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1.4-IMIDAZOLE DERIVATIVES OF BENZYL AND RESTRICTED BENZYL SULFONAMIDES, SULFAMIDES, UREAS, CARBAMATES AND AMIDES AND THEIR USE AS ALPHA-1A AGONISTS 审中-公开
Title translation: 苄基和LIMITED苄基磺酰胺,磺酰胺,脲,氨基甲酸酯和酰胺以及它们的使用AS ALPHA-1A激动剂4 - 咪唑衍生物公开(公告)号:EP1259491A1
公开(公告)日:2002-11-27
申请号:EP01908800.4
申请日:2001-02-01
Applicant: Abbott Laboratories
Inventor: ALTENBACH, Robert, J. , MEYER, Michael, D. , KERWIN, James, F. , KHILEVICH, Albert , KOLASA, Teodozyj , ROHDE, Jeffrey, J. , CARROLL, William, A. , SEARLE, Xenia, B. , YANG, Fan
IPC: C07D233/54 , C07D413/12 , C07D233/84 , C07D409/12 , C07D403/12 , C07D417/12 , C07D405/12 , C07D405/04 , C07D409/04 , A61K31/4164 , A61P13/00
CPC classification number: C07D233/64 , C07D233/84 , C07D401/12 , C07D403/12 , C07D405/04 , C07D409/04 , C07D409/12 , C07D417/12
Abstract: Compounds of formula (I) are useful in treating diseases prevented by or ameliorated with α1A agonists. Also disclosed are α1A agonist compositions and a method of activating α1 adrenoceptors in a mammal.
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2.IMIDAZOLES AND RELATED COMPOUNDS AS ALPHA-1A AGONISTS 审中-公开
Title translation: 咪唑和相关化合物如α-1A AGONISTE公开(公告)号:EP1102754A1
公开(公告)日:2001-05-30
申请号:EP99939019.8
申请日:1999-08-06
Applicant: ABBOTT LABORATORIES
Inventor: ALTENBACH, Robert, J. , MEYER, Michael, D. , KERWIN, James, F., Jr. , HOLLADAY, Mark, W. , KHILEVICH, Albert , KOLASA, Teodozyj , ROHDE, Jeffrey , CARROLL, William, A.
IPC: C07D233/61 , A61K31/4164 , C07D405/04 , C07D413/12 , C07D409/12 , C07D401/12 , C07D403/12 , C07D417/12 , C07D405/12 , C07D277/28 , C07D263/32 , C07D263/48 , C07D277/40
CPC classification number: C07D233/64 , C07D233/84 , C07D401/12 , C07D403/12 , C07D405/04 , C07D409/12 , C07D417/12
Abstract: Compounds having formula (I) are useful in treating diseases prevented by or ameliorated with α1A agonists. Also disclosed are α1A agonist compositions and a method of activating α1 adrenoceptors in a mammal.
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