示氢或烷基，烯基，炔基或链二烯基，卤代烷基，卤代烯基，环烷基，苯基，萘基或 含有1至4个氮原子或1至3个氮原子和1个硫或氧原子的5-或6-元杂环基，或者含有1-4个氮原子或1-3个氮原子的5-或6-元杂芳基， 硫或氧原子，或者其中R 1和R 2基团可以如说明书中所定义的那样未被取代或被取代，或者R 1和R 2与中间的氮原子一起表示5或6 - 含有1至4个氮原子或1至3个氮原子和1个硫或氧原子的可被取代的 - 元杂环; R 3是卤素，氰基，烷基，烷氧基，卤代烷基或C（= O）A，其中A是氢，羟基，烷基，氨基或单或二烷基氨基; n是1至4的整数; X是卤素，氰基，烷基，烷氧基，卤代烷氧基或烯氧基; 它们的制备方法，含有它们的组合物以及它们用于防治植物病原性真菌的用途。

公开(公告)号：WO02074753A3

公开(公告)日：2002-12-27

申请号：PCT/EP0202739

申请日：2002-03-13

Applicant: BASF AG ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SAUTER HUBERT ,  GEWEHR MARKUS ,  MUELLER BERND ,  TORMO I BLASCO JORDI ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

Inventor： GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SAUTER HUBERT ,  GEWEHR MARKUS ,  MUELLER BERND ,  TORMO I BLASCO JORDI ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N43/54 ,  A01N43/56 ,  A01N43/58 ,  A01N43/60 ,  A01N43/64 ,  A01N43/647 ,  A01N43/653 ,  A01N43/713 ,  A01N43/90 ,  C07D239/42 ,  C07D401/14 ,  C07D403/04 ,  C07D471/04 ,  C07D473/06 ,  C07D487/04 ,  C07D521/00 ,  C07D473/00

CPC classification number: C07D239/42 ,  A01N43/54 ,  A01N43/56 ,  A01N43/60 ,  A01N43/647 ,  A01N43/653 ,  A01N43/713 ,  A01N43/90 ,  C07D231/12 ,  C07D233/56 ,  C07D249/08 ,  C07D403/04 ,  C07D473/06 ,  C07D487/04

Abstract: The invention relates to 5-phenylpyrimidine of formula (I) wherein the substituents have the following designations: R represents a five to ten-membered saturated, partially unsaturated or aromatic monocyclic or bicyclic heterocycle which contains between one and four heteroatoms from the group 0, N or S, and which can be substituted as defined in the description; R represents hydrogen, halogen, cyano, alkyl, halogenalkyl or alkoxy; R and R represent hydrogen, alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, halogenalkenyl, cycloalkenyl, alkinyl, halogenalkinyl or cycloalkinyl; together with the nitrogen atom to which they are bonded, R and R can also form a five or six-membered ring which can be split by a heteroatom and can carry at least one substituent; R and R represent hydrogen, halogen, alkyl, halogenalkyl or alkoxy; R and R represent hydrogen, halogen, alkyl or halogenalkyl; and R represents hydrogen, halogen, alkyl, alkoxy, cycloalkoxy, halogenalkoxy or alkoxycarbonyl. The invention also relates to methods and intermediate products for producing said compounds and the use of the same for controlling pathogenic fungi.

Abstract translation: 式（I）其中取代基具有以下Begende含义的5-苯基嘧啶，R <1> 5〜10元饱和，部分不饱和或芳族单环或双环杂环，选自下组0含有一至四个杂原子，N或 如说明书中所定义的可被取代的S，R <2>为氢，卤素，氰基，烷基，卤代烷基或烷氧基; [R <3>，R <4>是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基，炔基，卤代炔基或环炔基，R <3>和R <4>可与氮原子一起他们 连接，形成可以被杂原子中断并且可以携带一个或多个取代基的五元或六元环; [R <5> - [R <6>是氢，卤素，烷基，卤代烷基或烷氧基; [R <7> - [R <8>是氢，卤素，烷基或卤代烷基; [R <9>是氢，卤素，烷基，烷氧基，环烷氧基，卤代烷氧基或烷氧基羰，卤代烷氧基或烷氧羰，涉及用于制备这些化合物和它们在防治有害真菌中的用途的方法和中间体。

公开(公告)号：WO02056685A2

公开(公告)日：2002-07-25

申请号：PCT/EP0200412

申请日：2002-01-17

Applicant: BASF AG ,  GROTE THOMAS ,  ROSE INGO ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  SCHERER MARIA ,  SCHELBERGER KLAUS ,  HADEN EGON

Inventor： GROTE THOMAS ,  ROSE INGO ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  SCHERER MARIA ,  SCHELBERGER KLAUS ,  HADEN EGON

IPC: A01N25/04 ,  A01N35/04 ,  A01N35/10 ,  A01N37/50 ,  A01N35/00

CPC classification number: A01N35/04 ,  A01N37/50 ,  A01N2300/00

Abstract: The invention relates to fungicidal mixtures containing a) benzophenones of formula (I), where R = chloro, methyl, methoxy, acetoxy, pivaloyloxy or hydroxy; R = chloro or methyl; R = H, halogen or methyl and R = C1-C6 alkyl or benzyl, where the phenyl moiety of the benzyl group may be halo- or methyl-substituted and b) trisoximethers of formula (II), where X = NH or O; R , R , independently = C1-C4 alkyl or cyclopropyl; R , R , independently = C1-C4 alkyl, C3-C4 alkenyl or cyclopropyl; in synergistically effective amounts. The invention further relates to the treatment of noxious fungi with mixtures of compounds (I) and (II) and agents containing the same.

Abstract translation: 含有式（I）中R <1>表示氯，甲基，甲氧基，乙酰氧基，新戊酰氧基或羟基的二苯甲酮类A9的杀真菌混合物; [R <2>是氯或甲基; [R <3>为氢，卤素或甲基; 且R <4>是氢，卤素或甲基; 并代表C1-C6烷基或苄基，其中基团，苄基的苯基部分可以带有卤素或甲基取代基，和b）式Trisoximether（II）其中取代基具有以下含义：X是NH或氧; [R <5>，R <7>独立地是C1-C4烷基或环丙基; [R <6>，R <8>独立地是C1-C4烷基，C3-C4链烯基或环丙基; 包含协同有效量的组合物，用于控制使用（I）和（II）的化合物的混合物和有害真菌的方法。

公开(公告)号：WO0248146A2

公开(公告)日：2002-06-20

申请号：PCT/EP0114577

申请日：2001-12-12

Applicant: BASF AG ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  MUELLER BERND ,  SAUTER HUBERT ,  GYPSER ANDREAS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHIEWECK FRANK ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

Inventor： CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  MUELLER BERND ,  SAUTER HUBERT ,  GYPSER ANDREAS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHIEWECK FRANK ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N43/90 ,  C07D471/04 ,  C07D487/04

CPC classification number: C07D471/04 ,  A01N43/90 ,  C07D487/04

Abstract: The invention relates to the use of substituted imidazoazines of formula (I), in which the variables have the following meanings: R represents alkyl, phenyl, phenylalkyl, naphthyl, anthracenyl, cycloalkyl, 5-membered or 6-membered hetaryl or 5-membered or 6-membered heterocyclyl, containing one to three N atoms and/or one O atom or S atom or one or two O atoms and/or S atoms, or condensed 8-membered to 12-membered hetaryl or condensed 8-membered to 12-membered heterocyclyl, containing one to four N atoms and/or one O atom or S atom or one or two O atoms and/or S atoms, whereby R can be unsubstituted or can be substituted as cited in the description; R and R represent hydrogen, alkyl, alkenyl, alkynyl, alkyl halide, alkenyl halide, alkynyl halide, trialkyl silylalkyl, phenyl, phenylalkyl or R and R , together with the bridging N atom, form a 5-membered or 6-membered heterocyclic or heteroaromatic ring, which can be interrupted by one to three N atoms and/or one O atom or S atom or by one or two O atoms and/or S atoms, and which can be substituted; A and B represent N or CR ; R , R and R represent hydrogen, halogen, cyano, nitro, hydroxy, alkyl, alkyl halide, cycloalkyl, alkoxy, alkoxy halide, alkylthio, amino, alkyl amino, dialkylamino, alkenyl, alkenyloxy, alkynyl or alkynyloxy. The inventive compounds are used for controlling phytopathogenic harmful fungi. The invention further relates to agents containing the inventive compounds, to novel imidazoazines, and to methods for the production thereof.

Abstract translation: 使用式（I）的取代的Imidazoazinen的，其中各变量具有以下含义：R t <1>是烷基，苯基，苯基烷基，萘基，蒽基，环烷基，5-或6-员杂芳基或5-或6-元杂环基 含有1至3个N原子和/或一个O或S原子或一个或两个O和/或S原子，或稠合8-12 gliederiges杂芳基或稠合的8-12 gliederiges杂环基， 含有一至四个N原子和/或一个O或S原子或一个或两个O和/或O原子，其中R是未取代的<1>或作为可在本说明书中被取代; [R <2>，R <3>是氢，烷基，烯基，炔基，卤代烷基，卤代烯基，卤代炔基，三烷基甲硅烷基，苯基，苯基烷基或R <2>，R <3>连同桥接氮原子的5-或6- 形成 - 元杂环基或可被一至三个N原子和/或一个O或S原子或一个或两个O和/或S原子被中断杂芳族环; A，B，N或CR <4>; [R <4>，R <5> - [R <6>为氢，卤素，氰基，硝基，羟基，烷基，卤代烷基，环烷基，烷氧基，卤代烷氧基，烷硫基，氨基，烷基氨基，二烷基氨基，烯基，烯氧基，炔氧基或炔氧基; 防治植物病原性有害真菌的，含有它们，它们的制备新imidazoazines和方法的组合物。

公开(公告)号：WO0167867A3

公开(公告)日：2002-03-14

申请号：PCT/EP0102957

申请日：2001-03-15

Applicant: BASF AG ,  JABS THORSTEN ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  LORENZ GISELA ,  BOLAND WILHELM ,  ENGELBERTH JUERGEN

Inventor： JABS THORSTEN ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  LORENZ GISELA ,  BOLAND WILHELM ,  ENGELBERTH JUERGEN

IPC: A01N37/46 ,  A01N63/04

CPC classification number: A01N37/46 ,  A01N63/04

Abstract: The invention relates to ion channel forming peptaibols from fungi which represent a novel class of highly effective elicitors of the secondary metabolism of plants, the coiling of touch-sensitive tendrils and the induced resistance to harmful fungi, bacteria, viruses, nematodes and insects.

Abstract translation: 离子通道形成从真菌peptaibols代表一类新的植物次生代谢的高度有效的诱导子，卷取触摸敏感卷须和有害真菌，细菌，病毒，线虫和昆虫的感应电阻。

公开(公告)号：CA2812887C

公开(公告)日：2016-02-23

申请号：CA2812887

申请日：2003-02-26

Applicant: BASF AG

Inventor： AMMERMANN EBERHARD ,  STIERL REINHARD ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  SCHELBERGER KLAUS ,  SPADAFORA V JAMES ,  CHRISTEN THOMAS

IPC: A01N43/653 ,  A01N25/04 ,  A01N37/06 ,  A01N37/18 ,  A01N37/50 ,  A01N43/40 ,  A01N47/24 ,  A01P3/00

Abstract: Disclosed is a fungicidal mixture containing (1) 2-[2-(1-chlorocyclopropyl)-3-(2-chlorophenyl)-2-hydroxypropyl]-2,4-dihydro-[1,2,4]-triazole-3-thion of formula (l) or the salts or adducts thereof, and an additional fungicidal compound or the salts or adducts thereof, which is pyraclostrobin, in a synergistically active quantity.