公开(公告)号：WO2007128480A3

公开(公告)日：2007-11-15

申请号：PCT/EP2007/003875

申请日：2007-05-02

Applicant: MAX-PLANCK-GESELLSCHAFT ZUR FÖRDERUNG DER WISSENSCHAFTEN E.V. ,  CASTANEDA, Francisco ,  KINNE, Rolf, K.-H. ,  BOLAND, Wilhelm ,  BURSE, Antje

Inventor： CASTANEDA, Francisco ,  KINNE, Rolf, K.-H. ,  BOLAND, Wilhelm ,  BURSE, Antje

IPC: C07H15/14 ,  C07H15/203 ,  A61K31/7028 ,  A61P3/10

Abstract: The present invention relates to thioglycosides and stereoisomeric forms, solvates, hydrates and/or pharmaceutically acceptable salts of these compounds, as well as pharmaceutical compositions containing at least one of these thioglycosides together with pharmaceutically acceptable carrier, excipient and/or diluents. Said thioglycosides have been identified as specific inhibitors of the sodium dependent glucose transporter 1 (SGLT1) and 2 (SGLT2), and are useful for the prophylaxis and/or treatment of hyperglycemia and hyperglycemia related diseases and conditions.

公开(公告)号：WO2007003346A3

公开(公告)日：2007-01-11

申请号：PCT/EP2006/006330

申请日：2006-06-29

Applicant: MAX-PLANCK-GESELLSCHAFT ZUR FÖRDERUNG DER WISSENSCHAFTEN E.V. ,  MENDGEN, Kurt ,  JUX, Andreas ,  WIRSEL, Stefan, G., R. ,  HOFFMANN, Jochen ,  BOLAND, Wilhelm ,  GIELE, Christine ,  VAHLENKAMP, Heinz ,  PIEL, Jörn

Inventor： MENDGEN, Kurt ,  JUX, Andreas ,  WIRSEL, Stefan, G., R. ,  HOFFMANN, Jochen ,  BOLAND, Wilhelm ,  GIELE, Christine ,  VAHLENKAMP, Heinz ,  PIEL, Jörn

IPC: A01N49/00 ,  A01H5/00 ,  C12N15/82 ,  A01P3/00

Abstract: The strongly negative effect of farnesol and its derivatives on the development of rust fungi is used to provide effective plant protection against pathogenic rust fungi.

公开(公告)号：WO2007003346A2

公开(公告)日：2007-01-11

申请号：PCT/EP2006006330

申请日：2006-06-29

Applicant: MAX PLANCK GESELLSCHAFT ,  MENDGEN KURT ,  JUX ANDREAS ,  WIRSEL STEFAN G R ,  HOFFMANN JOCHEN ,  BOLAND WILHELM ,  GIELE CHRISTINE ,  VAHLENKAMP HEINZ ,  PIEL JOERN

Inventor： MENDGEN KURT ,  JUX ANDREAS ,  WIRSEL STEFAN G R ,  HOFFMANN JOCHEN ,  BOLAND WILHELM ,  GIELE CHRISTINE ,  VAHLENKAMP HEINZ ,  PIEL JOERN

IPC: A01N49/00 ,  A01H5/00 ,  A01P3/00

CPC classification number: A01N49/00 ,  C12N15/8282

Abstract: The strongly negative effect of farnesol and its derivatives on the development of rust fungi is used to provide effective plant protection against pathogenic rust fungi.

Abstract translation: 法尼醇及其衍生物对锈菌发育的强烈负面影响被用于提供有效的植物保护以防止致病性锈菌。

公开(公告)号：WO0167867A3

公开(公告)日：2002-03-14

申请号：PCT/EP0102957

申请日：2001-03-15

Applicant: BASF AG ,  JABS THORSTEN ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  LORENZ GISELA ,  BOLAND WILHELM ,  ENGELBERTH JUERGEN

Inventor： JABS THORSTEN ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  LORENZ GISELA ,  BOLAND WILHELM ,  ENGELBERTH JUERGEN

IPC: A01N37/46 ,  A01N63/04

CPC classification number: A01N37/46 ,  A01N63/04

Abstract: The invention relates to ion channel forming peptaibols from fungi which represent a novel class of highly effective elicitors of the secondary metabolism of plants, the coiling of touch-sensitive tendrils and the induced resistance to harmful fungi, bacteria, viruses, nematodes and insects.

Abstract translation: 离子通道形成从真菌peptaibols代表一类新的植物次生代谢的高度有效的诱导子，卷取触摸敏感卷须和有害真菌，细菌，病毒，线虫和昆虫的感应电阻。

公开(公告)号：WO2002055480A3

公开(公告)日：2002-07-18

申请号：PCT/EP2002/000405

申请日：2002-01-16

Applicant: MAX-PLANCK-GESELLSCHAFT ZUR FÖRDERUNG DER WISSENSCHAFTEN E.V. ,  SCHÜLER, Göde ,  BOLAND, Wilhelm ,  LAUCHLI, Ryan

Inventor： SCHÜLER, Göde ,  BOLAND, Wilhelm ,  LAUCHLI, Ryan

IPC: C07C229/02

Abstract: Described are 6-substituted indanoyl amino acid conjugates of the chemical Formula (I) wherein R 1 = (II), R 2 R 5 have the meanings given in the description, and X = a halogen atom; as potent plant elicitors and efficient mimics of the phytotoxin coronatine. Also, processes for producing the improved elicitors are provided, which allow a rapid and convenient access to large quantities of the highly active compounds. Furthermore, there are compositions and plant protecting agents described, comprising as active ingredient a compound of the present invention. The plant protecting agents are useful for inducing resistance to pathogens in plants. The compositions may also be used to selectively induce senescence in fruit of plants.

公开(公告)号：WO2007128480A2

公开(公告)日：2007-11-15

申请号：PCT/EP2007003875

申请日：2007-05-02

Applicant: MAX PLANCK GESELLSCHAFT ,  CASTANEDA FRANCISCO ,  KINNE ROLF K-H ,  BOLAND WILHELM ,  BURSE ANTJE

Inventor： CASTANEDA FRANCISCO ,  KINNE ROLF K-H ,  BOLAND WILHELM ,  BURSE ANTJE

IPC: C07H15/14 ,  A61K31/7028 ,  A61P3/10 ,  C07H15/203

CPC classification number: C07H15/203 ,  C07H15/14

Abstract: The present invention relates to thioglycosides and stereoisomeric forms, solvates, hydrates and/or pharmaceutically acceptable salts of these compounds, as well as pharmaceutical compositions containing at least one of these thioglycosides together with pharmaceutically acceptable carrier, excipient and/or diluents. Said thioglycosides have been identified as specific inhibitors of the sodium dependent glucose transporter 1 (SGLT1) and 2 (SGLT2), and are useful for the prophylaxis and/or treatment of hyperglycemia and hyperglycemia related diseases and conditions.

Abstract translation: 本发明涉及这些化合物的硫代糖苷类和立体异构形式，溶剂合物，水合物和/或药学上可接受的盐，以及含有这些硫代糖苷类中的至少一种以及药学上可接受的载体，赋形剂和/或稀释剂的药物组合物。 所述硫代糖苷被鉴定为钠依赖性葡萄糖转运蛋白1（SGLT1）和2（SGLT2）的特异性抑制剂，可用于预防和/或治疗高血糖症和高血糖相关疾病和病症。

公开(公告)号：WO02055480A2

公开(公告)日：2002-07-18

申请号：PCT/EP0200405

申请日：2002-01-16

Applicant: MAX PLANCK GESELLSCHAFT ,  SCHUELER GOEDE ,  BOLAND WILHELM ,  LAUCHLI RYAN

Inventor： SCHUELER GOEDE ,  BOLAND WILHELM ,  LAUCHLI RYAN

IPC: A01N37/46 ,  C07B61/00 ,  C07C51/377 ,  C07C63/14 ,  C07C67/11 ,  C07C69/94 ,  C07C229/02 ,  C07C231/02 ,  C07C235/84

CPC classification number: C07C235/84 ,  A01N37/46 ,  C07C2602/08

Abstract: Described are 6-substituted indanoyl amino acid conjugates as defined in claim 1 of the present invention as potent plant elicitors and efficient mimics of the phytotoxin coronatine. Also, processes for producing the improved elicitors are provided, which allow a rapid and convenient access to large quantities of the highly active compounds. Furthermore, there are compositions and plant protecting agents described, comprising as active ingredient a compound of the present invention. The plant protecting agents are useful for inducing resistance to pathogens in plants. The compositions may also be used to selectively induce senescence in fruit of plants.

Abstract translation: 描述的是本发明权利要求1定义的6-取代的吲哚基氨基酸缀合物作为有效的植物诱导剂和植物毒素冠状病毒的有效模拟物。 此外，提供了用于生产改进的诱导剂的方法，其允许快速且方便地接近大量的高活性化合物。 此外，存在所述的组合物和植物保护剂，其包含本发明化合物作为活性成分。 植物保护剂可用于诱导植物中对病原体的抗性。 组合物还可用于选择性诱导植物果实中的衰老。