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公开(公告)号:EP0789688A4
公开(公告)日:1997-11-19
申请号:EP96930691
申请日:1996-08-30
Applicant: LILLY CO ELI
Inventor: BRITTON THOMAS C , BRUNS ROBERT F JR , GEHLERT DONALD R , HIPSKIND PHILIP A , LOBB KAREN L , NIXON JAMES A , ORNSTEIN PAUL L , SMITH EDWARD C R , ZARRINMAYEH HAMIDEH , ZIMMERMAN DENNIS M
IPC: C07D209/12 , C07D209/14 , C07D209/16 , C07D209/24 , C07D209/42 , C07D401/04 , C07D401/06 , C07D401/12 , C07D401/14 , C07D403/06 , C07D403/12 , C07D417/12 , C07D453/02 , C07D209/04 , A61K31/34
CPC classification number: C07D401/04 , C07D209/12 , C07D209/14 , C07D209/16 , C07D209/24 , C07D209/42 , C07D401/06 , C07D401/12 , C07D401/14 , C07D403/06 , C07D403/12 , C07D417/12 , C07D453/02
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2.2-ACYLAMINOPROPANAMIDES AS TACHYKININ RECEPTOR ANTAGONISTS 失效
Title translation: 2- ACYLAMINOPROPANAMIDE作为速激肽受体拮抗剂公开(公告)号:EP0819005A4
公开(公告)日:2001-03-21
申请号:EP96911557
申请日:1996-04-03
Applicant: LILLY CO ELI
Inventor: CHO SUNG-YONG S , HIPSKIND PHILIP A , HOWBERT JAMES JEFFRY , MUEHL BRIAN S , NIXON JAMES A
IPC: A61K38/00 , A61P25/04 , C07K5/06 , C07K5/062 , C07K5/08 , C07K5/097 , A61K31/495 , A61K31/445 , C07D209/08 , C07D401/04 , C07D401/12 , C07D403/04 , C07D403/12
CPC classification number: C07K5/0821 , A61K38/00 , C07K5/06026 , C07K5/06191 , C07K5/0827
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公开(公告)号:HU9701714A2
公开(公告)日:1999-06-28
申请号:HU9701714
申请日:1996-08-30
Applicant: LILLY CO ELI
Inventor: BRITTON THOMAS C , BRUNS ROBERT F , GEHLERT DONALD R , HIPSKIND PHILIP A , LOBB KAREN L , NIXON JAMES A , ORNSTEIN PAUL L , SMITH EDWARD C R , ZARRINMAYEH HAMIDEH , ZIMMERMAN DENNIS M
IPC: C07D209/12 , C07D209/14 , C07D209/16 , C07D209/24 , C07D209/42 , C07D401/04 , C07D401/06 , C07D401/12 , C07D401/14 , C07D403/06 , C07D403/12 , C07D417/12 , C07D453/02 , C07D209/04 , A61K31/34
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公开(公告)号:AU5440996A
公开(公告)日:1996-10-23
申请号:AU5440996
申请日:1996-04-03
Applicant: LILLY CO ELI
Inventor: CHO SUNG-YONG S , HIPSKIND PHILIP A , HOWBERT JAMES JEFFRY , MUEHL BRIAN S , NIXON JAMES A
IPC: A61K38/00 , A61P25/04 , C07K5/06 , C07K5/062 , C07K5/08 , C07K5/097 , A61K31/495 , A61K31/445 , C07D401/04 , C07D403/04
Abstract: This invention provides a series of novel substituted propanamides which are useful in the treatment or prevention of a physiological disorder associated with an excess of tachykinins. This invention also provides methods for the treatment of such physiological disorders as well as pharmaceutical formulations which employ these novel compounds.
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公开(公告)号:AU2242197A
公开(公告)日:1997-08-01
申请号:AU2242197
申请日:1997-01-09
Applicant: LILLY CO ELI
Inventor: ARNOLD MACKLIN B , BRITTON THOMAS C , BRUNS ROBERT F , CANTRELL BUDDY E , HAPP ANNE M , HIPSKIND PHILIP A , HOWBERT JAMES J , LOBB KAREN L , NIXON JAMES A , ORNSTEIN PAUL L , SMITH EDWARD C JR , ZARRINMAYEH HAMIDEH , ZIMMERMAN DENNIS M
IPC: A61K31/00 , A61K31/415 , A61K31/4184 , A61K31/4427 , A61K31/445 , A61K31/454 , A61K31/47 , A61K31/472 , A61K31/4725 , A61K31/495 , A61K31/496 , A61K31/505 , A61K31/506 , A61K31/535 , A61K31/5355 , A61K31/5375 , A61K31/5377 , A61P25/04 , C07D235/12 , C07D401/06 , C07D401/12 , C07D401/14 , C07D403/12 , C07D417/14
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公开(公告)号:AU6965096A
公开(公告)日:1997-03-27
申请号:AU6965096
申请日:1996-08-30
Applicant: LILLY CO ELI
Inventor: BRITTON THOMAS C , BRUNS ROBERT F , GEHLERT DONALD R , HIPSKIND PHILIP A , LOBB KAREN L , NIXON JAMES A , ORNSTEIN PAUL L , SMITH EDWARD C R , ZARRINMAYEH HAMIDEH , ZIMMERMAN DENNIS M
IPC: C07D209/12 , C07D209/14 , C07D209/16 , C07D209/24 , C07D209/42 , C07D401/04 , C07D401/06 , C07D401/12 , C07D401/14 , C07D403/06 , C07D403/12 , C07D417/12 , C07D453/02 , C07D209/04 , A61K31/34
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公开(公告)号:PL180866B1
公开(公告)日:2001-04-30
申请号:PL31832795
申请日:1995-06-30
Applicant: LILLY CO ELI
Inventor: CHO SUNG-YONG S , COPP JAMES D , GINAH FRANCIS O , HANSEN GUY J , HIPSKIND PHILIP A , HUFF BRET E , MARTINELLI MICHAEL J , STASZAK MICHAEL A , THARP-TAYLOR ROGER W
IPC: C07D401/14 , A61K31/4427 , A61K31/445 , A61P1/00 , A61P3/08 , A61P9/00 , A61P11/00 , A61P13/02 , A61P15/00 , A61P25/00 , A61P25/02 , A61P25/04 , A61P25/28 , A61P29/00 , A61P37/00 , A61P37/08 , A61P43/00 , C07D401/12
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公开(公告)号:AU717422B2
公开(公告)日:2000-03-23
申请号:AU6965096
申请日:1996-08-30
Applicant: LILLY CO ELI
Inventor: BRITTON THOMAS C , BRUNS ROBERT F JR , GEHLERT DONALD R , HIPSKIND PHILIP A , LOBB KAREN L , NIXON JAMES A , ORNSTEIN PAUL L , SMITH EDWARD C R , ZARRINMAYEH HAMIDEH , ZIMMERMAN DENNIS M
IPC: C07D209/12 , C07D209/14 , C07D209/16 , C07D209/24 , C07D209/42 , C07D401/04 , C07D401/06 , C07D401/12 , C07D401/14 , C07D403/06 , C07D403/12 , C07D417/12 , C07D453/02 , C07D209/04 , A61K31/34
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公开(公告)号:AU6772996A
公开(公告)日:1997-03-12
申请号:AU6772996
申请日:1996-08-14
Applicant: LILLY CO ELI
Inventor: DODGE JEFFREY A , HIPSKIND PHILIP A
IPC: A61K31/454 , A61K31/4545 , A61K31/496 , A61K31/50 , A61K31/445 , A61K31/495 , C07D401/00 , C07D401/04 , C07D401/06 , C07D401/14 , C07D403/00 , C07D403/04 , C07D403/06 , C07D403/14
Abstract: This invention provides a series of substituted propanamides which are useful in the treatment of a physiological condition which may be modulated by an increase in growth hormone. This invention also provides methods for the treatment of such physiological conditions which comprise administering a growth hormone secretagogue as described in the present invention in combination with growth hormone releasing hormone.
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公开(公告)号:AU6724496A
公开(公告)日:1997-03-12
申请号:AU6724496
申请日:1996-08-14
Applicant: LILLY CO ELI
Inventor: DODGE JEFFREY A , HIPSKIND PHILIP A
IPC: A61K31/137 , A61K31/165 , A61K31/166 , A61K31/4045 , A61K31/4439 , A61K31/454 , A61K31/4545 , A61K31/4725 , A61K31/495 , A61K31/496 , A61K31/506 , A61K31/5377 , A61K31/55 , C07D403/12 , A61K31/135 , A61K31/40 , A61K31/44 , A61K31/445 , A61K31/475 , A61K31/505 , A61K31/535 , C07C211/10 , C07C233/76 , C07C233/78 , C07D209/20 , C07D223/04 , C07D295/15 , C07D401/12 , C07D401/14 , C07D409/12 , C07D413/12
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