-
公开(公告)号:WO2008060767A2
公开(公告)日:2008-05-22
申请号:PCT/US2007080133
申请日:2007-10-02
Applicant: ABBOTT LAB , ALTENBACH ROBERT J , LIU HUAQING , DRIZIN IRENE , COWART MARLON D , WISHART NEIL , BABINSKI DAVID J , GREGG ROBERT J , ESBENSHADE TIMOTHY A , HSIEH GIN C , BRIONI JORGE D , HONORE MARIE P , BLACK LAWRENCE A , ZHAO CHEN , WAKEFIELD BRIAN D
Inventor: ALTENBACH ROBERT J , LIU HUAQING , DRIZIN IRENE , COWART MARLON D , WISHART NEIL , BABINSKI DAVID J , GREGG ROBERT J , ESBENSHADE TIMOTHY A , HSIEH GIN C , BRIONI JORGE D , HONORE MARIE P , BLACK LAWRENCE A , ZHAO CHEN , WAKEFIELD BRIAN D , HANCOCK ARTHUR A
IPC: C07D491/04 , C07D493/04 , C07H17/04
CPC classification number: C07H17/04 , C07D239/70 , C07D403/12 , C07D453/04 , C07D471/04 , C07D471/10 , C07D487/04 , C07D487/10 , C07D491/04 , C07D495/04 , C07D519/00
Abstract: Macrocyclic benzofused pyrimidine compounds, compositions comprising such compounds, methods for making the compounds, and methods of treating and preventing the progression of diseases, conditions and disorders using such compounds and compositions are described herein.
Abstract translation: 本文描述了大环苯并稠合的嘧啶化合物,包含此类化合物的组合物,制备所述化合物的方法以及使用此类化合物和组合物治疗和预防疾病,病症和障碍进展的方法。
-
公开(公告)号:WO2008060767A3
公开(公告)日:2008-05-22
申请号:PCT/US2007/080133
申请日:2007-10-02
Applicant: ABBOTT LABORATORIES , ALTENBACH, Robert J , LIU, Huaqing , DRIZIN, Irene , COWART, Marlon D , WISHART, Neil , BABINSKI, David J , GREGG, Robert J , ESBENSHADE, Timothy A , HSIEH, Gin C , BRIONI, Jorge D , HONORE, Marie P , BLACK, Lawrence A , ZHAO, Chen , WAKEFIELD, Brian D.
Inventor: ALTENBACH, Robert J , LIU, Huaqing , DRIZIN, Irene , COWART, Marlon D , WISHART, Neil , BABINSKI, David J , GREGG, Robert J , ESBENSHADE, Timothy A , HSIEH, Gin C , BRIONI, Jorge D , HONORE, Marie P , BLACK, Lawrence A , ZHAO, Chen , WAKEFIELD, Brian D.
IPC: C07D491/04 , C07D493/04 , C07H17/04
Abstract: Macrocyclic benzofused pyrimidine compounds, compositions comprising such compounds, methods for making the compounds, and methods of treating and preventing the progression of diseases, conditions and disorders using such compounds and compositions are described herein.
-
公开(公告)号:WO2008060766A2
公开(公告)日:2008-05-22
申请号:PCT/US2007/080132
申请日:2007-10-02
Applicant: ABBOTT LABORATORIES , COWART, Marlon D , ALTENBACH, Robert J , LIU, Huaqing , DRIZIN, Irene , WISHART, Neil , BABINSKI, David J , GREGG, Robert J , ESBENSHADE, Timothy A , HSIEH, Gin C , BRIONI, Jorge D , HONORE, Marie P , BLACK, Lawrence A , ZHAO, Chen , WAKEFIELD, Brian D
Inventor: ALTENBACH, Robert J , LIU, Huaqing , DRIZIN, Irene , WISHART, Neil , BABINSKI, David J , GREGG, Robert J , ESBENSHADE, Timothy A , HSIEH, Gin C , BRIONI, Jorge D , HONORE, Marie P , BLACK, Lawrence A , ZHAO, Chen , WAKEFIELD, Brian D
CPC classification number: A61K31/506 , A61K31/417 , A61K31/496 , A61K45/06
Abstract: This invention discloses a method of treating pain by administering histamine H 4 receptor ligands and compositions comprising the same.
Abstract translation: 本发明公开了一种通过施用组胺H 4受体配体和包含其的组合物来治疗疼痛的方法。
-
公开(公告)号:WO2011090669A1
公开(公告)日:2011-07-28
申请号:PCT/US2010/061713
申请日:2010-12-22
Applicant: ABBOTT LABORATORIES , LEE, CHIH-Hung , SCHRIMPF, Michael R. , ESBENSHADE, Timothy A. , ZHU, Chang Z.
Inventor: LEE, CHIH-Hung , SCHRIMPF, Michael R. , ESBENSHADE, Timothy A. , ZHU, Chang Z.
CPC classification number: A61K31/46 , A61K31/55 , A61K45/06 , A61K2300/00
Abstract: The present invention is directed to methods of treating pain by administering a therapeutically effective amount of an α7 nAChR ligand or a pharmaceutically acceptable salt thereof, to a mammal in need of treatment thereof and to pharmaceutical compositions comprising such a compound or salt.
Abstract translation: 本发明涉及通过向需要治疗的哺乳动物施用治疗有效量的a7 nAChR配体或其药学上可接受的盐和包含这种化合物或盐的药物组合物来治疗疼痛的方法。
-
5.HISTAMINE H4 RECEPTOR LIGANDS FOR USE IN PAIN TREATMENT 审中-公开
Title translation: HISTAMINE H4受体配体用于治疗疼痛公开(公告)号:WO2008060766A3
公开(公告)日:2009-02-19
申请号:PCT/US2007080132
申请日:2007-10-02
Applicant: ABBOTT LAB , COWART MARLON D , ALTENBACH ROBERT J , LIU HUAQING , DRIZIN IRENE , WISHART NEIL , BABINSKI DAVID J , GREGG ROBERT J , ESBENSHADE TIMOTHY A , HSIEH GIN C , BRIONI JORGE D , HONORE MARIE P , BLACK LAWRENCE A , ZHAO CHEN , WAKEFIELD BRIAN D
Inventor: COWART MARLON D , ALTENBACH ROBERT J , LIU HUAQING , DRIZIN IRENE , WISHART NEIL , BABINSKI DAVID J , GREGG ROBERT J , ESBENSHADE TIMOTHY A , HSIEH GIN C , BRIONI JORGE D , HONORE MARIE P , BLACK LAWRENCE A , ZHAO CHEN , WAKEFIELD BRIAN D , HANCOCK ARTHUR A
IPC: A61K31/417 , A61K31/496 , A61K31/506 , A61K45/06 , A61P29/00
CPC classification number: A61K31/506 , A61K31/417 , A61K31/496 , A61K45/06
Abstract: This invention discloses histamine H4 receptor ligands for use in a method of treating pain
Abstract translation: 本发明公开了用于治疗疼痛的方法中的组胺H 4受体配体
-
-
-
-