公开(公告)号：DE19755016A1

公开(公告)日：1999-06-17

申请号：DE19755016

申请日：1997-12-11

Applicant: BAYER AG ,  BAYER AGROCHEM KK

Inventor： VOIGT KATHARINA DR ,  RIEBEL HANS-JOCHEM DR ,  LEHR STEFAN DR ,  LENDER ANDREAS DR ,  KIRSTEN ROLF DR ,  DOLLINGER MARKUS DR ,  DREWES MARK WILHELM DR ,  WETCHOLOWSKY INGO DR ,  WATANABE YUKIYOSHI DR ,  GOTO TOSHIO ,  MYERS RANDY ALLEN DR

IPC: C07D251/18 ,  A01N43/68 ,  A01N43/70 ,  C07C279/26 ,  C07D251/42 ,  C07D251/48 ,  C07D405/12 ,  C07D409/12 ,  C07D413/12 ,  C07D417/12 ,  C07D401/12 ,  C07C277/08

Abstract: The invention relates to novel substituted 2,4-diamino-1,3,5-triazines of formula (I) in which Q represents O (oxygen), S (sulfur), SO, SO2, NH or N(alkyl), R represents hydrogen or optionally substituted alkyl, R represents hydrogen, formyl or respective optionally substituted alkyl, alkyl carbonyl, alkoxycarbonyl or alkyl amino carbonyl, R represents respective optionally substituted alkyl or cycloalkyl, R represents hydrogen or alkyl, R represents hydrogen or alkyl, Ar represents optionally substituted aryl or heteroaryl, and Z represents hydrogen, cyano, halogen, or respective substituted alkyl, alkoxyl, alkoxycarbonyl, alkylthio, alkyl sulfinyl, alkyl sulfonyl, alkenyl, alkynyl or cycloalkyl. The invention also relates to a method and novel intermediate products, to the production thereof, and the application thereof as herbicides.

公开(公告)号：DE19744711A1

公开(公告)日：1999-04-15

申请号：DE19744711

申请日：1997-10-10

Applicant: BAYER AG ,  BAYER AGROCHEM KK

Inventor： RIEBEL HANS-JOCHEM DR ,  DICKERSHOFF HANS-JOACHIM ,  KOTYSCH WOLF-RUEDIGER ,  LEHR STEFAN DIPL CHEM DR ,  LENDER ANDREAS DR ,  KIRSTEN ROLF DR ,  STELZER UWE DR ,  VOIGT KATHARINA DR ,  DOLLINGER MARKUS DR ,  GOTO TOSHIO ,  WATANABE YUKIYOSHI DR

IPC: A01N43/68 ,  C07D251/18 ,  C07D401/12 ,  C07D405/12 ,  C07D409/12 ,  A01N43/66

Abstract: 2,4-Diamino-1,3,5-triazine derivatives of formula (I) are new. R1 = H or optionally substituted alkyl, alkanoyl, alkoxycarbonyl, alkenoyl or alkynoyl; R2 = H or optionally substituted alkenyl or alkynyl; R3 = -A-Z; A = optionally substituted alkanediyl optionally terminated or interrupted by O, S, NH or alkylimino; and Z = optionally substituted cyclopentyl, cyclohexyl, phenyl, naphthyl, tetralinyl, decalinyl, indanyl, indenyl, furyl, benzofuryl, dihydrobenzofuryl, thienyl, benzothienyl, dihydrobenzothienyl, isobenzofuryl, dihydroisobenzofuryl, isobenzothienyl, dihydroisobenzothienyl, pyrrolyl, indolyl, isoindolyl, indolinyl, isoindolinyl, benzdioxolyl, oxazolyl, benzoxazolyl, thiazolyl, benzothiazolyl, benzimidazoly, indazolyl, oxadiazolyl, thiadiazolyl, pyrazolyl, pyridinyl, pyrimidinyl, pyrazinyl, pyridazinyl, quinolyl, isoquinolyl. quinoxalinyl, cinnolinyl and phthalazinyl. Also claimed are intermediates of formula (IV) (see 'Preparation').

公开(公告)号：DE19629144A1

公开(公告)日：1998-01-22

申请号：DE19629144

申请日：1996-07-19

Applicant: BAYER AG

Inventor： GESING ERNST R F DR ,  DREWES MARK WILHELM DR ,  JANSEN JOHANNES R DR ,  KIRSTEN ROLF DR ,  KLUTH JOACHIM DR ,  MUELLER KLAUS-HELMUT DR ,  PHILIPP ULRICH DR ,  RIEBEL HANS-JOCHEM DR ,  SCHALLNER OTTO DR ,  WOLLWEBER DETLEF DR ,  DOLLINGER MARKUS DR ,  STENZEL KLAUS DR ,  ERDELEN CHRISTOPH DR

IPC: A01N43/90 ,  C07D487/04 ,  C07D471/04

Abstract: The invention concerns novel substituted triazoloazine sulphonamides of formula (I) in which: Q stands for nitrogen or a CH group: Q stands for nitrogen or a CH group; R stands for hydrogen or halogen, or for C1-C4 alkyl, C1-C4 alkoxy, C1-C4 alkylthio, C1-C4 alkylamino or di(C1-C4 alkyl)amino, in each case optionally substituted by hydroxy, halogen or C1-C4 alkoxy; R stands for hydrogen or halogen, or for C1-C4 alkyl, C1-C4 alkoxy, C1-C4 alkylthio, C1-C4 alkylamino or di(C1-C4 alkyl)amino, in each case optionally substituted by halogen; and Ar stands for 4-cyano-2,5-difluoro-phenyl, 2,6-dimethoxy-phenyl, 2-bromo-3-trifluoro-methyl-phenyl, 2-bromo-5-trifluoromethyl-phenyl, 6-chloro-pyridine-3-yl-methyl or one of the 5- or 6-member (hetero)cyclic groups mentioned in the description. The invention also concerns salts of these substances, a process for preparing the novel compounds, and their use as plant-treatment agents.

公开(公告)号：DE19609059A1

公开(公告)日：1997-09-11

申请号：DE19609059

申请日：1996-03-08

Applicant: BAYER AG

Inventor： MUELLER KLAUS-HELMUT DR ,  DREWES MARK WILHELM DR ,  GESING ERNST R F DR ,  JANSEN JOHANNES R DR ,  KIRSTEN ROLF DR ,  KLUTH JOACHIM DR ,  KOENIG KLAUS DR ,  RIEBEL HANS-JOCHEM DR ,  SCHALLNER OTTO DR ,  FINDEISEN KURT PROF DR ,  DOLLINGER MARKUS DR

IPC: A01N47/38 ,  C07D249/12 ,  C07D249/14 ,  C07D403/12 ,  A01N43/653

Abstract: The invention relates to novel substituted aryl sulphonyl amino(thio)carbonyl-triazolin(thi)ones of the formula (I) in which: Q is oxygen or sulphur; Q is oxygen or sulphur; R is hydrogen, amino or possibly substituted alkyl, alkoxy, alkyl carbonyl, alkoxy carbonyl, alkyl thio, alkyl sulphinyl, alkyl sulphonyl, alkenyl, alkinyl or alkylidene amino; R is hydrogen or possibly substituted alkyl, alkyl carbonyl, alkoxy carbonyl, alkyl sulphonyl, alkenyl or alkinyl or, together with R , for alkane diyl possibly interrupted by oxygen and/or substituted alkandiyl; R is hydrogen, cyano, nitro, halogen or possibly substituted alkyl, alkyl carbonyl or alkoxycarbonyl; R is hydrogen, hydroxy, amino, alkylidene amino or a possibly substituted radical from the series alkyl, alkenyl, alkinyl, alkoxy, alkene oxy, alkyl amino, dialkyl amino, cycloalkyl, cycloalkyl alkyl, cycloalkyl amino, aryl, aryl alkyl; and R is hydrogen, hydroxy, mercapto, amino, cyano, halogen or a possibly substituted radical from the series alkyl, alkoxy, alkyl thio, alkyl amino, dialkyl amino, alkenyl, alkinyl, alkenyloxy, alkinyloxy, alkenyl thio, alkinylthio, alkenyl amino, alkinyl amino, cycloalkyl, cycloalkyloxy, cycloalkyl thio, cycloalkyl amino, cycloalkyl alkyl, aryl, aryloxy, aryl thio, aryl amino, aryl alkyl; and salts of compounds of formula (I), process for producing the novel compounds and their use as herbicides.

公开(公告)号：DE19525974A1

公开(公告)日：1997-01-23

申请号：DE19525974

申请日：1995-07-17

Applicant: BAYER AG

Inventor： MUELLER KLAUS-HELMUT DR ,  KIRSTEN ROLF DR ,  KLUTH JOACHIM DR ,  GESING ERNST R F DR ,  FINDEISEN KURT PROF DR ,  JANSEN JOHANNES R DR ,  KOENIG KLAUS DR ,  DREWES MARK WILHELM DR ,  RIEBEL HANS-JOCHEM DR ,  DOLLINGER MARKUS DR ,  SANTEL HANS-JOACHIM DR

IPC: A01N47/38 ,  C07D405/12 ,  C07D409/12 ,  A01N41/08 ,  A01N43/653 ,  C07D409/14

Abstract: The invention relates to novel substituted aryl sulphonyl amino (thio) carbonyl triazolin(thi)ones of formula (I) in which Ar is possibly substituted arylene or heteroarylene; Q is oxygen or sulphur; Q is oxygen or sulphur; R is hydrogen, hydroxy, amino, alkylidene amino or a possibly substitued radical from the series alkyl, alkenyl, alkinyl, alkoxy, alkenyloxy, alkylamino, dialkylamino, alkanoylamino, cycloalkyl, cycloalkyl alkyl, aryl, arylalkyl; R is hydrogen, hydroxy, mercapto, amino, halogen or a possibly substituted radical from the series alkyl, alkenyl, alkinyl, alkoxy, alkenyloxy, alkinyloxy, alkylthio, alkenylthio, alkinylthio, alkylamino, alkenylamino, alkinylamino, dialkylamino, alkanoylamino, aziridino, pyrrolidino, piperidino, morpholino, cycloalkyl, cycloalkenyl, cycloalkoxy, cycloalkylthio, cycloalkylamino, cycloalkyl alkyl, cycloalkyl alkoxy, cycloalkyl alkylthio, cycloalkyl alkylamino, aryl, aryloxy, arylthio, arylamino, arylalkyl, arylalkoxy, arylalkylthio, arylalkylamino, heterocyclyloxy, heterocyclylthio; or R and R together are possibly branched alkandiyl; and R is possibly substituted heterocyclyl; and salts of the compounds of formula (I), process for producing the novel compounds and their use as herbicides.

公开(公告)号：DE19508119A1

公开(公告)日：1996-09-12

申请号：DE19508119

申请日：1995-03-08

Applicant: BAYER AG

Inventor： MUELLER KLAUS-HELMUT DR ,  KIRSTEN ROLF DR ,  GESING ERNST R F DR ,  KLUTH JOACHIM DR ,  FINDEISEN KURT PROF DR ,  JANSEN JOHANNES R DR ,  KOENIG KLAUS DR ,  RIEBEL HANS-JOCHEM DR ,  BIELEFELDT DIETMAR DR ,  DOLLINGER MARKUS DR ,  SANTEL HANS-JOACHIM DR ,  STENZEL KLAUS DR

IPC: A01N47/38 ,  C07D249/12 ,  C07D249/14 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D417/12 ,  C07D401/14 ,  A01N43/653 ,  C07F19/00

Abstract: New sulphonylaminocarbonyltriazolinones have the formula (I), in which R stands for hydrogen, hydroxy, amino, alkylidene amino or for an optionally substituted residue from the series of alkyl, alkenyl, alkinyl, alkylamino, dialkylamino, alkanoylamino, cycloalkyl, cycloalkylalkyl, cycloalkylamino, aryl, arylalkyl; R stands for halogen-substituted alkyl or alkenyl; and R stands for an optionally substituted residue from the series of alkyl, aralkyl, aryl, heteroaryl. Also disclosed are salts of the compounds having the formula (I), a process and new intermediate products for preparing the compounds (I) and their use as herbicides and/or fungicides.

公开(公告)号：ES2054941T3

公开(公告)日：1994-08-16

申请号：ES89113013

申请日：1989-07-15

Applicant: BAYER AG

Inventor： MULLER KLAUS-HELMUT DR ,  KIRSTEN ROLF DR ,  KLUTH JOACHIM DR ,  KONIG KLAUS DR ,  RIEBEL HANS-JOCHEM DR ,  BABCZINSKI PETER DR ,  SANTEL HANS-JOACHIM DR ,  SCHMIDT ROBERT R DR ,  STRANG HARRY DR

IPC: A01N43/64 ,  A01N43/653 ,  A01N43/66 ,  A01N43/707 ,  A01N43/713 ,  C07D401/14 ,  C07D403/00 ,  C07D403/04 ,  C07D403/14 ,  C07D405/14 ,  C07D409/14 ,  C07D417/14 ,  C07D401/04

Abstract: The invention relates to new substituted 4-sulphonylamino-2-azinyl- 1,2,4-triazol-3-ones of the general formula … … (in which R , R , R , R , X, Y and Z have the meanings indicated in the description) and salts of compounds of the formula (I), a process for their preparation, new intermediates for their preparation and their use as herbicides.

公开(公告)号：BR9304117A

公开(公告)日：1994-04-12

申请号：BR9304117

申请日：1993-10-04

Applicant: BAYER AG

Inventor： KIRSTEN ROLF DR ,  SANTEL HANS-JOACHIM DR ,  LUERSSEN KLAUS DR ,  SCHMIDT ROBERT R DR

IPC: A01N43/707 ,  C07D253/07 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D417/12

公开(公告)号：DE4233338A1

公开(公告)日：1994-04-07

申请号：DE4233338

申请日：1992-10-05

Applicant: BAYER AG

Inventor： KIRSTEN ROLF DR ,  SANTEL HANS-JOACHIM DR ,  LUERSSEN KLAUS DR ,  SCHMIDT ROBERT RUDOLF DR

IPC: A01N43/707 ,  C07D253/07 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D417/12 ,  A01N43/80

公开(公告)号：DE4233195A1

公开(公告)日：1994-04-07

申请号：DE4233195

申请日：1992-10-02

Applicant: BAYER AG

Inventor： KIRSTEN ROLF DR ,  MUELLER KLAUS-HELMUTH DR ,  JANSEN JOHANNES R DR

IPC: A01N43/824 ,  C07D271/06 ,  A01N43/82 ,  C07D413/12 ,  C07D417/12

Abstract: Prodn. of N-sulphonyl 1,2,4-oxadiazole-3-carboxamides of formula (I) comprises reacting a 1,2,4-oxadiazole-3-carbonyl chloride of formula (II) with a sulphonamide of formula R1SO2NH2 (III) at 0-100 deg.C, opt. in the presence of an acid binder and/or a diluent: R1 is opt. substd. aryl, aralkyl or heteroaryl; R2 is H or opt. substd. alkyl, alkoxy, alkylthio, alkylsulphinyl, alkylsulphonyl, alkylamino, dialkylamino or phenyl. Also claimed are cpds. (II). The reaction is effected at 10-80 deg.C and 0.1-10 bar using a (III):(II) molar ratio of 0.5-1.5:1, esp. 0.8-1.2:1. USE/ADVANTAGE - (I) are useful as herbicides (see EP459244). The process gives higher yields (e.g. 75-79%) than processes involving reaction of carboxamides with sulphonyl chlorides or of carboxylate esters with sulphonamides (cf. EP459244).