PYRROLIN-2-YLAMINO COMPOUNDS FOR COMBATING ANIMAL PESTS
    52.
    发明申请
    PYRROLIN-2-YLAMINO COMPOUNDS FOR COMBATING ANIMAL PESTS 审中-公开
    用于组合动物饲料的吡咯啉-2-基亚氨基化合物

    公开(公告)号:WO2010029069A1

    公开(公告)日:2010-03-18

    申请号:PCT/EP2009/061624

    申请日:2009-09-08

    CPC classification number: C07D207/22 C07D209/54

    Abstract: The present invention relates to pyrrolin-2-ylamino compounds for combating animal pests. The invention also relates to a method for controlling animal pests by using these compounds, to plant propagation material and to an agricultural composition comprising said compounds. The invention also relates to a method for treating or protecting an animal from infestation or infection by parasites by using said compounds. Formula (I) wherein n is 0, 1, 2, 3, 4 or 5; m is 0, 1, 2, 3, 4 or 5; R 1 , R 2 are each independently selected from the group consisting of: halogen, CN, N 3 , NO 2 , C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl and C 2 -C 6 -alkynyl, where the last 3 radicals mentioned may be partly or completely halogenated and/or may carry any combination of 1, 2 or 3 radicals R # , etc.; R 3 and R 4 are selected each independently of one another from hydrogen, halogen, C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, wherein the last 3 radicals mentioned may be partly or completely halogenated and/or may carry any combination of 1, 2 or 3 radicals selected independently of one another from the group consisting of CN, NO 2 , -OR b , NR c R d , -SR e , -C(=O)R a and -C(=O)OR b , etc.; A is a radical of the formulae A.1 or A.2, wherein * indicates the point of attachment to the remaining part of the compound; R 5a , R 5b , R 5c , R 5d , R 5e and R 5f are selected independently from one another from hydrogen, halogen, C 1 -C 6 -alkyl, C 1 -C 6 -alkoxy, C 1 -C 6 -alkylamino, di(C 1 -C 6 -alkyl)amino, C 3 -C 6 - cycloalkyl and Ar 2 , etc.; R 6 and R 7 are selected each independently from one another from hydrogen, CN, NO 2 , C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 3 -C 8 -cycloalkyl, saturated or partially unsaturated 5-, 6- or 7-membered heterocyclic radicals, Ar 3 , etc.

    Abstract translation: 本发明涉及用于对抗动物害虫的吡咯啉-2-基氨基化合物。 本发明还涉及通过使用这些化合物,植物繁殖材料和包含所述化合物的农业组合物来控制动物害虫的方法。 本发明还涉及通过使用所述化合物治疗或保护动物免受寄生虫感染或感染的方法。 式(I)其中n为0,1,2,3,4或5; m为0,1,2,3,4或5; R 1,R 2各自独立地选自:卤素,CN,N 3,NO 2,C 1 -C 6 - 烷基,C 2 -C 6 - 烯基和C 2 -C 6 - 炔基,其中所述的最后3个基团可以部分或完全 卤化和/或可以携带1,2或3个基团R#等的任何组合; R 3和R 4彼此独立地选自氢,卤素,C 1 -C 6 - 烷基,C 2 -C 6 - 烯基,C 2 -C 6 - 炔基,其中所述的最后3个基团可以部分或完全卤化和/或可以携带 由CN,NO2,-ORb,NRcRd,-SRe,-C(= O)Ra和-C(= O)ORb等组成的组彼此独立地选择的1,2或3个基团的任意组合; A是式A.1或A.2的基团,其中*表示与化合物的其余部分的连接点; R5a,R5b,R5c,R5d,R5e和R5f彼此独立地选自氢,卤素,C1-C6-烷基,C1-C6-烷氧基,C1-C6-烷基氨基,二(C1-C6-烷基)氨基, C3-C6-环烷基和Ar2等; R 6和R 7彼此独立地选自氢,CN,NO 2,C 1 -C 6 - 烷基,C 2 -C 6 - 烯基,C 2 -C 6炔基,C 3 -C 8 - 环烷基,饱和或部分不饱和的5-, 或7元杂环基,Ar 3等

    AZOLIN-2-YLAMINO COMPOUNDS FOR COMBATING ANIMAL PESTS
    53.
    发明申请
    AZOLIN-2-YLAMINO COMPOUNDS FOR COMBATING ANIMAL PESTS 审中-公开
    用于组合动物饲料的AZOLIN-2-YLAMINO化合物

    公开(公告)号:WO2010007060A1

    公开(公告)日:2010-01-21

    申请号:PCT/EP2009/058981

    申请日:2009-07-14

    Abstract: The present invention relates to azolin-2-ylamino compounds of formula (I), wherein A is a radical of the formulae (A.1) or (A.2), wherein * denotes the binding site and wherein the indices and variables are as defined in the description. The present invention relates as well as to the precursor compounds thereof, which are both useful for combating animal pests selected from insects, arachnids and nematodes. The invention also relates to methods for controlling and/or combating such animal pests by using these compounds, to methods of protecting crops and plant propargation material, and further also to seeds and agricultural and veterinary composition comprising said compounds.

    Abstract translation: 本发明涉及式(I)的唑啉-2-基氨基化合物,其中A是式(A.1)或(A.2)的基团,其中*表示结合位点,其中指数和变量是 如说明书中所定义。 本发明涉及其前体化合物,它们都可用于对抗选自昆虫,蜘蛛和线虫的动物害虫。 本发明还涉及通过使用这些化合物来控制和/或对抗这种动物害虫的方法,以及用于保护作物和植物促进材料的方法,还涉及包含所述化合物的种子和农业和兽医组合物。

    PESTICIDAL ACTIVE MIXTURES COMPRISING AMINOTHIAZOLINE COMPOUNDS
    54.
    发明申请
    PESTICIDAL ACTIVE MIXTURES COMPRISING AMINOTHIAZOLINE COMPOUNDS 审中-公开
    包含氨基苯甲酸化合物的农药活性混合物

    公开(公告)号:WO2009118297A2

    公开(公告)日:2009-10-01

    申请号:PCT/EP2009/053402

    申请日:2009-03-24

    Abstract: The present invention relates to pesticidal mixtures comprising as active compounds 1 ) at least one aminothiazoline compound (I) of formula (I), tautomer a), b) wherein R 1 is selected from hydrogen, COCH 3 , COCH 2 CH 3 or COCH 2 C(CH 3 ) 3 ; R 2 and R 3 together with the carbon atoms of the phenyl ring to which they are attached form a ring which, depending on the tautomeric formula I a) or b) is depicted as: a benzene ring, a saturated 5-, 6-, or 7-membered carbocycle, a partially unsaturated 5-, 6-, or 7-membered carbocycle, a 5-, 6-, or 7-membered saturated heterocycle, a partially unsaturated 5-, 6-, or 7-membered heterocycle, which heterocycles contain 1, 2, or 3 heteroatoms selected from O, S and N as ring members, and a 5- or 6- membered heteroaromatic ring which contains 1, 2, or 3 heteroatoms selected from O, S and N as ring members, and wherein the ring is unsubstituted or may carry any combination of 1, 2, 3, or 4 radicals selected from the group consisting of halogen, CH 3 , CH 2 CH 3 , CF 3 , CH 3 O, cyano and (=0) (oxo); R 4 is selected from hydrogen, fluoro, chloro, bromo, CF 3 , CH 3 O or CH 3 ; R 5 , R 6 are selected from hydrogen, chloro, fluoro, bromo, CH 3 , CH 3 O or CF 3 , wherein at least one of R 5 or R 6 is not hydrogen; with the proviso that R 2 and R 3 together do not form a -OCH 2 -O- or a -OCF 2 O-group; or the tautomers, enantiomers, diastereomers or salts thereof, and 2) at least one active compound Il selected from group A as defined in the description, use of these mixtures for combating insects, acarids, or nematodes, and a method for treating, controlling, preventing or protecting animals against infestation or infection by parasites using these mixtures.

    Abstract translation: 本发明涉及包含作为活性化合物的至少一种式(I)的至少一种氨基噻唑啉化合物(I),互变异构体a),b)其中R 1选自氢,COCH 3,COCH 2 CH 3或COCH 2 C(CH 3)3的农药混合物; R2和R3与它们所连接的苯环的碳原子一起形成环,其取决于互变异构体式a a)或b)被描述为:苯环,饱和的5-,6-或 7元碳环,部分不饱和5-,6-或7-元碳环,5-,6-或7-元饱和杂环,部分不饱和5-,6-或7-元杂环,其中 杂环含有选自O,S和N作为环成员的1,2或3个杂原子,以及含有1,2或3个选自O,S和N作为环成员的杂原子的5-或6-元杂芳族环, 并且其中所述环是未取代的或可以携带选自卤素,CH 3,CH 2 CH 3,CF 3,CH 3 O,氰基和(= O)(氧代)的1,2,3或4个基团的任何组合。 R4选自氢,氟,氯,溴,CF 3,CH 3 O或CH 3; R5,R6选自氢,氯,氟,溴,CH3,CH3O或CF3,其中R5或R6中的至少一个不是氢; 条件是R2和R3一起不形成-OCH2-O-或-OCF2O-基团; 或其互变异构体,对映异构体,非对映异构体或其盐,以及2)选自如说明书中定义的组A的至少一种活性化合物II,这些混合物用于防治昆虫,螨虫或线虫的用途,以及治疗,控制 ,防止或保护动物免受使用这些混合物的寄生虫的感染或感染。

    AZOLIN-2-YLAMINO COMPOUNDS FOR COMBATING ANIMAL PESTS
    55.
    发明申请
    AZOLIN-2-YLAMINO COMPOUNDS FOR COMBATING ANIMAL PESTS 审中-公开
    用于组合动物饲料的AZOLIN-2-YLAMINO化合物

    公开(公告)号:WO2009115491A1

    公开(公告)日:2009-09-24

    申请号:PCT/EP2009/053079

    申请日:2009-03-16

    Abstract: The present invention relates to azolin-2-ylamino compounds of formulae (I) and (II), wherein n is 0 to 3; Ar is phenyl; A is a radical of formulae A 1 or A 2 , wherein * indicates the point of attachment; X is S, O or N(R 10 ); R 7a-d are H, halogen, C 1 -C 6 -alkyl, C 1 -C 6 -alkoxy, C 1 -C 6 -alkylamino or C 3 -C 6 -cycloalkyl; R 8-10 are H, CN, NO 2 , C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 3 -C 8 -cycloalkyl, Ar 3 , -B-C(=O)R a , -B-C(=S)R a , -B-C(=NR f )R a , etc., wherein B is a single bond or C 1 -C 4 -alkanediyl; R 1 is H, halogen, C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 3 -C 6 -cycloalkyl, phenyl or benzyl; R 2,3 are H, halogen, C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 3 -C 6 -cycloalkyl, phenyl or benzyl; R 4 is H, halogen, CN, N 3 , NO 2 , C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 3 -C 8 -cycloalkyl, a heterocycle, Ar 5 , -C(=O)R a, -C(=S)R a , -C(=NR f )R a , etc.; or R 4 and R 5 together form a carbocycle or heterocycle; R 5,6 are H, halogen, CN, N 3 , NO 2 , C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 3 -C 8 -cycloalkyl, heterocycle, Ar 8 , -C(=O)R a , -C(=S)R a , -C(=NR f )R a , etc.; or R 5 and R 6 together form a carbocycle or heterocycle; R a-h are H, C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 3 -C 8 -cycloalkyl, heterocycles or Ar 10 ; Ar 1 to 11 are phenyl, naphthyl or heteroaryl; and A' is a radical of formula A 3 , wherein W is halogen or OR 11 ; R 11 is H or -C(=O)-R i ; R i is H, C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C3-C8-cycloalkyl, heterocycle or Ar 12 ; and Ar 12 is phenyl, naphthyl or heteroaryl; as well as to agricultural composition containing such compounds, the use of such compounds for controlling animal pests, seed, comprising such compounds, a method for controlling animal pests and a method for treating or protecting an animal from infestation or infection by parasites.

    Abstract translation: 本发明涉及式(I)和(II)的唑啉-2-基氨基化合物,其中n为0至3; Ar是苯基; A是式A1或A2的基团,其中*表示连接点; X是S,O或N(R10); R7a-d为H,卤素,C1-C6-烷基,C1-C6-烷氧基,C1-C6-烷基氨基或C3-C6-环烷基; R8-10是H,CN,NO2,C1-C6-烷基,C2-C6-烯基,C2-C6-炔基,C3-C8-环烷基,Ar3,-BC(= O)Ra,-BC(= S) Ra,-BC(= NRf)Ra等,其中B为单键或C1-C4-烷二基; R1是H,卤素,C1-C6-烷基,C2-C6-烯基,C2-C6-炔基,C3-C6-环烷基,苯基或苄基; R2,3是H,卤素,C1-C6-烷基,C2-C6-烯基,C2-C6-炔基,C3-C6-环烷基,苯基或苄基; R4是H,卤素,CN,N3,NO2,C1-C6-烷基,C2-C6-烯基,C2-C6-炔基,C3-C8-环烷基,杂环,Ar5,-C(= O) C(= S)Ra,-C(= NRf)Ra等; 或R4和R5一起形成碳环或杂环; R5,6是H,卤素,CN,N3,NO2,C1-C6-烷基,C2-C6-烯基,C2-C6-炔基,C3-C8-环烷基,杂环,Ar8,-C(= O) -C(= S)R a,-C(= NR f)R a等; 或R5和R6一起形成碳环或杂环; R h为H,C 1 -C 6烷基,C 2 -C 6 - 烯基,C 2 -C 6炔基,C 3 -C 8 - 环烷基,杂环或Ar 10; Ar 1至11是苯基,萘基或杂芳基; 并且A'是式A3的基团,其中W是卤素或OR 11; R 11为H或-C(= O)-R i; R 1是H,C 1 -C 6烷基,C 2 -C 6 - 烯基,C 2 -C 6炔基,C 3 -C 8环烷基,杂环或Ar 12; 和Ar 12是苯基,萘基或杂芳基; 以及含有这种化合物的农业组合物,这些化合物用于控制动物害虫,种子,包含这些化合物的用途,控制动物害虫的方法以及用于治疗或保护动物不受寄生虫感染或感染的方法。

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