PYRIMIDINETRIONE DERIVATIVES, PROCESSES FOR THEIR PREPARATION, AGENTS CONTAINING THEM AND THEIR USE AS AGENTS FOR COMBATING PESTS

    公开(公告)号:CA2009301A1

    公开(公告)日:1990-08-06

    申请号:CA2009301

    申请日:1990-02-05

    Applicant: HOECHST AG

    Abstract: of the disclosure HOE 89/F 043 Pyrimidinetrione derivatives, processes for their preparation, agents containing them and their use as agents for combating pests Compounds of the formula I, tautomeric forms thereof of the formula Ia, stereoisomers thereof and the mixtures of these forms (I), (Ia), wherein R1 and R2 denote unsubstituted or substituted alkyl, alkenyl, alkynyl; alkoxy, alkylsulfonyl, alkylcarbonyl or cyano or optionally substituted phenyl, phenylsulfonyl or phenylcarbonyl, R3 denotes hydrogen, alkyl or optionally sub stituted phenyl, R4 denotes H, OH, unsubstituted or substituted alkyl, alkenyl, alkynyl, phenylsulfonyl, phenylcarbonyl, phenylcarbamoyl or phenyl; alkylsulfonyl or alkylcarbonyl, which can be halogenated, alkylcarbamoyl or cyano, R5 and R6 denote halogen, alkyl, alkoxy, alkylcarbonyl, alkoxycarbonyl, alkylsulfenyl, -sulfinyl or -sulfonyl, haloalkoxy, alkylamino, cyano, sulfo or nitro, A,X,Z and B denote oxygen, sulfur, sulfinyl, sulfonyl or nitrogen, which can be substituted by alkyl, or B denotes a double bond, C,D,E,F and G denote carbon or nitrogen, V denotes carbon or substituted phosphorus, W denotes alkylene or haloalkylene, both of which can be substituted, Y1 denotes H, halogen, alkyl, alkylamino or hydroxyl, Y2 denotes oxygen, sulfur or nitrogen which is optionally substituted by alkyl and n and m denote 0-4, and salts thereof which can be employed in agriculture or are physiologically tolerated, have advantageous actions against a broad spectrum of animal pests in agriculture and animal breeding.

    73.
    发明专利
    未知

    公开(公告)号:DK648489A

    公开(公告)日:1990-06-21

    申请号:DK648489

    申请日:1989-12-19

    Applicant: HOECHST AG

    Abstract: The present invention relates to agents for systemic combating of ectoperasites in host animals, containing a compound of the formul I (I) in which R1 denotes hydrogen, (C1-C5)-alkyl, (C1-C3)-halogenoalkyl or halogen; R2 and R3 independently of one another denote (c1-C5)-alkyl, (C2-C5)-alkenyl, (C2-C5)-alkynyl, (C3-C7)-cycloalkyl, (C3-C7)-cycloalkenyl, (C1-C3)-halogenoalkyl, halogen, cyano, nitro, (C1-C5)-alkoxy, (C1 -C3)-alkoxy-C1-C3)-alkyl, (C1-C3)-halogenoalkoxy or (C1-C3)-alkylthio, or R2 and R3 together form a polymethylene chain having 2 to 5 carbon atoms: R4 denotes hydrogen, (c1-C10)-alkyl, (C2-C5)-alkenyl or (C3-C7)-cycloalkyl; R5 denotes hydrogen, (C1-C10)-alkyl, (C3-C5)-alkenyl, C3-C5)-alkynyl, (C3-C7)- cycloalkyl, (C3-C7)-cycloalkenyl, (C1-C3)-halogenoalkyl or (C1-C3)-alkoxy-(C hd 1-C3)-alkyl; X denotes oxygen, sulfur or an -NR6-group; and R6 denotes hydrogen, (C1-C5)-alkyl, (C3-C5)-alkenyl, C3-C5)-alkynyl, (C3-C7)-cycloalkyl, C3-C7)-cycloalkenyl, (C1-C3)-halogenoalkyl or (C1-C3)-alkoxy-(C1 -C3)-alkyl, or biologically tolerated acid addition salts thereof. The compounds of the formulas I are novel in some cases and are likewise included in the invention.

    PROCESS FOR PRODUCING ORTHO-SUBSTITUTED ARYL-CARBOXIMIDO-ESTERS

    公开(公告)号:HUT49114A

    公开(公告)日:1989-08-28

    申请号:HU161888

    申请日:1988-04-01

    Applicant: HOECHST AG

    Abstract: The present invention describes a process for the preparation of compounds of the formula I (I) in which R denotes fluorine, chlorine, bromine or (C1-C4)alkyl, R1 denotes (C1-C4)alkyl, R2 denotes H, methyl, methoxy, fluorine, chlorine, bromine or trifluoromethyl, and X denotes Cl or Br, by reaction of nitriles of the formula II (II) R1OH (III) with alcohols of the formula III and hydrogen chloride or bromide, which comprises carrying out the reaction under pressure at temperatures from - DEG C. to +50 DEG C., if appropriate in the presence of a diluent, ad subsequently converting the resulting hydrochloride or hydrobromide into the free base.

    79.
    发明专利
    未知

    公开(公告)号:DD250043A5

    公开(公告)日:1987-09-30

    申请号:DD29557686

    申请日:1986-10-24

    Applicant: HOECHST AG

    Abstract: The compounds of the formula (I) (I) in which X denotes CH2, O, S or NR6, R1 denotes alkyl, cycloalkyl, alkenyl, (substituted) phenyl, or (substituted) naphthyl, R2 and R3 denote alkyl, alkenyl or phenyl, or R2 and R3 together denote an alkylene chain, R4 denotes -H, -CN, -CCl3, -C 3BOND CH, alkyl, F, or -C(S)-NH2, R5 denotes pyridyl, furyl, thienyl, phthalimidyl, di(C1-C4)alkylmaleinimidyl, thiophthalimidyl, dihydrophthalimidyl or tetrahydrophthalimidyl, which may all be substituted, or substituted phenyl, or R4 and R5-together with the carbon atom bridging them-denote an optionally substituted indanyl, cyclopentenoyl or cyclopentenyl radical, with the proviso that compounds of the formula I in which R1 denotes phenyl which is substituted in the para-position by (C1-C4)alkoxy, halogen or (C1-C4)alkyl; R2 and R3 denote CH3; X denotes O; R4 denotes H and R5 denotes 3-phenoxyphenyl or (4-fluoro-3-phenoxy)phenyl being excepted, have advantageous insecticidal, acaricidal and nematocidal properties.

    80.
    发明专利
    未知

    公开(公告)号:DK510186D0

    公开(公告)日:1986-10-24

    申请号:DK510186

    申请日:1986-10-24

    Applicant: HOECHST AG

    Abstract: The compounds of the formula (I) (I) in which X denotes CH2, O, S or NR6, R1 denotes alkyl, cycloalkyl, alkenyl, (substituted) phenyl, or (substituted) naphthyl, R2 and R3 denote alkyl, alkenyl or phenyl, or R2 and R3 together denote an alkylene chain, R4 denotes -H, -CN, -CCl3, -C 3BOND CH, alkyl, F, or -C(S)-NH2, R5 denotes pyridyl, furyl, thienyl, phthalimidyl, di(C1-C4)alkylmaleinimidyl, thiophthalimidyl, dihydrophthalimidyl or tetrahydrophthalimidyl, which may all be substituted, or substituted phenyl, or R4 and R5-together with the carbon atom bridging them-denote an optionally substituted indanyl, cyclopentenoyl or cyclopentenyl radical, with the proviso that compounds of the formula I in which R1 denotes phenyl which is substituted in the para-position by (C1-C4)alkoxy, halogen or (C1-C4)alkyl; R2 and R3 denote CH3; X denotes O; R4 denotes H and R5 denotes 3-phenoxyphenyl or (4-fluoro-3-phenoxy)phenyl being excepted, have advantageous insecticidal, acaricidal and nematocidal properties.

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