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公开(公告)号:KR20180054856A
公开(公告)日:2018-05-24
申请号:KR20187012166
申请日:2016-09-30
Applicant: SERVIER LAB , VERNALIS R&D LTD
Inventor: FIUMANA ANDREA , FOLOPPE NICOLAS , RAY STUART , WALMSLEY DAVID , KOTSCHY ANDRAS , BURBRIDGE MICHAEL FRANK , CRUZALEGUI FRANCISCO HUMBERTO
IPC: C07D487/04 , A61K31/437 , A61K31/519 , A61P25/00 , A61P25/16 , A61P25/28 , A61P35/00 , C07D471/04
CPC classification number: C07D471/04 , C07D487/04
Abstract: 암, 신경변성장애및 대사장애의치료에유용한하기화학식 (I)의화합물:(화학식 I)
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公开(公告)号:DK3027602T3
公开(公告)日:2018-09-24
申请号:DK14758604
申请日:2014-07-22
Applicant: SERVIER LAB , VERNALIS R&D LTD
Inventor: HENLIN JEAN-MICHEL , LETIRAN ARNAUD , DE NANTEUIL GUILLAUME , GENESTE OLIVIER , DAVIDSON JAMES EDWARD PAUL , MURRAY JAMES BROOKE , WALMSLEY CLAIRE , CASARA PATRICK , CHEN I-JEN , GRAHAM CHRISTOPHER JOHN , RAY STUART , MADDOX DANIEL , BEDFORD SIMON , LE DIGUARHER THIERRY , STARCK JÉRÔME-BENOÎT
IPC: C07D401/14 , A61K31/4709 , A61P35/00 , A61P37/00 , C07D401/10 , C07D405/14 , C07D471/04
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公开(公告)号:HK1255467A1
公开(公告)日:2019-08-16
申请号:HK18114640
申请日:2018-11-15
Applicant: SERVIER LAB , VERNALIS R&D LTD
Inventor: FIUMANA ANDREA , FOLOPPE NICOLAS , RAY STUART , WALMSLEY DAVID , KOTSCHY ANDRÁS , BURBRIDGE MICHAËL FRANK , CRUZALEGUI FRANCISCO HUMBERTO
IPC: C07D20060101 , A61K20060101 , A61P20060101
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4.
公开(公告)号:LT3027602T
公开(公告)日:2018-07-25
申请号:LT14758604
申请日:2014-07-22
Applicant: SERVIER LAB , VERNALIS R&D LTD
Inventor: CASARA PATRICK , LE DIGUARHER THIERRY , HENLIN JEAN-MICHEL , STARCK JÉRÔME-BENOÎT , LE TIRAN ARNAUD , DE NANTEUIL GUILLAUME , GENESTE OLIVIER , DAVIDSON JAMES EDWARD PAUL , MURRAY JAMES BROOKE , CHEN I-JEN , WALMSLEY CLAIRE , GRAHAM CHRISTOPHER JOHN , RAY STUART , MADDOX DANIEL , BEDFORD SIMON
IPC: C07D401/14 , A61K31/4709 , A61P35/00 , A61P37/00 , C07D401/10 , C07D405/14 , C07D471/04
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公开(公告)号:CO2018003466A2
公开(公告)日:2018-07-10
申请号:CO2018003466
申请日:2018-03-28
Applicant: SERVIER LAB , VERNALIS R&D LTD
Inventor: KOTSCHY ANDRÁS , BURBRIDGE MICHAËL FRANK , FIUMANA ANDREA , FOLOPPE NICOLAS , RAY STUART , WALMSLEY DAVID , CRUZALEGUI FRANCISCO HUMBERTO
IPC: C07D471/04 , A61K31/437 , A61K31/519 , A61P25/16 , A61P25/28 , A61P35/00 , C07D487/04
Abstract: Compuestos de fórmula (I) (Ver imagen adjunta) en la que R1, R2, W3, W4, A1, y A2 son como se definen en la descripción. Medicamentos.
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公开(公告)号:UA117020C2
公开(公告)日:2018-06-11
申请号:UAA201601398
申请日:2014-07-22
Applicant: SERVIER LAB , VERNALIS R&D LTD
Inventor: CASARA PATRICK , LE DIGUARHER THIERRY , HENLIN JEAN-MICHEL , STARCK JEROME-BENOIT , LE TIRAN ARNAUD , DE NANTEUIL GUILLAUME , GENESTE OLIVIER , DAVIDSON JAMES EDWARD PAUL , MURRAY JAMES BROOKE , CHEN I-JEN , WALMSLEY CLAIRE , GRAHAM CHRISTOPHER JOHN , RAY STUART , MADDOX DANIEL , BEDFORD SIMON
IPC: C07D401/14 , A61K31/4709 , A61P35/00 , A61P37/00 , C07D401/10 , C07D405/14 , C07D471/04
Abstract: Сполукаформули (І): ,(I) де Ra, Rb, Rc, Rd, R3, R4, R5, A1, А2, Тта W єтакими, яквизначенов описі. Медикаменти.
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公开(公告)号:CA2917965C
公开(公告)日:2018-03-06
申请号:CA2917965
申请日:2014-07-22
Applicant: SERVIER LAB , VERNALIS R&D LTD
Inventor: CASARA PATRICK , LE DIGUARHER THIERRY , HENLIN JEAN-MICHEL , STARCK JEROME-BENOIT , LE TIRAN ARNAUD , DE NANTEUIL GUILLAUME , GENESTE OLIVIER , DAVIDSON JAMES EDWARD PAUL , MURRAY JAMES BROOKE , CHEN I-JEN , WALMSLEY CLAIRE , GRAHAM CHRISTOPHER JOHN , RAY STUART , MADDOX DANIEL , BEDFORD SIMON
IPC: C07D401/14 , A61K31/4709 , A61P35/00 , A61P37/00 , C07D401/10 , C07D405/14 , C07D471/04
Abstract: Composés de formule (I) dans laquelle R a, R b, R c, R d, R3, R4, R5, A1, A2,T et W sont tels que définis dans la description. Médicaments.
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公开(公告)号:FR3008978A1
公开(公告)日:2015-01-30
申请号:FR1357277
申请日:2013-07-23
Applicant: SERVIER LAB , VERNALIS R & D LTD
Inventor: CASARA PATRICK , LE DIGUARHER THIERRY , HENLIN JEAN-MICHEL , STARCK JEROME-BENOIT , LE TIRAN ARNAUD , DE NANTEUIL GUILLAUME , GENESTE OLIVIER , DAVIDSON JAMES EDWARD PAUL , MURRAY JAMES BROOKE , CHEN I-JEN , WALMSLEY CLAIRE , GRAHAM CHRISTOPHER JOHN , RAY STUART , MADDOX DANIEL , BEDFORD SIMON
IPC: C07D471/04 , A61K31/437 , A61P35/00 , C07D207/30 , C07D209/04 , C07D213/02 , C07D215/14
Abstract: Composés de formule (I) : dans laquelle Ra, Rb, Rc, Rd, R3, R4, R5, A1, A2, T et W sont tels que définis dans la description.
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公开(公告)号:BR112016001333B1
公开(公告)日:2022-03-03
申请号:BR112016001333
申请日:2014-07-22
Applicant: SERVIER LAB , VERNALIS R&D LTD
Inventor: ARNAUD LE TIRAN , CHRISTOPHER JOHN GRAHAM , WALMSLEY CLAIRE , MADDOX DANIEL , GUILLAUME DE NANTEUIL , CHEN I-JEN , JAMES BROOKE MURRAY , JAMES EDWARD PAUL DAVIDSON , HENLIN JEAN-MICHEL , STARCK JÉRÔME-BENOÎT , GENESTE OLIVIER , CASARA PATRICK , BEDFORD SIMON , RAY STUART , THIERRY LE DIGUARHER
IPC: C07D401/10 , A61K31/4709 , A61P35/00 , A61P37/00 , C07D401/14 , C07D405/14 , C07D471/04
Abstract: derivados de indol e pirrol, processos para a produção dos mesmos e composições farmacêuticas contendo os mesmos. (i) a presente invenção refere-se aos compostos de fórmula (i), em que ra, rb, rc, rd, r3, r4, r5, a1, a2, t e w são como definidos na descrição. a invenção também se refere aos fármacos contendo os mesmos.
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公开(公告)号:AU2014294866B2
公开(公告)日:2018-09-27
申请号:AU2014294866
申请日:2014-07-22
Applicant: SERVIER LAB , VERNALIS R&D LTD
Inventor: CASARA PATRICK , LE DIGUARHER THIERRY , HENLIN JEAN-MICHEL , STARCK JEROME-BENOIT , LE TIRAN ARNAUD , DE NANTEUIL GUILLAUME , GENESTE OLIVIER , DAVIDSON JAMES EDWARD PAUL , MURRAY JAMES BROOKE , CHEN I-JEN , WALMSLEY CLAIRE , GRAHAM CHRISTOPHER JOHN , RAY STUART , MADDOX DANIEL , BEDFORD SIMON
IPC: C07D401/14 , A61K31/4709 , A61P35/00 , A61P37/00 , C07D401/10 , C07D405/14 , C07D471/04
Abstract: The invention relates to compounds of formula (I), wherein R
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