公开(公告)号：EP0243971A2

公开(公告)日：1987-11-04

申请号：EP87106296.4

申请日：1987-04-30

Applicant: STAUFFER CHEMICAL COMPANY

Inventor： Baker, Don Robert ,  Brownell, Keith Harvey

IPC: C07D213/82 ,  C07D213/83 ,  A01N53/00

CPC classification number: C07D213/75 ,  A01N53/00

Abstract: Novel fungicidal pyridyl cyclopropane carboxamides having the general structural formula
in which R is selected from the group halogen C 1 -C 3 alkoxy and C 1 -C 3 haloalkoxy, R, is selected from the group of-H and -C≡N; and R 2 is selected from the group of-H, 1-CH 3 ; and 2-CH 3 ; X is O or S; and fungicidally acceptable organic and inorganic salts thereof. These compounds provide excellent control of fungal growth.

Abstract translation: 具有通式结构式的新型杀真菌吡啶基环丙烷甲酰胺，其中R选自卤素C 1 -C 3烷氧基和C 1 -C 3卤代烷氧基，R 1选自-H和-CIDENTICAL N; 并且R 2选自-H，1-CH 3; 和2-CH 3; X为O或S; 和杀真菌可接受的有机和无机盐。 这些化合物提供了真菌生长的极好的控制。

公开(公告)号：EP0243971A3

公开(公告)日：1989-03-29

申请号：EP87106296.4

申请日：1987-04-30

Applicant: STAUFFER CHEMICAL COMPANY

Inventor： Baker, Don Robert ,  Brownell, Keith Harvey

IPC: C07D213/82 ,  C07D213/83 ,  A01N53/00

CPC classification number: C07D213/75 ,  A01N53/00

Abstract: Novel fungicidal pyridyl cyclopropane carboxamides having the general structural formula
in which R is selected from the group halogen C 1 -C 3 alkoxy and C 1 -C 3 haloalkoxy, R, is selected from the group of-H and -C≡N; and R 2 is selected from the group of-H, 1-CH 3 ; and 2-CH 3 ; X is O or S; and fungicidally acceptable organic and inorganic salts thereof. These compounds provide excellent control of fungal growth.

公开(公告)号：EP0243972A2

公开(公告)日：1987-11-04

申请号：EP87106297.2

申请日：1987-04-30

Applicant: STAUFFER CHEMICAL COMPANY

Inventor： Baker, Don Robert ,  Brownell, Keith Harvey ,  Kezerian, Charles

IPC: C07D213/82 ,  C07D405/12 ,  A01N53/00

CPC classification number: C07D213/75 ,  A01N53/00 ,  C07D213/76 ,  C07D405/12 ,  C07F7/10

Abstract: Novel fungicidal pyridyl cyclopropane carboxamides having the general structural formula
wherein Z is
R is selected from the group consisting of cycloalkyl, preferably cyclopropyl, hydrogen, alkyl, haloalkyl, substituted alkyl, aryl, substituted aryl, heteroalkyl, alkenyl, OR 1 , SR, and
wherein n is 0-10, preferably 0-2, ad R 1 is C 1 -C 4 alkyl; R 2 is selected from the group consisting of halogen such as chlorine, fluorine and bromine, preferably chlorine, C 1 -C 3 alkoxy such as propoxy ethoxy and methoxy, preferably methoxy and C 1 -C 3 haloalkoxy; R 3 is selected from the group consisting of hydrogen and methyl; X is oxygen or sulfur and Y is oxygen or sulfur; or Z is SR 9 wherein R 9 is selected from the group consisting of haloalkyl, preferably C 1 -C 3 haloalkyl, C 1 -C 8 alkyl, aryl, substituted aryl, and arylalkyl wherein the preferred aryl is phenyl, the alkyl is C 1 -C 3 alkyl and the preferred substitutions are Cl, Br, F and nitro, alkanoyl, preferably C 1 -C 4 alkanoyl,
wherein R 4 and R 5 can be alkyl, alkanoyl, alkoxycarbonyl, benzyl, pyridyl and substituted pyridyl; provided that when Z is -SR 9 Y is oxygen; and fungicidally acceptable organic and inorganic salts thereof which are highly effective fungicides for use both as preventive and curative fungicides are disclosed herein.

Abstract translation: 具有通式结构式的新型杀真菌吡啶基环丙烷甲酰胺，其中Z为-R; R选自环烷基，优选环丙基，氢，烷基，卤代烷基，取代的烷基，芳基，取代的芳基，杂烷基，烯基，OR 1，SR 1和 - （CH 2）n R OR 1，其中n为0-10， 优选0-2，并且R 1是C 1 -C 4烷基; R 2选自卤素如氯，氟和溴，优选氯，C 1 -C 3烷氧基如丙氧基乙氧基和甲氧基，优选甲氧基和C 1 -C 3卤代烷氧基; R3选自氢和甲基; X是氧或硫，Y是氧或硫; 或Z是SR 9，其中R 9选自卤代烷基，优选C 1 -C 3卤代烷基，C 1 -C 8烷基，芳基，取代的芳基和芳烷基，其中优选的芳基是苯基，所述烷基是C 1 -C 3烷基，优选的 取代基是Cl，Br，F和硝基，烷酰基，优选C 1 -C 4烷酰基，其中R 4和R 5可以是烷基，烷酰基，烷氧基羰基，苄基，吡啶基和取代的吡啶基; 条件是当Z为-SR 9时，Y为氧; 及其杀真菌可接受的有机和无机盐，它们是用作预防和治疗性杀真菌剂的高效杀真菌剂。

公开(公告)号：EP0243971B1

公开(公告)日：1994-08-03

申请号：EP87106296.4

申请日：1987-04-30

Applicant: STAUFFER CHEMICAL COMPANY

Inventor： Baker, Don Robert ,  Brownell, Keith Harvey

IPC: C07D213/82 ,  C07D213/83 ,  A01N53/00

CPC classification number: C07D213/75 ,  A01N53/00

公开(公告)号：EP0243972A3

公开(公告)日：1989-03-22

申请号：EP87106297.2

申请日：1987-04-30

Applicant: STAUFFER CHEMICAL COMPANY

Inventor： Baker, Don Robert ,  Brownell, Keith Harvey ,  Kezerian, Charles

IPC: C07D213/82 ,  C07D405/12 ,  A01N53/00

CPC classification number: C07D213/75 ,  A01N53/00 ,  C07D213/76 ,  C07D405/12 ,  C07F7/10

Abstract: Novel fungicidal pyridyl cyclopropane carboxamides having the general structural formula
wherein Z is
R is selected from the group consisting of cycloalkyl, preferably cyclopropyl, hydrogen, alkyl, haloalkyl, substituted alkyl, aryl, substituted aryl, heteroalkyl, alkenyl, OR 1 , SR, and
wherein n is 0-10, preferably 0-2, ad R 1 is C 1 -C 4 alkyl; R 2 is selected from the group consisting of halogen such as chlorine, fluorine and bromine, preferably chlorine, C 1 -C 3 alkoxy such as propoxy ethoxy and methoxy, preferably methoxy and C 1 -C 3 haloalkoxy; R 3 is selected from the group consisting of hydrogen and methyl; X is oxygen or sulfur and Y is oxygen or sulfur; or Z is SR 9 wherein R 9 is selected from the group consisting of haloalkyl, preferably C 1 -C 3 haloalkyl, C 1 -C 8 alkyl, aryl, substituted aryl, and arylalkyl wherein the preferred aryl is phenyl, the alkyl is C 1 -C 3 alkyl and the preferred substitutions are Cl, Br, F and nitro, alkanoyl, preferably C 1 -C 4 alkanoyl,
wherein R 4 and R 5 can be alkyl, alkanoyl, alkoxycarbonyl, benzyl, pyridyl and substituted pyridyl; provided that when Z is -SR 9 Y is oxygen; and fungicidally acceptable organic and inorganic salts thereof which are highly effective fungicides for use both as preventive and curative fungicides are disclosed herein.

公开(公告)号：EP0243970A1

公开(公告)日：1987-11-04

申请号：EP87106295.6

申请日：1987-04-30

Applicant: STAUFFER CHEMICAL COMPANY

Inventor： Baker, Don Robert ,  Brownell, Keith Harvey

IPC: C07D213/74 ,  C07D405/12 ,  C07F9/58 ,  A01N43/40 ,  A01N57/16

CPC classification number: C07D213/74 ,  A01N53/00 ,  A01N57/16 ,  C07D405/12 ,  C07F9/588

Abstract: Novel fungicidal pyridyl imidates having the general structural formula
wherein R is selected from the group consisting of C 1 -C 16 alkyl, C 3 -C 8 cycloalkyl, C 2 -C 8 alkenyl, C 2 -C 8 substituted alkenyl, C 3 -C 4 carboalkoxyalkyl, aryl, arylalkyl having C 1 -C 3 alkyl, substituted aryl and arylalkyl wherein the substituents are -Cl, -Br, -F and -N0 2 , furfuryl pyridyl, C 1 -C 6 alkyl substituted phosphorus, and
wherein R 3 and R 4 are C 1 -C 10 alkyl and can form a heterocyclic ring, R 1 is selected from the group consisting of halogen, C 1 -C 3 alkoxy and C 1 -C 3 haloalkoxy, R 2 is selected from the group consisting of methyl and hydrogen, and X is S or O; and fungicidally acceptable organic and inorganic salts thereof.

Abstract translation: 具有通式结构式的新型杀真菌吡啶基亚胺化物，其中R选自C1-C16烷基，C3-C8环烷基，C2-C8链烯基，C2-C8取代烯基，C3-C4烷氧羰基烷基，芳基，芳烷基 具有C 1 -C 3烷基，取代的芳基和芳基烷基，其中取代基是-Cl，-Br，-F和-NO 2，糠基吡啶基，C 1 -C 6烷基取代的磷和CHEM，其中R 3和R 4是C 1 -C 10烷基， 可以形成杂环，R 1选自卤素，C 1 -C 3烷氧基和C 1 -C 3卤代烷氧基，R 2选自甲基和氢，X是S或O; 和杀真菌可接受的有机和无机盐。