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公开(公告)号:AU4910590A
公开(公告)日:1990-08-09
申请号:AU4910590
申请日:1990-02-05
Applicant: HOECHST AG
Inventor: KRATT GUNTER , SALBECK GERHARD , BONIN WERNER , DUWEL DIETER
IPC: C07D239/557 , A01N43/54 , A01N57/36 , C07C217/84 , C07C265/12 , C07C323/36 , C07D239/54 , C07D239/545 , C07D239/553 , C07D239/60 , C07D239/62 , C07D319/12 , C07D401/12 , C07D403/12 , C07D405/12 , C07F9/6584 , C07D239/64
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公开(公告)号:CA2009301A1
公开(公告)日:1990-08-06
申请号:CA2009301
申请日:1990-02-05
Applicant: HOECHST AG
Inventor: KRATT GUNTER , SALBECK GERHARD , BONIN WERNER , DUWEL DIETER
IPC: C07D239/557 , A01N43/54 , A01N57/36 , C07C217/84 , C07C265/12 , C07C323/36 , C07D239/54 , C07D239/545 , C07D239/553 , C07D239/60 , C07D239/62 , C07D319/12 , C07D401/12 , C07D403/12 , C07D405/12 , C07F9/6584
Abstract: of the disclosure HOE 89/F 043 Pyrimidinetrione derivatives, processes for their preparation, agents containing them and their use as agents for combating pests Compounds of the formula I, tautomeric forms thereof of the formula Ia, stereoisomers thereof and the mixtures of these forms (I), (Ia), wherein R1 and R2 denote unsubstituted or substituted alkyl, alkenyl, alkynyl; alkoxy, alkylsulfonyl, alkylcarbonyl or cyano or optionally substituted phenyl, phenylsulfonyl or phenylcarbonyl, R3 denotes hydrogen, alkyl or optionally sub stituted phenyl, R4 denotes H, OH, unsubstituted or substituted alkyl, alkenyl, alkynyl, phenylsulfonyl, phenylcarbonyl, phenylcarbamoyl or phenyl; alkylsulfonyl or alkylcarbonyl, which can be halogenated, alkylcarbamoyl or cyano, R5 and R6 denote halogen, alkyl, alkoxy, alkylcarbonyl, alkoxycarbonyl, alkylsulfenyl, -sulfinyl or -sulfonyl, haloalkoxy, alkylamino, cyano, sulfo or nitro, A,X,Z and B denote oxygen, sulfur, sulfinyl, sulfonyl or nitrogen, which can be substituted by alkyl, or B denotes a double bond, C,D,E,F and G denote carbon or nitrogen, V denotes carbon or substituted phosphorus, W denotes alkylene or haloalkylene, both of which can be substituted, Y1 denotes H, halogen, alkyl, alkylamino or hydroxyl, Y2 denotes oxygen, sulfur or nitrogen which is optionally substituted by alkyl and n and m denote 0-4, and salts thereof which can be employed in agriculture or are physiologically tolerated, have advantageous actions against a broad spectrum of animal pests in agriculture and animal breeding.
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公开(公告)号:DK648489A
公开(公告)日:1990-06-21
申请号:DK648489
申请日:1989-12-19
Applicant: HOECHST AG
Inventor: STARK HERBERT , SALBECK GERHARD , BONIN WERNER
IPC: A61K31/415 , A61P33/00 , C07D233/20 , C07D233/22 , C07D233/24 , A01N43/50
Abstract: The present invention relates to agents for systemic combating of ectoperasites in host animals, containing a compound of the formul I (I) in which R1 denotes hydrogen, (C1-C5)-alkyl, (C1-C3)-halogenoalkyl or halogen; R2 and R3 independently of one another denote (c1-C5)-alkyl, (C2-C5)-alkenyl, (C2-C5)-alkynyl, (C3-C7)-cycloalkyl, (C3-C7)-cycloalkenyl, (C1-C3)-halogenoalkyl, halogen, cyano, nitro, (C1-C5)-alkoxy, (C1 -C3)-alkoxy-C1-C3)-alkyl, (C1-C3)-halogenoalkoxy or (C1-C3)-alkylthio, or R2 and R3 together form a polymethylene chain having 2 to 5 carbon atoms: R4 denotes hydrogen, (c1-C10)-alkyl, (C2-C5)-alkenyl or (C3-C7)-cycloalkyl; R5 denotes hydrogen, (C1-C10)-alkyl, (C3-C5)-alkenyl, C3-C5)-alkynyl, (C3-C7)- cycloalkyl, (C3-C7)-cycloalkenyl, (C1-C3)-halogenoalkyl or (C1-C3)-alkoxy-(C hd 1-C3)-alkyl; X denotes oxygen, sulfur or an -NR6-group; and R6 denotes hydrogen, (C1-C5)-alkyl, (C3-C5)-alkenyl, C3-C5)-alkynyl, (C3-C7)-cycloalkyl, C3-C7)-cycloalkenyl, (C1-C3)-halogenoalkyl or (C1-C3)-alkoxy-(C1 -C3)-alkyl, or biologically tolerated acid addition salts thereof. The compounds of the formulas I are novel in some cases and are likewise included in the invention.
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公开(公告)号:ZA892158B
公开(公告)日:1989-11-29
申请号:ZA892158
申请日:1989-03-22
Applicant: HOECHST AG
Inventor: SCHUBERT HANS HERBERT , HANS HERBERT SCHUBERT , SALBECK GERHARD , GERHARD SALBECK , KRAUSE HANS-PETER , HANS-PETER KRAUSE , KNAUF WERNER , WERNER KNAUF , WALTERSDORFER ANNA , ANNA WALTERSDORFER , KERN MANFRED , MANFRED KERN
IPC: C07D253/06 , A01N43/40 , A01N55/00 , A01N55/10 , C07D213/32 , C07D213/61 , C07D213/64 , C07D213/643 , C07D213/70 , C07D237/12 , C07D237/14 , C07D237/18 , C07D239/26 , C07D239/32 , C07D239/34 , C07D241/16 , C07D241/18 , C07D257/08 , C07D401/12 , C07D409/12 , C07D491/056 , C07F7/10 , C07D , C07F , A01N
Abstract: Compounds of the formula I, their optical isomers and mixtures thereof … … in which… M represents C or Si,… R represents unsubstituted or substituted pyridyl, unsubstituted or substituted pyrimidyl, and - when M = C - unsubstituted or substituted pyridazinyl, unsubstituted or substituted pyrazinyl, unsubstituted or substituted 1,2,4-triazinyl, unsubstituted or substituted 1,2,4,5-tetrazinyl,… R , R independently of one another represent alkyl, alkenyl, haloalkyl, phenyl, or R and R represent an alkylene chain which - together with the quaternary central atom (M)- forms an unsubstituted or fluorine-substituted ring having four to six ring members (when M = Si) or having three to six ring members (when M = C),… R represents H, F, -CN, -CCl3, -C IDENTICAL CH, (C1-C4)alkyl, - @ -NH2,… R represents pyridyl, furyl, thienyl, all of which can be substituted, phthalimidyl, dialkylmaleimidyl, thiophthalimidyl, dihydrophthalimidyl, tetrahydrophthalimidyl, substituted phenyl,… or R and R - together with the carbon atom linking them - form an optionally substituted indanyl, cyclopentenoyl or cyclopentenyl radical,… and their salts and quaternisation products have advantageous insecticidal, acaricidal or nematocidal properties.
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公开(公告)号:PT90102A
公开(公告)日:1989-11-10
申请号:PT9010289
申请日:1989-03-23
Applicant: HOECHST AG
Inventor: SCHUBERT HANS HERBERT , SALBECK GERHARD , KRAUSE HANS-PETER , KNAUF WERNER , KERN MANFRED , WALTERSDORFER ANNA
IPC: C07D253/06 , A01N43/40 , A01N55/00 , A01N55/10 , C07D213/32 , C07D213/61 , C07D213/64 , C07D213/643 , C07D213/70 , C07D237/12 , C07D237/14 , C07D237/18 , C07D239/26 , C07D239/32 , C07D239/34 , C07D241/16 , C07D241/18 , C07D257/08 , C07D401/12 , C07D409/12 , C07D491/056 , C07F7/10 , C07D401/00 , C07D403/00 , C07D405/00 , C07D409/00 , C07F7/00 , A01N43/54 , A01N43/66 , A01N43/64 , A01N43/08 , A01N43/10
Abstract: Compounds of the formula I, their optical isomers and mixtures thereof … … in which… M represents C or Si,… R represents unsubstituted or substituted pyridyl, unsubstituted or substituted pyrimidyl, and - when M = C - unsubstituted or substituted pyridazinyl, unsubstituted or substituted pyrazinyl, unsubstituted or substituted 1,2,4-triazinyl, unsubstituted or substituted 1,2,4,5-tetrazinyl,… R , R independently of one another represent alkyl, alkenyl, haloalkyl, phenyl, or R and R represent an alkylene chain which - together with the quaternary central atom (M)- forms an unsubstituted or fluorine-substituted ring having four to six ring members (when M = Si) or having three to six ring members (when M = C),… R represents H, F, -CN, -CCl3, -C IDENTICAL CH, (C1-C4)alkyl, - @ -NH2,… R represents pyridyl, furyl, thienyl, all of which can be substituted, phthalimidyl, dialkylmaleimidyl, thiophthalimidyl, dihydrophthalimidyl, tetrahydrophthalimidyl, substituted phenyl,… or R and R - together with the carbon atom linking them - form an optionally substituted indanyl, cyclopentenoyl or cyclopentenyl radical,… and their salts and quaternisation products have advantageous insecticidal, acaricidal or nematocidal properties.
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公开(公告)号:BR8901359A
公开(公告)日:1989-11-07
申请号:BR8901359
申请日:1989-03-22
Applicant: HOECHST AG
Inventor: SCHUBERT HANS HERBERT , SALBECK GERHARD , KRAUSE HANS-PETER , KNAUF WERNER , WALTERSDORFER ANNA , KERN MANFRED
IPC: C07D253/06 , A01N43/40 , A01N55/00 , A01N55/10 , C07D213/32 , C07D213/61 , C07D213/64 , C07D213/643 , C07D213/70 , C07D237/12 , C07D237/14 , C07D237/18 , C07D239/26 , C07D239/32 , C07D239/34 , C07D241/16 , C07D241/18 , C07D257/08 , C07D401/12 , C07D409/12 , C07D491/056 , C07F7/10 , C07D211/36 , C07D211/18
Abstract: Compounds of the formula I, their optical isomers and mixtures thereof … … in which… M represents C or Si,… R represents unsubstituted or substituted pyridyl, unsubstituted or substituted pyrimidyl, and - when M = C - unsubstituted or substituted pyridazinyl, unsubstituted or substituted pyrazinyl, unsubstituted or substituted 1,2,4-triazinyl, unsubstituted or substituted 1,2,4,5-tetrazinyl,… R , R independently of one another represent alkyl, alkenyl, haloalkyl, phenyl, or R and R represent an alkylene chain which - together with the quaternary central atom (M)- forms an unsubstituted or fluorine-substituted ring having four to six ring members (when M = Si) or having three to six ring members (when M = C),… R represents H, F, -CN, -CCl3, -C IDENTICAL CH, (C1-C4)alkyl, - @ -NH2,… R represents pyridyl, furyl, thienyl, all of which can be substituted, phthalimidyl, dialkylmaleimidyl, thiophthalimidyl, dihydrophthalimidyl, tetrahydrophthalimidyl, substituted phenyl,… or R and R - together with the carbon atom linking them - form an optionally substituted indanyl, cyclopentenoyl or cyclopentenyl radical,… and their salts and quaternisation products have advantageous insecticidal, acaricidal or nematocidal properties.
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公开(公告)号:HUT49114A
公开(公告)日:1989-08-28
申请号:HU161888
申请日:1988-04-01
Applicant: HOECHST AG
Inventor: KNORR HARALD , SALBECK GERHARD
IPC: C07C257/08 , C07C20060101 , C07C67/00 , C07C241/00 , C07C251/24 , C07C119/20
Abstract: The present invention describes a process for the preparation of compounds of the formula I (I) in which R denotes fluorine, chlorine, bromine or (C1-C4)alkyl, R1 denotes (C1-C4)alkyl, R2 denotes H, methyl, methoxy, fluorine, chlorine, bromine or trifluoromethyl, and X denotes Cl or Br, by reaction of nitriles of the formula II (II) R1OH (III) with alcohols of the formula III and hydrogen chloride or bromide, which comprises carrying out the reaction under pressure at temperatures from - DEG C. to +50 DEG C., if appropriate in the presence of a diluent, ad subsequently converting the resulting hydrochloride or hydrobromide into the free base.
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公开(公告)号:PT87246A
公开(公告)日:1988-05-01
申请号:PT8724688
申请日:1988-04-14
Applicant: HOECHST AG
Inventor: SCHUBERT HANS HERBERT , SALBECK GERHARD , KRAUSE HANS-PETER , LUEDERS WALTER , KNAUF WERNER , WALTERSDORFER ANNA , KERN MANFRED
IPC: A01N43/40 , A01N43/54 , A01N43/58 , A01N43/60 , A01N55/10 , A01P7/02 , A01P7/04 , C07D213/61 , C07D213/63 , C07D253/06 , C07D213/64 , C07D213/643 , C07D213/65 , C07D213/70 , C07D237/12 , C07D237/14 , C07D237/18 , C07D239/26 , C07D239/30 , C07D239/34 , C07D239/38 , C07D241/16 , C07D241/18 , C07D253/07 , C07D253/08 , C07D257/08 , C07D401/06 , C07D401/08 , C07D401/12 , C07D409/06 , C07D409/08 , C07D491/04 , C07D491/056 , C07D213/00 , C07D237/00 , C07D251/00 , C07D253/00 , C07D257/00 , A01N43/34 , A01N43/48 , A01N43/64 , A01N43/713
Abstract: Compounds of the formula (I) and their stereoisomers (I) wherein A, B, C' and D independently of one another denote CH or N, in which at least one of the symbols A, B, C' or D must correspond to a nitrogen atom, X denotes CH2 or oxygen, R1 denotes a radical bonded to a carbon atom from the series comprising H, trialkylsilyl, halogen, nitro, cyano, alkenyl, alkynyl, amino, cycloalkyl, phenyl, phenxy, alkoxy, alkenyloxy, alkynyloxy, hydroxycarbonyl, alkylthio, cycloalkyloxy, alkylcarbonyl, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, halogenoalkyl, alkoxyalkyl, halogenoalkoxy, halogenoalkylthio, halogenoalkoxyalkyl, alkylthioalkyl, alkoxyalkoxy, halogenoalkoxyalkoxy, alkenyloxyalkoxy, halogenoalkenyloxy, alkoxyalkylthio, alkylthioalkoxy, alkylthioalkylthio, halogenoalkoxycarbonyl, halogenoalkenyloxycarbonyl or dialkylamino or two radicals R1 when they are positioned ortho to one another together denote a methylenedioxy, ethylenedioxy or alkylene radical, R2 and R3 independently of one another denote alkyl, alkenyl or phenyl, or R2 and R3 denote an alkylene chain which-together with the quaternary carbon atom-forms an unsubstituted or fluorinesubstituted ring having three to six ring members, R4 denotes -H, F, -CN, -CCl3, -C 3BOND CH, (C1-C4)alkyl, -C-NH2, S R5 denotes pyridyl, furyl or thienyl which can all be substituted, phthalimidyl, dialkylmaleimidyl, thiophthalimidyl, dihydrophthalimidyl, tetrahydrophthalimidyl or substituted phenyl, or R4 and R5-together with the carbon atom bridging them-denote an optionally substituted indanyl, cyclopentenoyl or cyclopentenyl radical and n denotes 0, 1 or 2, possess advantageous properties for combating pests, in particular insects and acarids. Furthermore, processes for the preparation of compounds of the formula I are described.
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公开(公告)号:DD250043A5
公开(公告)日:1987-09-30
申请号:DD29557686
申请日:1986-10-24
Applicant: HOECHST AG
Inventor: SCHUBERT HANS H , SALBECK GERHARD , LUEDERS WALTER , KNAUF WERNER , WALTERSDORFER ANNA
IPC: A01N20060101 , A01N43/40 , A01N55/00 , A01N55/02 , A01N55/10 , A01P7/04 , A23K20060101 , A61K20060101 , C07C20060101 , C07C7/08 , C07C25/13 , C07C43/215 , C07C43/225 , C07D213/64 , C07F20060101 , C07F7/08 , C07F7/10
Abstract: The compounds of the formula (I) (I) in which X denotes CH2, O, S or NR6, R1 denotes alkyl, cycloalkyl, alkenyl, (substituted) phenyl, or (substituted) naphthyl, R2 and R3 denote alkyl, alkenyl or phenyl, or R2 and R3 together denote an alkylene chain, R4 denotes -H, -CN, -CCl3, -C 3BOND CH, alkyl, F, or -C(S)-NH2, R5 denotes pyridyl, furyl, thienyl, phthalimidyl, di(C1-C4)alkylmaleinimidyl, thiophthalimidyl, dihydrophthalimidyl or tetrahydrophthalimidyl, which may all be substituted, or substituted phenyl, or R4 and R5-together with the carbon atom bridging them-denote an optionally substituted indanyl, cyclopentenoyl or cyclopentenyl radical, with the proviso that compounds of the formula I in which R1 denotes phenyl which is substituted in the para-position by (C1-C4)alkoxy, halogen or (C1-C4)alkyl; R2 and R3 denote CH3; X denotes O; R4 denotes H and R5 denotes 3-phenoxyphenyl or (4-fluoro-3-phenoxy)phenyl being excepted, have advantageous insecticidal, acaricidal and nematocidal properties.
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公开(公告)号:DK510186D0
公开(公告)日:1986-10-24
申请号:DK510186
申请日:1986-10-24
Applicant: HOECHST AG
Inventor: SCHUBERT HANS H , SALBECK GERHARD , LUEDERS WALTER , KNAUF WERNER , WALTERSDORFER ANNA
IPC: A01N20060101 , A01N43/40 , A01N55/00 , A01N55/02 , A01N55/10 , A01P7/04 , A23K20060101 , A61K20060101 , C07C20060101 , C07C7/08 , C07C25/13 , C07C43/215 , C07C43/225 , C07D213/64 , C07F20060101 , C07F7/08 , C07F7/10 , C07F , A01N
Abstract: The compounds of the formula (I) (I) in which X denotes CH2, O, S or NR6, R1 denotes alkyl, cycloalkyl, alkenyl, (substituted) phenyl, or (substituted) naphthyl, R2 and R3 denote alkyl, alkenyl or phenyl, or R2 and R3 together denote an alkylene chain, R4 denotes -H, -CN, -CCl3, -C 3BOND CH, alkyl, F, or -C(S)-NH2, R5 denotes pyridyl, furyl, thienyl, phthalimidyl, di(C1-C4)alkylmaleinimidyl, thiophthalimidyl, dihydrophthalimidyl or tetrahydrophthalimidyl, which may all be substituted, or substituted phenyl, or R4 and R5-together with the carbon atom bridging them-denote an optionally substituted indanyl, cyclopentenoyl or cyclopentenyl radical, with the proviso that compounds of the formula I in which R1 denotes phenyl which is substituted in the para-position by (C1-C4)alkoxy, halogen or (C1-C4)alkyl; R2 and R3 denote CH3; X denotes O; R4 denotes H and R5 denotes 3-phenoxyphenyl or (4-fluoro-3-phenoxy)phenyl being excepted, have advantageous insecticidal, acaricidal and nematocidal properties.
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