-
公开(公告)号:BR9710897A
公开(公告)日:1999-08-17
申请号:BR9710897
申请日:1997-07-18
Applicant: BAYER AG
Inventor: HEIL MARKUS DR , BRETSCHNEIDER THOMAS DR , KLEEFELD GERD DR , ERDELEN CHRISTOPH DR
IPC: A01N43/90 , A61K31/429 , A61K31/4365 , A61P33/14 , C07D513/04
Abstract: New N-isothiazolyl-(thio)amides have the formula (I), in which Q stands for the grouping (a), in which Het stands for an optionally substituted heterocycle, and R, X, Y and A have the meanings given in the description. Also disclosed are several processes for preparing the same and their use for controlling animal pests.
-
公开(公告)号:DE19800400A1
公开(公告)日:1999-07-15
申请号:DE19800400
申请日:1998-01-08
Applicant: BAYER AG
Inventor: WAGNER KLAUS DR , ERDELEN CHRISTOPH DR , ANDERSCH WOLFRAM DR , WACHENDORFF-NEUMANN ULRIKE DR , TURBERG ANDREAS DR , MENCKE NORBERT DR
IPC: A01N43/50 , A01N43/78 , A01N47/40 , A01N51/00 , C07D401/06 , C07D417/06 , A61K31/41
Abstract: The present invention relates to novel guanidine derivatives of formula (1), wherein R represents a five or six membered heterocyclic group containing 1, 2, 3 or 4 nitrogen atoms and/or one or two oxygen or sulphur atoms as heteroatom ring members, whereby the number of heteroatoms is 1, 2, 3 or 4 and is optionally substituted by halogen, cyano, nitro, alkyl, halogen alkane, alkenyl, halogen alkenyl, alkinyl, alkoxy, halogen alkoxy, alkenyloxy, halogen alkenyloxy, alkinyloxy, alkylthio, halogen alkanethio, alkenylthio, halogen alkenylthio, alkinylthio, alkylsulphinyl, halogen alkanesulphinyl, alkylsulphonyl, amino, alkylamino, dialkylamino, aryl, arylthio, arylamino, aralkyl, formylamino, alkylcarbonylamino, formyl, carbamoyl, alkylcarbonyl and or alkoxycarbonyl, R represents hydrogen or alkyl, R represents groups -OCR , -OCOR , OCOOR , OCONR R and -OSO R , whereby R and R represent independently of each other alkyl, alkoxyalkyl, halogen alkane, alkenyl, alkinyl, alkylaminoalkyl, dialkylaminoalkyl, optionally substituted cycloalkyl and optionally substituted phenyl or benzyl, R and R represent independently of each other hydrogen, alkyl, alkenyl and optionally substituted phenyl or benzyl and R represents alkyl or optionally substituted pheyl, A represents groups -CH2CH2-, (CH2)3 and -CH=CH- and Z represents cyano or nitro, with the proviso that when Z represents NO2 and A represents -CH2CH2, the radical R represents hydrogen and the compound of formula (1), wherein R corresponds to formula (II), R = H, R = OCH3, A = -CH2CH2- and Z = NO2, is excluded.
-
公开(公告)号:BR9611475A
公开(公告)日:1999-07-13
申请号:BR9611475
申请日:1996-11-04
Applicant: BAYER AG
Inventor: HEIL MARKUS DR , ERDELEN CHRISTOPH DR , WACHENDORFF-NEUMANN ULRIKE DR , TURBERG ANDREAS DR , MENCKE NORBERT DR
IPC: C07C327/52 , A01N43/80 , C07C233/91 , C07D275/02 , C07D275/03
Abstract: PCT No. PCT/EP96/04796 Sec. 371 Date May 11, 1998 Sec. 102(e) Date May 11, 1998 PCT Filed Nov. 4, 1996 PCT Pub. No. WO97/18198 PCT Pub. Date May 22, 1997The present invention relates to novel acylated 5-aminoisothiazoles of the formula (I) in which R1, R2, R3, R4 and Y have the meaning given in the description, processes for their preparation and their use for controlling animal pests.
-
公开(公告)号:DE19750402A1
公开(公告)日:1999-05-20
申请号:DE19750402
申请日:1997-11-14
Applicant: BAYER AG
Inventor: BRETSCHNEIDER THOMAS DR , HEIL MARKUS DR , ALIG BERND DR , KLEEFELD GERD DR , ERDELEN CHRISTOPH DR
IPC: A01N47/18 , C07D213/75 , C07D213/89 , C07D213/74 , A01N43/40 , A61K31/44
Abstract: 2-(1-Oxyalkyl)-4-(N-(hydrocarbyloxycarbonyl)-N-(phenylacetyl)-amino)-p yridine derivatives (I) are new. Pyridine derivatives of formula (I) and their N-oxides and pyridine N-protonated salts are new. Several classes of intermediates are also new. R1 = COY1, COOY2, COSY3, CONH2, CONHY4, CONY5Y6 or SO2Y7; Y1-Y7 = alkyl, haloalkyl, optionally substituted cycloalkyl or optionally substituted phenyl; R2 = H or alkyl; R3 = H, alkyl, halo, CN, CSNH2 or optionally substituted phenyl; R5 = phenyl (optionally substituted, e.g. by 1-4 of halo, alkyl, alkoxy, haloalkyl, haloalkoxy, NO2, CN, CSNH2, alkylthio, alkylsulfinyl and alkylsulfonyl); X = halo, alkyl, alkoxy or haloalkyl; n = 0-3. Independent claims are included for the preparation of (I); and for novel intermediates of formulae (II), (IV), (VI), (IV') and (VI'), including analogues of (II) and (IV) in which R1 is replaced by H.
-
公开(公告)号:DE59309357D1
公开(公告)日:1999-03-18
申请号:DE59309357
申请日:1993-08-30
Applicant: BAYER AG
Inventor: FISCHER REINER DR , KREBS ANDREAS DR , LIEB FOLKER DR , RUTHER MICHAEL DR , STETTER JOERG DR , ERDELEN CHRISTOPH DR , WACHENDORFF-NEUMANN ULRIKE , LUERSSEN KLAUS DR , SANTEL HANS-JOACHIM DR , SCHMIDT ROBERT R DR
IPC: A01N43/16 , A01N43/40 , A01N43/90 , A01N47/06 , A01N57/24 , A61K31/35 , A61K31/351 , A61K31/365 , A61K31/44 , A61K31/443 , A61K31/4433 , A61P33/00 , C07D309/36 , C07D309/38 , C07D311/74 , C07D311/94 , C07D405/04 , C07D405/06 , C07D407/04 , C07D407/06 , C07D407/12 , C07D409/04 , C07D413/06 , C07D493/04 , C07D495/04 , C07F9/655
Abstract: The invention relates to 3-arylpyrone derivatives of the general formula (I) in which A represents hydrogen, halogen, optionally substituted radicals from the series comprising alkyl, cycloalkyl, alkenyl, alkynyl, arylalkyl, aryl, hetarylalkyl and hetaryl, or the groups -COR , -COR2R , -CN, -CONR R , -SO2R and -P(O)(OR )(OR ) in which R and R independently of one another represent hydrogen or optionally substituted radicals from the series comprising alkyl, alkenyl, arylalkyl, aryl, hetarylalkyl and hetaryl or R and R together represent an optionally substituted alkylene group which can be interrupted by one or more hetero atoms; B represents hydrogen or optionally substituted radicals from the series comprising alkyl, cycloalkyl, alkenyl, alkynyl, arylalkyl, aryl, hetarylalkyl and hetaryl; A and B together form an optionally substituted alkylene or alkenylene group which can be interrupted by, or contain, one or more hetero atoms or hetero groups; X represents halogen, alkyl or alkoxy; Y represents hydrogen, halogen, alkyl, haloalkyl or alkoxy; Z represents hydrogen, halogen, alkyl or alkoxy; n represents an integer 1, 2 or 3; and G represents hydrogen, a metal ion equivalent and an ammonium ion or a group -COR -SO2-R and -CONR R , in which R represents optionally substituted radicals from the series comprising alkyl, alkenyl, alkoxyalkyl, polyalkoxyalkyl, alkylthioalkyl, or cycloalkyl, arylalkyl, aryl, hetarylalkyl, hetaryl, aryloxyalkyl and hetaryloxyalkyl, it being possible for each of the seven last-mentioned radicals to be interrupted by one or more hetero atoms; R represents optionally substituted radicals from the series comprising alkyl, alkenyl, alkoxyalkyl, polyalkoxyalkyl, aryl and arylalkyl; R , R and R independently of one another represent optionally substituted radicals from the series comprising alkyl, alkoxy, alkylthio, alkylamino, dialkylamino, alkenylthio, alkynylthio, cycloalkylthio, aryl, aryloxy and arylthio; R and R independently of one another represent hydrogen or optionally substituted radicals from the series comprising alkyl, alkenyl, alkoxy, cycloalkyl, alkoxyalkyl, aryl or arylalkyl, or together form an optionally substituted alkylene group which can be interrupted by one or more hetero atoms or hetero groups; L represents oxygen or sulphur; and M represents oxygen or sulphur, which can be used as pesticides.t
-
公开(公告)号:DE59504876D1
公开(公告)日:1999-03-04
申请号:DE59504876
申请日:1995-08-04
Applicant: BAYER AG , YASHIMA KAGAKU KOGYO KK
Inventor: LANTZSCH REINHARD DR , MARHOLD ALBRECHT DR , KRAEMER WOLFGANG DR , ERDELEN CHRISTOPH DR , WACHENDORFF-NEUMANN ULRIKE DR , TURBERG ANDREAS DR , MENCKE NORBERT DR
IPC: A01N43/76 , C07C43/205 , C07C43/225 , C07C45/46 , C07C45/63 , C07C45/64 , C07C45/71 , C07C49/84 , C07C217/64 , C07C233/67 , C07C233/73 , C07C233/87 , C07C251/44 , C07C251/48 , C07D263/14
-
公开(公告)号:DE19715017A1
公开(公告)日:1998-10-15
申请号:DE19715017
申请日:1997-04-11
Applicant: BAYER AG
Inventor: ANDREE ROLAND DR , DOLLINGER MARKUS DR , ERDELEN CHRISTOPH DR
IPC: A01N43/54 , A01N43/76 , A01N43/78 , A01N43/80 , A01N43/836 , C07D401/12 , C07D403/12 , C07D405/12 , C07D413/12 , C07D417/12
Abstract: The invention relates to novel substituted aryluracils of general formula (I), wherein n stands for 0, 1, 2 or 3; Q stands for O, S, SO, or SO2; R stands for hydrogen, amino or optionally substituted alkyl; R stands for carboxy, cyano, carbamoyl, thiocarbamoyl or for respectively optionally substituted alkyl or alkoxycarbonyl; R stands for hydrogen, halogen or optionally substituted alkyl; Y stands for nitro, amino, hydroxy, carboxy, cyano, carbamoyl, thiocarbamoyl, sulfo, chlorosulfonyl, aminosulfonyl, halogen, or for respectively optionally substituted alkyl, alkoxy, alkylthio, alkylsulfinyl, alkylsulfonyl, alkylamino, alkylcarbonyl, alkoxycarbonyl, alkylaminocarbonyl, alkylcarbonylamino, alkoxycarbonylamino or alkylsulfonylamino and Z stands for optionally substituted heterocyclyl from the series of furyl, tetrahydrofuryl, benzofuryl, dihydrobensofuryl, dioxolanyl, dioxanyl, benzodioxanyl, pyrrolyl, pyrazolyl, imidazolyl, triazolyl, oxazolyl, isoxazolyl, benzoxazolyl, pyridinyl, chinolinyl, isochinolinyl, pyrimidinyl, pyrazinyl, pyradazinyl, chinazolinyl, chinoxalinyl, or for respectively substituted thiazolyl, isothiazolyl, benzothiazolyl or benzimidazolyl. The invention also relates to methods for the production and use thereof as phytosanitary products.
-
公开(公告)号:DE19651686A1
公开(公告)日:1998-06-18
申请号:DE19651686
申请日:1996-12-12
Applicant: BAYER AG
Inventor: HAGEMANN HERMANN DR , FISCHER REINER DR , BRETSCHNEIDER THOMAS DR , ERDELEN CHRISTOPH DR , WACHENDORFF-NEUMANN ULRIKE DR , DAHMEN PETER DR , DOLLINGER MARKUS DR , GRAFF ALAN DR , ANDERSCH WOLFRAM DR
IPC: A01N43/90 , A01N47/06 , C07D309/08 , C07D309/10 , C07D309/14 , C07D405/12 , C07D491/10 , C07D491/107 , C07D493/10 , C07D495/10 , C07F9/6561
Abstract: This invention concerns new phenyl-substituted cyclic ketoenols of formula (I) in which Het stand for one of the groups (1), (2) or (3), and G, V, W, Y, and Z have the meaning given in the description, processes and intermediate products for their production and their us as pesticides and herbicides.
-
公开(公告)号:DE19648011A1
公开(公告)日:1998-05-28
申请号:DE19648011
申请日:1996-11-20
Applicant: BAYER AG
Inventor: PLANT ANDREW DR , KLEEFELD GERD DR , POETTER THORSTEN DR , ERDELEN CHRISTOPH DR , MENCKE NORBERT DR , TURBERG ANDREAS DR , WACHENDORFF-NEUMANN ULRIKE DR
IPC: C12N15/09 , A01N43/34 , A01N43/36 , A61K38/00 , A61P31/12 , A61P31/14 , C07C205/04 , C07C205/45 , C07C271/18 , C07D207/12 , C07D207/20 , C07D211/70 , C07D223/04 , C07D227/04 , C07D405/10 , C07D407/10 , C07D409/10 , C07K7/06 , C07D207/26
Abstract: The invention relates to novel cyclic imines of formula (I) wherein Ar , Ar mean in each case substituted phenyl and n is 1,2 or 3; several methods for the production and the use thereof as pesticides.
-
公开(公告)号:AU688401B2
公开(公告)日:1998-03-12
申请号:AU8043894
申请日:1994-12-14
Applicant: BAYER AG
Inventor: STETTER JORG DR , MENCKE NORBERT DR , TURBERG ANDREAS DR , WACHENDORFF ULRIKE DR , HARTWIG JURGEN DR , ERDELEN CHRISTOPH DR , OOMS PIETER DR , BERTSCH ACHIM DR , BOHM STEFAN DR , ALIG BERND DR
IPC: C07D231/46 , A01N43/36 , A01N43/40 , A01N43/56 , A01P7/04 , C07C255/30 , C07D231/18 , C07D231/38 , C07D231/44 , C07D401/04 , C07D403/04 , C07C255/26
Abstract: 1-(Phenyl or pyridyl)-4-(trifluoroethylthio, -sulfinyl or -sulfonyl)-pyrazole derivatives (I) are new. Pyrazole derivatives of formula (I) are new. R1 = H, CN, 1-6C alkyl, (1-4C) alkoxy-(1-4C) alkyl, 1-4C haloalkyl or cyano-(1-2C) alkyl; R2 = trifluoroethyl; R3 = H, NH2, halo, -NHCOR4, -N=C(R5)-NR5R6, 1H-pyrrol-1-yl, -N=CR5R6 or -N=C(R5)-OR7; R4 = 1-6C alkyl (optionally substituted by 1-3 halo), (1-6C) alkoxy-(1-6C) alkyl or phenyl (optionally mono-, di- or trisubstituted); R5 = H or 1-6C alkyl; R6 = H, 1-6C alkyl or phenyl (optionally mono-, di- or trisubstituted); or CR5R6 = optionally substituted pyridyl; R7 = 1-6C alkyl; Ar = phenyl or pyridyl (both optionally substituted by 1-3 of halo, 1-6C haloalkyl, 1-6C haloalkylthio, 1-6C haloalkoxy, alkoxy, hydrazino, di-(1-6C alkyl)-hydrazino, NH2, 1-6C mono- or diaminoalkyl, 1-6C iminoalkyl, CN, 1-6C alkylthio or -CONR9R10); R9, R10 = H or alkyl; and n = 0-2. AN Independent claim is also included for the preparation of (I).
-
-
-
-
-
-
-
-
-