公开(公告)号：US6410486B2

公开(公告)日：2002-06-25

申请号：US86752401

申请日：2001-05-31

Applicant: BASF AG

Inventor： WETTERICH FRANK ,  EICKEN KARL ,  LORENZ GISELA ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  ROSE INGO

IPC: A01N37/34 ,  C07C255/31 ,  C07C255/58 ,  C07C255/00

CPC classification number: C07C255/58 ,  A01N37/34 ,  C07C255/31 ,  C07C2601/02 ,  C07C2601/08

Abstract: The present invention relates to novel cycloalkylalkane-carboxamides of the formula Iwhere the substituents have the following meanings:A is C3-C6-cycloalkyl;R1 is C1-C6-alkyl or C2-C6-alkenyl;R2, R3 and R4 are hydrogen or, independently of this meaning, have one of the meanings of the radical R1;n is 0 or 1;Y is cyano or halogen;w is phenyl, naphthyl or heteroaryl.

Abstract translation: 本发明涉及式I的新的环烷基烷烃 - 甲酰胺，其中取代基具有以下含义：A为C 3 -C 6 - 环烷基; R 1为C 1 -C 6 - 烷基或C 2 -C 6 - 烯基; R 2，R 3和R 4为氢或 独立于该含义，具有基团R 1的含义之一; n为0或1; Y为氰基或卤素; w为苯基，萘基或杂芳基。

公开(公告)号：JP2002220307A

公开(公告)日：2002-08-09

申请号：JP2001380603

申请日：2001-12-13

Applicant: BASF AG

Inventor： EICKEN KARL ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  SCHERER MARIA ,  SCHELBERGER KLAUS ,  HAMPEL MANFRED

IPC: A01N43/30 ,  A01N43/40

Abstract: PROBLEM TO BE SOLVED: To provide a mixture (a synergistic mixture), in which reduction of the total amount of active compounds included and an improvement of their fugicidal activities are achieved, in order to reduce the proportion of known compounds I and II included within the mixture and to improve their spectra of activity. SOLUTION: The fungicidal mixture contains an amide compound represented by formula I and an amino compound represented by formula II in synergistically effective amounts [wherein, R1 and R2 are halogen, nitro, cyano, alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, haloalkynyl, alkoxy, haloalkoxy, haloalkylthio, alkyl sulfynyl, or alkyl sulfonyl; x is an integer of 1-4; and y is an integer of 1-5.].

公开(公告)号：JP2002047262A

公开(公告)日：2002-02-12

申请号：JP2001207021

申请日：2001-07-06

Applicant: BASF AG

Inventor： GYPSER ANDREAS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  MUELLER BERND ,  SAUTER HUBERT ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: C07C251/80 ,  A01N33/26 ,  A01N37/50 ,  C07C249/16 ,  C07C251/86

Abstract: PROBLEM TO BE SOLVED: To provide a compound that has increased controlling effect against harmful fungi. SOLUTION: The objective salicylic acid derivative is represented by formula I [wherein X is a halogen, NO2, cyano, an alkyl or an alkoxy; (m) is 0, 1, 2 or 3 where in the case m >=2, X may differ from each other; A is OH, an alkoxy, NH2, NHCH3 or N(CH3)2, R1 is phenyl, naphthyl, cycloalkyl, one to three N-atoms and/or one O or S atom or one or two O and/or S atoms- including 5-membered or 5-membered ring heteroaryl or 5-membered or 6-membered heterocyclyl where the ring structure may be unsubstituted or substituted; and R2 is H, cyano, an alkyl, an alkenyl, an alkynyl, a haloalkyl, an alkoxy or an alkylthio]. This invention further provides a method of producing the derivative, a composition including the derivative and the use of the composition for controlling harmful fungi.

公开(公告)号：JP2003206252A

公开(公告)日：2003-07-22

申请号：JP2002313232

申请日：2002-10-28

Applicant: BASF AG

Inventor： ROSE INGO ,  BLASCO JORDI TORMO I ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  GROTE THOMAS ,  GYPSER ANDREAS ,  AMMERMANN EBERHARD ,  LORENZ GISELA ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED ,  CARTER PAUL ,  CURTZE JUERGEN

IPC: A01N31/14 ,  A01N31/16 ,  A01N33/10 ,  A01N37/38 ,  A01N37/40 ,  C07B61/00 ,  C07C39/42 ,  C07C41/26 ,  C07C43/23 ,  C07C69/017 ,  C07C69/14 ,  C07C323/19 ,  C07C323/25

Abstract: PROBLEM TO BE SOLVED: To provide a benzhydryl derivative that exhibits high effect in the control of deleterious fungi. SOLUTION: The benzhydryl derivative is represented by formula I (wherein X is O or S; R 1 , R 3 are each a halogen, cyano, nitro, hydroxyl, mercapto, an amino, an alkyl, an alkenyl, an alkynyl, an alkoxy, an alkenyloxy, an alkynyloxy, an alkyklcarbonyloxy, formyloxy or alkylthio or the like; R 2 is a halogen, cyano, nitro, hydroxyl, mercapto, an amino, an alkyl, an alkoxy, a haloalkyl, or a haloalkoxy wherein in the case that n=2, R 2 may differ from each other; R 4 is an alkyl, an alkenyl or an alkynyl; R 5 and R 6 are each hydroxyl, an alkyl, an alkenyl, a haloalkyl, a haloalkenyl, an alkoxy or an alkenyloxy; m is 0, 1 or 2). COPYRIGHT: (C)2003,JPO

公开(公告)号：JP2002193708A

公开(公告)日：2002-07-10

申请号：JP2001379292

申请日：2001-12-12

Applicant: BASF AG

Inventor： EICKEN KARL ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  SCHERER MARIA ,  SCHELBERGER KLAUS ,  HAMPEL MANFRED

IPC: A01N37/06 ,  A01N43/40

Abstract: PROBLEM TO BE SOLVED: To provide a mixture (synergistic action mixture) which intends the reduction in the application rates of known compounds I and II and the improvement in activity spectrum and achieves the reduction in the total amount of the applied active compounds and the improvement in activities to harmful fungi. SOLUTION: This fungicidal mixture contains an amide compound of formula I (R1 and R2 are each a halogen, nitro, cyano, an alkyl, an alkenyl, an alkynyl, a haloalkyl, a haloalkenyl, a haloalkynyl, an alkoxy, a haloalkoxy, a haloalkylthio, an alkylsulfinyl or an alkylsulfonyl; (x) is an integer of 1 to 4; (y) is an integer of 1 to 5) and dinitrophenol derivatives of formulas II.a and II.b [(n) is an integer of 0 to 2] in synergistic effective amounts.

公开(公告)号：JPH11335361A

公开(公告)日：1999-12-07

申请号：JP2568099

申请日：1999-02-03

Applicant: BASF AG

Inventor： GYPSER ANDREAS ,  SAUTER HUBERT ,  BAYER HERBERT ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GOETZ ROLAND ,  MUELLER BERND ,  PTOCK ARNE ,  ROEHL FRANZ ,  HARRIES VOLKER ,  AMMERMANN EBERHARD ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED

IPC: A01N43/653 ,  A01N43/76 ,  C07C271/10 ,  C07D249/12 ,  C07D263/44 ,  C07D403/12 ,  C07D413/12

Abstract: PROBLEM TO BE SOLVED: To obtain the subject new compound useful for controlling harmful animals and harmful fungi. SOLUTION: This compound is shown by formula I Y is a halogen, a 1-4C alkyl or the like; (n) is 0-2; E is a group of formula II (V is O or the like); T is O or oxymethylene; Z is a group X [X is a (substituted) heterocyclyl, a (substituted) aryl or the like], N=CWR [W is a (substituted) 1-6C alkyl or the like; R is H, cyano or the like] or the like} such as N-methyl-5-[2-(o-tolyloxymethylene)phenyl]-1,3- oxazolidine-2,4-dione.The compound of formula I, for example, in the case in which it is a compound of formula III, is obtained by a process for acylating an alkyl α- hydroxy-α-phenylacetate with phosgene or the like to give a compound of formula IV and further reacting the compound with a primary amine of the formula H2 N-R αto cause a ring formation and in the case of not advancing the ring formation by the strength of the amine, by a process for hydrolyzing an ester amide of formula V, then treating the resultant substance with an acid and reacting the treated substance with a compound of the formula Z-OH.

公开(公告)号：JP2003201289A

公开(公告)日：2003-07-18

申请号：JP2002272397

申请日：2002-09-19

Applicant: BASF AG

Inventor： ROSE INGO ,  BLASCO JORDI TORMO I ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  GROTE THOMAS ,  GYPSER ANDREAS ,  AMMERMANN EBERHARD ,  LORENZ GISELA ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED

IPC: A01N43/16 ,  C07C45/46 ,  C07C45/54 ,  C07C49/84 ,  C07D311/86

Abstract: PROBLEM TO BE SOLVED: To provide a compound effective for controlling hazardous phytopathogenic fungi, to provide a method for producing the compound, to provide a composition containing the compound, and to provide a method for using the composition. SOLUTION: This compound comprises a xanthone derivative expressed by general formula (I) (n is 0, 1 or 2; R 1 is an alkyl or the like; R 2 and R 3 are each an alkoxy or the like, or together form an oxyalkyleneoxy which may be substituted; R 4 is a halogen or the like; R 5 is equal to the R 4 , provided that R 5 s may be different from each other when n is 2; and X and Y are each O or S). The method for producing the compound and the composition containing the compound are provided in the specification, respectively. The composition is used for controlling the hazardous phytopathogenic fungi. COPYRIGHT: (C)2003,JPO

公开(公告)号：JP2002030058A

公开(公告)日：2002-01-29

申请号：JP2001182539

申请日：2001-06-15

Applicant: BASF AG

Inventor： GYPSER ANDREAS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  MUELLER BERND ,  SAUTER HUBERT ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N37/28 ,  A01N37/34 ,  A01N37/40 ,  A01N37/46 ,  A01N47/20 ,  A01N47/30 ,  C07B61/00 ,  C07C249/16 ,  C07C251/86 ,  C07C253/30 ,  C07C255/59 ,  C07C255/64 ,  C07C255/66 ,  C07C269/04 ,  C07C271/28 ,  C07C273/18 ,  C07C275/42

Abstract: PROBLEM TO BE SOLVED: To provide a compound improved in controlling actions on noxious fungi. SOLUTION: This salicylohydrazide derivative is represented by the formula I (wherein, X is a halogen, NO2, cyano, a 1-4C alkyl or a 1-4C alkoxy; (m) is 0, 1, 2 or 3; R1 is NO2, NH2 or NH-CO-A; A is hydrogen, 1-4C alkyl, a 1-4C alkoxy, NH2, NHCH3 or N(CH3)2; R2 is hydrogen, cyano, a 1-6C alkyl, a 2-6C alkeiyl, a 2-6C alkynyl, a 1-6C haloalkyl, a 1-6C alkoxy or a 1-6C alkylthio; and R3 is phenyl, naphthyl, a 3-10C cycloalkyl, a 5- or a 6-membered ring heteroaryl or a 5- or a 6-membered ring heterocyclyl). The method for producing the salicylohydrazide derivative is provided and an intermediate for producing the derivative is obtained. The composition for controlling the noxious fungi comprises the derivative.

公开(公告)号：WO2005018328A8

公开(公告)日：2006-03-09

申请号：PCT/EP2004007397

申请日：2004-07-07

Applicant: BASF AG ,  TORMO I BLASCO JORDI ,  GROTE THOMAS ,  SCHERER MARIA ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH

Inventor： TORMO I BLASCO JORDI ,  GROTE THOMAS ,  SCHERER MARIA ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH

IPC: A01N43/90 ,  A01N43

CPC classification number: A01N43/90 ,  A01N2300/00

Abstract: Disclosed are fungicidal mixtures containing 1) a triazolopyrimidine derivative of formula (I) and 2) epoxiconazole of formula (II) as active components at a synergistically effective quantity, a method for controlling harmful fungi of the class

Abstract translation: 一种杀真菌混合物，其包含作为活性组分1）式（I）的三唑并嘧啶衍生物，以及2）在协同有效量的式（II）的氟环唑，对于从类<我的防治有害真菌的方法

公开(公告)号：WO2005087770A3

公开(公告)日：2005-12-08

申请号：PCT/EP2005002424

申请日：2005-03-08

Applicant: BASF AG ,  TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  NIEDENBRUECK MATTHIAS ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD ,  HUENGER UDO

Inventor： TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  NIEDENBRUECK MATTHIAS ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD ,  HUENGER UDO

IPC: C07D487/04

CPC classification number: C07D487/04

Abstract: The invention relates to 5,6-dialkyl-7-amino-triazolopyrimidines of formula (I), in which the substituents are defined as follows: R represents alkyl, alkoxyalkyl, alkenyl or alkynyl; R represents alkyl, alkoxyalkyl, alkenyl or alkynyl, R and/or R being substituted according to the description. The invention also relates to a method for producing said compounds, to agents containing the latter and to their use for controlling plant-pathogenic fungi.

Abstract translation: 5,6-二烷基 - 7-氨基三唑并嘧啶，其中取代基具有式（I）的以下含义：R t <1>是烷基，烷氧基烷基，烯基或炔基; [R <2>是烷基，烷氧基烷基，烯基或炔基; 其中R <1>和/或R <2>取代根据描述; 一种用于制备这些化合物，含有它们和它们在防治植物病原性有害真菌的用途的组合物的过程。