公开(公告)号：US20150299144A1

公开(公告)日：2015-10-22

申请号：US14691279

申请日：2015-04-20

Applicant: KUREHA CORPORATION

Inventor： Nobuyuki ARAKI ,  Taiji MIYAKE ,  Eiyu IMAI ,  Emiko OBATA

IPC: C07D249/12 ,  C07D405/04

CPC classification number: C07D249/12 ,  A01N43/50 ,  A01N43/653 ,  A01N43/80 ,  C07D233/56 ,  C07D233/60 ,  C07D249/08 ,  C07D405/04 ,  C07D405/06 ,  A01N25/04 ,  A01N25/28

Abstract: Provided is an azole derivative superior in disease-controlling activity contained as an active ingredient in agricultural or horticultural chemical agents.The azole derivative according to the present invention is represented by the following General Formula (I): (in Formula (I), R1 represents an unsubstituted or substituted C1-C6-alkyl group; R2 represents a carbonyl group-containing functional group, wherein the carbon atom in the carbonyl group is bound to the carbon atom in the cyclopentane ring substituted with R1 and to a hydrogen atom, a hydroxyl group, R3, OR3, or NR3R4; R3 and R4 each represent a C1-C6-alkyl group, a C2-C6-alkenyl group, or a C2-C2-alkynyl group; Y represents a halogen atom, a C1-C4-alkyl group, a C1-C4-haloalkyl group, a C1-C4-alkoxy group, a C1-C4-haloalkoxy group, a phenyl group, a cyano group, or a nitro group; m is 0 to 5; and A represents a nitrogen atom or a methine group).

Abstract translation: 提供在农业或园艺化学试剂中作为活性成分含有的疾病控制活性优异的唑衍生物。 根据本发明的唑衍​​生物由以下通式（I）表示：（在式（I）中，R 1表示未取代或取代的C 1 -C 6 - 烷基; R 2表示含羰基的官能团，其中 羰基中的碳原子与被R 1取代的环戊烷环中的碳原子结合，并与氢原子，羟基，R3，OR3或NR3R4结合; R3和R4各自表示C1-C6-烷基， C2-C6-烯基或C2-C2-炔基; Y表示卤素原子，C1-C4-烷基，C1-C4-卤代烷基，C1-C4-烷氧基，C1- C4卤代烷氧基，苯基，氰基或硝基; m为0-5; A表示氮原子或次甲基）。