公开(公告)号：DE4029648A1

公开(公告)日：1992-03-26

申请号：DE4029648

申请日：1990-09-19

Applicant: HOECHST AG

Inventor： MINN KLEMENS DR ,  BRAUN PETER DR ,  SACHSE BURKHARD DR ,  WICKE HEINRICH DR

IPC: A01N43/54 ,  C07D239/46 ,  C07D401/12 ,  C07D405/12 ,  C07D409/12 ,  C07D491/048

Abstract: Compounds have the formula (I), in which R , R represent independently from each other hydrogen or (C1-C4)alkyl; R and R if necessary form together a saturated or partially unsaturated carbocyclic or heterocyclic moiety with the heteroatoms O, N or S and 5 or 6 cyclic members; R represents hydrogen or halogen; R , R , R represent independently from each other hydrogen, halogen, (C1-C4)alkyl, (C1-C4)alkoxy or phenoxy eventually substituted in the phenyl moiety by halogen, (C1-C4)alkyl or (C1-C4)alkoxy; R , R and R form together a saturated, partially insaturated or aromatic carbocyclic or heterocyclic moiety with the heteroatoms O, N or S and 5 to 7 cyclic members; R is hydrogen or (C1-C4)alkyl; R is hydrogen, (C1-C4)alkyl, (C1-C4)alkoxy, phenyl-(C1-C4)alkoxy or halogen; R is hydrogen, (C1-C4)alkyl, perhalo-(C1-C4)alkyl, (C1-C4)alkoxy-(C1-C4)alkyl or phenyl-(C1-C4)alkyl; R and R if necessary form together a saturated or partially unsaturated carbocycle or heterocycle with the heteroatoms O, N or S and 5 to 6 cyclic members; X is oxygen or sulphur and n equals 0 or 1. These compounds have advantageous pesticide properties, in particular against fungus pests. A process for producing compounds having formula (I) is also disclosed.

公开(公告)号：DE4029654A1

公开(公告)日：1992-04-02

申请号：DE4029654

申请日：1990-09-19

Applicant: HOECHST AG

Inventor： MINN KLEMENS DR ,  BRAUN PETER DR ,  SACHSE BURKHARD DR ,  WICKE HEINRICH DR

IPC: A01N43/54 ,  A01N43/90 ,  C07D239/28 ,  C07D401/12 ,  C07D495/04

Abstract: Compounds have formula (I), in which R , R , R represent independently from each other hydrogen, chlorine, bromine, nitro or (C1-C4)alkoxy; R represents hydrogen, iodine, bromine, (C1-C4)alkyl, dialkylamino-(C1-C4)alkyl, phenyl-(C1-C4)alkyl(C1-C4)alkylamino-(C1-C4)alkyl, phenyl or pyridinyl eventually substituted in the phenyl (heteroaromatic) moiety by halogen, (C1-C4)alkyl, (C1-C4)alkoxy or perhalo-(C1-C4)alkyl; R represents halogen, (C1-C4)alkyl, (C1-C4)alkoxy, phenyl-(C1-C4)alkoxy, (C1-C4)alkinyloxy, (C1-C4)alkylmercapto or (C1-C4)alkylsulfonyl; R represents hydrogen, (C1-C4)alkyl, (C1-C4)alkoxy-(C1-C4)alkyl or (C1-C4)alkoxy-carbonyl; R and R if necessary form together a saturated or insaturated ring moiety with 5 or 6 members, in which a carbon can be substituted by an S; X represents C=O or NH; Y represents O or NH when X represents C=O; Y is absent when X represents O or NH; and n is a number from 0 to 2. These compounds have advantageous pesticide properties, in particular against fungus pests. A process for producing compounds having formula (I) is also disclosed.

公开(公告)号：DE4029650A1

公开(公告)日：1992-03-26

申请号：DE4029650

申请日：1990-09-19

Applicant: HOECHST AG

Inventor： MINN KLEMENS DR ,  BRAUN PETER DR ,  SACHSE BURKHARD DR ,  WICKE HEINRICH DR

IPC: A01N43/54 ,  A01N43/90 ,  C07D239/46 ,  C07D239/48 ,  C07D239/52 ,  C07D239/70 ,  C07D239/95 ,  C07D403/04 ,  C07D403/14 ,  C07D491/048 ,  C07D495/04

Abstract: 2-arylaminopyrimidine derivs. of formula (I) are new: R1 = H, halogen, R, alkoxy, alkylamino, dialkylamino or cycloalkylamino; R = alkyl, hydroxyalkyl, dihydroxyalkyl, cyanoalkyl, haloalkyl, alkoxyalkyl, haloalkoxyalkyl, alkylthio, haloalkylthio, haloalkylthioalkyl, alkylthioalkyl, alkenyl, alkynyl, (di)alkylaminoalkyl, cycloalkylaminoalkyl, cycloalkyl, cycloalkylalkyl, heterocycloalkylalkyl, (di)alkylcarbamoylalkyl, alkanoyl, haloalkanoyl, alkoxycarbonyl, haloalkoxycarbonyl, alkylthiocarbonyl, haloalkylthiocarbonyl, CONH2, (di)alkylcarbamoyl, haloalkylcarbamoyl, alkoxycarbonylalkyl or opt. substd. phenyl, phenylalkyl, benzoylalkyl, phenoxy, phenoxyalkyl, phenylthioalkyl, phenoxycarbonylalkyl, anilinoalkyl or phenoxyphenylalkyl; R2 = H, CHO or R; R3-R5 = H, halogen, OH, NH2, NO2, CN, SCN, alkoxy, R, (di)alkylamino or alkanoylamino; R6 and R7 = H or R; R8 = H, halogen or R; R9 = halogen, alkoxy, R, (di)alkylamino or cycloalkylamino; X = O, S, NH or alkylimino; n = 0-8; or R1+R9, R3+R4, R3+R5, R2+R3, R2+R4 and/or R6+R7 form a 4- to 10-membered ring opt. contg. O, N, S, Si or P. USE - (I) are fungicides useful for plant protection and for technical purposes, e.g. as wood preservatives or preservatives for paints or metal working fluids. They are active, e.g., against Pseudocercosporella herpotrichoides on wheat.