公开(公告)号：EP0936213A1

公开(公告)日：1999-08-18

申请号：EP99300573.5

申请日：1999-01-26

Applicant: ROHM AND HAAS COMPANY

Inventor： Lixin, Zhang ,  Zongcheng, Li ,  Zhinian, Li ,  Hong, Zhang ,  Changling, Liu ,  Bin, Li ,  Shaber, Steven Howard

IPC: C07C251/60 ,  A01N33/24 ,  C07D307/52 ,  C07D213/53 ,  A01N43/08 ,  A01N43/40

CPC classification number: C07D213/53 ,  A01N37/36 ,  A01N37/50 ,  A01N43/40 ,  C07C251/60 ,  C07D307/52

Abstract: Compounds with fungicidal and insecticidal properties having formula
wherein X is N or CH; Y is O, S or NR 6 ;

A is independently hydrogen, halo, cyano, (C 1 -C 12 )alkyl, or (C 1 -C 12 )alkoxy;
R 1 and R 6 is independently hydrogen or (C 1 -C 4 )alkyl;
R 2 is independently hydrogen, (C 1 -C 12 )alkyl, halo(C 1- C 12 )alkyl, (C 3 -C 7 )cycloalkyl, (C 2 -C 8 )alkenyl, halo(C 2 -C 8 )alkenyl, (C 2 -C 8 )alkynyl, halo(C 2 -C 8 )alkynyl, aryl, aralkyl, heterocyclic, or heterocyclic(C 1 -C 4 )alkyl;
R 3 is independently hydrogen or (C 1 -C 4 )alkyl;
R 4 and R 5 is independently hydrogen, (C 1 -C 4 )alkyl, aryl, aralkyl, aryl(C 2 -C 8 )alkenyl, aryl(C 2 -C 8 )alkynyl, heterocyclic, or heterocyclic(C 1 -C 4 )alkyl wherein if one of R 4 and R 5 is hydrogen or (C 1 -C 4 )alkyl than the other of R 4 and R 5 is other than hydrogen or (C 1 -C 4 )alkyl,
   and its enantiomers and stereoisomers and agronomically acceptable salts.

Abstract translation: 具有杀菌和杀虫性质的具有式CHEM的化合物，其中X是N或CH; Y是O，S或NR6; A独立地是氢，卤素，氰基，（C 1 -C 12）烷基或（C 1 -C 12）烷氧基; R1和R6独立地是氢或（C1-C4）烷基; （C 1 -C 12）烷基，（C 3 -C 7）环烷基，（C 2 -C 8）烯基，卤代（C 2 -C 8）烯基，（C 2 -C 8）炔基，卤代 （C 2 -C 8）炔基，芳基，芳烷基，杂环或杂环（C 1 -C 4）烷基; R3独立地为氢或（C1-C4）烷基; R4和R5独立地是氢，（C1-C4）烷基，芳基，芳烷基，芳基（C2-C8）烯基，芳基（C2-C8）炔基，杂环或杂环（C1-C4）烷基，其中如果R4和 R 5是氢或（C 1 -C 4）烷基，而R 4和R 5不是氢或（C 1 -C 4）烷基，其对映异构体和立体异构体和农艺学上可接受的盐。