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公开(公告)号:EP0874625A4
公开(公告)日:2001-03-14
申请号:EP97903904
申请日:1997-01-22
Applicant: LILLY CO ELI
Inventor: HOLLINSHEAD SEAN P , HUFF BRET E , HUGHES PHILIP F , MENDOZA JOSE S , MITCH CHARLES H , STASZAK MICHAEL A , WARD JOHN S , WILSON JOSEPH W
IPC: C07D295/12 , A61K31/00 , A61K31/16 , A61K31/165 , A61K31/18 , A61K31/275 , A61K31/34 , A61K31/38 , A61K31/381 , A61K31/40 , A61K31/44 , A61K31/445 , A61K31/4453 , A61P25/18 , A61P43/00 , C07B61/00 , C07C231/02 , C07C233/41 , C07C233/43 , C07C233/44 , C07C233/62 , C07C233/65 , C07C233/79 , C07C233/80 , C07C235/22 , C07C235/24 , C07C235/54 , C07C235/56 , C07C255/50 , C07C255/57 , C07C257/12 , C07C275/26 , C07C275/28 , C07C275/40 , C07C311/01 , C07C311/20 , C07C311/21 , C07C311/28 , C07C311/29 , C07C311/46 , C07D201/10 , C07D207/06 , C07D209/40 , C07D211/06 , C07D213/16 , C07D213/81 , C07D213/82 , C07D215/36 , C07D261/18 , C07D295/13 , C07D307/68 , C07D333/10 , C07D333/24 , C07D333/38 , C07D333/40 , C07D333/52 , C07D333/70 , C07D401/02 , C08F8/30 , C08G85/00 , C40B20/02 , C40B30/00 , C40B40/04 , C40B40/14 , C40B50/00 , C40B60/04 , G01N33/15 , G01N33/50 , G01N37/00
CPC classification number: C07D213/82 , C07C257/12 , C07C311/20 , C07C2602/08 , C07C2602/10 , C07D295/13 , C07D333/38 , C07D333/70 , C40B40/00
Abstract: The present invention provides novel indane-like compounds which can be useful for treating psychosis and other conditions associated with the modulation of a muscarinic receptor. The invention provides formulations and methods for using the novel compounds.
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公开(公告)号:EP0971885A4
公开(公告)日:2001-03-07
申请号:EP98902664
申请日:1998-01-21
Applicant: LILLY CO ELI
Inventor: HUFF BRET E , STASZAK MICHAEL A , WARD JOHN S
IPC: C07D295/12 , A61K31/166 , A61K31/40 , A61K31/4453 , A61P13/10 , A61P25/08 , A61P25/16 , A61P25/18 , A61P25/22 , A61P25/28 , A61P27/06 , A61P43/00 , C07B61/00 , C07C209/36 , C07C211/60 , C07C215/70 , C07C219/32 , C07C257/12 , C07C257/14 , C07C271/24 , C07C317/24 , C07C317/28 , C07D213/82 , C07D215/48 , C07D295/195 , C07D333/24 , C07D333/38 , C07D333/70 , C07C257/00 , C07C211/00 , C07C237/00 , C07C239/00 , C07C249/00 , C07C251/00 , C07C263/00 , C07C267/00
CPC classification number: C07D213/82 , C07C257/12 , C07C271/24 , C07C2601/08 , C07C2601/14 , C07C2602/08 , C07D215/48 , C07D295/195 , C07D333/24 , C07D333/38 , C07D333/70 , C40B40/00
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公开(公告)号:EP0817797A4
公开(公告)日:2000-12-06
申请号:EP96909713
申请日:1996-03-14
Applicant: LILLY CO ELI
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公开(公告)号:PT874625E
公开(公告)日:2005-07-29
申请号:PT97903904
申请日:1997-01-22
Applicant: LILLY CO ELI
Inventor: WARD JOHN S , MITCH CHARLES H , HOLLINSHEAD SEAN P , HUFF BRET E , HUGHES PHILIP F , MENDOZA JOSE S , STASZAK MICHAEL A , WILSON JOSEPH W
IPC: A61K31/00 , A61K31/16 , A61K31/165 , A61K31/18 , A61K31/275 , A61K31/34 , A61K31/38 , A61K31/381 , A61K31/40 , A61K31/44 , A61K31/445 , A61K31/4453 , A61P25/18 , A61P43/00 , C07B61/00 , C07C231/02 , C07D295/12 , C07C233/41 , C07C233/43 , C07C233/44 , C07C233/62 , C07C233/65 , C07C233/79 , C07C233/80 , C07C235/22 , C07C235/24 , C07C235/54 , C07C235/56 , C07C255/50 , C07C255/57 , C07C257/12 , C07C275/26 , C07C275/28 , C07C275/40 , C07C311/01 , C07C311/20 , C07C311/21 , C07C311/28 , C07C311/29 , C07C311/46 , C07D201/10 , C07D207/06 , C07D209/40 , C07D211/06 , C07D213/16 , C07D213/81 , C07D213/82 , C07D215/36 , C07D261/18 , C07D295/13 , C07D307/68 , C07D333/10 , C07D333/24 , C07D333/38 , C07D333/40 , C07D333/52 , C07D333/70 , C07D401/02 , C08F8/30 , C08G85/00 , C40B20/02 , C40B30/00 , C40B40/04 , C40B40/14 , C40B50/00 , C40B60/04 , G01N33/15 , G01N33/50 , G01N37/00
Abstract: The present invention provides novel indane-like compounds which can be useful for treating psychosis and other conditions associated with the modulation of a muscarinic receptor. The invention provides formulations and methods for using the novel compounds.
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公开(公告)号:CA2042346A1
公开(公告)日:1991-11-18
申请号:CA2042346
申请日:1991-05-10
Applicant: LILLY CO ELI
Inventor: STASZAK MICHAEL A , STATEN GILBERT S , WEIGEL LELAND O
IPC: C07C215/30 , C07C213/00 , C07D333/20 , C07C213/08
Abstract: X-7392 DOM This invention is directed to a process for preparing chiral l-ary1-3-amino-pxopan-1-ols. These compounds are important intermediates in the synthesis of pharmacologically active compounds.
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公开(公告)号:PL180961B1
公开(公告)日:2001-05-31
申请号:PL30697695
申请日:1995-01-27
Applicant: LILLY CO ELI
Inventor: COOPER ROBIN D G , NICAS THALIA I , RODRIGUEZ MICHAEL J , SNYDER NANCY J , THOMPSON RICHARD C , ZWEIFEL MARK J , HUFF BRET E , QUATROCHE JOHN T , STASZAK MICHAEL A , WILKIE STEPHEN C
Abstract: A new glycopeptide molecule is inserted into the antibiotic group and both components are mixed with a standard pharmaceutical carrier.
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公开(公告)号:AU1834997A
公开(公告)日:1997-08-11
申请号:AU1834997
申请日:1997-01-22
Applicant: LILLY CO ELI
Inventor: HOLLINSHEAD SEAN P , HUFF BRET E , HUGHES PHILIP F , MENDOZA JOSE S , MITCH CHARLES H , STASZAK MICHAEL A , WARD JOHN S , WILSON JOSEPH W
IPC: C07D295/12 , A61K31/00 , A61K31/16 , A61K31/165 , A61K31/18 , A61K31/275 , A61K31/34 , A61K31/38 , A61K31/381 , A61K31/40 , A61K31/44 , A61K31/445 , A61K31/4453 , A61P25/18 , A61P43/00 , C07B61/00 , C07C231/02 , C07C233/41 , C07C233/43 , C07C233/44 , C07C233/62 , C07C233/65 , C07C233/79 , C07C233/80 , C07C235/22 , C07C235/24 , C07C235/54 , C07C235/56 , C07C255/50 , C07C255/57 , C07C257/12 , C07C275/26 , C07C275/28 , C07C275/40 , C07C311/01 , C07C311/20 , C07C311/21 , C07C311/28 , C07C311/29 , C07C311/46 , C07D201/10 , C07D207/06 , C07D209/40 , C07D211/06 , C07D213/16 , C07D213/81 , C07D213/82 , C07D215/36 , C07D261/18 , C07D295/13 , C07D307/68 , C07D333/10 , C07D333/24 , C07D333/38 , C07D333/40 , C07D333/52 , C07D333/70 , C07D401/02 , C08F8/30 , C08G85/00 , C40B20/02 , C40B30/00 , C40B40/04 , C40B40/14 , C40B50/00 , C40B60/04 , G01N33/15 , G01N33/50 , G01N37/00
Abstract: The present invention provides novel indane-like compounds which can be useful for treating psychosis and other conditions associated with the modulation of a muscarinic receptor. The invention provides formulations and methods for using the novel compounds.
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公开(公告)号:DK0817797T3
公开(公告)日:2007-05-07
申请号:DK96909713
申请日:1996-03-14
Applicant: LILLY CO ELI
Inventor: COOPER ROBIN D G , HUFF BRET E , NICAS THALIA I , RODRIGUEZ MICHAEL J , ZWEIFEL MARK J , STASZAK MICHAEL A , WILKIE STEPHEN C , QUATROCHE JOHN T , SNYDER NANCY J , THOMPSON RICHARD C
Abstract: The present invention provides glycopeptide antibiotic derivative compounds. These derivative compounds possess antibacterial activity against a wide variety of bacteria, including activity against vancomycin-resistant isolates. Methods of making and using these glycopeptide antibiotic derivative compounds are also provided.
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公开(公告)号:AT349464T
公开(公告)日:2007-01-15
申请号:AT96909713
申请日:1996-03-14
Applicant: LILLY CO ELI
Inventor: COOPER ROBIN D G , HUFF BRET E , NICAS THALIA I , QUATROCHE JOHN T , RODRIGUEZ MICHAEL J , SNYDER NANCY J , STASZAK MICHAEL A , THOMPSON RICHARD C , WILKIE STEPHEN C , ZWEIFEL MARK J
Abstract: The present invention provides glycopeptide antibiotic derivative compounds. These derivative compounds possess antibacterial activity against a wide variety of bacteria, including activity against vancomycin-resistant isolates. Methods of making and using these glycopeptide antibiotic derivative compounds are also provided.
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公开(公告)号:AT290859T
公开(公告)日:2005-04-15
申请号:AT97903904
申请日:1997-01-22
Applicant: LILLY CO ELI
Inventor: HOLLINSHEAD SEAN P , HUFF BRET E , HUGHES PHILIP F , MENDOZA JOSE S , MITCH CHARLES H , STASZAK MICHAEL A , WARD JOHN S , WILSON JOSEPH W
IPC: C07D295/12 , A61K31/00 , A61K31/16 , A61K31/165 , A61K31/18 , A61K31/275 , A61K31/34 , A61K31/38 , A61K31/381 , A61K31/40 , A61K31/44 , A61K31/445 , A61K31/4453 , A61P25/18 , A61P43/00 , C07B61/00 , C07C231/02 , C07C233/41 , C07C233/43 , C07C233/44 , C07C233/62 , C07C233/65 , C07C233/79 , C07C233/80 , C07C235/22 , C07C235/24 , C07C235/54 , C07C235/56 , C07C255/50 , C07C255/57 , C07C257/12 , C07C275/26 , C07C275/28 , C07C275/40 , C07C311/01 , C07C311/20 , C07C311/21 , C07C311/28 , C07C311/29 , C07C311/46 , C07D201/10 , C07D207/06 , C07D209/40 , C07D211/06 , C07D213/16 , C07D213/81 , C07D213/82 , C07D215/36 , C07D261/18 , C07D295/13 , C07D307/68 , C07D333/10 , C07D333/24 , C07D333/38 , C07D333/40 , C07D333/52 , C07D333/70 , C07D401/02 , C08F8/30 , C08G85/00 , C40B20/02 , C40B30/00 , C40B40/04 , C40B40/14 , C40B50/00 , C40B60/04 , G01N33/15 , G01N33/50 , G01N37/00
Abstract: The present invention provides novel indane-like compounds which can be useful for treating psychosis and other conditions associated with the modulation of a muscarinic receptor. The invention provides formulations and methods for using the novel compounds.
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