公开(公告)号：WO2008043835A2

公开(公告)日：2008-04-17

申请号：PCT/EP2007060879

申请日：2007-10-12

Applicant: BASF AG ,  SCHMIDT THOMAS ,  GEBHARDT JOACHIM ,  LOEHR SANDRA ,  KEIL MICHAEL ,  WEVERS JAN HENDRIK ,  ERK PETER ,  SAXELL HEIDI EMILIA ,  HAMPRECHT GERHARD ,  SEITZ WERNER ,  MAYER GUIDO ,  WOLF BERND ,  COX GERHARD ,  MICHEL ALFRED ,  ZAGAR CYRILL ,  REINHARD ROBERT ,  SIEVERNICH BERND

Inventor： SCHMIDT THOMAS ,  GEBHARDT JOACHIM ,  LOEHR SANDRA ,  KEIL MICHAEL ,  WEVERS JAN HENDRIK ,  ERK PETER ,  SAXELL HEIDI EMILIA ,  HAMPRECHT GERHARD ,  SEITZ WERNER ,  MAYER GUIDO ,  WOLF BERND ,  COX GERHARD ,  MICHEL ALFRED ,  ZAGAR CYRILL ,  REINHARD ROBERT ,  SIEVERNICH BERND

CPC classification number: C07D239/54

Abstract: The present invention relates to a crystalline form of 2-chloro-5-[3,6-dihydro-3-methyl-2,6-dioxo-4-(trifluoromethyl)-1-(2H)-pyrimidinyl]-4-fluoro-N-[[methyl-(1-methylethyl)amino]sulphonyl]benzamide. The invention also relates to a method for preparing this crystalline form and to formulations for crop protection which comprise this crystalline form of the phenyluracil.

Abstract translation: 本发明涉及2-氯-5- [3,6-二氢-3-甲基-2,6-二氧-4-（三氟甲基）-1（2H） - 嘧啶基] -4-氟的结晶形式 N - [[甲基 - （1-甲基乙基）氨基]磺酰基]苯甲酰胺。 本发明还涉及一种用于该结晶形式的制备以及制剂，其包含苯基尿嘧啶的该晶形的作物保护的方法。

公开(公告)号：WO2007063028A3

公开(公告)日：2007-08-23

申请号：PCT/EP2006068832

申请日：2006-11-23

Applicant: BASF AG ,  SCHMIDT THOMAS ,  GEBHARDT JOACHIM ,  LOEHR SANDRA ,  KEIL MICHAEL ,  WEVERS JAN HENDRIK ,  RACK MICHAEL ,  MAYER GUIDO ,  PLESCHKE AXEL

Inventor： SCHMIDT THOMAS ,  GEBHARDT JOACHIM ,  LOEHR SANDRA ,  KEIL MICHAEL ,  WEVERS JAN HENDRIK ,  RACK MICHAEL ,  MAYER GUIDO ,  PLESCHKE AXEL

IPC: C07C303/38 ,  C07C201/12 ,  C07C205/58 ,  C07C303/40 ,  C07C311/51

CPC classification number: C07C303/38 ,  C07C201/12 ,  C07C303/40 ,  C07C311/51 ,  C07C205/58

Abstract: The invention relates to methods for producing sulfonamides of formula I, wherein the variables have the designations cited in the description, by reacting m-nitro-benzoic acid chlorides of formula II with aminosulfons of formula III, under the influence of B equivalents of base IV. Said method is characterised in that, during step a) the aminosulfon of formula III is reacted with B1 equivalents of base IV, and during step b), the reaction mixture resulting from step a) is reacted with m-nitro-benzoic acid chlorides of formula II and B2 equivalents of base IV; B, B1 and B2 having the designations cited in the description.

Abstract translation: 一种用于磺酰胺的制备（I）其中各变量具有说明书中给出的含义，由间硝基 - 苯甲酰氯II与aminosulfones III的反应中，碱IV的乙等同物的影响下，其特征在于在步骤a工艺）包括一 氨基砜III用碱IV的B1当量反应，和在步骤b），其从步骤a）的反应混合物结果与间 - 硝基 - 苯甲酰氯Ⅱ和的碱IV发生反应B2当量; 其中B，B1和B2具有说明书中给出的含义。

公开(公告)号：WO2006125641A3

公开(公告)日：2007-02-15

申请号：PCT/EP2006004992

申请日：2006-05-24

Applicant: BASF AG ,  PUHL MICHAEL ,  RACK MICHAEL ,  SCHMIDT THOMAS ,  HOFMANN MICHAEL ,  BAUMANN ERNST ,  KORDES MARKUS ,  DEYN WOLFGANG VON ,  KUHN DAVID G ,  CULBERTSON DEBORAH L ,  ANSPAUGH DOUGLAS ,  COTTER HENRY VAN TUYL ,  OLOUMI-SADEGHI HASSAN ,  BUCCI TONI ,  BASTIAANS HENRICUS M M

Inventor： PUHL MICHAEL ,  RACK MICHAEL ,  SCHMIDT THOMAS ,  HOFMANN MICHAEL ,  BAUMANN ERNST ,  KORDES MARKUS ,  VON DEYN WOLFGANG ,  KUHN DAVID G ,  CULBERTSON DEBORAH L ,  ANSPAUGH DOUGLAS ,  COTTER HENRY VAN TUYL ,  OLOUMI-SADEGHI HASSAN ,  BUCCI TONI ,  BASTIAANS HENRICUS M M

IPC: C07D401/12 ,  A01N43/40

CPC classification number: A01N43/40 ,  C07D401/12

Abstract: The present invention relates to new pyridine compounds which are useful for combating animal pests, in particular insects, arachnids and nematodes. The invention also relates to a method for combating insects, nematodes and arachnids. The pyridine compounds have the formula I as defined below. Likewise, compounds of the formula Il are suitable for combating pests. In formulae I and Il n is 1 or 2, and R1, R2, R3, R4 and R5 are as defined in the claims and in the specification.

Abstract translation: 本发明涉及可用于对抗动物害虫，特别是昆虫，蜘蛛和线虫的新的吡啶化合物。 本发明还涉及一种防治昆虫，线虫和蜘蛛的方法。 吡啶化合物具有如下定义的式I。 同样地，式II化合物适用于防治害虫。 在式I和II中，n为1或2，R1，R2，R3，R4和R5如权利要求书和说明书中所定义。

公开(公告)号：WO2005063724B1

公开(公告)日：2005-08-25

申请号：PCT/EP2004014623

申请日：2004-12-22

Applicant: BASF AG ,  KORDES MARKUS ,  HOFMANN MICHAEL ,  PUHL MICHAEL ,  GOETZ NORBERT ,  RACK MICHAEL ,  BAUMANN ERNST ,  DEYN WOLFGANG VON ,  SCHMIDT THOMAS ,  TEDESCHI LIVIO ,  TREACY MICHAEL F ,  CULBERTSON DEBORAH L ,  BUCCI TONI ,  KUHN DAVID G

Inventor： KORDES MARKUS ,  HOFMANN MICHAEL ,  PUHL MICHAEL ,  GOETZ NORBERT ,  RACK MICHAEL ,  BAUMANN ERNST ,  VON DEYN WOLFGANG ,  SCHMIDT THOMAS ,  TEDESCHI LIVIO ,  TREACY MICHAEL F ,  CULBERTSON DEBORAH L ,  BUCCI TONI ,  KUHN DAVID G

IPC: A01N43/76 ,  A01N43/78 ,  C07D263/28 ,  C07D277/18

CPC classification number: C07D263/28 ,  A01N43/76 ,  A01N43/78 ,  C07D277/18

Abstract: The present invention relates to 1 -(azolin-2-yl)amino-1,2-diphenylethane compounds of the general formula (I) wherein A is a radical of the formulae A' or A : N R A' A and wherein m is 0, 1, 2, 3, 4 or 5, n is 0, 1, 2, 3, 4 or 5, X is sulfur or oxygen, and wherein the variables R , R , R , R , R , R , R , R are as defined in the claims, and to the agriculturally acceptable salts thereof. The invention relates also to a method of combating animal pests, selected from in­sects, arachnids and nematodes and to a method for protecting crops from attack or infestation by insects, arachnids or nematodes, which comprises contacting a crop with a pesticidally effective amount of a 1 -(azolin-2-yl)amino-1,2-diphenylethane com­pounds of the general formula I and/or at least one salt thereof.

Abstract translation: 本发明涉及通式（I）的1-（唑啉-2-基）氨基-1,2-二苯基乙烷化合物，其中A是式A'或A 2的基团：NRA'A <2 并且其中m是0,1,2,3,4或5，n是0,1,2,3,4或5，X是硫或氧，并且其中变量R 1，R 2， R 3，R 4，R 5a，R 5b，R 5c，R 5如权利要求中所定义，以及其农业上可接受的盐。 本发明还涉及一种对抗昆虫，蜘蛛和线虫的动物害虫的方法，还涉及一种保护作物免受昆虫，蜘蛛或线虫袭击或侵染的方法，其中包括使农作物与杀虫有效量的1 - （唑啉-2-基）氨基-1,2-二苯基乙烷化合物和/或其至少一种盐。

公开(公告)号：WO2007060220A3

公开(公告)日：2007-08-02

申请号：PCT/EP2006068880

申请日：2006-11-24

Applicant: BASF AG ,  POHLMAN MATTHIAS ,  DEYN WOLFGANG VON ,  SCHMIDT THOMAS ,  KAISER FLORIAN ,  ANSPAUGH DOUGLAS D ,  CULBERTSON DEBORAH L ,  COTTER HENRY VAN TUYL

Inventor： POHLMAN MATTHIAS ,  VON DEYN WOLFGANG ,  SCHMIDT THOMAS ,  KAISER FLORIAN ,  ANSPAUGH DOUGLAS D ,  CULBERTSON DEBORAH L ,  COTTER HENRY VAN TUYL

IPC: A01N43/10 ,  A01N41/04 ,  A01N41/06 ,  A01N43/36 ,  A01N43/40 ,  A01N43/48 ,  A01N43/50 ,  A01N43/653 ,  A01N47/34 ,  C07C311/48 ,  C07C311/51 ,  C07C311/53 ,  C07C311/65 ,  C07D207/48 ,  C07D333/46

CPC classification number: C07C311/51 ,  A01N41/06 ,  A01N43/10 ,  A01N43/36 ,  A01N43/50 ,  A01N43/56 ,  A01N43/653 ,  A01N47/24 ,  A01N47/34 ,  A01N47/42 ,  A01N51/00 ,  C07C311/16 ,  C07C311/53 ,  C07C311/58 ,  C07C381/10 ,  C07D207/48 ,  C07D231/12 ,  C07D231/26 ,  C07D233/54 ,  C07D333/46

Abstract: The present invention relates to a method of combating animal pests which comprises contacting the animal pests, their habit, breeding ground, food supply, plant, seed, soil, area, material or environment in which the animal pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from animal attack or infestation with a pesticidally effective amount of at least one cyanobenzene compound of the formula (I) and/or at least one agriculturally acceptable salt thereof: where m is 0, 1 or 2; is a radical of the formulae N=CR 5 R 6 , N=SR 7 R 8 , NR 10 -C(=X)-R 9 , where X is O, S A or NR 11 , or A is a N-bound 5-, 6- or 7-membered heterocycle, which is ethylenically unsaturated or aromatic, and which additionally may contain 1, 2, or 3 further heteroatoms or heteroatom groups, selected from O, S, SO, SO 2 , N, and NR 12 , and/or 1, 2 or 3 carbonyl groups as ring members and which may carry 1, 2, 3 or 4 radicals R 13 , where the radicals R 1 to R 13 are as defined in the claims or the description. The invention further relates to specific compounds I and to agricultural compositions comprising them.

Abstract translation: 本发明涉及一种对抗动物害虫的方法，其包括使动物害虫，其习惯，繁殖地，食物供应，植物，种子，土壤，面积，材料或动物害虫生长或可能生长的环境接触;或 用农药有效量的至少一种式（I）的氰基苯化合物和/或其至少一种农业上可接受的盐保护免受动物攻击或侵染的材料，植物，种子，土壤，表面或空间：其中m 是0，1或2; 是下式的基团：N = CR 5 R 6，N = SR 7 R 8，NR 6， 其中X是O，SA或NR 11，或者A是N键的5-位， 6或7元杂环，其为烯属不饱和或芳族的，并且另外可以含有1,2或3个选自O，S，SO，SO 2的杂原子或杂原子基团。 ，N和NR 12，和/或1,2或3个羰基作为环成员，并且可以带有1,2,3或4个基团R 13，其中 基团R 1至R 13如权利要求或说明书所定义。 本发明还涉及特定的化合物I和包含它们的农业组合物。

公开(公告)号：WO2004047534A3

公开(公告)日：2004-07-08

申请号：PCT/EP0313108

申请日：2003-11-21

Applicant: BASF AG ,  KORDES MARKUS ,  DEYN WOLFGANG VON ,  HOFMANN MICHAEL ,  SCHMIDT THOMAS ,  STEINER GERD ,  TREACY MICHAEL F ,  VAN TUYL COTTER HENRY ,  CULBERTSON DEBORAH ,  SHIEH HONG-MING

Inventor： KORDES MARKUS ,  VON DEYN WOLFGANG ,  HOFMANN MICHAEL ,  SCHMIDT THOMAS ,  STEINER GERD ,  TREACY MICHAEL F ,  VAN TUYL COTTER HENRY ,  CULBERTSON DEBORAH ,  SHIEH HONG-MING

IPC: A01N47/06

CPC classification number: A01N47/06

Abstract: The present invention relates to the use of compounds of formula (I), wherein R is C1-C8-alkyl, unsubstituted or substituted with 1, 2 or 3 radicals selected from the group consisting of halogen, amino, nitro, cyano, C1-C4-alkenyl, C1-C4-haloalkenyl, C1-C4-alkoxy, C1-C4-haloalkoxy, C1-C4-alkylthio, 5- to 10-membered heteroaryl containing as ring members 1, 2, 3 or 4 heteroatoms selected from oxygen, sulfur and nitrogen, and phenyl, wherein the heteroaryl and phenyl radicals may be substituted for the control of nematodes, a method for the control of nematodes, and a method for the protection of plants from infestation or attack by nematodes.

Abstract translation: 本发明涉及式（I）化合物的用途，其中R是未取代或被1,2或3个选自卤素，氨基，硝基，氰基，C1- C 4 - 烯基，C 1 -C 4卤代链烯基，C 1 -C 4 - 烷氧基，C 1 -C 4卤代烷氧基，C 1 -C 4 - 烷硫基，含有作为环成员1,2,3或4的选自氧的杂原子的5至10元杂芳基 ，硫和氮和苯基，其中杂芳基和苯基可以代替线虫的控制，控制线虫的方法，以及保护植物免受线虫侵袭或侵袭的方法。

公开(公告)号：WO2004080170A3

公开(公告)日：2004-11-04

申请号：PCT/EP2004001677

申请日：2004-02-20

Applicant: BASF AG ,  STEINER GERD ,  SCHMIDT THOMAS ,  KORDES MARKUS ,  DEYN WOLFGANG VON ,  HOFMANN MICHAEL ,  BAUMANN ERNEST ,  PUHL MICHAEL ,  HEFFERNAN GAVIN ,  CULBERTSON DEBORAH L ,  TREACY MICHAEL F

Inventor： STEINER GERD ,  SCHMIDT THOMAS ,  KORDES MARKUS ,  VON DEYN WOLFGANG ,  HOFMANN MICHAEL ,  BAUMANN ERNEST ,  PUHL MICHAEL ,  HEFFERNAN GAVIN ,  CULBERTSON DEBORAH L ,  TREACY MICHAEL F

IPC: A01N43/60 ,  A01N43/72

CPC classification number: A01N43/72 ,  A01N43/60

Abstract: Use of compounds Formula (I), A = a 5- to 7-membered ring which may contain 1-3 heteroatoms and which may be saturated or partially or completely unsaturated; R = OH, SH, NH2, CN, NO2, halogen, C1-C6-alkyl, C1-C6-haloalkyl; C1-C6- alkoxy, C1-C6-haloalkoxy, C1-C6-alkylthio, C1-C6-haloalkylthio, C2-C6-alkenyl, C2-C6-alkenyloxy, C2-C6-alkenylthio, C2-C6-alkynyl, C2-C6­alkynyloxy, C2-C6-alkynylthio, C1-C6-alkylsulfonyl, C1-C6-alkylsulfoxyl, C2-C6-alkenylsulfonyl, C2-C6-alkynylsulfoxyl, C1-C6-alkylcarbonyl, C1-C6- alkoxycarbonyl, C1-C6-alkylcarbonyloxy; R = C1-C6-alkyl or a mono- or bicyclic 5- to 10-membered aromatic ringsystem which may contain 1 to 4 heteroatoms and which is either bonded directly or through an O, S, C1-C6-alkylene or C1-C6-alkyleneoxy linkage to A or fused to A and which may be substituted; R , R = H, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkylamino, C1-C6-alkoxy, C3-C6 cycloalkyl, or R and R together with the nitrogen atom to which they are attached form a saturated or partially saturated mono- or bicyclic 5- to 10-membered ring system con-taining 1 to 3 heteroatoms or a 5-membered hetaryl containing 1 to 4 nitro-gen atoms, wherein the carbon and/or nitrogen atoms in the ring systems may be substituted or phenyl or benzyl which may be substituted; or R and R together form the chains -(CH2)2N (O-)(CH2)2- or -(CH2)3N (O )(CH2)2 ; m = 0 to 4; n is 0 to 4; and the enantiomers, diastereomers, cis/trans isomers or salts thereof for combatting insects, arachnids or nematodes, methods for the control of these pests and of protecting growing plants attack or infestation by these pests by applying a pesticidally effective amount of a compound of formula (I), processes for preparing them, and compositions comprising them.

Abstract translation: 式（I）化合物的用途，A =可含有1-3个杂原子且可以是饱和或部分或完全不饱和的5至7元环; R 1 = OH，SH，NH 2，CN，NO 2，卤素，C 1 -C 6烷基，C 1 -C 6卤代烷基; C 1 -C 6烷氧基，C 1 -C 6卤代烷氧基，C 1 -C 6烷硫基，C 1 -C 6卤代烷硫基，C 2 -C 6烯基，C 2 -C 6烯氧基，C 2 -C 6烯硫基， C 1 -C 6烷基磺酰基，C 1 -C 6烷基亚磺酰基，C 2 -C 6烯基磺酰基，C 2 -C 6炔基亚磺酰基，C 1 -C 6烷基羰基，C 1 -C 6烷氧基羰基， R 2 = C 1 -C 6烷基或可含有1至4个杂原子并且直接键合或通过O，S，C 1 -C 6亚烷基键合的单环或双环5至10元芳环体系或 与A相连的C1-C6-亚烷氧基键或者与A相连并可以被取代的; R 3，R 4 = H，C 1 -C 6烷基，C 1 -C 6卤代烷基，C 1 -C 6烷基氨基，C 1 -C 6烷氧基，C 3 -C 6环烷基或R 3和 R 4与它们所连接的氮原子一起形成饱和或部分饱和的含有1至3个杂原子的5至10元环系统或含有1至4个硝基的5元杂芳基 其中环系统中的碳和/或氮原子可以被取代或者可以被取代的苯基或苄基; 或者R 3和R 4一起形成链 - （CH 2）2 N +（O-）（CH 2）2 - 或 - （CH 2）3 N +（O-）（CH 2）2 < - >; m = 0至4; n是0至4; 以及用于防治昆虫，蛛形纲动物或线虫的对映异构体，非对映异构体，顺式/反式异构体或其盐，控制这些害虫的方法以及通过施用农药有效量的式（I）化合物来保护生长中的植物对这些害虫的侵袭或侵染 （I），制备它们的方法以及包含它们的组合物。

公开(公告)号：CA2574406C

公开(公告)日：2013-02-19

申请号：CA2574406

申请日：2005-07-13

Applicant: BASF AG

Inventor： LOEHR SANDRA ,  GEBHARDT JOACHIM ,  MAYER GUIDO ,  KEIL MICHAEL ,  SCHMIDT THOMAS ,  WOLF BERND

IPC: C07D239/54 ,  C07C307/06

Abstract: The invention relates to a method for the production of 3-phenyl(thio)uracils and dithiouracils of formula I, wherein the variables have the meanings cited in the description, characterized in that carbamates of formula II, wherein variables X1, X3, Ar and A have the above-mentioned meanings and L1 represents a nucleophilically displaceable nucleofuge, can be reacted with enamines of formula III, wherein variables X2, R1, R2 and R3 have the above-mentioned meanings and L2 represents a nucleophilically displaceable nucleofuge. The invention also relates to intermediate products for the production thereof.

公开(公告)号：EG25540A

公开(公告)日：2012-02-12

申请号：EG2008010013

申请日：2008-01-03

Applicant: BASF AG

Inventor： SCHMIDT THOMAS ,  PUHL MICHAEL ,  DICKHAUT JOACHIM ,  BASTIAANS HENRICUS MARIA MARTINUS ,  RACK MICHAEL ,  CULBERTSON DEBORAH L ,  ANSPAUGH DOUGLAS D ,  BRAUN FRANZ-JOSEF ,  BUCCL TONI ,  COTTER HENRY VAN TUYL ,  KUHN DAVID G ,  OLOUMI-SADEGHI HASSAN

IPC: C07D401/04 ,  A01N43/56

Abstract: wherein the variables and the indices are as defined per the description, processes for preparing the compounds I, pesticidal compositions comprising compounds I, use of compounds I for the control of insects, acarids or nematodes, and methods for treating, controlling, preventing or protecting animals against infestation or infection by parasites by use of compounds of formula I.

公开(公告)号：AU2004271715B2

公开(公告)日：2010-08-26

申请号：AU2004271715

申请日：2004-09-10

Applicant: BASF AG

Inventor： SCHIEWECK FRANK ,  OLOUMI-SADEGHI HASSAN ,  RACK MICHAEL ,  CULBERTSON DEBORAH L ,  DEYN WOLFGANG VON ,  PUHL MICHAEL ,  COTTER HENRY VAN TUYL ,  KORDES MARKUS ,  GOTZ NORBERT ,  BUCCI TONI ,  HOFMANN MICHAEL ,  BAUMANN ERNST ,  SCHMIDT THOMAS ,  GROTE THOMAS

IPC: A01N43/90 ,  C07D487/04

Abstract: The present invention relates to a method of combating animal pests which comprises contacting the animal pests, their habit, breeding ground, food supply, plant, seed, soil, area, material or environment in which the animal pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from animal attack or infestation with a pesticidally effective amount of at least one 6-halogeno[1,2,4]triazolo[1,5-a]-pyrimidine of the general formula (I), wherein X, R1, R2, R3 and R4 are as defined in claim 1 and/or the agriculturally useful salts thereof.