Abstract:
PROBLEM TO BE SOLVED: To provide an aniline derivative as an intermediate of a pyrazolecarboxylic acid anilide compound with high microbicidal activity.SOLUTION: The aniline derivative is an aniline compound represented by formula (III) (wherein, the variable part is defined as follows: n is 0; m is 3; and Xis a halogen atom, being meant indefinitely).
Abstract translation:待解决的问题:提供苯胺衍生物作为具有高杀微生物活性的吡唑甲酰苯胺化合物的中间体。 苯胺衍生物是由式(III)表示的苯胺化合物(其中,可变部分定义如下:n为0; m为3; X 2 < SP>是卤素原子,意思是无限期)。 版权所有(C)2013,JPO&INPIT
Abstract:
The present invention relates to fungicidal pyrimidine compounds, to their use and to methods for combating phytopathogenic fungi. The present invention also relates to seeds treated with at least one such compound. Furthermore the invention relates to processes for preparing compounds of formula I.
Abstract:
The invention relates to fungicidal mixtures which comprise 1) azolylmethyloxiranes of general formula I, wherein the variables are defined as in the application, 2) a fungicidal compound II, and 3) optionally another fungicidal compound II as the active components, the compounds II of components 2 and 3 being independently selected from among the compounds described in the application with the proviso that components 2 and components 3 are not the same. The invention also relates to the use of the fungicidal mixtures for the control of phytopathogenic fungi and to agents containing said mixtures.
Abstract:
The present invention relates to mixtures comprising, as active components, 1) a fungicidal compound of formula (I) wherein: R1 is alkyl; alkoxyalkyl; haloalkyl; arylalkyl; aryl; or heteroaryl; R2 is alkyl; alkoxyalkyl; haloalkyl; arylalkyl; aryl; heteroaryl; 5-pyrimidinyl; or 2-or 5-thiazolyl; R3 is H; alkyl; alkoxyalkyl; haloalkyl; arylalkyl; aryloxyalkyl; arylthioalkyl; aryl; heteroaryl; or alkylsilyl; R4 is H; acyl; haloacyl, alkoxycarbonyl; aryloxycarbonyl; alkylaminocarbonyl; or dialkylaminocarbonyl; or a salt thereof; and 2) a fungicidal compound II selected from azoles, strobilurins, carboxamides, heterocylic compounds, carbamates, and other active compounds in synergistically effective amounts.
Abstract:
The present invention relates to fungicidal mixtures, comprising, as active components, 1 ) at least one 5-hydroxypyrazoline of Formula (I), in which the substituents are defined according to the description, and 2) at least one active compound Il selected from the groups of the azoles, strobilurins, carboxamides, nitrogenous heterocyclyl compounds, carbamates and dithiocarbamates, and other active compounds according to the description in a synergistically effective amount, to methods for controlling harmful fungi using mixtures of a compound I and active compounds Il and to preparations comprising these mixtures, and also to processes for preparing these preparations.
Abstract:
The present invention relates to compounds of the formula (I) wherein the variables are as defined in the claims and description, their preparation and the uses of compounds(I).
Abstract:
Fungicidal mixtures comprising, as active components, 1) a triazolyl compound selected from the compounds of the formula (I) in which the variables have the meanings as defined in the description and the claims, and a component 2.
Abstract:
The invention relates to fungicidal mixtures which comprise 1) sulphur-containing triazole compounds I as described in the application, and 2) a fungicidal compound II as the active components, the compounds II of component 2 being selected from among the compounds described in the application. The invention also relates to the use of the fungicidal mixtures for the control of phytopathogenic fungi and to agents containing said mixtures.
Abstract:
The invention relates to a method for producing 3-difluoromethyl-substituted pyrazole compounds of formula (I), wherein R1 represents H, halogen, nitro, C1-C8 alkyl, C1-C8 haloalkyl, C3-C8 cycloalkyl, phenyl, naphthyl, hetaryl, cyano, -C(=O)-OR1a, -C(=O)-NR1bR1c, -C(=O)-SR1d or -C(=S)-SR1 e; R2 represents H, C1-C4 alkyl, benzyl or phenyl; R3 represents H, halogen, C1-C8 alkoxy, C1-C8 haloalkoxy, C3-C8 cycloalkoxy, C2-C8 alkenyloxy, C1-C8 alkylthio, C1-C8 haloalkylthio, C3-C8 cycloalkylthio or C2-C8 alkenylthio; to compounds of formula (II.a) or (II.b), wherein R1 and R3 have one of the above definitions; R4 represents halogen, -OR4a, -SR4a , -O-SO2-R4a or a group -NR4bR4c; R5 and R6 represent C1-C8 alkyl, C1-C8 haloalkyl, C3-C8 cycloalkyl, benzyl or phenyl or together with the nitrogen atom to which they are bound represent a 3- to 8-membered heterocycle; to Lewis acid adducts of compounds of formula (II.b); to the use of compounds of formula (II.a) or (II.b) and of the Lewis acid adducts thereof for producing compounds of formula (I) or (VI); and to a method for converting said compounds to the corresponding 3-difluoromethylpyrazole-4-yl carboxylic acids.
Abstract translation:本发明涉及一种用于制备式-3-二氟甲基吡唑(I)化合物其中R1是H,卤素,硝基,C1-C8烷基,C1-C8卤代烷基,C3-C8环烷基,苯基,萘基,杂芳基, 氰基,-C(= O)-OR1a,-C(= O)-NR1bR1c,-C(= O)-SR1d或-C(= S)-SR1e基; R2是H,C1-C4烷基,苄基或苯基; R 3为H,卤素,C1-C8烷氧基,C1-C8卤代烷氧基,C3-C8环烷氧基,C2-C8链烯氧基,C1-C8烷硫基,C1-C8卤代烷硫基,C3-C8-环烷硫基或C 2 -C C8-烯硫基;式(二.a)或(二.b)的化合物,其中R 1和R 3具有以上给出的含义之一; R 4是卤素,-OR4a,-SR4a,-O-SO2-R4A或一组-NR4bR4c基; R5和R6是C1-C8烷基,C1-C8卤代烷基,C3-C8环烷基,苄基或苯基或一起与氮原子到它们所键合的,代表3-至8-元杂环; 式(二.b)化合物的路易斯酸加合物;使用(二.a)或(二.b)和路易斯酸加合物,式I化合物的对式(I)或(VI)的化合物的制备方法; 并且这些化合物转变成相应的3-二氟甲基吡唑-4-基甲磺酸的方法。