公开(公告)号：US20230192630A1

公开(公告)日：2023-06-22

申请号：US17905446

申请日：2021-03-05

Applicant: Kureha Corporation

Inventor： Taiga MASANO ,  Tsutomu MUKADE ,  Tomoyuki KOUGE ,  Taiji MIYAKE ,  Junya HIRATA

IPC: C07D249/08 ,  A01N43/653 ,  A01P3/00

CPC classification number: C07D249/08 ,  A01N43/653 ,  A01P3/00

Abstract: Provided is a plant disease controlling agent that has low toxicity to humans and animals, that is excellent in handling safety, and that has an excellent controlling effect against a wide range of plant diseases and a high antimicrobial action against plant disease fungi. The present invention is a compound represented by general formula (I) below, or N-oxide or a pesticidally acceptable salt thereof: [Chem. 1]

公开(公告)号：US20160270398A1

公开(公告)日：2016-09-22

申请号：US15035514

申请日：2014-10-08

Applicant: KUREHA CORPORATION

Inventor： Taiji MIYAKE ,  Nobuyuki ARAKI

IPC: A01N43/653 ,  A01N37/34 ,  A01N47/08 ,  A01N43/56 ,  A01N43/40

CPC classification number: A01N43/653 ,  A01N37/34 ,  A01N43/40 ,  A01N43/50 ,  A01N43/56 ,  A01N47/08 ,  A01N45/02 ,  A01N47/34

Abstract: An agricultural or horticultural chemical according to the present invention is an agricultural or horticultural chemical containing a plurality of active ingredients, the agricultural or horticultural chemical comprises, as one of the active ingredients, an azole derivative represented by general formula (I) below, and can be used as a plant disease controlling agent that can reduce the content of an active ingredient, (In the general formula, R1 represents an alkyl group having from 1 to 6 carbons, R2 represents a hydrogen atom, an alkyl group having from 1 to 3 carbons, an alkenyl group or an alkynyl group having from 2 to 3 carbons, A represents a nitrogen atom or a methine group, Y1 represents a halogen atom, and n represents either 0 or 1).

Abstract translation: （通式中，R 1表示碳原子数1〜6的烷基，R 2表示氢原子，碳原子数1〜3的烷基，烯基或碳原子数2〜3的炔基，A表示 氮原子或次甲基，Y1表示卤素原子，n表示0或1）。

公开(公告)号：US20160295865A1

公开(公告)日：2016-10-13

申请号：US15038574

申请日：2014-10-08

Applicant: Kureha Corporation

Inventor： Taiji MIYAKE ,  Nobuyuki ARAKI

IPC: A01N43/653 ,  A01N43/84

CPC classification number: A01N43/653 ,  A01N43/50 ,  A01N43/84 ,  A01N43/40

Abstract: An agricultural or horticultural chemical according to the present invention is an agricultural or horticultural chemical containing a plurality of active ingredients, the agricultural or horticultural chemical comprises, as one of the active ingredients, an azole derivative represented by general formula (I), and can be used as a plant disease controlling agent that can reduce the content of an active ingredient: wherein, R1 represents an alkyl group having from 1 to 6 carbons, R2 represents a hydrogen atom, an alkyl group having from 1 to 3 carbons, an alkenyl group or an alkynyl group having from 2 to 3 carbons, A represents a nitrogen atom or a methine group, Y1 represents a halogen atom, and n represents either 0 or 1.

Abstract translation: 其中，R1表示碳原子数1〜6的烷基，R2表示氢原子，碳原子数1〜3的烷基，烯基或碳原子数2〜3的炔基，A表示氮原子或 次甲基，Y1表示卤素原子，n表示0或1。

公开(公告)号：US20150299144A1

公开(公告)日：2015-10-22

申请号：US14691279

申请日：2015-04-20

Applicant: KUREHA CORPORATION

Inventor： Nobuyuki ARAKI ,  Taiji MIYAKE ,  Eiyu IMAI ,  Emiko OBATA

IPC: C07D249/12 ,  C07D405/04

CPC classification number: C07D249/12 ,  A01N43/50 ,  A01N43/653 ,  A01N43/80 ,  C07D233/56 ,  C07D233/60 ,  C07D249/08 ,  C07D405/04 ,  C07D405/06 ,  A01N25/04 ,  A01N25/28

Abstract: Provided is an azole derivative superior in disease-controlling activity contained as an active ingredient in agricultural or horticultural chemical agents.The azole derivative according to the present invention is represented by the following General Formula (I): (in Formula (I), R1 represents an unsubstituted or substituted C1-C6-alkyl group; R2 represents a carbonyl group-containing functional group, wherein the carbon atom in the carbonyl group is bound to the carbon atom in the cyclopentane ring substituted with R1 and to a hydrogen atom, a hydroxyl group, R3, OR3, or NR3R4; R3 and R4 each represent a C1-C6-alkyl group, a C2-C6-alkenyl group, or a C2-C2-alkynyl group; Y represents a halogen atom, a C1-C4-alkyl group, a C1-C4-haloalkyl group, a C1-C4-alkoxy group, a C1-C4-haloalkoxy group, a phenyl group, a cyano group, or a nitro group; m is 0 to 5; and A represents a nitrogen atom or a methine group).

Abstract translation: 提供在农业或园艺化学试剂中作为活性成分含有的疾病控制活性优异的唑衍生物。 根据本发明的唑衍​​生物由以下通式（I）表示：（在式（I）中，R 1表示未取代或取代的C 1 -C 6 - 烷基; R 2表示含羰基的官能团，其中 羰基中的碳原子与被R 1取代的环戊烷环中的碳原子结合，并与氢原子，羟基，R3，OR3或NR3R4结合; R3和R4各自表示C1-C6-烷基， C2-C6-烯基或C2-C2-炔基; Y表示卤素原子，C1-C4-烷基，C1-C4-卤代烷基，C1-C4-烷氧基，C1- C4卤代烷氧基，苯基，氰基或硝基; m为0-5; A表示氮原子或次甲基）。

公开(公告)号：US20200288714A1

公开(公告)日：2020-09-17

申请号：US16636502

申请日：2018-11-13

Applicant: Kureha Corporation

Inventor： Ryo HARIGAE ,  Atsushi ITO ,  Taiji MIYAKE ,  Toru YAMAZAKI

IPC: A01N43/653 ,  C07D249/08

Abstract: It is provided a plant disease controlling agent having low toxicity to human and animals and excellent handling safety, and showing excellent controlling effects on various plant diseases and high antibiotic action to plant disease germs.A compound represented by the following the general formula (I), or an N-oxide or agrochemically acceptable salt thereof.

公开(公告)号：US20140213794A1

公开(公告)日：2014-07-31

申请号：US14213240

申请日：2014-03-14

Applicant: KUREHA CORPORATION

Inventor： Nobuyuki ARAKI ,  Toru YAMAZAKI ,  Nobuyuki KUSANO ,  Eiyu IMAI ,  Hisashi KANNO ,  Masaru MORI ,  Taiji MIYAKE

IPC: C07D405/06 ,  C07C201/12 ,  C07C67/31

CPC classification number: C07C67/31 ,  A01N37/10 ,  A01N43/50 ,  A01N43/653 ,  C07C201/12 ,  C07C2601/08 ,  C07D405/06

Abstract: An azole derivative according to the invention is represented by Formula (I), wherein each of Ra and Rb denotes a hydrogen atom, or a C1-C6 alkyl group, a C2-C6 alkenyl group or a C2-C6 alkynyl group; Ra and Rb may be substituted with Xa or Xb which is a halogen atom; each of na and nb denotes 0 or the number of Xa- or Xb-substituted hydrogen atoms among the hydrogen atoms in Ra or Rb; each Y denotes a halogen atom, a C1-C4 alkyl group, a C1-C4 haloalkyl group, a C1-C4 alkoxy group, a C1-C4 haloalkoxy group, a phenyl group, a cyano group or a nitro group; m denotes 0 to 5; and A denotes a nitrogen atom or a methyne group. As a result, an azole derivative contained as an active ingredient in an agro-horticultural agent having an excellent controlling effect on diseases can be provided.

Abstract translation: 根据本发明的唑衍​​生物由式（I）表示，其中R a和R b各自表示氢原子或C 1 -C 6烷基，C 2 -C 6烯基或C 2 -C 6炔基; Ra和Rb可以被Xa或Xb取代，Xb或Xb是卤素原子; na和nb中的每一个表示0或Ra或Rb中的氢原子中的X a或X b取代的氢原子的数目; 每个Y表示卤素原子，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，苯基，氰基或硝基; m表示0〜5; A表示氮原子或甲炔基。 结果，可以提供在对疾病具有优异控制作用的农业园艺剂中作为活性成分含有的唑衍生物。

公开(公告)号：US20140200352A1

公开(公告)日：2014-07-17

申请号：US14213043

申请日：2014-03-14

Applicant: KUREHA CORPORATION

Inventor： Nobuyuki ARAKI ,  Toru YAMAZAKI ,  Nobuyuki KUSANO ,  Eiyu IMAI ,  Hisashi KANNO ,  Masaru MORI ,  Taiji MIYAKE

IPC: A01N43/50 ,  A01N43/653 ,  A01N37/10

CPC classification number: C07C67/31 ,  A01N37/10 ,  A01N43/50 ,  A01N43/653 ,  C07C201/12 ,  C07C2601/08 ,  C07D405/06

Abstract: An azole derivative according to the invention is represented by Formula (I), wherein each of Ra and Rb denotes a hydrogen atom, or a C1-C6 alkyl group, a C2-C6 alkenyl group or a C2-C6 alkynyl group; Ra and Rb may be substituted with Xa or Xb which is a halogen atom; each of na and nb denotes 0 or the number of Xa- or Xb-substituted hydrogen atoms among the hydrogen atoms in Ra or Rb; each Y denotes a halogen atom, a C1-C4 alkyl group, a C1-C4 haloalkyl group, a C1-C4 alkoxy group, a C1-C4 haloalkoxy group, a phenyl group, a cyano group or a nitro group; m denotes 0 to 5; and A denotes a nitrogen atom or a methyne group.As a result, an azole derivative contained as an active ingredient in an agro-horticultural agent having an excellent controlling effect on diseases can be provided.